Ligand source activities (1 row/activity)





Ligands Receptor Assay information Chemical information
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name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Potency)
# tested GPCRs
(Potency)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI
101635584 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
1458 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
16136567 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
3794 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
91898963 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
CHEMBL525634 2548 26 None - 1 Human 10.4 pEC50 = 10.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL None None None None 10.1021/jm801332q
10010118 100952 0 None - 1 Human 10.3 pEC50 = 10.3 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL297494 100952 0 None - 1 Human 10.3 pEC50 = 10.3 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL2372767 208530 0 None - 1 Human 9.8 pEC50 = 9.8 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](N)Cc1ccccc1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](CCSC)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)O 10.1021/jm0304865
11181688 100852 0 None - 1 Human 9.7 pEC50 = 9.7 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 721 13 4 11 1.5 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL296748 100852 0 None - 1 Human 9.7 pEC50 = 9.7 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 721 13 4 11 1.5 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
23728661 88388 0 None - 1 Human 9.6 pEC50 = 9.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 Cc1cc(N(C)C(=O)c2ccc(-c3cccc(F)c3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364292 88388 0 None - 1 Human 9.6 pEC50 = 9.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 Cc1cc(N(C)C(=O)c2ccc(-c3cccc(F)c3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
23728772 88409 0 None - 1 Human 9.6 pEC50 = 9.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 448 6 1 5 4.4 Cc1cc(N(C)C(=O)c2ccc(Oc3ccc(F)cc3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364312 88409 0 None - 1 Human 9.6 pEC50 = 9.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 448 6 1 5 4.4 Cc1cc(N(C)C(=O)c2ccc(Oc3ccc(F)cc3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
23728875 88414 0 None - 1 Human 9.5 pEC50 = 9.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 468 6 1 5 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)cc2Cl)CCN1 10.6019/CHEMBL2364262
CHEMBL2364317 88414 0 None - 1 Human 9.5 pEC50 = 9.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 468 6 1 5 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)cc2Cl)CCN1 10.6019/CHEMBL2364262
10010118 100952 0 None - 1 Human 9.5 pEC50 = 9.5 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL297494 100952 0 None - 1 Human 9.5 pEC50 = 9.5 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
23728544 88381 0 None - 1 Human 9.4 pEC50 = 9.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 446 5 1 4 4.7 Cc1nc(-c2ccc(F)cc2)ccc1C(=O)N(C)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364285 88381 0 None - 1 Human 9.4 pEC50 = 9.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 446 5 1 4 4.7 Cc1nc(-c2ccc(F)cc2)ccc1C(=O)N(C)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.6019/CHEMBL2364262
23728806 88415 0 None - 1 Human 9.4 pEC50 = 9.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 448 7 1 5 4.5 CCN(C(=O)c1ccc(Oc2ccc(F)cc2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364318 88415 0 None - 1 Human 9.4 pEC50 = 9.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 448 7 1 5 4.5 CCN(C(=O)c1ccc(Oc2ccc(F)cc2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
23729106 88378 0 None - 1 Human 9.2 pEC50 = 9.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 Cc1nc(-c2cccc(F)c2)ccc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364282 88378 0 None - 1 Human 9.2 pEC50 = 9.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 Cc1nc(-c2cccc(F)c2)ccc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
23728770 88398 0 None - 1 Human 9.1 pEC50 = 9.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 6 1 4 4.3 CCN(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364302 88398 0 None - 1 Human 9.1 pEC50 = 9.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 6 1 4 4.3 CCN(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
16749783 88427 0 None - 1 Human 9.1 pEC50 = 9.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 450 6 1 7 3.2 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4cccc(F)c4)CC3)n2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364330 88427 0 None - 1 Human 9.1 pEC50 = 9.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 450 6 1 7 3.2 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4cccc(F)c4)CC3)n2)CCN1 10.6019/CHEMBL2364262
101635584 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
1458 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
16136567 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
3794 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
91898963 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
CHEMBL525634 2548 26 None - 1 Human 9.0 pEC50 = 9.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL None None None None 10.1016/j.bmcl.2022.128554
23728693 88393 0 None - 1 Human 9.0 pEC50 = 9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 434 6 1 5 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(F)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364297 88393 0 None - 1 Human 9.0 pEC50 = 9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 434 6 1 5 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(F)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
16040758 88423 0 None - 1 Human 9.0 pEC50 = 9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 487 6 2 5 4.4 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364326 88423 0 None - 1 Human 9.0 pEC50 = 9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 487 6 2 5 4.4 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23729022 88377 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364281 88377 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728731 88397 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 436 5 1 4 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)cc2F)CCN1 10.6019/CHEMBL2364262
CHEMBL2364301 88397 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 436 5 1 4 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)cc2F)CCN1 10.6019/CHEMBL2364262
16749753 88426 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4ccc(F)cc4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364329 88426 0 None - 1 Human 8.9 pEC50 = 8.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4ccc(F)cc4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
23729025 88373 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364277 88373 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728541 88380 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 439 5 1 5 4.0 Cc1nc(-c2cccc(C#N)c2)ccc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364284 88380 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 439 5 1 5 4.0 Cc1nc(-c2cccc(C#N)c2)ccc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
23728581 88384 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 5 1 5 3.7 Cc1nc(-c2ccc(F)cc2)ncc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364288 88384 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 5 1 5 3.7 Cc1nc(-c2ccc(F)cc2)ncc1C(=O)N(C)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
42623380 88412 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.8 Cc1cc(NS(=O)(=O)c2ccc(-c3ccc(F)cc3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364315 88412 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.8 Cc1cc(NS(=O)(=O)c2ccc(-c3ccc(F)cc3)nc2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
42623463 88417 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 508 6 2 5 4.5 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2C(F)(F)F)CCN1 10.6019/CHEMBL2364262
CHEMBL2364320 88417 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 508 6 2 5 4.5 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2C(F)(F)F)CCN1 10.6019/CHEMBL2364262
56959013 190795 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 534 9 2 5 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CC(=O)NC(C)C)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5192530 190795 0 None - 1 Human 8.8 pEC50 = 8.8 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 534 9 2 5 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CC(=O)NC(C)C)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
89723534 189923 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 499 7 2 5 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(Cl)c(CO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5179573 189923 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 499 7 2 5 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(Cl)c(CO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
16041119 177819 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465917 177819 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
23728546 88382 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364286 88382 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 5 1 4 4.3 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
59262141 88395 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 441 6 1 6 3.8 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(C#N)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364299 88395 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 441 6 1 6 3.8 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(C#N)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
23728915 88418 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 449 6 1 6 3.8 Cc1cc(N(C)C(=O)c2ccc(Oc3ccc(F)cc3)nc2)ncc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364321 88418 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 449 6 1 6 3.8 Cc1cc(N(C)C(=O)c2ccc(Oc3ccc(F)cc3)nc2)ncc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
16122912 88420 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 463 6 2 7 3.7 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Nc4ccc(F)cc4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364323 88420 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 463 6 2 7 3.7 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Nc4ccc(F)cc4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
15984938 186195 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.1021/jm801332q
CHEMBL489094 186195 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.1021/jm801332q
46882521 5620 0 None 158 2 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 458 6 2 4 4.5 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(-c2ccccc2)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078207 5620 0 None 158 2 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 458 6 2 4 4.5 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(-c2ccccc2)cc1 10.1016/j.bmcl.2009.09.027
16752689 187774 0 None 5 3 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.072
CHEMBL501315 187774 0 None 5 3 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.072
16752689 187774 0 None 5 3 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL501315 187774 0 None 5 3 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
16040941 177703 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2F)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465094 177703 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2F)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
11993730 177822 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 500 6 1 4 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465925 177822 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 500 6 1 4 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570412 177836 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 505 8 1 5 4.0 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)CS(=O)(=O)c3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465948 177836 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 505 8 1 5 4.0 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)CS(=O)(=O)c3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570489 182467 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 499 6 1 3 5.8 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL479418 182467 0 None - 1 Human 8.0 pEC50 = 8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 499 6 1 3 5.8 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15985000 88364 0 None - 1 Human 8.0 pEC50 = 8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C(F)(F)F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364268 88364 0 None - 1 Human 8.0 pEC50 = 8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C(F)(F)F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
44571939 180024 0 None - 1 Human 7.0 pEC50 = 7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 540 10 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL475467 180024 0 None - 1 Human 7.0 pEC50 = 7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 540 10 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
52946479 17034 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 794 9 7 15 1.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256547 17034 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 794 9 7 15 1.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
52946426 17042 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 778 9 6 14 2.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1256558 17042 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 778 9 6 14 2.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
54584627 61883 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 794 9 7 15 1.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778155 61883 0 None - 1 Rabbit 7.0 pEC50 = 7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 794 9 7 15 1.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
42623375 88389 0 None - 1 Human 7.0 pEC50 = 7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 429 6 2 6 2.7 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(N4CCCCC4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364293 88389 0 None - 1 Human 7.0 pEC50 = 7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 429 6 2 6 2.7 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(N4CCCCC4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
44570112 176845 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 513 7 2 6 4.7 COc1ccc(NC2CCN(C(=O)c3ncccc3-c3ccc(CN4C[C@H](C)N[C@H](C)C4)cc3)CC2)cc1 10.1016/j.bmcl.2008.10.072
CHEMBL463861 176845 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 513 7 2 6 4.7 COc1ccc(NC2CCN(C(=O)c3ncccc3-c3ccc(CN4C[C@H](C)N[C@H](C)C4)cc3)CC2)cc1 10.1016/j.bmcl.2008.10.072
44570452 189230 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 446 7 1 5 4.0 Cc1cc(CC(=O)N(C)Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)on1 10.1016/j.bmcl.2008.10.072
CHEMBL516551 189230 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 446 7 1 5 4.0 Cc1cc(CC(=O)N(C)Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)on1 10.1016/j.bmcl.2008.10.072
44571990 189094 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 533 11 1 4 5.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)Cc2ccccc2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL515434 189094 0 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 533 11 1 4 5.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)Cc2ccccc2)c1 10.1016/j.bmcl.2008.10.071
1048 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmc.2010.08.035
1048 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
12560 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmc.2010.08.035
12560 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
1456 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmc.2010.08.035
1456 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL532 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmc.2010.08.035
CHEMBL532 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
DB00199 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmc.2010.08.035
DB00199 1548 72 None 5 2 Human 6.0 pEC50 = 6 Functional
Agonist activity at motilin receptorAgonist activity at motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
52944056 17038 0 None - 1 Rabbit 7.0 pEC50 = 7.0 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 748 8 5 13 3.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1256554 17038 0 None - 1 Rabbit 7.0 pEC50 = 7.0 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 748 8 5 13 3.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
168288449 191090 0 None - 1 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 475 7 1 6 4.0 CC[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccnc(C#N)c4)CC3)cc2C)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5196819 191090 0 None - 1 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 475 7 1 6 4.0 CC[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccnc(C#N)c4)CC3)cc2C)CCN1 10.1016/j.bmcl.2022.128554
15984937 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1021/jm801332q
4035 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1021/jm801332q
CHEMBL489095 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1021/jm801332q
DB12567 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1021/jm801332q
46882713 5639 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 395 4 1 3 4.2 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)cc2)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078345 5639 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 395 4 1 3 4.2 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)cc2)cc1 10.1016/j.bmcl.2009.09.027
15984136 88359 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364263 88359 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
15984135 88367 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 442 6 2 4 3.4 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364271 88367 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 442 6 2 4 3.4 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
15984138 88369 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 6 1 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364273 88369 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 432 6 1 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728769 88404 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 446 6 1 4 4.7 CC(C)N(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364308 88404 0 None - 1 Human 7.9 pEC50 = 7.9 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 446 6 1 4 4.7 CC(C)N(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
54583621 61867 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 760 8 5 13 3.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778046 61867 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 760 8 5 13 3.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542067 197046 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 865 13 7 16 1.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCCO)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL582871 197046 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 865 13 7 16 1.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCCO)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542068 197047 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 905 12 6 16 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CCOCC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL582872 197047 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 905 12 6 16 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CCOCC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
1048 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2010.08.030
12560 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2010.08.030
1456 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL532 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2010.08.030
DB00199 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2010.08.030
1048 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
1048 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm901107f
12560 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
12560 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm901107f
1456 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
1456 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm901107f
CHEMBL532 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL532 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm901107f
DB00199 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2011.04.078
DB00199 1548 72 None -5 2 Rabbit 5.9 pEC50 = 5.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm901107f
46882672 5544 0 None - 1 Human 6.9 pEC50 = 6.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 357 6 1 3 3.7 CCCCc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1077736 5544 0 None - 1 Human 6.9 pEC50 = 6.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 357 6 1 3 3.7 CCCCc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
46882711 5637 0 None - 1 Human 5.9 pEC50 = 5.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 351 3 1 3 3.5 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc2ccccc2c1 10.1016/j.bmcl.2009.09.027
CHEMBL1078343 5637 0 None - 1 Human 5.9 pEC50 = 5.9 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 351 3 1 3 3.5 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc2ccccc2c1 10.1016/j.bmcl.2009.09.027
54583623 61869 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 9 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778049 61869 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 9 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542518 196475 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 863 12 6 15 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL574848 196475 0 None - 1 Rabbit 6.9 pEC50 = 6.9 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 863 12 6 15 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
16041292 183019 0 None 31 2 Human 7.8 pEC50 = 7.8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 490 6 2 6 3.9 C[C@H]1CN(Cc2ccc(-n3ccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL480219 183019 0 None 31 2 Human 7.8 pEC50 = 7.8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 490 6 2 6 3.9 C[C@H]1CN(Cc2ccc(-n3ccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984137 88368 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364272 88368 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
15984184 88370 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364274 88370 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728771 88410 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 462 8 1 5 4.0 COCCN(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364313 88410 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 462 8 1 5 4.0 COCCN(C(=O)c1ccc(-c2cccc(F)c2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
59262173 88413 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 478 9 1 6 4.1 COCCN(C(=O)c1ccc(Oc2ccc(F)cc2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364316 88413 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 478 9 1 6 4.1 COCCN(C(=O)c1ccc(Oc2ccc(F)cc2)nc1)c1ccc(CN2CCN[C@@H](C)C2)cc1 10.6019/CHEMBL2364262
15984243 88429 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 6 2 4 4.2 CC(C(=O)N1CCC(Nc2cccc(F)c2)CC1)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.6019/CHEMBL2364262
CHEMBL2364332 88429 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 6 2 4 4.2 CC(C(=O)N1CCC(Nc2cccc(F)c2)CC1)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.6019/CHEMBL2364262
44542965 197081 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 891 15 6 15 3.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL583097 197081 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 891 15 6 15 3.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542966 196233 0 None - 1 Rabbit 5.8 pEC50 = 5.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 12 6 15 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCc2ccc(C(=O)NC)cc2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL572998 196233 0 None - 1 Rabbit 5.8 pEC50 = 5.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 12 6 15 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCc2ccc(C(=O)NC)cc2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
46882754 5629 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 403 4 1 5 3.3 N#Cc1ccc(-c2ccc(S(=O)(=O)Cc3ccc4c(c3)CCNCC4)cn2)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078269 5629 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 403 4 1 5 3.3 N#Cc1ccc(-c2ccc(S(=O)(=O)Cc3ccc4c(c3)CCNCC4)cn2)cc1 10.1016/j.bmcl.2009.09.027
46882794 5656 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 360 5 1 5 2.5 CC(C)Oc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
CHEMBL1078461 5656 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 360 5 1 5 2.5 CC(C)Oc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
42623379 88411 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.9 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364314 88411 0 None - 1 Human 6.8 pEC50 = 6.8 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.9 C[C@H]1CN(Cc2ccc(NS(=O)(=O)c3ccc(-c4ccc(F)cc4)nc3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
46882623 5759 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 388 4 2 6 1.4 O=S(=O)(Nc1ccc2c(c1)CCNCC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079260 5759 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 388 4 2 6 1.4 O=S(=O)(Nc1ccc2c(c1)CCNCC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
9863611 96469 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 358 6 2 3 3.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL266018 96469 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 358 6 2 3 3.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
44571376 183469 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 510 9 2 3 5.8 O=C(NC1CCCCC1)N(CCc1ccccc1)Cc1ccccc1-c1cccc(CN2CCNCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL482307 183469 0 None - 1 Human 5.8 pEC50 = 5.8 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 510 9 2 3 5.8 O=C(NC1CCCCC1)N(CCc1ccccc1)Cc1ccccc1-c1cccc(CN2CCNCC2)c1 10.1016/j.bmcl.2008.10.071
44542519 197236 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 903 12 6 15 3.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCC(F)(F)F)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL584553 197236 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 903 12 6 15 3.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCC(F)(F)F)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
54583624 61872 0 None - 1 Rabbit 7.8 pEC50 = 7.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 819 11 5 14 3.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778052 61872 0 None - 1 Rabbit 7.8 pEC50 = 7.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 819 11 5 14 3.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
168274082 189691 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 459 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5175905 189691 0 None - 1 Human 7.8 pEC50 = 7.8 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 459 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1016/j.bmcl.2022.128554
52941569 17040 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 9 6 14 2.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1256556 17040 0 None - 1 Rabbit 6.8 pEC50 = 6.8 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 9 6 14 2.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
15984134 192658 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1021/jm801332q
CHEMBL523933 192658 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 424 6 2 4 3.3 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1021/jm801332q
46882712 5638 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 411 4 1 3 4.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(Cl)cc2)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078344 5638 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 411 4 1 3 4.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(Cl)cc2)cc1 10.1016/j.bmcl.2009.09.027
46882797 5659 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 411 5 2 5 3.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(Nc2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078464 5659 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 411 5 2 5 3.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(Nc2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
44570450 177155 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 534 9 2 5 3.8 Cc1ccc(S(=O)(=O)NCC(=O)N(C)Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)cc1 10.1016/j.bmcl.2008.10.072
CHEMBL464247 177155 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 534 9 2 5 3.8 Cc1ccc(S(=O)(=O)NCC(=O)N(C)Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)cc1 10.1016/j.bmcl.2008.10.072
16041481 178217 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL469098 178217 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
16040587 178794 0 None 14 2 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL473921 178794 0 None 14 2 Human 7.7 pEC50 = 7.7 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984997 88362 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364266 88362 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
59262241 88407 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 495 6 1 4 5.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(C(=O)c4ccc(C(F)(F)F)cc4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364310 88407 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 495 6 1 4 5.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(C(=O)c4ccc(C(F)(F)F)cc4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
42623461 88419 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.8 Cc1cc(NS(=O)(=O)c2cncc(-c3ccc(F)cc3)c2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364322 88419 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 6 2 5 3.8 Cc1cc(NS(=O)(=O)c2cncc(-c3ccc(F)cc3)c2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
16041291 88422 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 555 7 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3S(=O)(=O)N3CCC(Nc4ccccc4F)CC3)cc2F)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364325 88422 0 None - 1 Human 7.7 pEC50 = 7.7 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 555 7 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3S(=O)(=O)N3CCC(Nc4ccccc4F)CC3)cc2F)C[C@@H](C)N1 10.6019/CHEMBL2364262
54581677 61873 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 833 11 4 14 3.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778053 61873 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 833 11 4 14 3.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL388812 210663 0 None - 1 Rat 5.7 pEC50 = 5.7 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None CC(C)c1nc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1016/j.bmc.2006.09.045
46882302 5674 0 None - 1 Human 6.7 pEC50 = 6.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 426 7 1 3 5.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(C2CCCC2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078558 5674 0 None - 1 Human 6.7 pEC50 = 6.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 426 7 1 3 5.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(C2CCCC2)CC3)cc1 10.1016/j.bmcl.2009.09.027
46882755 5630 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 439 5 2 5 3.1 O=C(Nc1ccc(F)cc1)c1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
CHEMBL1078270 5630 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 439 5 2 5 3.1 O=C(Nc1ccc(F)cc1)c1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
46882303 5677 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 442 8 1 4 4.3 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(CC2CCOC2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078586 5677 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 442 8 1 4 4.3 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(CC2CCOC2)CC3)cc1 10.1016/j.bmcl.2009.09.027
89723541 189921 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 473 6 1 4 4.9 C[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2Cl)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5179543 189921 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 473 6 1 4 4.9 C[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2Cl)CCN1 10.1016/j.bmcl.2022.128554
56960874 190510 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 453 6 1 4 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cc3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5187928 190510 0 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 453 6 1 4 4.5 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cc3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL223972 207692 0 None 2 2 Rat 8.6 pEC50 = 8.6 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None Cn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
46882458 5886 0 None 31 2 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 438 8 2 4 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1080046 5886 0 None 31 2 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 438 8 2 4 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44570527 190375 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 500 6 2 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL518618 190375 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 500 6 2 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984186 88372 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C(F)(F)F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364276 88372 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C(F)(F)F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23729107 88379 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 6 1 4 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(F)c4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364283 88379 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 6 1 4 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(F)c4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
16749782 88425 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4cccc(F)c4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364328 88425 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4cccc(F)c4)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
89723498 190801 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 492 9 2 5 5.0 CCOCc1cccc(N[C@H]2CC[C@H](C(=O)N(C)c3ccc(CN4CCN[C@@H](C)C4)c(C)c3)CC2)c1 10.1016/j.bmcl.2022.128554
CHEMBL5192584 190801 0 None - 1 Human 8.6 pEC50 = 8.6 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 492 9 2 5 5.0 CCOCc1cccc(N[C@H]2CC[C@H](C(=O)N(C)c3ccc(CN4CCN[C@@H](C)C4)c(C)c3)CC2)c1 10.1016/j.bmcl.2022.128554
CHEMBL390942 210691 0 None 5 2 Rat 8.6 pEC50 = 8.6 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None CCn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
CHEMBL389037 210666 0 None 8 2 Rat 5.7 pEC50 = 5.7 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1cn(Cc2ccccc2)cn1)NC(=O)[C@@H]1CCCC(=O)N1 10.1016/j.bmc.2006.09.045
52942786 17026 0 None - 1 Rabbit 5.7 pEC50 = 5.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 790 9 6 14 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC3(C)CC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256538 17026 0 None - 1 Rabbit 5.7 pEC50 = 5.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 790 9 6 14 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC3(C)CC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
52943975 17029 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256542 17029 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
54586525 61875 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778055 61875 0 None - 1 Rabbit 6.7 pEC50 = 6.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542215 195446 0 None - 1 Rabbit 5.7 pEC50 = 5.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 12 6 15 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCc2cccc(C(=O)NC)c2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL567808 195446 0 None - 1 Rabbit 5.7 pEC50 = 5.7 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 12 6 15 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCc2cccc(C(=O)NC)c2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
54582662 61870 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 778 9 6 14 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778050 61870 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 778 9 6 14 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)(C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
168278248 190498 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 453 6 1 4 4.5 Cc1cc(CN2CCN[C@@H](C)C2)ccc1N(C)C(=O)[C@H]1CC[C@H](Oc2ccc(F)cc2)CC1 10.1016/j.bmcl.2022.128554
CHEMBL5187776 190498 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 453 6 1 4 4.5 Cc1cc(CN2CCN[C@@H](C)C2)ccc1N(C)C(=O)[C@H]1CC[C@H](Oc2ccc(F)cc2)CC1 10.1016/j.bmcl.2022.128554
52942785 17024 0 None - 1 Rabbit 5.6 pEC50 = 5.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 9 6 14 2.5 C=C(C)CN(C)[C@H]1C[C@@H](C)O[C@@H](O[C@@H]2[C@@H](C)[C@H](O[C@@H]3C[C@@](C)(OC)[C@@H](O)[C@H](C)O3)[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)[C@@H](O)[C@H](C)C[C@@]2(C)O)[C@@H]1O 10.1016/j.bmcl.2010.08.030
CHEMBL1256536 17024 0 None - 1 Rabbit 5.6 pEC50 = 5.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 9 6 14 2.5 C=C(C)CN(C)[C@H]1C[C@@H](C)O[C@@H](O[C@@H]2[C@@H](C)[C@H](O[C@@H]3C[C@@](C)(OC)[C@@H](O)[C@H](C)O3)[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)[C@@H](O)[C@H](C)C[C@@]2(C)O)[C@@H]1O 10.1016/j.bmcl.2010.08.030
16088034 197078 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 899 12 6 17 2.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)Nc2ccncn2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL583094 197078 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 899 12 6 17 2.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)Nc2ccncn2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
15984241 178933 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 7 2 4 3.7 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1021/jm801332q
CHEMBL474130 178933 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 7 2 4 3.7 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1 10.1021/jm801332q
46882714 5600 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 413 4 1 3 4.3 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)c(F)c2)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1077991 5600 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 413 4 1 3 4.3 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)c(F)c2)cc1 10.1016/j.bmcl.2009.09.027
15984998 88363 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364267 88363 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 6 1 4 3.2 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
15984187 88366 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 7 2 5 3.3 COc1cc(CC(=O)N2CCC(Nc3cccc(F)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
CHEMBL2364270 88366 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 454 7 2 5 3.3 COc1cc(CC(=O)N2CCC(Nc3cccc(F)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.6019/CHEMBL2364262
16749728 88421 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 479 6 2 6 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3N3CCC(Nc4ccc(F)cc4)CC3)s2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364324 88421 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 479 6 2 6 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3N3CCC(Nc4ccc(F)cc4)CC3)s2)C[C@@H](C)N1 10.6019/CHEMBL2364262
15984319 88430 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 466 6 2 4 4.4 C[C@H]1CN(Cc2ccc(C(C)(C)C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364333 88430 0 None - 1 Human 7.6 pEC50 = 7.6 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 466 6 2 4 4.4 C[C@H]1CN(Cc2ccc(C(C)(C)C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
52948855 17035 0 None - 1 Rabbit 5.6 pEC50 = 5.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 795 10 8 16 0.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(O)CO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256548 17035 0 None - 1 Rabbit 5.6 pEC50 = 5.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 795 10 8 16 0.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(O)CO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
44593551 37519 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 549 12 1 5 5.4 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)COc2ccccc2)c1 10.1016/j.bmcl.2008.10.072
CHEMBL14581 37519 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 549 12 1 5 5.4 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)COc2ccccc2)c1 10.1016/j.bmcl.2008.10.072
44570451 189900 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 421 8 1 3 4.9 CC(C)CCC(=O)N(C)Cc1ccccc1-c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1016/j.bmcl.2008.10.072
CHEMBL517934 189900 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 421 8 1 3 4.9 CC(C)CCC(=O)N(C)Cc1ccccc1-c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1016/j.bmcl.2008.10.072
44593551 37519 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 549 12 1 5 5.4 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)COc2ccccc2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL14581 37519 0 None - 1 Human 6.6 pEC50 = 6.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 549 12 1 5 5.4 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)COc2ccccc2)c1 10.1016/j.bmcl.2008.10.071
46882350 5714 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 454 8 1 4 5.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cccs2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078882 5714 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 454 8 1 4 5.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cccs2)CC3)cc1 10.1016/j.bmcl.2009.09.027
46882624 5760 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 372 6 1 3 3.5 CCCCc1ccc(S(=O)(=O)N(C)c2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079261 5760 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 372 6 1 3 3.5 CCCCc1ccc(S(=O)(=O)N(C)c2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
46882625 5761 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 388 4 2 6 1.4 O=S(=O)(Nc1ccc(N2CCOCC2)nc1)c1ccc2c(c1)CCNCC2 10.1016/j.bmcl.2009.09.027
CHEMBL1079262 5761 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 388 4 2 6 1.4 O=S(=O)(Nc1ccc(N2CCOCC2)nc1)c1ccc2c(c1)CCNCC2 10.1016/j.bmcl.2009.09.027
46882460 6218 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 396 6 2 4 3.0 O=S(=O)(Cc1ccccc1)Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2 10.1016/j.bmcl.2009.09.027
CHEMBL1081859 6218 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 396 6 2 4 3.0 O=S(=O)(Cc1ccccc1)Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2 10.1016/j.bmcl.2009.09.027
44570013 176283 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 526 7 3 6 3.7 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(C(N)=O)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL461446 176283 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 526 7 3 6 3.7 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(C(N)=O)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570608 190130 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 493 6 2 5 4.1 C[C@H]1CN(Cc2ccc(N3CCCC3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL518261 190130 0 None - 1 Human 5.6 pEC50 = 5.6 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 493 6 2 5 4.1 C[C@H]1CN(Cc2ccc(N3CCCC3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
52947632 17022 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256534 17022 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
44542667 197232 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542667 197232 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL584549 197232 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL584549 197232 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 764 8 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542964 197080 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 877 14 6 15 3.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL583096 197080 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 877 14 6 15 3.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542520 197045 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 875 12 6 15 3.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CCC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL582870 197045 0 None - 1 Rabbit 7.6 pEC50 = 7.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 875 12 6 15 3.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CCC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
52942801 17041 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 9 6 14 2.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1256557 17041 0 None - 1 Rabbit 6.6 pEC50 = 6.6 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 764 9 6 14 2.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL224525 207693 0 None 13 2 Rat 7.5 pEC50 = 7.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None CCCc1nc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1016/j.bmc.2006.09.045
2139 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
2316 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
3836 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
638678 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
CHEMBL1472 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
DB09421 3782 51 None -57 3 Rat 8.5 pEC50 = 8.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
46882395 5751 0 None 1 2 Human 8.5 pEC50 = 8.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 2 4 4.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2[nH]cnc2C)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079186 5751 0 None 1 2 Human 8.5 pEC50 = 8.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 2 4 4.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2[nH]cnc2C)CC3)cc1 10.1016/j.bmcl.2009.09.027
44570411 177781 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 473 8 1 4 5.3 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)CSc3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465271 177781 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 473 8 1 4 5.3 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)CSc3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984185 88371 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364275 88371 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728695 88391 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 441 6 1 6 3.8 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(C#N)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364295 88391 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 441 6 1 6 3.8 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4cccc(C#N)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728694 88394 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 6 1 5 4.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)c(F)c2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364298 88394 0 None - 1 Human 8.5 pEC50 = 8.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 6 1 5 4.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)c(F)c2)CCN1 10.6019/CHEMBL2364262
16040587 178794 0 None 14 2 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
CHEMBL473921 178794 0 None 14 2 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
15984939 186260 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 431 6 2 5 3.0 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)CCN1 10.1021/jm801332q
CHEMBL489480 186260 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 431 6 2 5 3.0 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C#N)c4)CC3)cc2)CCN1 10.1021/jm801332q
46882522 5621 0 None 39 2 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 440 7 2 5 3.6 CC(C)Oc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078208 5621 0 None 39 2 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 440 7 2 5 3.6 CC(C)Oc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
16040939 190101 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2F)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL518229 190101 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 519 6 2 5 4.9 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2F)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
52946425 17039 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 760 8 5 13 3.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1256555 17039 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 760 8 5 13 3.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
44541929 197044 0 None - 1 Rabbit 7.5 pEC50 = 7.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 861 12 6 15 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL582869 197044 0 None - 1 Rabbit 7.5 pEC50 = 7.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 861 12 6 15 2.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC2CC2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
15984242 186221 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 452 6 2 4 4.2 CC(C(=O)N1CCC(Nc2ccc(F)cc2)CC1)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1021/jm801332q
CHEMBL489297 186221 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 452 6 2 4 4.2 CC(C(=O)N1CCC(Nc2ccc(F)cc2)CC1)c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1021/jm801332q
15984318 186259 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 466 6 2 4 4.4 C[C@H]1CN(Cc2ccc(C(C)(C)C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
CHEMBL489479 186259 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 466 6 2 4 4.4 C[C@H]1CN(Cc2ccc(C(C)(C)C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
46882583 5664 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 453 5 2 6 2.6 CN1CCOc2cc(S(=O)(=O)Nc3ccc4c(c3)CCN(Cc3cc[nH]n3)CC4)ccc21 10.1016/j.bmcl.2009.09.027
CHEMBL1078491 5664 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 453 5 2 6 2.6 CN1CCOc2cc(S(=O)(=O)Nc3ccc4c(c3)CCN(Cc3cc[nH]n3)CC4)ccc21 10.1016/j.bmcl.2009.09.027
44570365 177584 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 475 8 1 4 4.7 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)COc3ccc(F)cc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL464909 177584 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 475 8 1 4 4.7 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)COc3ccc(F)cc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984994 88360 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364264 88360 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 431 6 2 5 3.0 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728774 88399 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 435 6 1 6 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)nc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364303 88399 0 None - 1 Human 7.5 pEC50 = 7.5 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 435 6 1 6 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccc(F)cc4)nc3)nc2)CCN1 10.6019/CHEMBL2364262
52950053 17025 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 9 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC3CC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256537 17025 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 9 6 14 2.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC3CC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
46882710 5636 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 357 3 1 3 3.6 CC(C)(C)c1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078342 5636 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 357 3 1 3 3.6 CC(C)(C)c1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cc1 10.1016/j.bmcl.2009.09.027
46882457 5859 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 1 5 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cncn2C)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079868 5859 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 1 5 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cncn2C)CC3)cc1 10.1016/j.bmcl.2009.09.027
44572092 179954 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 487 14 0 4 5.0 COCCCN(Cc1ccccc1-c1ccc(CN(C)CCN(C)C)cc1)C(=O)Cc1ccccc1 10.1016/j.bmcl.2008.10.071
CHEMBL475380 179954 0 None - 1 Human 5.5 pEC50 = 5.5 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 487 14 0 4 5.0 COCCCN(Cc1ccccc1-c1ccc(CN(C)CCN(C)C)cc1)C(=O)Cc1ccccc1 10.1016/j.bmcl.2008.10.071
CHEMBL224655 207695 0 None - 1 Rat 5.5 pEC50 = 5.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None CC(C)(C)c1nc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1016/j.bmc.2006.09.045
CHEMBL388528 210661 0 None 15 2 Rat 6.5 pEC50 = 6.5 Functional
Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityAgonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity
ChEMBL None None None C=CCn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
89872388 189883 0 None - 1 Human 6.5 pEC50 = 6.5 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 467 7 1 4 4.9 CC[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2C)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5179060 189883 0 None - 1 Human 6.5 pEC50 = 6.5 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 467 7 1 4 4.9 CC[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2C)CCN1 10.1016/j.bmcl.2022.128554
52941620 17027 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 8 6 14 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256539 17027 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 776 8 6 14 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
54587558 61874 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 776 8 6 14 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778054 61874 0 None - 1 Rabbit 6.5 pEC50 = 6.5 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 776 8 6 14 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
54580662 61871 0 None - 1 Rabbit 7.4 pEC50 = 7.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 805 11 5 14 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778051 61871 0 None - 1 Rabbit 7.4 pEC50 = 7.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 805 11 5 14 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
52942788 17032 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256545 17032 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
54584626 61882 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778154 61882 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
52946408 17023 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 778 9 6 14 2.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256535 17023 0 None - 1 Rabbit 6.4 pEC50 = 6.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 778 9 6 14 2.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
52942789 17036 0 None - 1 Rabbit 5.4 pEC50 = 5.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 767 9 6 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCF)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256549 17036 0 None - 1 Rabbit 5.4 pEC50 = 5.4 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 767 9 6 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCF)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
15604512 179596 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 6 2 4 3.7 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
CHEMBL474934 179596 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 6 2 4 3.7 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
46882795 5657 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 374 6 1 5 2.8 CC(C)COc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
CHEMBL1078462 5657 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 374 6 1 5 2.8 CC(C)COc1ccc(S(=O)(=O)Cc2ccc3c(c2)CCNCC3)cn1 10.1016/j.bmcl.2009.09.027
46882520 5764 0 None 1 2 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 430 5 2 4 3.8 Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1Cl 10.1016/j.bmcl.2009.09.027
CHEMBL1079311 5764 0 None 1 2 Human 7.4 pEC50 = 7.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 430 5 2 4 3.8 Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1Cl 10.1016/j.bmcl.2009.09.027
23729060 88374 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 417 5 1 3 4.6 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364278 88374 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 417 5 1 3 4.6 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)cc3)cc2)CCN1 10.6019/CHEMBL2364262
23728733 88400 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 445 6 1 5 3.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4cccc(C#N)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364304 88400 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 445 6 1 5 3.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4cccc(C#N)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728840 88405 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(C#N)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364309 88405 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(C#N)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
15984239 88428 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 7 2 4 4.0 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364331 88428 0 None - 1 Human 7.4 pEC50 = 7.4 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 452 7 2 4 4.0 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.6019/CHEMBL2364262
44571375 189073 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 539 10 2 3 7.0 COc1cccc(CCN(Cc2ccccc2-c2ccc(CC3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL515275 189073 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 539 10 2 3 7.0 COc1cccc(CCN(Cc2ccccc2-c2ccc(CC3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
44593552 177723 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 487 12 1 5 4.2 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)COc1ccccc1 10.1016/j.bmcl.2008.10.072
CHEMBL465104 177723 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 487 12 1 5 4.2 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)COc1ccccc1 10.1016/j.bmcl.2008.10.072
44570568 183310 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 507 6 2 6 4.8 C[C@H]1CN(Cc2cnc(-c3ccccc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)s2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL481192 183310 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 507 6 2 6 4.8 C[C@H]1CN(Cc2cnc(-c3ccccc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)s2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44593552 177723 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 487 12 1 5 4.2 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)COc1ccccc1 10.1016/j.bmcl.2008.10.071
CHEMBL465104 177723 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 487 12 1 5 4.2 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)COc1ccccc1 10.1016/j.bmcl.2008.10.071
53322109 55961 0 None 1 2 Human 8.4 pEC50 = 8.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm0304865
CHEMBL1628277 55961 0 None 1 2 Human 8.4 pEC50 = 8.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm0304865
89723511 189441 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 507 8 2 5 4.7 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CC(C)(C)O)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5171964 189441 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 507 8 2 5 4.7 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CC(C)(C)O)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
56960875 190267 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 454 6 1 5 3.9 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cn3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5184722 190267 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 454 6 1 5 3.9 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cn3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
56961016 191103 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 479 8 2 5 3.9 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CCO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5196982 191103 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 479 8 2 5 3.9 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cccc(CCO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
1048 1548 72 None 5 2 Human 6.4 pEC50 = 6.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
12560 1548 72 None 5 2 Human 6.4 pEC50 = 6.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
1456 1548 72 None 5 2 Human 6.4 pEC50 = 6.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
CHEMBL532 1548 72 None 5 2 Human 6.4 pEC50 = 6.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
DB00199 1548 72 None 5 2 Human 6.4 pEC50 = 6.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
44292287 186987 0 None - 1 Human 5.4 pEC50 = 5.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 546 7 3 10 -0.0 NC(=O)[C@@H](Cc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL49464 186987 0 None - 1 Human 5.4 pEC50 = 5.4 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 546 7 3 10 -0.0 NC(=O)[C@@H](Cc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
89723443 189913 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 439 6 1 4 4.1 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cc3)CC2)ccc1CN1CCNCC1 10.1016/j.bmcl.2022.128554
CHEMBL5179463 189913 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 439 6 1 4 4.1 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)cc3)CC2)ccc1CN1CCNCC1 10.1016/j.bmcl.2022.128554
52950055 17033 0 None - 1 Rabbit 6.3 pEC50 = 6.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256546 17033 0 None - 1 Rabbit 6.3 pEC50 = 6.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 9 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C[C@@H](C)O)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
46882753 5628 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 396 4 1 4 3.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078268 5628 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 396 4 1 4 3.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
46882582 5663 0 None 125 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 466 5 2 5 3.9 CC1(C)CCc2cc(S(=O)(=O)Nc3ccc4c(c3)CCN(Cc3cc[nH]n3)CC4)ccc2O1 10.1016/j.bmcl.2009.09.027
CHEMBL1078490 5663 0 None 125 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 466 5 2 5 3.9 CC1(C)CCc2cc(S(=O)(=O)Nc3ccc4c(c3)CCN(Cc3cc[nH]n3)CC4)ccc2O1 10.1016/j.bmcl.2009.09.027
16041121 177704 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 531 7 2 6 4.8 COc1cc(-c2cccnc2C(=O)N2CCC(Nc3ccc(F)cc3)CC2)ccc1CN1C[C@H](C)N[C@H](C)C1 10.1016/j.bmcl.2008.10.072
CHEMBL465095 177704 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 531 7 2 6 4.8 COc1cc(-c2cccnc2C(=O)N2CCC(Nc3ccc(F)cc3)CC2)ccc1CN1C[C@H](C)N[C@H](C)C1 10.1016/j.bmcl.2008.10.072
44570491 182468 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 482 6 2 4 5.3 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccccc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL479419 182468 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 482 6 2 4 5.3 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccccc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
23729063 88375 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 438 6 1 4 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364279 88375 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 438 6 1 4 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4cccc(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23729103 88376 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccccc4F)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364280 88376 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccccc4F)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728578 88383 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 6 1 4 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccccc4F)cc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364287 88383 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 433 6 1 4 4.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccccc4F)cc3)cc2)CCN1 10.6019/CHEMBL2364262
23728582 88385 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 419 5 1 5 3.4 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3cnc(-c4ccc(F)cc4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364289 88385 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 419 5 1 5 3.4 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3cnc(-c4ccc(F)cc4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
57586303 88386 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 458 6 2 4 3.9 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2Cl)CCN1 10.6019/CHEMBL2364262
CHEMBL2364290 88386 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 458 6 2 4 3.9 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2Cl)CCN1 10.6019/CHEMBL2364262
11902 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 10.1016/j.bmcl.2022.128554
56960876 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5201797 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 10.1016/j.bmcl.2022.128554
89723482 191495 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 479 7 2 5 4.2 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cc(CO)ccc3C)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5203126 191495 0 None - 1 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 479 7 2 5 4.2 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3cc(CO)ccc3C)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
44542816 196382 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 879 14 6 16 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCCOC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL574205 196382 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 879 14 6 16 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCCOC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
1048 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm801332q
12560 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm801332q
1456 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm801332q
CHEMBL532 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm801332q
DB00199 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm801332q
15984238 188968 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 452 7 2 4 4.0 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
CHEMBL514475 188968 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 452 7 2 4 4.0 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm801332q
1048 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
12560 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
1456 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
CHEMBL532 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
DB00199 1548 72 None 5 2 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
46882393 5748 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 511 9 2 5 5.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2ccc(NC(C)=O)s2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079170 5748 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 511 9 2 5 5.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2ccc(NC(C)=O)s2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44571939 180024 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 540 10 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL475467 180024 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 540 10 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
44570409 177829 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 459 7 1 3 4.9 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)Cc3ccc(F)cc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465940 177829 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 459 7 1 3 4.9 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)Cc3ccc(F)cc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570492 183357 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 516 6 2 4 5.9 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccc(Cl)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL481575 183357 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 516 6 2 4 5.9 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Nc4ccc(Cl)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
16752689 187774 0 None 5 3 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.072
CHEMBL501315 187774 0 None 5 3 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.072
16041483 190317 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccccc4F)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL518540 190317 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccccc4F)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
46882671 5543 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 387 4 1 6 1.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1077735 5543 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 387 4 1 6 1.6 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
46882756 5673 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 412 5 1 5 3.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(Oc2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078555 5673 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 412 5 1 5 3.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(Oc2ccc(F)cc2)nc1 10.1016/j.bmcl.2009.09.027
46882349 5713 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 505 9 2 4 5.4 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cccc(NC(C)=O)c2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078881 5713 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 505 9 2 4 5.4 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cccc(NC(C)=O)c2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44571989 179627 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 478 10 2 4 4.6 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)NC1CCCCC1 10.1016/j.bmcl.2008.10.071
CHEMBL474978 179627 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 478 10 2 4 4.6 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)NC1CCCCC1 10.1016/j.bmcl.2008.10.071
44571373 179323 0 None - 1 Human 5.3 pEC50 = 5.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 526 9 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(N3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL474606 179323 0 None - 1 Human 5.3 pEC50 = 5.3 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 526 9 2 4 5.9 COc1cccc(CCN(Cc2ccccc2-c2ccc(N3CCNCC3)cc2)C(=O)NC2CCCCC2)c1 10.1016/j.bmcl.2008.10.071
44571940 180339 0 None - 1 Human 5.3 pEC50 = 5.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 415 9 2 4 4.1 COc1cccc(CCNCc2ccccc2-c2ccc(CN3CCNCC3)cc2)c1 10.1016/j.bmcl.2008.10.071
CHEMBL475808 180339 0 None - 1 Human 5.3 pEC50 = 5.3 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 415 9 2 4 4.1 COc1cccc(CCNCc2ccccc2-c2ccc(CN3CCNCC3)cc2)c1 10.1016/j.bmcl.2008.10.071
11993730 177822 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 500 6 1 4 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2022.128554
CHEMBL465925 177822 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 500 6 1 4 5.2 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Cc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2022.128554
44542367 196409 0 None - 1 Rabbit 6.3 pEC50 = 6.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 847 11 6 15 2.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL574429 196409 0 None - 1 Rabbit 6.3 pEC50 = 6.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 847 11 6 15 2.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3CCC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542368 197233 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 821 11 6 15 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542368 197233 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 821 11 6 15 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL584550 197233 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 821 11 6 15 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL584550 197233 0 None - 1 Rabbit 7.3 pEC50 = 7.3 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 821 11 6 15 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(N)=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
56960873 191110 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 439 6 1 4 4.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2)CCN1 10.1016/j.bmcl.2022.128554
CHEMBL5197045 191110 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 439 6 1 4 4.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)[C@H]3CC[C@H](Oc4ccc(F)cc4)CC3)cc2)CCN1 10.1016/j.bmcl.2022.128554
11398860 175461 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL45905 175461 0 None - 1 Human 6.3 pEC50 = 6.3 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
52947633 17028 0 None - 1 Rabbit 5.2 pEC50 = 5.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 777 8 6 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3COC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256540 17028 0 None - 1 Rabbit 5.2 pEC50 = 5.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 777 8 6 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C3COC3)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
45483679 196231 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 835 11 6 15 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
45483679 196231 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 835 11 6 15 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL572996 196231 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 835 11 6 15 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL572996 196231 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 835 11 6 15 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
54584601 61866 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 748 8 5 13 3.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778045 61866 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 748 8 5 13 3.4 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
45102708 5678 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 468 6 2 7 2.0 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078595 5678 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 468 6 2 7 2.0 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(N2CCOCC2)nc1 10.1016/j.bmcl.2009.09.027
16040940 176866 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL463881 176866 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
15984999 88365 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C(F)(F)F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364269 88365 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 474 6 2 4 4.1 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(C(F)(F)F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728692 88392 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 436 5 1 4 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)c(F)c2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364296 88392 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 436 5 1 4 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)nc3)c(F)c2)CCN1 10.6019/CHEMBL2364262
16749781 88424 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4ccccc4F)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
CHEMBL2364327 88424 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 464 6 1 7 3.6 C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4ccccc4F)CC3)n2)C[C@@H](C)N1 10.6019/CHEMBL2364262
54582661 61868 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 749 9 6 14 2.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL1778047 61868 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 749 9 6 14 2.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
15984240 178932 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 7 2 4 3.7 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.1021/jm801332q
CHEMBL474129 178932 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells assessed as increase in intracellular calcium by FLIPR assay
ChEMBL 438 7 2 4 3.7 C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1 10.1021/jm801332q
46882796 5658 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 385 4 1 5 2.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(N2CCCCC2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078463 5658 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 385 4 1 5 2.7 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(N2CCCCC2)nc1 10.1016/j.bmcl.2009.09.027
46882396 5752 0 None -3 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 2 4 4.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cnc(C)[nH]2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079187 5752 0 None -3 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 452 8 2 4 4.5 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cnc(C)[nH]2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44570528 183014 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 513 6 1 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(C(=O)c4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL480210 183014 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 513 6 1 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(C(=O)c4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570490 190043 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 1 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL518142 190043 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 501 6 1 4 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3C(=O)N3CCC(Oc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
23728734 88401 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 445 6 1 5 3.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364305 88401 0 None - 1 Human 7.2 pEC50 = 7.2 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 445 6 1 5 3.2 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4ccc(C#N)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
1048 1548 72 None 5 2 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
12560 1548 72 None 5 2 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
1456 1548 72 None 5 2 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
CHEMBL532 1548 72 None 5 2 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
DB00199 1548 72 None 5 2 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/j.bmcl.2008.10.072
44569919 178216 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL469097 178216 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(C#N)cc4)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44572029 178816 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 511 11 1 5 4.1 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)S(=O)(=O)c1ccc(F)cc1 10.1016/j.bmcl.2008.10.071
CHEMBL474008 178816 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 511 11 1 5 4.1 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)S(=O)(=O)c1ccc(F)cc1 10.1016/j.bmcl.2008.10.071
44571991 180353 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 395 9 1 4 3.1 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(C)=O 10.1016/j.bmcl.2008.10.071
CHEMBL475823 180353 0 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by calcium mobilization-based FLIPR assay
ChEMBL 395 9 1 4 3.1 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(C)=O 10.1016/j.bmcl.2008.10.071
44542369 197234 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 11 5 15 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
44542369 197234 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 11 5 15 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL584551 197234 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 11 5 15 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2011.04.078
CHEMBL584551 197234 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 11 5 15 2.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)N(C)C)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44541928 197235 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 12 6 15 2.5 CCNC(=O)CO[C@H]1[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H]1C 10.1021/jm901107f
CHEMBL584552 197235 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 849 12 6 15 2.5 CCNC(=O)CO[C@H]1[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H]1C 10.1021/jm901107f
44542069 196232 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 899 12 6 17 2.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)Nc2cnccn2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL572997 196232 0 None - 1 Rabbit 7.2 pEC50 = 7.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 899 12 6 17 2.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)Nc2cnccn2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
53322109 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
CHEMBL1628277 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2010.08.030
53322109 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2011.04.078
53322109 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm901107f
CHEMBL1628277 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1016/j.bmcl.2011.04.078
CHEMBL1628277 55961 0 None -1 2 Rabbit 8.2 pEC50 = 8.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm901107f
44292517 101048 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@@H](CCc1ccccc1)NC(=O)[C@@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL298224 101048 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
In vitro effective concentration towards human motilin receptorIn vitro effective concentration towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@@H](CCc1ccccc1)NC(=O)[C@@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
89723612 190684 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 483 7 2 5 4.0 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)c(CO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
CHEMBL5190786 190684 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 483 7 2 5 4.0 Cc1cc(N(C)C(=O)[C@H]2CC[C@H](Oc3ccc(F)c(CO)c3)CC2)ccc1CN1CCN[C@@H](C)C1 10.1016/j.bmcl.2022.128554
46882752 5627 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 412 4 1 4 4.1 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(Cl)cc2)nc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078267 5627 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 412 4 1 4 4.1 O=S(=O)(Cc1ccc2c(c1)CCNCC2)c1ccc(-c2ccc(Cl)cc2)nc1 10.1016/j.bmcl.2009.09.027
45102707 5665 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 465 6 2 6 3.9 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(-c2ccccn2)s1 10.1016/j.bmcl.2009.09.027
CHEMBL1078492 5665 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 465 6 2 6 3.9 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(-c2ccccn2)s1 10.1016/j.bmcl.2009.09.027
46882394 5750 0 None -1 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 438 8 2 4 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cnc[nH]2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1079185 5750 0 None -1 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 438 8 2 4 4.2 CCCCc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cnc[nH]2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44570453 177789 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 455 8 1 3 5.2 CCN(CCc1ccccc1)C(=O)c1ccccc1-c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1016/j.bmcl.2008.10.072
CHEMBL465289 177789 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 455 8 1 3 5.2 CCN(CCc1ccccc1)C(=O)c1ccccc1-c1ccc(CN2C[C@H](C)N[C@H](C)C2)cc1 10.1016/j.bmcl.2008.10.072
15984995 88361 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 442 6 2 4 3.4 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364265 88361 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 442 6 2 4 3.4 C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(F)c4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728626 88387 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 434 6 1 5 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccccc4F)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364291 88387 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 434 6 1 5 4.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(Oc4ccccc4F)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728691 88390 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(C#N)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364294 88390 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.7 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(C#N)c4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
23728730 88396 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 438 6 1 4 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364300 88396 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 438 6 1 4 3.5 C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4ccc(F)cc4)CC3)cc2)CCN1 10.6019/CHEMBL2364262
23728871 88402 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364306 88402 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4cccc(F)c4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
23728838 88403 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364307 88403 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 418 5 1 4 4.0 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(-c4ccc(F)cc4)cn3)cc2)CCN1 10.6019/CHEMBL2364262
23728841 88408 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 430 6 1 5 3.8 COc1cccc(-c2ccc(C(=O)N(C)c3ccc(CN4CCN[C@@H](C)C4)cc3)nc2)c1 10.6019/CHEMBL2364262
CHEMBL2364311 88408 0 None - 1 Human 8.1 pEC50 = 8.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 430 6 1 5 3.8 COc1cccc(-c2ccc(C(=O)N(C)c3ccc(CN4CCN[C@@H](C)C4)cc3)nc2)c1 10.6019/CHEMBL2364262
52946409 17031 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 10 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256544 17031 0 None - 1 Rabbit 6.2 pEC50 = 6.2 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 10 7 15 1.3 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCCO)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
52945184 17037 0 None - 1 Rabbit 5.1 pEC50 = 5.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCN)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256550 17037 0 None - 1 Rabbit 5.1 pEC50 = 5.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 765 9 7 15 0.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCN)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
52950054 17030 0 None - 1 Rabbit 5.1 pEC50 = 5.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 10 6 15 1.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCOC)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
CHEMBL1256543 17030 0 None - 1 Rabbit 5.1 pEC50 = 5.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contraction
ChEMBL 780 10 6 15 1.6 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CCOC)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/j.bmcl.2010.08.030
44542817 197048 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 13 6 15 3.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCc2ccccc2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL582873 197048 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 911 13 6 15 3.7 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NCc2ccccc2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44570364 177775 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 457 8 1 4 4.6 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)COc3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465244 177775 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 457 8 1 4 4.6 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)COc3ccccc3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
44570410 177830 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 475 7 1 3 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)Cc3cccc(Cl)c3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL465941 177830 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 475 7 1 3 5.4 C[C@H]1CN(Cc2ccc(-c3ccccc3CN(C)C(=O)Cc3cccc(Cl)c3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
23728916 88416 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(N4CCC(F)CC4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
CHEMBL2364319 88416 0 None - 1 Human 7.1 pEC50 = 7.1 Functional
SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680SUPPLEMENTARY: Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay. Same assay as CHEMBL942680
ChEMBL 425 5 1 5 3.1 C[C@H]1CN(Cc2ccc(N(C)C(=O)c3ccc(N4CCC(F)CC4)nc3)cc2)CCN1 10.6019/CHEMBL2364262
46882519 5616 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 416 5 2 4 3.5 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(Cl)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1078104 5616 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 416 5 2 4 3.5 O=S(=O)(Nc1ccc2c(c1)CCN(Cc1cc[nH]n1)CC2)c1ccc(Cl)cc1 10.1016/j.bmcl.2009.09.027
44572030 178826 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 471 11 1 4 4.4 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)Cc1ccccc1 10.1016/j.bmcl.2008.10.071
CHEMBL474018 178826 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by calcium mobilization-based FLIPR assay
ChEMBL 471 11 1 4 4.4 COCCCN(Cc1ccccc1-c1ccc(CN2CCNCC2)cc1)C(=O)Cc1ccccc1 10.1016/j.bmcl.2008.10.071
44569920 188814 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccccc4C#N)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
CHEMBL513183 188814 0 None - 1 Human 6.1 pEC50 = 6.1 Functional
Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assay
ChEMBL 508 6 2 6 4.5 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccccc4C#N)CC3)cc2)C[C@@H](C)N1 10.1016/j.bmcl.2008.10.072
46882461 6220 0 None - 1 Human 5.1 pEC50 = 5.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 407 5 2 5 2.7 N#Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
CHEMBL1081860 6220 0 None - 1 Human 5.1 pEC50 = 5.1 Functional
Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayAgonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assay
ChEMBL 407 5 2 5 2.7 N#Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(Cc2cc[nH]n2)CC3)cc1 10.1016/j.bmcl.2009.09.027
44542214 197079 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 863 13 6 15 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL583095 197079 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 863 13 6 15 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCCCC(=O)NC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
44542666 197082 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 819 11 5 14 3.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm901107f
CHEMBL583098 197082 0 None - 1 Rabbit 7.1 pEC50 = 7.1 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 819 11 5 14 3.0 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NC)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm901107f
44542815 196557 0 None - 1 Rabbit 7.0 pEC50 = 7.0 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 851 12 6 16 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NOC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
CHEMBL575518 196557 0 None - 1 Rabbit 7.0 pEC50 = 7.0 Functional
Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionAgonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contraction
ChEMBL 851 12 6 16 2.1 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)[C@H](OCC(=O)NOC)[C@H](C)[C@@H](O)[C@]1(C)O 10.1021/jm901107f
15984937 771 27 None - 1 Human 6.0 pEC50 = 6.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1016/j.bmcl.2022.128554
4035 771 27 None - 1 Human 6.0 pEC50 = 6.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1016/j.bmcl.2022.128554
CHEMBL489095 771 27 None - 1 Human 6.0 pEC50 = 6.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1016/j.bmcl.2022.128554
DB12567 771 27 None - 1 Human 6.0 pEC50 = 6.0 Functional
Agonist activity at human GPR38 expressed in COS-7 cellsAgonist activity at human GPR38 expressed in COS-7 cells
ChEMBL 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 10.1016/j.bmcl.2022.128554
23656869 147311 0 None - 1 Human 8.7 pIC50 = 8.7 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 631 5 4 6 3.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN2CCCC2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393315 147311 0 None - 1 Human 8.7 pIC50 = 8.7 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 631 5 4 6 3.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN2CCCC2)NC1=O 10.1016/j.bmcl.2007.05.043
23557214 140539 0 None 6 2 Rabbit 7.7 pIC50 = 7.7 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382613 140539 0 None 6 2 Rabbit 7.7 pIC50 = 7.7 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
23557214 140539 0 None -6 2 Human 6.6 pIC50 = 6.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382613 140539 0 None -6 2 Human 6.6 pIC50 = 6.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
11341873 140960 0 None - 1 Human 7.6 pIC50 = 7.6 Functional
Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseActivity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium release
ChEMBL 552 6 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(OC)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL384501 140960 0 None - 1 Human 7.6 pIC50 = 7.6 Functional
Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseActivity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium release
ChEMBL 552 6 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(OC)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
23557218 139013 0 None 38 2 Rabbit 7.6 pIC50 = 7.6 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL379665 139013 0 None 38 2 Rabbit 7.6 pIC50 = 7.6 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
12016400 168383 0 None -11 2 Human 5.6 pIC50 = 5.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL438962 168383 0 None -11 2 Human 5.6 pIC50 = 5.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44412878 140538 0 None -5 2 Human 6.6 pIC50 = 6.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382612 140538 0 None -5 2 Human 6.6 pIC50 = 6.6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
44412861 77506 0 None - 1 Rabbit 7.6 pIC50 = 7.6 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 673 11 0 4 7.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL209333 77506 0 None - 1 Rabbit 7.6 pIC50 = 7.6 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 673 11 0 4 7.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
44432977 151136 0 None - 1 Human 7.6 pIC50 = 7.6 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 619 5 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL396413 151136 0 None - 1 Human 7.6 pIC50 = 7.6 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 619 5 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
44432975 87298 0 None - 1 Human 8.5 pIC50 = 8.5 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 591 5 5 6 2.2 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL233711 87298 0 None - 1 Human 8.5 pIC50 = 8.5 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 591 5 5 6 2.2 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
44432974 87122 0 None - 1 Human 7.5 pIC50 = 7.5 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 557 5 5 6 1.8 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL233560 87122 0 None - 1 Human 7.5 pIC50 = 7.5 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 557 5 5 6 1.8 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
9895192 77487 0 None -38 2 Human 6.5 pIC50 = 6.5 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL209301 77487 0 None -38 2 Human 6.5 pIC50 = 6.5 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44412878 140538 0 None 5 2 Rabbit 7.4 pIC50 = 7.4 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382612 140538 0 None 5 2 Rabbit 7.4 pIC50 = 7.4 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
44412894 138368 0 None -1 2 Human 7.3 pIC50 = 7.3 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL378317 138368 0 None -1 2 Human 7.3 pIC50 = 7.3 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
25114977 146464 0 None - 1 Human 7.3 pIC50 = 7.3 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2cccn2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL392657 146464 0 None - 1 Human 7.3 pIC50 = 7.3 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2cccn2)NC1=O 10.1016/j.bmcl.2007.05.043
12016400 168383 0 None 11 2 Rabbit 6.2 pIC50 = 6.2 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL438962 168383 0 None 11 2 Rabbit 6.2 pIC50 = 6.2 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44412894 138368 0 None 1 2 Rabbit 7.1 pIC50 = 7.1 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL378317 138368 0 None 1 2 Rabbit 7.1 pIC50 = 7.1 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
11994554 80145 0 None - 1 Human 7.1 pIC50 = 7.1 Functional
Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseActivity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium release
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL214935 80145 0 None - 1 Human 7.1 pIC50 = 7.1 Functional
Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseActivity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium release
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11994554 80145 0 None - 1 Human 7.1 pIC50 = 7.1 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL214935 80145 0 None - 1 Human 7.1 pIC50 = 7.1 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1016/j.bmcl.2007.05.043
9895192 77487 0 None 38 2 Rabbit 8.1 pIC50 = 8.1 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL209301 77487 0 None 38 2 Rabbit 8.1 pIC50 = 8.1 Functional
Activity at rabbit duodenum motilin receptor by tissue contractility assayActivity at rabbit duodenum motilin receptor by tissue contractility assay
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44432973 97847 0 None - 1 Human 8.1 pIC50 = 8.1 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 577 4 5 6 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL274876 97847 0 None - 1 Human 8.1 pIC50 = 8.1 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 577 4 5 6 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
44432976 154313 0 None - 1 Human 7.0 pIC50 = 7.0 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL400635 154313 0 None - 1 Human 7.0 pIC50 = 7.0 Functional
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayAntagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
23557218 139013 0 None -38 2 Human 6.0 pIC50 = 6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL379665 139013 0 None -38 2 Human 6.0 pIC50 = 6 Functional
Activity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilizationActivity at human motilin receptor transfected in HEK293 cells assessed as inhibition of motilin-induced intracellular calcium mobilization
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL496391 212302 0 None - 1 Rabbit 7.9 pKd = 7.9 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)[C@@H](C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
CHEMBL496389 212300 0 None - 1 Rabbit 6.9 pKd = 6.9 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
CHEMBL497004 212303 0 None - 1 Rabbit 7.8 pKd = 7.8 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)(C)c1cc(C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](N)Cc2ccccc2)c2ccccc2)C(N)=O)ccc1O 10.1016/j.bmcl.2009.05.059
44583348 187247 0 None - 1 Rabbit 8.6 pKd = 8.6 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 510 10 3 5 2.6 CC(C)[C@@H](C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
CHEMBL496190 187247 0 None - 1 Rabbit 8.6 pKd = 8.6 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 510 10 3 5 2.6 CC(C)[C@@H](C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
9956253 187248 0 None - 1 Rabbit 8.4 pKd = 8.4 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 467 9 3 4 3.8 CC(C)[C@@H](C(=O)N[C@H](C)Cc1ccc(O)c(C(C)(C)C)c1)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
CHEMBL496191 187248 0 None - 1 Rabbit 8.4 pKd = 8.4 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 467 9 3 4 3.8 CC(C)[C@@H](C(=O)N[C@H](C)Cc1ccc(O)c(C(C)(C)C)c1)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
44583286 192837 0 None - 1 Rabbit 7.4 pKd = 7.4 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 564 6 5 6 2.8 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCCC(=O)CCNC2=O)ccc1O 10.1016/j.bmcl.2009.05.059
CHEMBL526496 192837 0 None - 1 Rabbit 7.4 pKd = 7.4 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 564 6 5 6 2.8 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCCC(=O)CCNC2=O)ccc1O 10.1016/j.bmcl.2009.05.059
CHEMBL496390 212301 0 None - 1 Rabbit 7.3 pKd = 7.3 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)C[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
44583347 187227 0 None - 1 Rabbit 7.2 pKd = 7.2 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 496 10 4 5 2.3 CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
CHEMBL495994 187227 0 None - 1 Rabbit 7.2 pKd = 7.2 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL 496 10 4 5 2.3 CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
CHEMBL502792 212377 0 None - 1 Rabbit 7.2 pKd = 7.2 Functional
Antagonist activity at MTL receptor in rabbit duodenum homogenateAntagonist activity at MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)(C)c1cc(C[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](N)Cc2ccccc2)C(N)=O)ccc1O 10.1016/j.bmcl.2009.05.059
1466 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10081621
1466 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7752063
9850904 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10081621
9850904 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7752063
CHEMBL3143516 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10081621
CHEMBL3143516 1790 0 None - 1 Rabbit 7.4 pA2 = 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7752063
4036 2409 0 None - 1 Human 9.2 pA2 = 9.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 592 12 4 5 3.7 CCNC(=O)[C@@H](NC(=O)[C@@H](N(C(=O)[C@H](Cc1ccc(cc1)F)NC)C)C(C)C)Cc1ccc(c(c1)C(C)(C)C)O.Cl 18164286
73755070 2409 0 None - 1 Human 9.2 pA2 = 9.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 592 12 4 5 3.7 CCNC(=O)[C@@H](NC(=O)[C@@H](N(C(=O)[C@H](Cc1ccc(cc1)F)NC)C)C(C)C)Cc1ccc(c(c1)C(C)(C)C)O.Cl 18164286
138107041 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
276 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
447043 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
6510 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
CHEMBL529 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
DB00207 555 63 None 60 3 Human 8.3 pEC50 = 8.3 Functional
NoneNone
Drug Central 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O None
138107041 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
276 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
447043 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
6510 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
CHEMBL529 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
DB00207 555 63 None 60 3 Human 5.5 pEC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 749 7 5 14 1.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](CN([C@@H]([C@H]([C@]1(C)O)O)C)C)C)(C)O 23190027
177964 2498 2 None -3 2 Rabbit 7.7 pEC50 = 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 17183187
3511 2498 2 None -3 2 Rabbit 7.7 pEC50 = 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 17183187
CHEMBL1778156 2498 2 None -3 2 Rabbit 7.7 pEC50 = 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 17183187
15984937 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 19374732
15984937 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 25341626
4035 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 19374732
4035 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 25341626
CHEMBL489095 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 19374732
CHEMBL489095 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 25341626
DB12567 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 19374732
DB12567 771 27 None - 1 Human 7.9 pEC50 = 7.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology 424 6 2 4 3.3 C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F 25341626
11902 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 35051575
56960876 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 35051575
CHEMBL5201797 1454 5 None - 1 Human 8.3 pEC50 = 8.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 465 7 2 5 3.9 C[C@H]1CN(Cc2ccc(cc2C)N(C)C(=O)[C@H]2CC[C@@H](CC2)Oc2cc(CO)ccc2)CCN1 35051575
139592915 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
1465 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
2410 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
6915744 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
CHEMBL1214185 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
DB00778 3310 31 None 16 2 Human 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C None
1048 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10381885
1048 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 15764739
12560 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10381885
12560 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 15764739
1456 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10381885
1456 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 15764739
CHEMBL532 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10381885
CHEMBL532 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 15764739
DB00199 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10381885
DB00199 1548 72 None 5 2 Human 6.0 pIC50 = 6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 15764739
1444 338 0 None - 1 Human 7.2 pIC50 = 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 697 8 2 11 5.2 CCN([C@H]1C[C@@H](C)O[C@H]([C@@H]1O)O[C@@H]1[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@@H](C)C(=O)O[C@@H]([C@@H]([C@@H]([C@H](C2=C(C[C@@]1(C)O2)C)C)O)C)CC)C 15764739
9918079 338 0 None - 1 Human 7.2 pIC50 = 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 697 8 2 11 5.2 CCN([C@H]1C[C@@H](C)O[C@H]([C@@H]1O)O[C@@H]1[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@@H](C)C(=O)O[C@@H]([C@@H]([C@@H]([C@H](C2=C(C[C@@]1(C)O2)C)C)O)C)CC)C 15764739
CHEMBL300049 338 0 None - 1 Human 7.2 pIC50 = 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 697 8 2 11 5.2 CCN([C@H]1C[C@@H](C)O[C@H]([C@@H]1O)O[C@@H]1[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@@H](C)C(=O)O[C@@H]([C@@H]([C@@H]([C@H](C2=C(C[C@@]1(C)O2)C)C)O)C)CC)C 15764739
1466 1790 0 None - 1 Rabbit 8.0 pIC50 = 8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11806718
9850904 1790 0 None - 1 Rabbit 8.0 pIC50 = 8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11806718
CHEMBL3143516 1790 0 None - 1 Rabbit 8.0 pIC50 = 8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11806718
177964 2498 2 None -3 2 Rabbit 8.2 pIC50 = 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10081621
3511 2498 2 None -3 2 Rabbit 8.2 pIC50 = 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10081621
CHEMBL1778156 2498 2 None -3 2 Rabbit 8.2 pIC50 = 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10081621
1447 2433 0 None - 1 Human 4.7 pIC50 None 4.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 747 8 5 14 2.2 CCN(C1CC(C)OC(C1O)OC1C(C)C(OC2OC(C)C(C(C2)(C)OC)O)C(C)C(=O)OC(CC)C(C(C(C(=O)C(CC1(C)O)C)C)O)(C)O)C 15764739
14487390 2433 0 None - 1 Human 4.7 pIC50 None 4.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 747 8 5 14 2.2 CCN(C1CC(C)OC(C1O)OC1C(C)C(OC2OC(C)C(C(C2)(C)OC)O)C(C)C(=O)OC(CC)C(C(C(C(=O)C(CC1(C)O)C)C)O)(C)O)C 15764739
139592915 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
1465 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
2410 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
6915744 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
CHEMBL1214185 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
DB00778 3310 31 None 16 2 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 837 13 5 17 2.2 COCCOCO/N=C/1\[C@H](C)C[C@@](C)(O)[C@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C(=O)O[C@@H]([C@@]([C@@H]([C@H]1C)O)(C)O)CC)C 10381885
1448 2434 29 None -2 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
83954 2434 29 None -2 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
CHEMBL300004 2434 29 None -2 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
10032648 2435 0 None - 1 Human 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 699 7 3 12 3.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H]([C@H]([C@@H]1C)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
1449 2435 0 None - 1 Human 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 699 7 3 12 3.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H]([C@H]([C@@H]1C)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
1445 1515 0 None - 1 Human 6.6 pIC50 None 6.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 729 8 4 13 3.3 CCN([C@H]1C[C@@H](C)O[C@H]([C@@H]1O)O[C@@H]1[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@@H](C)C(=O)O[C@@H]([C@@]([C@@H]([C@H](C2=C(C[C@]1(C)O2)C)C)O)(C)O)CC)C 15764739
184178 1515 0 None - 1 Human 6.6 pIC50 None 6.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology 729 8 4 13 3.3 CCN([C@H]1C[C@@H](C)O[C@H]([C@@H]1O)O[C@@H]1[C@@H](C)[C@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@@H](C)C(=O)O[C@@H]([C@@]([C@@H]([C@H](C2=C(C[C@]1(C)O2)C)C)O)(C)O)CC)C 15764739
1460 2551 0 None - 1 Human 6.8 pIC50 None 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817408 2551 0 None - 1 Human 6.8 pIC50 None 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
10259168 2159 0 None - 1 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 699 7 3 12 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
1446 2159 0 None - 1 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 699 7 3 12 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
CHEMBL51522 2159 0 None - 1 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology 699 7 3 12 3.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)C[C@](C2)(C)OC)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 15764739
1464 2555 0 None - 1 Human 7.5 pIC50 None 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817411 2555 0 None - 1 Human 7.5 pIC50 None 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1454 3044 0 None - 1 Human 8.9 pIC50 None 8.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
101650014 2257 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1453 2257 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
16198245 2257 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
91898971 2257 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
101930759 2552 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1461 2552 0 None - 1 Human 9.0 pIC50 None 9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1457 2549 0 None - 1 Human 9.3 pIC50 None 9.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817406 2549 0 None - 1 Human 9.3 pIC50 None 9.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
16139289 2549 0 None - 1 Human 9.3 pIC50 None 9.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
71311666 2549 0 None - 1 Human 9.3 pIC50 None 9.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1462 2553 0 None - 1 Human 9.5 pIC50 None 9.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817409 2553 0 None - 1 Human 9.5 pIC50 None 9.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1463 2554 0 None - 1 Human 9.5 pIC50 None 9.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817410 2554 0 None - 1 Human 9.5 pIC50 None 9.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1455 2777 0 None - 1 Human 9.5 pIC50 None 9.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1459 2550 0 None - 1 Human 9.7 pIC50 None 9.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
155817407 2550 0 None - 1 Human 9.7 pIC50 None 9.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885




Ligands Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Affinity)
# tested GPCRs
(Affinity)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI
16752689 187774 0 None - 0 Human 8.0 pEC50 = 8 Binding
Agonist activity at MLNR (unknown origin)Agonist activity at MLNR (unknown origin)
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1021/jm301653f
CHEMBL501315 187774 0 None - 0 Human 8.0 pEC50 = 8 Binding
Agonist activity at MLNR (unknown origin)Agonist activity at MLNR (unknown origin)
ChEMBL 568 10 2 4 6.6 COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1 10.1021/jm301653f
CHEMBL382080 210537 0 None - 0 Rat 6.0 pEC50 = 6.0 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.21-5.7 uMSignaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.21-5.7 uM
ChEMBL None None None NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1c[nH]c(C2CCCCC2)n1)NC(=O)[C@@H]1CCC(=O)N1 10.1021/jm0505462
CHEMBL382714 210554 0 None - 0 Rat 5.9 pEC50 = 5.9 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.76-2.2 uMSignaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.76-2.2 uM
ChEMBL None None None CC(C)(C)c1nc(C[C@H](NC(=O)[C@@H]2CCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1021/jm0505462
CHEMBL381666 210534 0 None - 0 Rat 5.8 pEC50 = 5.8 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 h at 37 degree C and pH 7.8; Range = 0.69-3.2 uMSignaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 h at 37 degree C and pH 7.8; Range = 0.69-3.2 uM
ChEMBL None None None CC(C)c1nc(C[C@H](NC(=O)[C@@H]2CCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1021/jm0505462
CHEMBL197149 207351 0 None - 1 Rat 7.6 pEC50 = 7.6 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.011-0.052 uMSignaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.011-0.052 uM
ChEMBL None None None CCCc1nc(C[C@H](NC(=O)[C@@H]2CCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1021/jm0505462
2139 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
2316 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
3836 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
638678 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
CHEMBL1472 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
DB09421 3782 51 None 1 4 Rat 8.5 pEC50 = 8.5 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8
ChEMBL None None None None 10.1021/jm0505462
CHEMBL198263 207352 0 None - 0 Rat 6.4 pEC50 = 6.4 Binding
Signaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.19-0.85 uMSignaling (activation) potency for thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells with CREB-luciferase reporter upon incubation with the compound for 6 hr at 37 degree C and pH 7.8; Range = 0.19-0.85 uM
ChEMBL None None None NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1c[nH]c(C2CC2)n1)NC(=O)[C@@H]1CCC(=O)N1 10.1021/jm0505462
CHEMBL496391 212302 0 None - 1 Rabbit 9.0 pIC50 = 9.0 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)[C@@H](C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
11018075 99909 0 None - 0 Rabbit 8.8 pIC50 = 8.8 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 739 9 1 12 5.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL289955 99909 0 None - 0 Rabbit 8.8 pIC50 = 8.8 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 739 9 1 12 5.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44290233 172247 0 None - 0 Rabbit 8.7 pIC50 = 8.7 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 723 9 0 11 6.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2CC(N(C)C(C)C)CC(C)O2)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL45141 172247 0 None - 0 Rabbit 8.7 pIC50 = 8.7 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 723 9 0 11 6.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2CC(N(C)C(C)C)CC(C)O2)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
9956253 187248 0 None - 1 Rabbit 8.7 pIC50 = 8.7 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 467 9 3 4 3.8 CC(C)[C@@H](C(=O)N[C@H](C)Cc1ccc(O)c(C(C)(C)C)c1)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
CHEMBL496191 187248 0 None - 1 Rabbit 8.7 pIC50 = 8.7 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 467 9 3 4 3.8 CC(C)[C@@H](C(=O)N[C@H](C)Cc1ccc(O)c(C(C)(C)C)c1)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
9895192 77487 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL209301 77487 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@@H]1CCC[C@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44412981 137799 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 704 11 2 5 7.3 O=C(Nc1ccccc1)N(CC1=C[C@@](Cc2cccc(Cl)c2)(NC(=O)C(Cl)(Cl)Cl)CC1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL377137 137799 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 704 11 2 5 7.3 O=C(Nc1ccccc1)N(CC1=C[C@@](Cc2cccc(Cl)c2)(NC(=O)C(Cl)(Cl)Cl)CC1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
1466 1790 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL None None None None 10.1021/jm010332u
9850904 1790 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL None None None None 10.1021/jm010332u
CHEMBL3143516 1790 0 None - 0 Rabbit 8.0 pIC50 = 8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL None None None None 10.1021/jm010332u
10122749 77894 0 None - 0 Rabbit 5.9 pIC50 = 5.9 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 691 13 1 7 7.2 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)c2cccc([N+](=O)[O-])c2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL210899 77894 0 None - 0 Rabbit 5.9 pIC50 = 5.9 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 691 13 1 7 7.2 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)c2cccc([N+](=O)[O-])c2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
44583286 192837 0 None - 1 Rabbit 7.9 pIC50 = 7.9 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 564 6 5 6 2.8 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCCC(=O)CCNC2=O)ccc1O 10.1016/j.bmcl.2009.05.059
CHEMBL526496 192837 0 None - 1 Rabbit 7.9 pIC50 = 7.9 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 564 6 5 6 2.8 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCCC(=O)CCNC2=O)ccc1O 10.1016/j.bmcl.2009.05.059
CHEMBL497004 212303 0 None - 1 Rabbit 7.9 pIC50 = 7.9 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)(C)c1cc(C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](N)Cc2ccccc2)c2ccccc2)C(N)=O)ccc1O 10.1016/j.bmcl.2009.05.059
44412894 138368 0 None - 0 Rabbit 7.9 pIC50 = 7.9 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL378317 138368 0 None - 0 Rabbit 7.9 pIC50 = 7.9 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 718 12 0 6 7.8 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
44380651 119614 0 None - 0 Human 7.8 pIC50 = 7.8 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 757 9 3 13 4.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL351216 119614 0 None - 0 Human 7.8 pIC50 = 7.8 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 757 9 3 13 4.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
44276703 98814 0 None - 0 Human 6.8 pIC50 = 6.8 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/0960-894X(95)00122-A
CHEMBL281952 98814 0 None - 0 Human 6.8 pIC50 = 6.8 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/0960-894X(95)00122-A
44276703 98814 0 None - 0 Rabbit 6.8 pIC50 = 6.8 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/S0960-894X(01)80359-0
CHEMBL281952 98814 0 None - 0 Rabbit 6.8 pIC50 = 6.8 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/S0960-894X(01)80359-0
44276703 98814 0 None - 0 Human 6.8 pIC50 = 6.8 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/0960-894X(95)00122-A
CHEMBL281952 98814 0 None - 0 Human 6.8 pIC50 = 6.8 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/0960-894X(95)00122-A
44276703 98814 0 None - 0 Rabbit 6.8 pIC50 = 6.8 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/S0960-894X(01)80359-0
CHEMBL281952 98814 0 None - 0 Rabbit 6.8 pIC50 = 6.8 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 715 7 3 13 3.0 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)C3(O2)O[C@]1(C)[C@H](O)[C@H]3C 10.1016/S0960-894X(01)80359-0
11767227 106196 0 None - 0 Rabbit 7.8 pIC50 = 7.8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 607 6 6 6 2.7 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3143521 106196 0 None - 0 Rabbit 7.8 pIC50 = 7.8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 607 6 6 6 2.7 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCCCNC2=O)ccc1O 10.1021/jm010332u
10940742 114903 0 None - 0 Rabbit 5.8 pIC50 = 5.8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3350348 114903 0 None - 0 Rabbit 5.8 pIC50 = 5.8 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL524083 213814 0 None - 0 Rabbit 6.7 pIC50 = 6.7 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None C[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
24878741 187346 1 None - 0 Rat 4.7 pIC50 = 4.7 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL 522 8 4 7 6.1 Cc1c(O)c(C(=O)CCc2ccccc2)c(O)c(C(CC(C)C)C2=C(O)C(C)(C)C(=O)C(C)(C)C2=O)c1O 10.1021/np0706567
CHEMBL496930 187346 1 None - 0 Rat 4.7 pIC50 = 4.7 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL 522 8 4 7 6.1 Cc1c(O)c(C(=O)CCc2ccccc2)c(O)c(C(CC(C)C)C2=C(O)C(C)(C)C(=O)C(C)(C)C2=O)c1O 10.1021/np0706567
44290232 100901 0 None - 0 Rabbit 8.6 pIC50 = 8.6 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 711 8 1 12 4.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL297168 100901 0 None - 0 Rabbit 8.6 pIC50 = 8.6 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 711 8 1 12 4.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
11018075 99909 0 None - 0 Rabbit 8.6 pIC50 = 8.6 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 739 9 1 12 5.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL289955 99909 0 None - 0 Rabbit 8.6 pIC50 = 8.6 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 739 9 1 12 5.6 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
9809991 138979 0 None - 0 Rabbit 7.7 pIC50 = 7.7 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 670 11 2 5 6.6 O=C(Nc1ccccc1)N(CC1=C[C@@](Cc2ccccc2)(NC(=O)C(Cl)(Cl)Cl)CC1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL379519 138979 0 None - 0 Rabbit 7.7 pIC50 = 7.7 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 670 11 2 5 6.6 O=C(Nc1ccccc1)N(CC1=C[C@@](Cc2ccccc2)(NC(=O)C(Cl)(Cl)Cl)CC1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
10211030 77377 0 None - 0 Rabbit 7.7 pIC50 = 7.7 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptor at 1 uMInhibition of [125]I-motilin binding to rabbit motilin receptor at 1 uM
ChEMBL 610 11 1 4 7.8 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)Nc2ccccc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL209024 77377 0 None - 0 Rabbit 7.7 pIC50 = 7.7 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptor at 1 uMInhibition of [125]I-motilin binding to rabbit motilin receptor at 1 uM
ChEMBL 610 11 1 4 7.8 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)Nc2ccccc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44374025 51886 0 None - 0 Rabbit 5.7 pIC50 = 5.7 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(CC2NC(=O)[C@@H](NC(=O)C(N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL158821 51886 0 None - 0 Rabbit 5.7 pIC50 = 5.7 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(CC2NC(=O)[C@@H](NC(=O)C(N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
1448 2434 29 None - 0 Human 6.7 pIC50 = 6.7 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
83954 2434 29 None - 0 Human 6.7 pIC50 = 6.7 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
CHEMBL300004 2434 29 None - 0 Human 6.7 pIC50 = 6.7 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
1448 2434 29 None - 0 Rabbit 6.7 pIC50 = 6.7 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
83954 2434 29 None - 0 Rabbit 6.7 pIC50 = 6.7 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
CHEMBL300004 2434 29 None - 0 Rabbit 6.7 pIC50 = 6.7 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
2139 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
2316 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
3836 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
638678 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
CHEMBL1472 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
DB09421 3782 51 None 1 4 Rat 7.6 pIC50 = 7.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np070658r
2139 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
2316 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
3836 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
638678 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
CHEMBL1472 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
DB09421 3782 51 None 1 4 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL None None None None 10.1021/np0706567
24878685 171594 1 None - 0 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL 570 9 4 7 6.7 Cc1c(O)c(C(=O)CCc2ccccc2)c(O)c(C(CCc2ccccc2)C2=C(O)C(C)(C)C(=O)C(C)(C)C2=O)c1O 10.1021/np0706567
CHEMBL447346 171594 1 None - 0 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cells
ChEMBL 570 9 4 7 6.7 Cc1c(O)c(C(=O)CCc2ccccc2)c(O)c(C(CCc2ccccc2)C2=C(O)C(C)(C)C(=O)C(C)(C)C2=O)c1O 10.1021/np0706567
24878743 188771 0 None - 0 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL 360 3 1 4 4.2 CC(=O)OC[C@]12CCC[C@](C)(CO)[C@@H]1CC[C@@]1(C)c3cocc3CC[C@H]21 10.1021/np070658r
CHEMBL512825 188771 0 None - 0 Rat 4.6 pIC50 = 4.6 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL 360 3 1 4 4.2 CC(=O)OC[C@]12CCC[C@](C)(CO)[C@@H]1CC[C@@]1(C)c3cocc3CC[C@H]21 10.1021/np070658r
44583347 187227 0 None - 1 Rabbit 7.6 pIC50 = 7.6 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 496 10 4 5 2.3 CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
CHEMBL495994 187227 0 None - 1 Rabbit 7.6 pIC50 = 7.6 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 496 10 4 5 2.3 CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
11081770 89015 0 None - 0 Rabbit 4.6 pIC50 = 4.6 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 509 6 6 6 0.3 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCCCNC(=O)CCNC(=O)[C@H](Cc2ccc(O)cc2)NC1=O 10.1021/jm010332u
CHEMBL2371260 89015 0 None - 0 Rabbit 4.6 pIC50 = 4.6 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 509 6 6 6 0.3 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCCCNC(=O)CCNC(=O)[C@H](Cc2ccc(O)cc2)NC1=O 10.1021/jm010332u
CHEMBL496390 212301 0 None - 1 Rabbit 7.6 pIC50 = 7.6 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)C[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
23557218 139013 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL379665 139013 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44380970 119881 0 None - 0 Human 8.5 pIC50 = 8.5 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 8 4 13 3.0 CCC1OC(=O)C(C)C(OC2C[C@@](C)(OC)[C@@H](O)C(C)O2)C[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/0960-894X(95)00122-A
CHEMBL353526 119881 0 None - 0 Human 8.5 pIC50 = 8.5 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 8 4 13 3.0 CCC1OC(=O)C(C)C(OC2C[C@@](C)(OC)[C@@H](O)C(C)O2)C[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/0960-894X(95)00122-A
44276737 96916 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
CHEMBL26966 96916 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
44276737 96916 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80583-7
CHEMBL26966 96916 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80583-7
1448 2434 29 None - 0 Human 8.5 pIC50 = 8.5 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
83954 2434 29 None - 0 Human 8.5 pIC50 = 8.5 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
CHEMBL300004 2434 29 None - 0 Human 8.5 pIC50 = 8.5 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/0960-894X(95)00122-A
1448 2434 29 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
83954 2434 29 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
CHEMBL300004 2434 29 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 715 7 4 13 2.9 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@@]2(OC(=C(C)C2)[C@@H]([C@H]([C@]1(C)O)O)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C)C 10.1016/S0960-894X(01)80359-0
44290012 167587 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 725 9 1 12 5.2 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL43313 167587 0 None - 0 Rabbit 8.5 pIC50 = 8.5 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 725 9 1 12 5.2 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44276779 96410 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL265495 96410 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44290012 167587 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 725 9 1 12 5.2 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL43313 167587 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 725 9 1 12 5.2 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44276779 96410 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL265495 96410 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44290232 100901 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 711 8 1 12 4.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL297168 100901 0 None - 0 Rabbit 8.4 pIC50 = 8.4 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 711 8 1 12 4.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)CC(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
177964 2498 2 None - 0 Human 8.4 pIC50 = 8.4 Binding
Antagonist activity at MLNR (unknown origin)Antagonist activity at MLNR (unknown origin)
ChEMBL 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10.1021/jm301653f
3511 2498 2 None - 0 Human 8.4 pIC50 = 8.4 Binding
Antagonist activity at MLNR (unknown origin)Antagonist activity at MLNR (unknown origin)
ChEMBL 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10.1021/jm301653f
CHEMBL1778156 2498 2 None - 0 Human 8.4 pIC50 = 8.4 Binding
Antagonist activity at MLNR (unknown origin)Antagonist activity at MLNR (unknown origin)
ChEMBL 755 9 2 13 4.5 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@H]([C@]2(OC(=C(C)C2)[C@@H](C(=O)[C@]1(C)OC)C)C)O[C@@H]1O[C@H](C)C[C@@H]([C@H]1O)N(C(C)C)C 10.1021/jm301653f
16040587 178794 0 None - 0 Human 8.4 pIC50 = 8.4 Binding
Antagonist activity at MLNR (unknown origin)Antagonist activity at MLNR (unknown origin)
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm301653f
CHEMBL473921 178794 0 None - 0 Human 8.4 pIC50 = 8.4 Binding
Antagonist activity at MLNR (unknown origin)Antagonist activity at MLNR (unknown origin)
ChEMBL 501 6 2 5 4.8 C[C@H]1CN(Cc2ccc(-c3cccnc3C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@@H](C)N1 10.1021/jm301653f
44380970 119881 0 None - 0 Human 6.5 pIC50 = 6.5 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 8 4 13 3.0 CCC1OC(=O)C(C)C(OC2C[C@@](C)(OC)[C@@H](O)C(C)O2)C[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/0960-894X(95)00122-A
CHEMBL353526 119881 0 None - 0 Human 6.5 pIC50 = 6.5 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 715 8 4 13 3.0 CCC1OC(=O)C(C)C(OC2C[C@@](C)(OC)[C@@H](O)C(C)O2)C[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/0960-894X(95)00122-A
44276737 96916 0 None - 0 Rabbit 6.5 pIC50 = 6.5 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
CHEMBL26966 96916 0 None - 0 Rabbit 6.5 pIC50 = 6.5 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
44276737 96916 0 None - 0 Rabbit 6.5 pIC50 = 6.5 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80583-7
CHEMBL26966 96916 0 None - 0 Rabbit 6.5 pIC50 = 6.5 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 729 8 4 13 3.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80583-7
10897050 106192 0 None - 0 Rabbit 5.5 pIC50 = 5.5 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(C[C@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3143517 106192 0 None - 0 Rabbit 5.5 pIC50 = 5.5 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 6 6 6 1.6 CC(C)(C)c1cc(C[C@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)ccc1O 10.1021/jm010332u
11146277 106193 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 579 6 6 6 2.0 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3143518 106193 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 579 6 6 6 2.0 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL2371264 208272 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL None None None CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CNC2=O)ccc1O 10.1021/jm010332u
44413071 77896 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 731 12 1 7 7.3 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL210906 77896 0 None - 0 Rabbit 7.5 pIC50 = 7.5 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 731 12 1 7 7.3 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2cccc([N+](=O)[O-])c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
44380971 57256 0 None - 0 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 729 8 3 13 3.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL166642 57256 0 None - 0 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 729 8 3 13 3.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
44583348 187247 0 None - 1 Rabbit 8.4 pIC50 = 8.4 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 510 10 3 5 2.6 CC(C)[C@@H](C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
CHEMBL496190 187247 0 None - 1 Rabbit 8.4 pIC50 = 8.4 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL 510 10 3 5 2.6 CC(C)[C@@H](C(=O)N(C)[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O)N(C)C(=O)[C@@H](N)Cc1ccccc1 10.1016/j.bmcl.2009.05.059
44380610 95966 0 None - 0 Human 8.3 pIC50 = 8.3 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 743 9 3 13 3.9 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL262052 95966 0 None - 0 Human 8.3 pIC50 = 8.3 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 743 9 3 13 3.9 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
11081770 89015 0 None - 0 Rabbit 4.4 pIC50 = 4.4 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 509 6 6 6 0.3 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCCCNC(=O)CCNC(=O)[C@H](Cc2ccc(O)cc2)NC1=O 10.1021/jm010332u
CHEMBL2371260 89015 0 None - 0 Rabbit 4.4 pIC50 = 4.4 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 509 6 6 6 0.3 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCCCNC(=O)CCNC(=O)[C@H](Cc2ccc(O)cc2)NC1=O 10.1021/jm010332u
1048 1548 72 None - 1 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
12560 1548 72 None - 1 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
1456 1548 72 None - 1 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
CHEMBL532 1548 72 None - 1 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
DB00199 1548 72 None - 1 Human 7.4 pIC50 = 7.4 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
10897911 155724 0 None - 0 Rabbit 7.4 pIC50 = 7.4 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 733 7 5 14 1.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
CHEMBL406517 155724 0 None - 0 Rabbit 7.4 pIC50 = 7.4 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 733 7 5 14 1.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
CHEMBL496389 212300 0 None - 1 Rabbit 7.3 pIC50 = 7.3 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)=O 10.1016/j.bmcl.2009.05.059
11135894 106197 0 None - 0 Rabbit 6.3 pIC50 = 6.3 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 621 6 6 6 2.9 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc(C(C)(C)C)c1O 10.1021/jm010332u
CHEMBL3143523 106197 0 None - 0 Rabbit 6.3 pIC50 = 6.3 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 621 6 6 6 2.9 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc(C(C)(C)C)c1O 10.1021/jm010332u
10995344 106194 0 None - 0 Rabbit 6.3 pIC50 = 6.3 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 9 5 6 1.8 CCC(C)Oc1ccc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc1 10.1021/jm010332u
CHEMBL3143519 106194 0 None - 0 Rabbit 6.3 pIC50 = 6.3 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 9 5 6 1.8 CCC(C)Oc1ccc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc1 10.1021/jm010332u
44412861 77506 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 673 11 0 4 7.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL209333 77506 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 673 11 0 4 7.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
44412878 140538 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382612 140538 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 707 11 0 4 8.6 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCC2)c1 10.1016/j.bmcl.2006.04.017
11146277 106193 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 579 6 6 6 2.0 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3143518 106193 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 579 6 6 6 2.0 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL502792 212377 0 None - 1 Rabbit 8.2 pIC50 = 8.2 Binding
Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateDisplacement of [125I]motilin from MTL receptor in rabbit duodenum homogenate
ChEMBL None None None CC(C)(C)c1cc(C[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](N)Cc2ccccc2)C(N)=O)ccc1O 10.1016/j.bmcl.2009.05.059
44276778 97741 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL27424 97741 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44276778 97741 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL27424 97741 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44276779 96410 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL265495 96410 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44276779 96410 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL265495 96410 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 741 9 2 13 4.1 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44380651 119614 0 None - 0 Human 8.2 pIC50 = 8.2 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 757 9 3 13 4.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL351216 119614 0 None - 0 Human 8.2 pIC50 = 8.2 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 757 9 3 13 4.3 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
23557214 140539 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL382613 140539 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 721 11 0 4 8.9 O=C(c1ccc(F)cc1)N(CC1CCCC(N(Cc2cccc(Cl)c2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCCCC2)c1 10.1016/j.bmcl.2006.04.017
11767227 106196 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 607 6 6 6 2.7 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCCCNC2=O)ccc1O 10.1021/jm010332u
CHEMBL3143521 106196 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 607 6 6 6 2.7 CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCCCCNC2=O)ccc1O 10.1021/jm010332u
44412941 139787 0 None - 0 Rabbit 6.2 pIC50 = 6.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 710 13 1 6 8.0 COc1cccc(C(=O)N(Cc2cccc(Cl)c2)C2CCCC(CN(C(=O)Nc3ccccc3)c3cccc(OCCN4CCOCC4)c3)C2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL380678 139787 0 None - 0 Rabbit 6.2 pIC50 = 6.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 710 13 1 6 8.0 COc1cccc(C(=O)N(Cc2cccc(Cl)c2)C2CCCC(CN(C(=O)Nc3ccccc3)c3cccc(OCCN4CCOCC4)c3)C2)c1 10.1016/j.bmcl.2006.04.017
44413072 77898 0 None - 0 Rabbit 6.2 pIC50 = 6.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 636 12 1 6 6.9 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)c2ccco2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL210923 77898 0 None - 0 Rabbit 6.2 pIC50 = 6.2 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 636 12 1 6 6.9 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)c2ccco2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL2371264 208272 0 None - 0 Rabbit 8.2 pIC50 = 8.2 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL None None None CC(C)(C)c1cc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CNC2=O)ccc1O 10.1021/jm010332u
44380971 57256 0 None - 0 Human 8.1 pIC50 = 8.1 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 729 8 3 13 3.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL166642 57256 0 None - 0 Human 8.1 pIC50 = 8.1 Binding
Compound was tested for in vitro motilin receptor binding affinityCompound was tested for in vitro motilin receptor binding affinity
ChEMBL 729 8 3 13 3.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
44276778 97741 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL27424 97741 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44276778 97741 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL27424 97741 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 755 9 2 13 4.5 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
1048 1548 72 None - 1 Human 7.2 pIC50 = 7.2 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
12560 1548 72 None - 1 Human 7.2 pIC50 = 7.2 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
1456 1548 72 None - 1 Human 7.2 pIC50 = 7.2 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
CHEMBL532 1548 72 None - 1 Human 7.2 pIC50 = 7.2 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
DB00199 1548 72 None - 1 Human 7.2 pIC50 = 7.2 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1016/0960-894X(95)00122-A
10897911 155724 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 733 7 5 14 1.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
CHEMBL406517 155724 0 None - 0 Rabbit 7.2 pIC50 = 7.2 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 733 7 5 14 1.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O 10.1016/S0960-894X(01)80359-0
24878742 178180 0 None - 0 Rat 4.2 pIC50 = 4.2 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL 360 3 1 4 4.2 CC(=O)OC[C@@]1(C)CCC[C@@]2(CO)[C@H]1CC[C@@]1(C)c3cocc3CC[C@H]21 10.1021/np070658r
CHEMBL468803 178180 0 None - 0 Rat 4.2 pIC50 = 4.2 Binding
Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsDisplacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cells
ChEMBL 360 3 1 4 4.2 CC(=O)OC[C@@]1(C)CCC[C@@]2(CO)[C@H]1CC[C@@]1(C)c3cocc3CC[C@H]21 10.1021/np070658r
12016400 168383 0 None - 0 Rabbit 7.1 pIC50 = 7.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL438962 168383 0 None - 0 Rabbit 7.1 pIC50 = 7.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 613 11 0 4 7.6 CC(C)(C)C(=O)N(Cc1ccccc1)[C@H]1CCC[C@@H](CN(C(=O)c2ccc(F)cc2)c2cccc(OCCN3CCCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44412951 77792 0 None - 0 Rabbit 6.1 pIC50 = 6.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 674 14 1 5 7.7 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)CCc2ccccc2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL210447 77792 0 None - 0 Rabbit 6.1 pIC50 = 6.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 674 14 1 5 7.7 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)CCc2ccccc2)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
10875453 106195 0 None - 0 Rabbit 5.1 pIC50 = 5.1 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 7 5 6 1.8 CC(C)(C)Oc1ccc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc1 10.1021/jm010332u
CHEMBL3143520 106195 0 None - 0 Rabbit 5.1 pIC50 = 5.1 Binding
Inhibition of the motilin receptor (MTL-R)Inhibition of the motilin receptor (MTL-R)
ChEMBL 565 7 5 6 1.8 CC(C)(C)Oc1ccc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H](N)Cc3ccccc3)CCCCNC(=O)CCNC2=O)cc1 10.1021/jm010332u
44412982 58736 0 None - 0 Rabbit 6.1 pIC50 = 6.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 644 11 1 5 7.2 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)Nc2ccc(F)cc2)c2cccc(OCCN3CCOCC3)c2)C1 10.1016/j.bmcl.2006.04.017
CHEMBL169509 58736 0 None - 0 Rabbit 6.1 pIC50 = 6.1 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 644 11 1 5 7.2 CC(C)(C)C(=O)N(Cc1ccccc1)C1CCCC(CN(C(=O)Nc2ccc(F)cc2)c2cccc(OCCN3CCOCC3)c2)C1 10.1016/j.bmcl.2006.04.017
44380610 95966 0 None - 0 Human 8.1 pIC50 = 8.1 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 743 9 3 13 3.9 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
CHEMBL262052 95966 0 None - 0 Human 8.1 pIC50 = 8.1 Binding
Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)
ChEMBL 743 9 3 13 3.9 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)CC)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@]1(C)OC 10.1016/0960-894X(95)00122-A
44276817 97737 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL27419 97737 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor bindingConcentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution for motilin receptor binding
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44276817 97737 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL27419 97737 0 None - 0 Rabbit 8.1 pIC50 = 8.1 Binding
In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44276817 97737 0 None - 0 Rabbit 8.0 pIC50 = 8.0 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
CHEMBL27419 97737 0 None - 0 Rabbit 8.0 pIC50 = 8.0 Binding
Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80359-0
44276817 97737 0 None - 0 Rabbit 8.0 pIC50 = 8.0 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
CHEMBL27419 97737 0 None - 0 Rabbit 8.0 pIC50 = 8.0 Binding
In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateIn vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenate
ChEMBL 727 8 2 13 3.8 CCC1OC(=O)C(C)C(O[C@H]2C[C@@](C)(OC)[C@@H](O)C(C)O2)C(C)[C@@H](OC2OC(C)CC(N(C)C)[C@H]2O)[C@]2(C)CC(C)=C(O2)[C@H](C)C(=O)[C@]1(C)OC 10.1016/S0960-894X(01)80583-7
44412977 79389 0 None - 0 Rabbit 6.0 pIC50 = 6.0 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 686 11 1 5 7.4 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL212044 79389 0 None - 0 Rabbit 6.0 pIC50 = 6.0 Binding
Inhibition of [125]I-motilin binding to rabbit motilin receptorInhibition of [125]I-motilin binding to rabbit motilin receptor
ChEMBL 686 11 1 5 7.4 O=C(Nc1ccccc1)N(CC1CCCC(N(Cc2ccccc2)C(=O)C(Cl)(Cl)Cl)C1)c1cccc(OCCN2CCOCC2)c1 10.1016/j.bmcl.2006.04.017
CHEMBL2372767 208530 0 None - 1 Human 9.4 pKi = 9.4 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](N)Cc1ccccc1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](CCSC)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)O 10.1021/jm0606600
10010118 100952 0 None - 1 Human 9.2 pKi = 9.2 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL297494 100952 0 None - 1 Human 9.2 pKi = 9.2 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
10010118 100952 0 None - 1 Human 9.0 pKi = 9 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL297494 100952 0 None - 1 Human 9.0 pKi = 9 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
2139 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
2316 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
3836 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
638678 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
CHEMBL1472 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
DB09421 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None None 10.1016/j.bmc.2006.09.045
2139 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
2316 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
3836 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
638678 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
CHEMBL1472 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
DB09421 3782 51 None 1 4 Rat 8.0 pKi = 8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
ChEMBL None None None None 10.1021/jm0505462
25115428 160204 0 None - 1 Human 7.0 pKi = 7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 610 5 6 7 1.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN/C(N)=N/C#N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL411408 160204 0 None - 1 Human 7.0 pKi = 7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 610 5 6 7 1.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN/C(N)=N/C#N)NC1=O 10.1016/j.bmcl.2007.05.043
11444593 172147 0 None - 1 Human 8.0 pKi = 8.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 578 5 4 6 4.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2csc3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL450634 172147 0 None - 1 Human 8.0 pKi = 8.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 578 5 4 6 4.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2csc3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
44432981 87531 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 595 5 4 7 2.8 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cc2cscn2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL234191 87531 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 595 5 4 7 2.8 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cc2cscn2)NC1=O 10.1016/j.bmcl.2007.05.043
11995356 80126 0 None - 1 Human 5.9 pKi = 5.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 488 5 5 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCCCCCCNC1=O 10.1021/jm0606600
CHEMBL214869 80126 0 None - 1 Human 5.9 pKi = 5.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 488 5 5 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCCCCCCNC1=O 10.1021/jm0606600
CHEMBL223972 207692 0 None -3 2 Rat 7.9 pKi = 7.9 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None Cn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
11994554 80145 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL214935 80145 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11994554 80145 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL214935 80145 0 None - 1 Human 6.9 pKi = 6.9 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 536 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1016/j.bmcl.2007.05.043
11994677 141355 0 None - 1 Human 5.9 pKi = 5.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 508 3 5 6 1.8 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](C)NC1=O 10.1021/jm0606600
CHEMBL386854 141355 0 None - 1 Human 5.9 pKi = 5.9 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 508 3 5 6 1.8 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](C)NC1=O 10.1021/jm0606600
11995358 80173 0 None - 1 Human 5.8 pKi = 5.8 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 6 4 5 3.1 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](CCc2ccccc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL215043 80173 0 None - 1 Human 5.8 pKi = 5.8 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 6 4 5 3.1 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](CCc2ccccc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
44432973 97847 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 577 4 5 6 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL274876 97847 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 577 4 5 6 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
11995155 141364 0 None - 1 Human 5.8 pKi = 5.8 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 584 6 5 6 3.1 CCC[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL386906 141364 0 None - 1 Human 5.8 pKi = 5.8 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 584 6 5 6 3.1 CCC[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11410548 87123 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL233561 87123 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
25115652 96824 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 643 5 4 8 2.6 Cc1cnnn1C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL269007 96824 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 643 5 4 8 2.6 Cc1cnnn1C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL197149 207351 0 None - 1 Rat 4.8 pKi = 4.8 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH; Range = 0.12-0.24 uMInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH; Range = 0.12-0.24 uM
ChEMBL None None None CCCc1nc(C[C@H](NC(=O)[C@@H]2CCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1021/jm0505462
44432969 147058 0 None - 1 Human 6.8 pKi = 6.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 525 4 6 7 0.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393112 147058 0 None - 1 Human 6.8 pKi = 6.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 525 4 6 7 0.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
25114977 146464 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2cccn2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL392657 146464 0 None - 1 Human 7.8 pKi = 7.8 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2cccn2)NC1=O 10.1016/j.bmcl.2007.05.043
11994680 168189 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 584 5 5 6 3.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](Cc2ccccc2)NC1=O 10.1021/jm0606600
CHEMBL437326 168189 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 584 5 5 6 3.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](Cc2ccccc2)NC1=O 10.1021/jm0606600
11995359 168389 0 None - 1 Human 5.7 pKi = 5.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 539 5 4 7 2.9 CCC[C@@H]1OC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL438998 168389 0 None - 1 Human 5.7 pKi = 5.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 539 5 4 7 2.9 CCC[C@@H]1OC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
44467360 124002 0 None -3 2 Human 4.7 pKi = 4.7 Binding
Inhibition of human motilin receptorInhibition of human motilin receptor
ChEMBL 420 3 2 6 1.5 COc1nc(N2C[C@H]3C(=O)N(C)C(=N)N[C@@]3(c3ccc(F)cc3F)C2)nc(C)c1F 10.1021/acs.jmedchem.5b01995
CHEMBL3640290 124002 0 None -3 2 Human 4.7 pKi = 4.7 Binding
Inhibition of human motilin receptorInhibition of human motilin receptor
ChEMBL 420 3 2 6 1.5 COc1nc(N2C[C@H]3C(=O)N(C)C(=N)N[C@@]3(c3ccc(F)cc3F)C2)nc(C)c1F 10.1021/acs.jmedchem.5b01995
11994928 141325 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 539 5 4 7 2.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)OC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL386626 141325 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 539 5 4 7 2.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)OC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
44432971 86596 0 None - 1 Human 5.7 pKi = 5.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 567 5 6 7 0.8 CC(=O)NC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL232551 86596 0 None - 1 Human 5.7 pKi = 5.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 567 5 6 7 0.8 CC(=O)NC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
11995153 141091 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 508 4 5 6 1.9 CCC[C@@H]1NC(=O)[C@@H](C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL385293 141091 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 508 4 5 6 1.9 CCC[C@@H]1NC(=O)[C@@H](C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11181688 100852 0 None - 1 Human 8.7 pKi = 8.7 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 721 13 4 11 1.5 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL296748 100852 0 None - 1 Human 8.7 pKi = 8.7 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 721 13 4 11 1.5 NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
71720372 88610 0 None - 1 Human 8.6 pKi = 8.6 Binding
Agonist activity at MLNR (unknown origin)Agonist activity at MLNR (unknown origin)
ChEMBL 570 13 4 6 3.3 CCNC(=O)[C@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](Cc1ccc(F)cc1)NC 10.1021/jm301653f
CHEMBL2313632 88610 0 None - 1 Human 8.6 pKi = 8.6 Binding
Agonist activity at MLNR (unknown origin)Agonist activity at MLNR (unknown origin)
ChEMBL 570 13 4 6 3.3 CCNC(=O)[C@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](Cc1ccc(F)cc1)NC 10.1021/jm301653f
CHEMBL2364821 88610 0 None - 1 Human 8.6 pKi = 8.6 Binding
Agonist activity at MLNR (unknown origin)Agonist activity at MLNR (unknown origin)
ChEMBL 570 13 4 6 3.3 CCNC(=O)[C@H](Cc1ccc(O)c(C(C)(C)C)c1)C(N)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](Cc1ccc(F)cc1)NC 10.1021/jm301653f
44292517 101048 0 None - 1 Human 8.6 pKi = 8.6 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@@H](CCc1ccccc1)NC(=O)[C@@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL298224 101048 0 None - 1 Human 8.6 pKi = 8.6 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 723 13 4 11 1.7 NC(=O)[C@@H](CCc1ccccc1)NC(=O)[C@@H](CCc1ccccc1)NC(=O)C1CCC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
25115429 86259 0 None - 1 Human 7.7 pKi = 7.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 655 6 5 8 2.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNc2ncccn2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL231744 86259 0 None - 1 Human 7.7 pKi = 7.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 655 6 5 8 2.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNc2ncccn2)NC1=O 10.1016/j.bmcl.2007.05.043
25115653 146462 0 None - 1 Human 7.7 pKi = 7.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 644 5 4 9 2.0 Cc1nnnn1C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL392656 146462 0 None - 1 Human 7.7 pKi = 7.7 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 644 5 4 9 2.0 Cc1nnnn1C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL388528 210661 0 None -2 2 Rat 4.7 pKi = 4.7 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None C=CCn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
11250008 79988 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 566 5 4 6 3.0 CC(C)C[C@H]1C(=O)NCCCc2ccccc2OCCN[C@H](Cc2ccc(O)cc2)C(=O)N[C@H](C(C)C)C(=O)N1C 10.1021/jm0606600
CHEMBL214570 79988 0 None - 1 Human 6.7 pKi = 6.7 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 566 5 4 6 3.0 CC(C)C[C@H]1C(=O)NCCCc2ccccc2OCCN[C@H](Cc2ccc(O)cc2)C(=O)N[C@H](C(C)C)C(=O)N1C 10.1021/jm0606600
25115654 159445 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 657 5 4 8 2.9 Cc1nnn(C[C@@H]2NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc3cccc(C(F)(F)F)c3)NCCOc3ccccc3CCCNC2=O)c1C 10.1016/j.bmcl.2007.05.043
CHEMBL410786 159445 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 657 5 4 8 2.9 Cc1nnn(C[C@@H]2NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc3cccc(C(F)(F)F)c3)NCCOc3ccccc3CCCNC2=O)c1C 10.1016/j.bmcl.2007.05.043
11995042 141343 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 553 5 6 7 2.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NNC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL386735 141343 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 553 5 6 7 2.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NNC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11192254 141165 0 None - 1 Human 6.6 pKi = 6.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 561 5 5 5 3.2 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL385673 141165 0 None - 1 Human 6.6 pKi = 6.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 561 5 5 5 3.2 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11995157 168747 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 5 6 7 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CC(=O)O)NC1=O 10.1021/jm0606600
CHEMBL441697 168747 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 5 6 7 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CC(=O)O)NC1=O 10.1021/jm0606600
11995157 168747 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 552 5 6 7 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CC(=O)O)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL441697 168747 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 552 5 6 7 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CC(=O)O)NC1=O 10.1016/j.bmcl.2007.05.043
25115200 87803 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 584 6 6 6 2.3 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CCC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL234810 87803 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 584 6 6 6 2.3 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CCC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
44432976 154313 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL400635 154313 0 None - 1 Human 7.6 pKi = 7.6 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 571 5 4 6 2.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN(C)C)NC1=O 10.1016/j.bmcl.2007.05.043
11995454 141230 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 5 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)N(C)CCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL386086 141230 0 None - 1 Human 5.6 pKi = 5.6 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 5 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)N(C)CCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL224525 207693 0 None 1 2 Rat 6.5 pKi = 6.5 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None CCCc1nc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c[nH]1 10.1016/j.bmc.2006.09.045
CHEMBL2372767 208530 0 None - 1 Human 8.5 pKi = 8.5 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](N)Cc1ccccc1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](CCSC)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)O 10.1021/jm0304865
53322109 55961 0 None - 1 Human 8.5 pKi = 8.5 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm0304865
CHEMBL1628277 55961 0 None - 1 Human 8.5 pKi = 8.5 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 697 8 2 11 5.2 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)C[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)CC)[C@H]2O)[C@@]2(C)CC(C)=C(O2)[C@H](C)[C@@H](O)[C@H]1C 10.1021/jm0304865
44432974 87122 0 None - 1 Human 7.5 pKi = 7.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 557 5 5 6 1.8 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL233560 87122 0 None - 1 Human 7.5 pKi = 7.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 557 5 5 6 1.8 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
11995041 80057 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 5 5 6 2.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL214685 80057 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 5 5 6 2.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11995357 140907 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 528 5 4 5 3.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](CC2CCCCC2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL384204 140907 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 528 5 4 5 3.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](CC2CCCCC2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
25114744 160206 0 None - 1 Human 7.5 pKi = 7.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 599 6 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CCNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL411409 160206 0 None - 1 Human 7.5 pKi = 7.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 599 6 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CCNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
11994678 140844 0 None - 1 Human 6.5 pKi = 6.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 6 2.5 CCC[C@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL383881 140844 0 None - 1 Human 6.5 pKi = 6.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 6 2.5 CCC[C@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL390942 210691 0 None -3 2 Rat 7.5 pKi = 7.5 Binding
Displacement of [3H]N(1)-Me-His-TRH from TRHR2Displacement of [3H]N(1)-Me-His-TRH from TRHR2
ChEMBL None None None CCn1cnc(C[C@H](NC(=O)[C@@H]2CCCC(=O)N2)C(=O)N2CCC[C@H]2C(N)=O)c1 10.1016/j.bmc.2006.09.045
44432968 86507 0 None - 1 Human 6.5 pKi = 6.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 539 5 6 7 1.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CCN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL232342 86507 0 None - 1 Human 6.5 pKi = 6.5 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 539 5 6 7 1.0 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CCN)NC1=O 10.1016/j.bmcl.2007.05.043
11994556 80063 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 472 4 4 5 2.2 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](C(C)C)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL214703 80063 0 None - 1 Human 5.5 pKi = 5.5 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 472 4 4 5 2.2 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](C(C)C)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
1048 1548 72 None - 1 Human 4.4 pKi = 4.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
12560 1548 72 None - 1 Human 4.4 pKi = 4.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
1456 1548 72 None - 1 Human 4.4 pKi = 4.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
CHEMBL532 1548 72 None - 1 Human 4.4 pKi = 4.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
DB00199 1548 72 None - 1 Human 4.4 pKi = 4.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O 10.1021/jm0304865
44432970 86595 0 None - 1 Human 6.4 pKi = 6.4 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 567 6 6 7 1.7 CC(C)NC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL232550 86595 0 None - 1 Human 6.4 pKi = 6.4 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 567 6 6 7 1.7 CC(C)NC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
23656869 147311 0 None - 1 Human 8.3 pKi = 8.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 631 5 4 6 3.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN2CCCC2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393315 147311 0 None - 1 Human 8.3 pKi = 8.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 631 5 4 6 3.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN2CCCC2)NC1=O 10.1016/j.bmcl.2007.05.043
44432979 147973 0 None - 1 Human 7.4 pKi = 7.4 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 626 6 5 8 3.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNc2nccs2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393842 147973 0 None - 1 Human 7.4 pKi = 7.4 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 626 6 5 8 3.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNc2nccs2)NC1=O 10.1016/j.bmcl.2007.05.043
11398860 175461 0 None - 1 Human 5.4 pKi = 5.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL45905 175461 0 None - 1 Human 5.4 pKi = 5.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
11995154 80661 0 None - 1 Human 5.3 pKi = 5.3 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 566 7 6 7 1.7 CCC[C@@H]1NC(=O)[C@@H](CCC(=O)O)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL215532 80661 0 None - 1 Human 5.3 pKi = 5.3 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 566 7 6 7 1.7 CCC[C@@H]1NC(=O)[C@@H](CCC(=O)O)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
25115201 158216 0 None - 1 Human 7.3 pKi = 7.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 611 5 6 8 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC2=NCCN2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL409410 158216 0 None - 1 Human 7.3 pKi = 7.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 611 5 6 8 1.2 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC2=NCCN2)NC1=O 10.1016/j.bmcl.2007.05.043
44432978 86532 0 None - 1 Human 6.3 pKi = 6.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 586 5 6 6 1.3 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(N)=O)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL232359 86532 0 None - 1 Human 6.3 pKi = 6.3 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 586 5 6 6 1.3 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(N)=O)NC1=O 10.1016/j.bmcl.2007.05.043
11226476 80748 0 None - 1 Human 7.3 pKi = 7.3 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 538 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL215825 80748 0 None - 1 Human 7.3 pKi = 7.3 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 538 5 5 6 2.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11994925 80638 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 522 5 4 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccccc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL215440 80638 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 522 5 4 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccccc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
44432980 146351 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 585 5 7 6 1.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL392553 146351 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 585 5 7 6 1.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
11398860 175461 0 None - 1 Human 5.2 pKi = 5.2 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
CHEMBL45905 175461 0 None - 1 Human 5.2 pKi = 5.2 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
ChEMBL 560 8 3 10 0.4 NC(=O)[C@H](CCc1ccccc1)NC(=O)C1C=CC2(CCNCC2)n2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)n21 10.1021/jm0304865
11204067 86344 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 585 5 7 6 1.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL232154 86344 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 585 5 7 6 1.1 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
44432975 87298 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 591 5 5 6 2.2 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL233711 87298 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 591 5 5 6 2.2 CNC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC1=O 10.1016/j.bmcl.2007.05.043
44432977 151136 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 619 5 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL396413 151136 0 None - 1 Human 8.2 pKi = 8.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 619 5 7 6 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(C(F)(F)F)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC(=N)N)NC1=O 10.1016/j.bmcl.2007.05.043
11168753 144406 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 543 4 5 6 1.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL391045 144406 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 543 4 5 6 1.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(Cl)cc2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
11994802 81031 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 5 3.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCCc2ccccc2CCNC1=O 10.1021/jm0606600
CHEMBL215963 81031 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 5 3.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCCc2ccccc2CCNC1=O 10.1021/jm0606600
11994800 141248 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 5 3.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCc2ccccc2CCCCNC1=O 10.1021/jm0606600
CHEMBL386187 141248 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 536 5 5 5 3.0 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCc2ccccc2CCCCNC1=O 10.1021/jm0606600
11180385 80990 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 550 5 5 6 2.8 CC(C)C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL215946 80990 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 550 5 5 6 2.8 CC(C)C[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
25114976 147469 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2ccnc2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393439 147469 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 594 5 4 7 2.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2ccnc2)NC1=O 10.1016/j.bmcl.2007.05.043
44417633 140905 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 580 5 4 6 2.7 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)N(C(C)=O)CCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL384188 140905 0 None - 1 Human 5.2 pKi = 5.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 580 5 4 6 2.7 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)N(C(C)=O)CCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11398651 147586 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 543 4 5 6 1.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL393541 147586 0 None - 1 Human 7.2 pKi = 7.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 543 4 5 6 1.6 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CN)NC1=O 10.1016/j.bmcl.2007.05.043
11995156 141220 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 4 6 7 0.7 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CO)NC1=O 10.1021/jm0606600
CHEMBL386036 141220 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 4 6 7 0.7 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CO)NC1=O 10.1021/jm0606600
11994679 79969 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 565 7 6 7 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCCN)NC1=O 10.1021/jm0606600
CHEMBL214508 79969 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 565 7 6 7 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCCN)NC1=O 10.1021/jm0606600
11994679 79969 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 565 7 6 7 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCCN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL214508 79969 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 565 7 6 7 1.9 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCCN)NC1=O 10.1016/j.bmcl.2007.05.043
11994924 79985 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 444 5 5 5 1.4 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NC/C=C/CCNC1=O 10.1021/jm0606600
CHEMBL214555 79985 0 None - 1 Human 6.2 pKi = 6.2 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 444 5 5 5 1.4 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NC/C=C/CCNC1=O 10.1021/jm0606600
44417743 165543 0 None - 1 Human 5.1 pKi = 5.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 548 5 5 5 3.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCc2ccccc2/C=C\CCNC1=O 10.1021/jm0606600
CHEMBL425988 165543 0 None - 1 Human 5.1 pKi = 5.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 548 5 5 5 3.5 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCCc2ccccc2/C=C\CCNC1=O 10.1021/jm0606600
11203197 80166 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 520 5 4 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccccc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL215016 80166 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 520 5 4 5 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccccc2)NCCOc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11994927 81338 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 572 5 4 5 3.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL216400 81338 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 572 5 4 5 3.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11341873 140960 0 None - 1 Human 8.1 pKi = 8.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 6 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(OC)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL384501 140960 0 None - 1 Human 8.1 pKi = 8.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 552 6 4 6 2.8 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(OC)cc2)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
11433096 141059 0 None - 1 Human 8.1 pKi = 8.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 572 5 4 5 3.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
CHEMBL385087 141059 0 None - 1 Human 8.1 pKi = 8.1 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 572 5 4 5 3.9 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2cccc3ccccc23)NCCOc2ccccc2CCCNC1=O 10.1021/jm0606600
25115427 98192 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 625 5 6 8 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC2=NCCCN2)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL277329 98192 0 None - 1 Human 7.1 pKi = 7.1 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 625 5 6 8 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(Cl)c2)NCCOc2ccccc2CCCNC(=O)[C@H](CNC2=NCCCN2)NC1=O 10.1016/j.bmcl.2007.05.043
44432967 145026 0 None - 1 Human 6.1 pKi = 6.1 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 551 6 6 7 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCN)NC1=O 10.1016/j.bmcl.2007.05.043
CHEMBL391524 145026 0 None - 1 Human 6.1 pKi = 6.1 Binding
Displacement of [125I]motilin from human motilin receptor expressed in CHO cellsDisplacement of [125I]motilin from human motilin receptor expressed in CHO cells
ChEMBL 551 6 6 7 1.5 CC(C)[C@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2/C=C/CNC(=O)[C@H](CCCN)NC1=O 10.1016/j.bmcl.2007.05.043
11995259 80341 0 None - 1 Human 5.0 pKi = 5.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 520 5 5 5 2.7 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
CHEMBL215177 80341 0 None - 1 Human 5.0 pKi = 5.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 520 5 5 5 2.7 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCc2ccccc2/C=C/CNC1=O 10.1021/jm0606600
11995261 80339 0 None - 1 Human 6.0 pKi = 6.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 5 5 6 2.1 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCNC1=O 10.1021/jm0606600
CHEMBL215169 80339 0 None - 1 Human 6.0 pKi = 6.0 Binding
Displacement of [125I]motilin from human MOTRDisplacement of [125I]motilin from human MOTR
ChEMBL 524 5 5 6 2.1 CCC[C@@H]1NC(=O)[C@@H](C(C)C)NC(=O)[C@@H](Cc2ccc(O)cc2)NCCOc2ccccc2CCNC1=O 10.1021/jm0606600
101635584 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1458 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
16136567 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
3794 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
91898963 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
CHEMBL525634 2548 26 None - 1 Human 10.0 pKd = 10 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10381885
1048 1548 72 None - 1 Human 8.4 pKi = 8.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
Drug Central 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O None
12560 1548 72 None - 1 Human 8.4 pKi = 8.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
Drug Central 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O None
1456 1548 72 None - 1 Human 8.4 pKi = 8.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
Drug Central 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O None
CHEMBL532 1548 72 None - 1 Human 8.4 pKi = 8.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
Drug Central 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O None
DB00199 1548 72 None - 1 Human 8.4 pKi = 8.4 Binding
In vitro binding affinity towards human motilin receptorIn vitro binding affinity towards human motilin receptor
Drug Central 733 7 5 14 1.8 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2O[C@@H](C)[C@@H]([C@](C2)(C)OC)O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C[C@H](C(=O)[C@@H]([C@H]([C@]1(C)O)O)C)C)(C)O None
2139 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
2316 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
3836 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
638678 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
CHEMBL1472 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
DB09421 3782 51 None 1 4 Rat 8.1 pKi = 8.1 Binding
Inhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRHInhibitory constant against thyrotropin releasing hormone receptor 2 expressed in HEK 293EM cells upon incubation at 37 degree C for 1 hr at pH 7.4 using [3H]Ntau(1)-Me-His-TRH
Drug Central None None None None None
101635584 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
101635584 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
101635584 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
101635584 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
1458 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
1458 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
1458 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
1458 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
16136567 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
16136567 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
16136567 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
16136567 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
3794 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
3794 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
3794 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
3794 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
91898963 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
91898963 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
91898963 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
91898963 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
CHEMBL525634 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914
CHEMBL525634 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11781320
CHEMBL525634 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
CHEMBL525634 2548 26 None - 1 Human 8.6 pKi = 8.6 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 16531413
1450 3555 0 None - 1 Human 6.4 pKi None 6.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
1451 3558 0 None - 1 Human 7.3 pKi None 7.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15677347
1452 700 0 None - 1 Human 7.9 pKi None 7.9 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11461914