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Ligand source activities (1 row/activity)

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	90012275	133115	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	416	6	2	3	5.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(C)(C)C)c1	nan
	CHEMBL3714858	133115	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	416	6	2	3	5.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(C)(C)C)c1	nan
	56593334	133585	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716462	133585	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90011833	133765	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc([N+](=O)[O-])c1	nan
	CHEMBL3717071	133765	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc([N+](=O)[O-])c1	nan
	56593330	133850	0	None	-	1	Human	6.9	pAC50	=	6.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717389	133850	0	None	-	1	Human	6.9	pAC50	=	6.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593346	133795	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	nan
	CHEMBL3717178	133795	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	nan
	90010727	133278	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	487	6	2	4	4.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cncc(I)c1	nan
	CHEMBL3715451	133278	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	487	6	2	4	4.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cncc(I)c1	nan
	118037864	133346	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	3	3	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2nc[nH]c12	nan
	CHEMBL3715676	133346	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	3	3	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2nc[nH]c12	nan
	2806493	133582	4	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	nan
	CHEMBL3716450	133582	4	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	nan
	118037922	134150	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	612	8	2	6	6.1	CC(C)(C)OC(=O)N1CCN(CCOc2ccccc2C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	CHEMBL3718384	134150	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	612	8	2	6	6.1	CC(C)(C)OC(=O)N1CCN(CCOc2ccccc2C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	90010869	134329	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	392	6	2	4	4.9	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC)c1	nan
	CHEMBL3718995	134329	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	392	6	2	4	4.9	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC)c1	nan
	38269206	134144	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718363	134144	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010751	133836	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C\c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	CHEMBL3717338	133836	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C\c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	90012348	134050	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3718077	134050	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc([N+](=O)[O-])cc1	nan
	90010773	133375	0	None	-1	2	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	375	4	2	4	4.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccno1	nan
	CHEMBL3715750	133375	0	None	-1	2	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	375	4	2	4	4.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccno1	nan
	90011033	134337	0	None	-	1	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2ccccc2c1	nan
	CHEMBL3719015	134337	0	None	-	1	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2ccccc2c1	nan
	56593309	133226	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715203	133226	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90011788	133290	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3715489	133290	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	90012098	134044	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Br)c1	nan
	CHEMBL3718061	134044	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Br)c1	nan
	56593314	133804	0	None	-	1	Human	6.7	pAC50	=	6.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717211	133804	0	None	-	1	Human	6.7	pAC50	=	6.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593340	133564	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3716394	133564	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1313624	133912	8	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Cl)c1	nan
	CHEMBL3717590	133912	8	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Cl)c1	nan
	56593311	133951	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717723	133951	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	24671974	134256	2	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	3	5.3	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccs1	nan
	CHEMBL3718728	134256	2	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	3	5.3	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccs1	nan
	90012130	133149	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3714976	133149	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	90010778	133677	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C/c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	CHEMBL3716808	133677	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C/c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	56593317	134412	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	nan
	CHEMBL3719257	134412	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	nan
	40622265	133344	2	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	374	4	2	3	4.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccco1	nan
	CHEMBL3715664	133344	2	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	374	4	2	3	4.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccco1	nan
	127024729	133940	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	500	7	2	6	4.0	CCOc1ccccc1C(=O)NC1SC=CC1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717683	133940	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	500	7	2	6	4.0	CCOc1ccccc1C(=O)NC1SC=CC1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010630	134261	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.7	CC1CCC(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	CHEMBL3718740	134261	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.7	CC1CCC(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	5298634	134422	10	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	nan
	CHEMBL3719295	134422	10	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	nan
	56593335	133769	0	None	-	1	Human	6.6	pAC50	=	6.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717089	133769	0	None	-	1	Human	6.6	pAC50	=	6.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011775	133136	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Cl)cc1	nan
	CHEMBL3714926	133136	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Cl)cc1	nan
	90011735	133234	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	511	8	2	4	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCCCC1	nan
	CHEMBL3715244	133234	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	511	8	2	4	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCCCC1	nan
	56593308	133623	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716596	133623	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593324	133680	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	8	2	5	5.2	CCOc1ccccc1C(=O)Nc1ccccc1CNc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3716811	133680	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	8	2	5	5.2	CCOc1ccccc1C(=O)Nc1ccccc1CNc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593333	133699	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716871	133699	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593350	134111	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3718273	134111	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	56593315	133776	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3717103	133776	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	90010752	133159	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	448	4	2	2	5.1	O=C(Nc1cccc(I)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3714999	133159	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	448	4	2	2	5.1	O=C(Nc1cccc(I)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90011874	133176	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1	nan
	CHEMBL3715040	133176	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1	nan
	56593323	133200	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715105	133200	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593318	133596	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	nan
	CHEMBL3716512	133596	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	nan
	90010791	133736	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccccn1	nan
	CHEMBL3716987	133736	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccccn1	nan
	56593313	134315	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	nan
	CHEMBL3718895	134315	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	nan
	56593329	133897	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717553	133897	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593336	133307	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715551	133307	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593337	133196	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	nan
	CHEMBL3715097	133196	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	nan
	127024591	133207	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	457	8	3	4	4.8	CNCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715139	133207	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	457	8	3	4	4.8	CNCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	2233108	133933	9	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3717655	133933	9	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1511185	133301	12	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3715535	133301	12	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	4795548	133701	6	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3716878	133701	6	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	32157880	133707	5	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1ccc(F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716901	133707	5	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1ccc(F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010785	133151	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	574	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1I	nan
	CHEMBL3714984	133151	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	574	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1I	nan
	118043134	133199	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	4	2	2	7.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	CHEMBL3715104	133199	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	4	2	2	7.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	21179517	133413	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	2	2	6.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715901	133413	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	2	2	6.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1cccc(C(F)(F)F)c1	nan
	56593306	133758	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717045	133758	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90012794	133976	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Br)cc1	nan
	CHEMBL3717803	133976	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Br)cc1	nan
	54784887	134146	2	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1ccccc1	nan
	CHEMBL3718373	134146	2	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1ccccc1	nan
	1313916	39841	8	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1479446	39841	8	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593322	133189	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715081	133189	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593331	134190	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718541	134190	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011206	133273	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	513	8	2	5	4.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCOCC1	nan
	CHEMBL3715429	133273	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	513	8	2	5	4.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCOCC1	nan
	56593347	133303	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715539	133303	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010797	133329	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	4	2	2	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C12CC3CC(CC(C3)C1)C2	nan
	CHEMBL3715615	133329	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	4	2	2	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C12CC3CC(CC(C3)C1)C2	nan
	4484023	133733	6	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3716976	133733	6	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	56593338	134195	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	8	2	5	3.1	CCOc1ccccc1C(=O)NCCC(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3718557	134195	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	8	2	5	3.1	CCOc1ccccc1C(=O)NCCC(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593307	134285	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	386	5	2	3	5.7	COc1ccccc1Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718811	134285	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	386	5	2	3	5.7	COc1ccccc1Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011315	133669	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	370	5	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1ccccc1	nan
	CHEMBL3716765	133669	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	370	5	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1ccccc1	nan
	127024076	133953	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	308	4	2	2	3.5	O=CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717734	133953	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	308	4	2	2	3.5	O=CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010896	133993	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	438	5	2	2	6.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717869	133993	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	438	5	2	2	6.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1cccc(C(F)(F)F)c1	nan
	56593316	133232	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715235	133232	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593341	133299	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	508	7	2	5	5.6	CCSc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715526	133299	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	508	7	2	5	5.6	CCSc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010758	133281	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	5	2	2	6.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(-c2ccccc2)c1	nan
	CHEMBL3715462	133281	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	5	2	2	6.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(-c2ccccc2)c1	nan
	56593299	133477	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3716127	133477	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	56593339	133589	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716488	133589	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593319	133681	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716813	133681	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010729	133687	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	6	2	4	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(N2CCCCC2)c1	nan
	CHEMBL3716829	133687	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	6	2	4	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(N2CCCCC2)c1	nan
	90010865	134186	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	380	3	2	3	5.3	CC(C)(C)OC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718514	134186	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	380	3	2	3	5.3	CC(C)(C)OC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010599	134426	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	5	2	2	5.6	CC(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3719301	134426	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	5	2	2	5.6	CC(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	90011364	133523	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	5	2	2	6.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCC1CCCCC1	nan
	CHEMBL3716260	133523	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	5	2	2	6.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCC1CCCCC1	nan
	90011496	133613	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2ccccc12	nan
	CHEMBL3716563	133613	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2ccccc12	nan
	90011579	133734	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(C(F)(F)F)cc1	nan
	CHEMBL3716978	133734	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(C(F)(F)F)cc1	nan
	56593303	134081	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	nan
	CHEMBL3718178	134081	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	nan
	60288826	134112	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	426	5	2	3	5.4	CC(=O)c1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3718279	134112	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	426	5	2	3	5.4	CC(=O)c1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	56593326	134211	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718612	134211	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593302	133240	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715266	133240	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011338	133256	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	485	9	2	4	5.5	CN(C)CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715346	133256	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	485	9	2	4	5.5	CN(C)CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593298	133946	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	6	2	3	5.6	COc1ccccc1CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717700	133946	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	6	2	3	5.6	COc1ccccc1CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010708	133759	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	6	2	4	4.5	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C#N)c1	nan
	CHEMBL3717047	133759	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	6	2	4	4.5	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C#N)c1	nan
	118043136	134389	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	7	2	4	6.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3719197	134389	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	7	2	4	6.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	90010848	133198	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	6	2	5	3.6	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(C)(=O)=O)c1	nan
	CHEMBL3715101	133198	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	6	2	5	3.6	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(C)(=O)=O)c1	nan
	90010777	134041	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	346	4	2	2	4.4	C#Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3718054	134041	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	346	4	2	2	4.4	C#Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	118037818	134173	0	None	-1	2	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	4	2	4	4.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL3718470	134173	0	None	-1	2	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	4	2	4	4.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)OCO2	nan
	56593305	134154	0	None	-	1	Human	7.2	pAC50	=	7.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	CHEMBL3718400	134154	0	None	-	1	Human	7.2	pAC50	=	7.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	90010645	133255	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	486	6	2	3	5.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(I)c1	nan
	CHEMBL3715345	133255	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	486	6	2	3	5.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(I)c1	nan
	56593345	133371	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715743	133371	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593320	133606	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716540	133606	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011367	134238	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	476	6	2	3	7.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1Oc1ccccc1	nan
	CHEMBL3718664	134238	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	476	6	2	3	7.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1Oc1ccccc1	nan
	56593296	133621	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716581	133621	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011087	133737	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1C(F)(F)F	nan
	CHEMBL3716990	133737	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1C(F)(F)F	nan
	90011219	134122	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	510	4	2	2	5.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1I	nan
	CHEMBL3718291	134122	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	510	4	2	2	5.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1I	nan
	90011247	134180	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Br	nan
	CHEMBL3718498	134180	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Br	nan
	52764307	134332	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccncc1	nan
	CHEMBL3719005	134332	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccncc1	nan
	90010748	133201	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1ccc([N+](=O)[O-])cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715107	133201	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1ccc([N+](=O)[O-])cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010731	133358	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccncc1	nan
	CHEMBL3715708	133358	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccncc1	nan
	3348337	133913	1	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	3	2	2	3.9	CC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717591	133913	1	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	3	2	2	3.9	CC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	29448220	134326	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	366	4	2	4	4.2	O=C(Nc1ccc2c(c1)OCO2)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718975	134326	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	366	4	2	4	4.2	O=C(Nc1ccc2c(c1)OCO2)c1ccccc1NC(=O)C1CCCCC1	nan
	56593344	133161	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715001	133161	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593325	134231	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	nan
	CHEMBL3718643	134231	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	nan
	56593349	2524	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	8322	2524	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	CHEMBL3716980	2524	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	90011702	133216	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.9	O=C(Nc1ccc2c(c1)CCC2)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715166	133216	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.9	O=C(Nc1ccc2c(c1)CCC2)c1ccccc1NC(=O)C1CCCCC1	nan
	56593321	133950	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717718	133950	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	nan
	90011489	134063	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	6	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCCc1ccccc1	nan
	CHEMBL3718114	134063	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	6	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCCc1ccccc1	nan
	60589025	134259	1	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	5	2	4	4.6	CS(=O)(=O)c1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3718735	134259	1	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	5	2	4	4.6	CS(=O)(=O)c1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1320335	134286	9	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3718813	134286	9	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	730108	41283	15	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1491180	41283	15	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593342	133881	0	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717485	133881	0	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	162654489	180043	0	None	4	2	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180043	0	None	4	2	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162648163	179283	0	None	-	1	Human	10.0	pEC50	=	10	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4745611	179283	0	None	-	1	Human	10.0	pEC50	=	10	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672427	182607	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4795810	182607	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162667576	181892	0	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4786789	181892	0	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654489	180043	0	None	4	2	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180043	0	None	4	2	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162677247	182938	0	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	CHEMBL4799907	182938	0	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	162661030	180857	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4764326	180857	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162674882	182760	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797641	182760	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593316	133232	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715235	133232	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593334	133585	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716462	133585	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593305	134154	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	CHEMBL3718400	134154	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	56593346	133795	0	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	10.1016/j.ejmech.2018.06.008
	CHEMBL3717178	133795	0	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	10.1016/j.ejmech.2018.06.008
	162664297	181489	0	None	-2	2	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781560	181489	0	None	-2	2	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593322	133189	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715081	133189	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	162649438	179462	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3412	125	54	48	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4747756	179462	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3412	125	54	48	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	2806493	133582	4	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716450	133582	4	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	10.1016/j.ejmech.2018.06.008
	38269206	134144	0	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718363	134144	0	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	162659815	180608	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2785	100	45	39	-13.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4761130	180608	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2785	100	45	39	-13.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162666079	181721	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2855	106	46	40	-12.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4784237	181721	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2855	106	46	40	-12.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162656358	180297	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3355	121	53	47	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4757578	180297	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3355	121	53	47	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162677445	182951	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3139	113	49	43	-12.2	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4800116	182951	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3139	113	49	43	-12.2	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593309	133226	0	None	-	1	Human	5.8	pEC50	=	5.8	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715203	133226	0	None	-	1	Human	5.8	pEC50	=	5.8	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162646950	179089	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3195	119	50	44	-12.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4743539	179089	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3195	119	50	44	-12.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162643258	181150	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3411	126	53	47	-12.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NCC(C)C(=O)NCC(C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4777259	181150	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3411	126	53	47	-12.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NCC(C)C(=O)NCC(C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/acs.jmedchem.0c01533
	162674863	182721	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3509	135	52	47	-9.4	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797258	182721	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3509	135	52	47	-9.4	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162662427	181366	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3383	123	53	47	-14.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4779982	181366	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3383	123	53	47	-14.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162648609	179225	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3292	122	50	45	-12.0	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4744987	179225	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3292	122	50	45	-12.0	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672427	182607	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4795810	182607	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593314	133804	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717211	133804	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593330	133850	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717389	133850	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	1313916	39841	8	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL1479446	39841	8	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593340	133564	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716394	133564	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	10.1016/j.ejmech.2018.06.008
	56593311	133951	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717723	133951	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	162650672	179566	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3152	116	49	43	-12.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748931	179566	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3152	116	49	43	-12.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162648163	179283	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4745611	179283	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593349	2524	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	8322	2524	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	CHEMBL3716980	2524	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	162659417	180634	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3257	114	52	46	-15.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4761424	180634	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3257	114	52	46	-15.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162670766	182360	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3097	111	49	43	-13.1	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4792874	182360	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3097	111	49	43	-13.1	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593317	134412	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3719257	134412	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	10.1016/j.ejmech.2018.06.008
	162654519	180078	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2828	103	46	40	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4755239	180078	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2828	103	46	40	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654037	180082	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3424	126	53	47	-12.7	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4755289	180082	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3424	126	53	47	-12.7	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	5298634	134422	10	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3719295	134422	10	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	10.1016/j.ejmech.2018.06.008
	56593332	161689	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	498	7	2	6	4.9	CCOc1ccccc1C(=O)Nc1sccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL4163593	161689	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	498	7	2	6	4.9	CCOc1ccccc1C(=O)Nc1sccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162667576	181892	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4786789	181892	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593335	133769	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717089	133769	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593308	133623	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716596	133623	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593333	133699	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716871	133699	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593350	134111	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718273	134111	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	162672610	182424	0	None	-35	2	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182424	0	None	-35	2	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593323	133200	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715105	133200	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593318	133596	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716512	133596	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	10.1016/j.ejmech.2018.06.008
	56593313	134315	0	None	-	1	Human	4.5	pEC50	=	4.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718895	134315	0	None	-	1	Human	4.5	pEC50	=	4.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162652974	179826	0	None	-	1	Human	8.5	pEC50	=	8.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4163	175	54	60	-9.4	CCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4752287	179826	0	None	-	1	Human	8.5	pEC50	=	8.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4163	175	54	60	-9.4	CCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672610	182424	0	None	-35	2	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182424	0	None	-35	2	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162674882	182760	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797641	182760	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162669540	182047	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2867	105	45	40	-11.9	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4788675	182047	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2867	105	45	40	-11.9	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162670803	182244	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3314	119	53	47	-14.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4791290	182244	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3314	119	53	47	-14.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593329	133897	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717553	133897	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593336	133307	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715551	133307	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593314	133804	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717211	133804	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593330	133850	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717389	133850	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	162648114	179325	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4489	180	64	59	-8.3	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4746080	179325	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4489	180	64	59	-8.3	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162649375	179530	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3327	120	53	47	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748601	179530	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3327	120	53	47	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593337	133196	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	10.1016/j.ejmech.2018.06.008
	CHEMBL3715097	133196	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	10.1016/j.ejmech.2018.06.008
	56593300	161640	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	471	8	2	4	5.2	CN(C)CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL4162685	161640	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	471	8	2	4	5.2	CN(C)CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	1511185	133301	12	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715535	133301	12	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	4795548	133701	6	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716878	133701	6	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	162646638	179124	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3055	109	49	43	-14.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4743958	179124	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3055	109	49	43	-14.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593306	133758	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717045	133758	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162644941	178810	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2883	107	46	40	-11.8	CC[C@H](C)[C@H](NC(=O)C(C)CNC(=O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4739969	178810	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2883	107	46	40	-11.8	CC[C@H](C)[C@H](NC(=O)C(C)CNC(=O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162649856	179549	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3481	130	54	48	-12.8	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748830	179549	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3481	130	54	48	-12.8	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162663002	181456	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3122	115	48	43	-11.7	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781139	181456	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3122	115	48	43	-11.7	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162655145	180166	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3166	116	49	43	-11.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4756139	180166	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3166	116	49	43	-11.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	56593322	133189	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715081	133189	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	47936	192809	82	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	410	2	3	7	1.5	C=C[C@@]1(C)CC(=O)[C@@]2(O)[C@](C)(O1)[C@@H](OC(C)=O)[C@@H](O)[C@H]1C(C)(C)CC[C@H](O)[C@@]12C	10.1016/j.ejmech.2018.06.008
	CHEMBL52606	192809	82	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	410	2	3	7	1.5	C=C[C@@]1(C)CC(=O)[C@@]2(O)[C@](C)(O1)[C@@H](OC(C)=O)[C@@H](O)[C@H]1C(C)(C)CC[C@H](O)[C@@]12C	10.1016/j.ejmech.2018.06.008
	56593331	134190	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718541	134190	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593335	133769	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717089	133769	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593347	133303	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715539	133303	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162654330	179164	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3299	116	52	46	-14.6	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4744303	179164	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3299	116	52	46	-14.6	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593316	133232	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715235	133232	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162654892	180028	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3083	110	49	43	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754697	180028	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3083	110	49	43	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593315	133776	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3717103	133776	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	56593299	133477	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716127	133477	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	56593339	133589	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716488	133589	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593319	133681	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716813	133681	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162670817	182257	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3209	121	50	44	-11.0	CC[C@H](C)[C@H](NC[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4791486	182257	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3209	121	50	44	-11.0	CC[C@H](C)[C@H](NC[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	56593303	134081	1	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718178	134081	1	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	10.1016/j.ejmech.2018.06.008
	56593326	134211	0	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718612	134211	0	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593302	133240	0	None	-	1	Human	4.2	pEC50	=	4.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715266	133240	0	None	-	1	Human	4.2	pEC50	=	4.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593305	134154	0	None	-	1	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	10.1016/j.ejmech.2018.06.008
	CHEMBL3718400	134154	0	None	-	1	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	10.1016/j.ejmech.2018.06.008
	162656612	180325	0	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3041	106	48	42	-13.3	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4757890	180325	0	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3041	106	48	42	-13.3	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593345	133371	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715743	133371	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593320	133606	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716540	133606	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593296	133621	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716581	133621	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162662592	181377	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4780098	181377	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162675717	182685	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4461	178	64	59	-9.0	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4796713	182685	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4461	178	64	59	-9.0	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593344	133161	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715001	133161	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593325	134231	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718643	134231	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	10.1016/j.ejmech.2018.06.008
	162661030	180857	0	None	-	1	Human	7.1	pEC50	=	7.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4764326	180857	0	None	-	1	Human	7.1	pEC50	=	7.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162661521	180938	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3341	120	53	47	-14.6	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4765167	180938	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3341	120	53	47	-14.6	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162677247	182938	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	CHEMBL4799907	182938	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	162666829	181833	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3069	110	49	43	-13.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4785899	181833	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3069	110	49	43	-13.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162664515	181483	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3027	105	48	42	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781482	181483	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3027	105	48	42	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593349	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	8322	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	CHEMBL3716980	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	56593321	133950	0	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717718	133950	0	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	1320335	134286	9	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718813	134286	9	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	10.1016/j.ejmech.2018.06.008
	730108	41283	15	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL1491180	41283	15	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593342	133881	0	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717485	133881	0	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	820020	21611	7	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	2	2	3	1.6	O=C(NN=C1CCCC1)c1[nH]nc2c1CCC2	nan
	CHEMBL1319564	21611	7	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	2	2	3	1.6	O=C(NN=C1CCCC1)c1[nH]nc2c1CCC2	nan
	2146184	44300	10	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	4	2.4	CN(C)c1ccc(C(=S)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc1	nan
	CHEMBL1519935	44300	10	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	4	2.4	CN(C)c1ccc(C(=S)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc1	nan
	1761	99202	9	None	-	1	Human	6.0	pPotency	=	6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	4	9	-1.7	Nc1ncnc2c1ncn2C1OC(C(=O)NC2CC2)C(O)C1O	nan
	CHEMBL28449	99202	9	None	-	1	Human	6.0	pPotency	=	6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	4	9	-1.7	Nc1ncnc2c1ncn2C1OC(C(=O)NC2CC2)C(O)C1O	nan
	16019574	10765	10	None	-14	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(F)cc1)c1sccc12	nan
	CHEMBL1172596	10765	10	None	-14	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(F)cc1)c1sccc12	nan
	4132952	19456	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	11	0.2	CCOP1(=O)OCC2OC(n3cnc4c(N)ncnc43)C(O)C2O1	nan
	CHEMBL1300691	19456	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	11	0.2	CCOP1(=O)OCC2OC(n3cnc4c(N)ncnc43)C(O)C2O1	nan
	54677759	20875	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	3	4.1	O=c1c(Cc2ccccc2)c(O)c2cccc3c4c(n1c23)CCCC4	nan
	CHEMBL1312172	20875	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	3	4.1	O=c1c(Cc2ccccc2)c(O)c2cccc3c4c(n1c23)CCCC4	nan
	16027480	21308	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	CHEMBL1316197	21308	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	941768	21876	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	3	7	-0.5	O=C1NC(=O)C(=NNc2ccc3c(c2)COC3=O)C(=O)N1	nan
	CHEMBL1321879	21876	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	3	7	-0.5	O=C1NC(=O)C(=NNc2ccc3c(c2)COC3=O)C(=O)N1	nan
	2764158	22431	30	None	-2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	2	1	5	2.7	CSc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1326901	22431	30	None	-2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	2	1	5	2.7	CSc1ccccc1-c1nnc(S)o1	nan
	2810145	25716	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	3.6	COc1cc2nc(NC(=O)c3ccc(Cl)cc3)sc(=O)c2cc1OC	nan
	CHEMBL1354031	25716	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	3.6	COc1cc2nc(NC(=O)c3ccc(Cl)cc3)sc(=O)c2cc1OC	nan
	16010496	25890	2	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	6	0.6	Cc1ccc2ncc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c(=O)n2c1	nan
	CHEMBL1356009	25890	2	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	6	0.6	Cc1ccc2ncc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c(=O)n2c1	nan
	2140949	25891	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	7	4.8	COc1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1OC	nan
	CHEMBL1356037	25891	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	7	4.8	COc1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1OC	nan
	2137373	27034	15	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	7	4.5	Cc1cccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccccc23)c1C	nan
	CHEMBL1366864	27034	15	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	7	4.5	Cc1cccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccccc23)c1C	nan
	16027547	27322	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	8	4.5	CC(C)CC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CCCCC4)sc3n2)cc1	nan
	CHEMBL1369113	27322	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	8	4.5	CC(C)CC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CCCCC4)sc3n2)cc1	nan
	16009802	27655	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	5	4.9	CCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1371530	27655	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	5	4.9	CCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	17581362	28606	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1cccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)c1	nan
	CHEMBL1379032	28606	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1cccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)c1	nan
	4875840	29409	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	2	4	2.5	COc1ccc(CNC(=O)CN2C(=O)NC(C)(c3cccc(Br)c3)C2=O)cc1	nan
	CHEMBL1386021	29409	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	2	4	2.5	COc1ccc(CNC(=O)CN2C(=O)NC(C)(c3cccc(Br)c3)C2=O)cc1	nan
	1486264	29776	13	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	Cc1ccc(Sc2ccc(NC(=O)c3ccc(S(C)(=O)=O)cc3Cl)cc2)cc1	nan
	CHEMBL1388862	29776	13	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	Cc1ccc(Sc2ccc(NC(=O)c3ccc(S(C)(=O)=O)cc3Cl)cc2)cc1	nan
	2810230	30206	6	None	2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	1	4	3.9	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)C1CCC1	nan
	CHEMBL1392489	30206	6	None	2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	1	4	3.9	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)C1CCC1	nan
	16012884	30685	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	7	3.1	COc1ccc(-n2ncc3c2ncn2nc(Cc4ccccc4)nc32)cc1	nan
	CHEMBL1397962	30685	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	7	3.1	COc1ccc(-n2ncc3c2ncn2nc(Cc4ccccc4)nc32)cc1	nan
	16021838	30715	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cccc(Cl)c2C)c(-c2ccccc2)n1	nan
	CHEMBL1398407	30715	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cccc(Cl)c2C)c(-c2ccccc2)n1	nan
	2135605	30892	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	4.6	c1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1400053	30892	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	4.6	c1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	15990902	31615	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	2	3	5.7	Cc1cc(C)cc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	CHEMBL1406771	31615	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	2	3	5.7	Cc1cc(C)cc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	963186	32043	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	3	4.2	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)cc1	nan
	CHEMBL1410023	32043	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	3	4.2	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)cc1	nan
	15989908	32045	9	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1410062	32045	9	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	15988850	32146	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	3.6	O=C(Nc1ccc(F)cc1F)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	CHEMBL1410908	32146	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	3.6	O=C(Nc1ccc(F)cc1F)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	1128972	32254	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	0	5	4.3	CCOC(=O)CSc1nc(-c2ccccc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1411854	32254	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	0	5	4.3	CCOC(=O)CSc1nc(-c2ccccc2)cc(C(F)(F)F)c1C#N	nan
	3361436	34017	2	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	4	4	4.2	Cc1ccc(NC(=S)NC(=O)c2ccccc2)cc1NC(=S)NC(=O)c1ccccc1	nan
	CHEMBL1426572	34017	2	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	4	4	4.2	Cc1ccc(NC(=S)NC(=O)c2ccccc2)cc1NC(=S)NC(=O)c1ccccc1	nan
	1627636	34695	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	6	1.6	NN=C(S)Nc1cccc(-c2nnc(S)o2)c1	nan
	CHEMBL1432353	34695	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	6	1.6	NN=C(S)Nc1cccc(-c2nnc(S)o2)c1	nan
	8087251	34845	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1433615	34845	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccc(F)cc2)CC1	nan
	16023146	35004	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	7	4.9	CCOc1ccc(CNC(=O)CSc2nnc(C)c3c(C)n(-c4ccc(Cl)cc4)nc23)cc1	nan
	CHEMBL1435835	35004	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	7	4.9	CCOc1ccc(CNC(=O)CSc2nnc(C)c3c(C)n(-c4ccc(Cl)cc4)nc23)cc1	nan
	1741544	37413	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccccc1C(=O)Nc1ccc2oc(-c3cccc4c(Br)cccc34)nc2c1	nan
	CHEMBL1457270	37413	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccccc1C(=O)Nc1ccc2oc(-c3cccc4c(Br)cccc34)nc2c1	nan
	2136370	37898	4	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	3.3	CCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccccc12	nan
	CHEMBL1461369	37898	4	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	3.3	CCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccccc12	nan
	3594053	39317	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Cl)c1	nan
	CHEMBL1473447	39317	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Cl)c1	nan
	16241285	40229	2	None	1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	2.3	CN(C)C=O.CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	CHEMBL1482781	40229	2	None	1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	2.3	CN(C)C=O.CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	1241177	41018	11	None	-1	3	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	0	8	2.4	c1ccc(COn2nnc3ccccc32)c(COn2nnc3ccccc32)c1	nan
	CHEMBL1489236	41018	11	None	-1	3	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	0	8	2.4	c1ccc(COn2nnc3ccccc32)c(COn2nnc3ccccc32)c1	nan
	16009541	41738	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccc(F)cc4)cc3)cc(=O)n12	nan
	CHEMBL1495115	41738	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccc(F)cc4)cc3)cc(=O)n12	nan
	2978485	42458	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	2	4.1	CCC(C)NC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1501669	42458	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	2	4.1	CCC(C)NC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	7514097	42504	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	4	6	2.2	O=C(O)CCNc1ccc(NCCC(=O)O)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1502018	42504	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	4	6	2.2	O=C(O)CCNc1ccc(NCCC(=O)O)c2c1C(=O)c1ccccc1C2=O	nan
	5777938	42599	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	10	1	8	4.1	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1502864	42599	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	10	1	8	4.1	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	1256983	43330	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	3	5.3	O=C(Nc1ccc(F)cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	CHEMBL1509228	43330	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	3	5.3	O=C(Nc1ccc(F)cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	16017574	43660	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	8	1	6	2.5	CCCCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1512435	43660	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	8	1	6	2.5	CCCCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	15988274	43761	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	CHEMBL1513838	43761	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	4921215	43915	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	2	4	6.7	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)Nc3ccc(C)c(C)c3)sc2n1	nan
	CHEMBL1516149	43915	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	2	4	6.7	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)Nc3ccc(C)c(C)c3)sc2n1	nan
	135466071	45980	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	6	4.5	CCc1cc2c(s1)N1Cc3ccccc3C(C(=O)c3cccc([N+](=O)[O-])c3)=C1NC2=O	nan
	CHEMBL1535161	45980	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	6	4.5	CCc1cc2c(s1)N1Cc3ccccc3C(C(=O)c3cccc([N+](=O)[O-])c3)=C1NC2=O	nan
	16024942	47980	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.7	CCc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1553067	47980	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.7	CCc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16015892	47994	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(-c2nc3cc(NC(=O)COc4ccc(C)c(C)c4)ccc3o2)cc1	nan
	CHEMBL1553238	47994	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(-c2nc3cc(NC(=O)COc4ccc(C)c(C)c4)ccc3o2)cc1	nan
	16028168	48662	4	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(F)c3)cc21	nan
	CHEMBL1560108	48662	4	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(F)c3)cc21	nan
	16009056	49116	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	3.7	COC(=O)c1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(C(=O)OC)c1	nan
	CHEMBL1564251	49116	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	3.7	COC(=O)c1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(C(=O)OC)c1	nan
	626021	50058	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	4	3.0	CNC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	CHEMBL1572204	50058	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	4	3.0	CNC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	2462898	50479	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	0	5	3.4	COc1ccc(C(C)=O)cc1COc1ncnc2ccccc12	nan
	CHEMBL1576381	50479	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	0	5	3.4	COc1ccc(C(C)=O)cc1COc1ncnc2ccccc12	nan
	16024893	52119	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	4.2	COc1ccc(OC)c(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	CHEMBL1590399	52119	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	4.2	COc1ccc(OC)c(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	16010832	52150	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.0	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3cccnc32)cc1C	nan
	CHEMBL1590845	52150	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.0	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3cccnc32)cc1C	nan
	16019294	52233	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	1	8	5.2	Cc1cc(C)cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)c1	nan
	CHEMBL1591857	52233	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	1	8	5.2	Cc1cc(C)cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)c1	nan
	3854561	52310	15	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	N#Cc1c(C(F)(F)F)cc(-c2ccc(F)cc2)nc1SCC(=O)Nc1ccccc1	nan
	CHEMBL1592912	52310	15	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	N#Cc1c(C(F)(F)F)cc(-c2ccc(F)cc2)nc1SCC(=O)Nc1ccccc1	nan
	16018208	53212	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1601478	53212	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	16025642	53363	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	6	1	6	5.9	Cc1cccc(C)c1NC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	CHEMBL1603009	53363	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	6	1	6	5.9	Cc1cccc(C)c1NC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	4402705	54435	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	8	-0.5	CN1C(=O)C(=NNc2cccc(S(=O)(=O)N3CCOCC3)c2)C(=O)N(C)C1=O	nan
	CHEMBL1611899	54435	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	8	-0.5	CN1C(=O)C(=NNc2cccc(S(=O)(=O)N3CCOCC3)c2)C(=O)N(C)C1=O	nan
	16018210	54449	3	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	4	5.8	Cc1ccccc1NC(=O)c1oc2c(c1C)-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1612043	54449	3	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	4	5.8	Cc1ccccc1NC(=O)c1oc2c(c1C)-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	2795741	79455	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	5	5.4	Cc1nc(-c2ccc(S(=O)(=O)Nc3ccc(Br)cc3Cl)s2)cs1	nan
	CHEMBL212314	79455	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	5	5.4	Cc1nc(-c2ccc(S(=O)(=O)Nc3ccc(Br)cc3Cl)s2)cs1	nan
	3127110	107248	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	1	8	2.9	C/C(=N\CCCn1ccnc1)c1c(C)nn(-c2ccc([N+](=O)[O-])cc2)c1O	nan
	CHEMBL3191381	107248	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	1	8	2.9	C/C(=N\CCCn1ccnc1)c1c(C)nn(-c2ccc([N+](=O)[O-])cc2)c1O	nan
	1528721	107855	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	3.4	CC(=O)/N=c1\scc(-c2ccccc2)n1-c1cccc(O)c1	nan
	CHEMBL3198106	107855	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	3.4	CC(=O)/N=c1\scc(-c2ccccc2)n1-c1cccc(O)c1	nan
	414	3318	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	93205	3318	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	CHEMBL139000	3318	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	24818570	20988	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	3	4	3.8	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)cc1	nan
	CHEMBL1312949	20988	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	3	4	3.8	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)cc1	nan
	3138147	21457	14	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	0	5	5.7	O=C(CSc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1)c1ccccc1	nan
	CHEMBL1318270	21457	14	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	0	5	5.7	O=C(CSc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1)c1ccccc1	nan
	5428505	22848	24	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	0	1	3	3.3	O=c1oc2cc(O)c(Cl)cc2c2ccccc12	nan
	CHEMBL1330383	22848	24	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	0	1	3	3.3	O=c1oc2cc(O)c(Cl)cc2c2ccccc12	nan
	5913370	23790	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	6	1	5	2.8	COCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1337918	23790	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	6	1	5	2.8	COCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	3694202	24138	19	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Cl)c2)no1	nan
	CHEMBL1341012	24138	19	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Cl)c2)no1	nan
	7190321	24513	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	7	2.6	O=C(CSc1ccc2nnc(-c3cccs3)n2n1)N1CCCC1	nan
	CHEMBL1344120	24513	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	7	2.6	O=C(CSc1ccc2nnc(-c3cccs3)n2n1)N1CCCC1	nan
	661441	24559	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1344527	24559	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1530959	24559	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	16017580	25094	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	7	2.9	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Cl)s1	nan
	CHEMBL1349094	25094	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	7	2.9	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Cl)s1	nan
	3239502	26748	10	None	1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	9	0.3	COc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	CHEMBL1364442	26748	10	None	1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	9	0.3	COc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	7189863	29104	8	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.9	O=C(Nc1nc2cc3c(cc2s1)OCO3)c1ccc(N2C(=O)CCC2=O)cc1	nan
	CHEMBL1383330	29104	8	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.9	O=C(Nc1nc2cc3c(cc2s1)OCO3)c1ccc(N2C(=O)CCC2=O)cc1	nan
	16189478	29138	2	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	0	6	2.2	CCCCN(Cc1ccccc1)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1383621	29138	2	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	0	6	2.2	CCCCN(Cc1ccccc1)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	2457625	30100	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	7	-0.0	CN(CC(=O)c1c(N)n(C)c(=O)n(C)c1=O)c1ccccc1	nan
	CHEMBL1391543	30100	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	7	-0.0	CN(CC(=O)c1c(N)n(C)c(=O)n(C)c1=O)c1ccccc1	nan
	686152	30275	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1393131	30275	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1576064	30275	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	16009717	30574	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	Fc1ccc(CNc2nc3c(-c4ccc(F)cc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1396454	30574	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	Fc1ccc(CNc2nc3c(-c4ccc(F)cc4)nnn3c3ccccc23)cc1	nan
	24892133	30755	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	11	1.7	COc1ccccc1-c1nc(SCC(=O)Nc2cc(C)on2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1398694	30755	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	11	1.7	COc1ccccc1-c1nc(SCC(=O)Nc2cc(C)on2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	1115170	32944	15	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	5	4.8	Cc1cccc(OCC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)c1	nan
	CHEMBL1417596	32944	15	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	5	4.8	Cc1cccc(OCC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)c1	nan
	15988646	35135	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	4.9	COc1ccccc1NC(=O)c1sc(-c2ccc(Cl)cc2)cc1N	nan
	CHEMBL1437533	35135	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	4.9	COc1ccccc1NC(=O)c1sc(-c2ccc(Cl)cc2)cc1N	nan
	1341231	35250	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	5	5.5	COc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	CHEMBL1438558	35250	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	5	5.5	COc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	2999623	36345	7	None	-1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	9	0	8	2.9	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(CCC(=O)OCc1c(C)noc1C)n2C	nan
	CHEMBL1448461	36345	7	None	-1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	9	0	8	2.9	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(CCC(=O)OCc1c(C)noc1C)n2C	nan
	2609971	38508	7	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	7	3.2	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccccc2c1=O	nan
	CHEMBL1466287	38508	7	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	7	3.2	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccccc2c1=O	nan
	16024828	41410	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5F)CC4)ccc3c2)CC1	nan
	CHEMBL1492051	41410	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5F)CC4)ccc3c2)CC1	nan
	3276076	42104	9	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	7	3.1	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	CHEMBL1498535	42104	9	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	7	3.1	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	3494087	43545	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	7	2.0	Cc1sc2ncnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)c2c1C	nan
	CHEMBL1511159	43545	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	7	2.0	Cc1sc2ncnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)c2c1C	nan
	22513173	43865	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	7	2.0	COc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccccc4F)ncn3n2)cc1	nan
	CHEMBL1515462	43865	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	7	2.0	COc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccccc4F)ncn3n2)cc1	nan
	16025349	44404	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.6	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccccc1)S2(=O)=O)Nc1ccccc1	nan
	CHEMBL1520822	44404	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.6	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccccc1)S2(=O)=O)Nc1ccccc1	nan
	16017252	45651	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.1	Cc1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	CHEMBL1532051	45651	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.1	Cc1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	659886	45955	13	None	1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	5	5.4	CCc1ccccc1NC(=O)CSc1nc2c(c(-c3ccco3)c1C#N)CCCC2	nan
	CHEMBL1534846	45955	13	None	1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	5	5.4	CCc1ccccc1NC(=O)CSc1nc2c(c(-c3ccco3)c1C#N)CCCC2	nan
	790785	45995	11	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	3	2	3	3.5	CCCc1c(C)nc2ccc(C(=O)O)cc2c1S	nan
	CHEMBL1535349	45995	11	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	3	2	3	3.5	CCCc1c(C)nc2ccc(C(=O)O)cc2c1S	nan
	3767937	46434	11	None	-3	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	6	5.6	N#Cc1c(N)nc(SCC(=O)C23CC4CC(CC(C4)C2)C3)c(C#N)c1-c1ccc(Cl)cc1	nan
	CHEMBL1539280	46434	11	None	-3	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	6	5.6	N#Cc1c(N)nc(SCC(=O)C23CC4CC(CC(C4)C2)C3)c(C#N)c1-c1ccc(Cl)cc1	nan
	24792845	50100	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	1.3	Cc1nn(CC(=O)NCC2CCCO2)c(=O)c2cc3ccccc3n12	nan
	CHEMBL1572639	50100	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	1.3	Cc1nn(CC(=O)NCC2CCCO2)c(=O)c2cc3ccccc3n12	nan
	319257	50118	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	4	2	2	3.0	C=C(C)C(=O)Nc1ccc(NC(C)C)cc1	nan
	CHEMBL1572793	50118	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	4	2	2	3.0	C=C(C)C(=O)Nc1ccc(NC(C)C)cc1	nan
	2100389	51406	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	2.5	O=C(COc1ncnc2scc(-c3ccccc3)c12)NCCN1C(=O)CSC1=O	nan
	CHEMBL1584231	51406	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	2.5	O=C(COc1ncnc2scc(-c3ccccc3)c12)NCCN1C(=O)CSC1=O	nan
	16019541	52148	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	8	5.1	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(Nc2ccc(C)c(C)c2)c2sccc23)c1	nan
	CHEMBL1590799	52148	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	8	5.1	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(Nc2ccc(C)c(C)c2)c2sccc23)c1	nan
	16025640	52205	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	5.6	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1591452	52205	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	5.6	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	1189472	52660	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	2.9	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCN1CCOCC1	nan
	CHEMBL1596394	52660	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	2.9	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCN1CCOCC1	nan
	1115820	54399	22	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	6	5.4	COc1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1611566	54399	22	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	6	5.4	COc1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	9581898	72227	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	5	2.0	Cc1cccc(C(=O)N/N=C2\CS(=O)(=O)N(C)c3ccsc32)c1	nan
	CHEMBL1992883	72227	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	5	2.0	Cc1cccc(C(=O)N/N=C2\CS(=O)(=O)N(C)c3ccsc32)c1	nan
	17584449	108612	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	0	7	2.6	COc1cc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2c2ccccc2)cc(OC)c1OC	nan
	CHEMBL3213657	108612	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	0	7	2.6	COc1cc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2c2ccccc2)cc(OC)c1OC	nan
	CHEMBL1411485	207012	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL		None	None	None		None	nan
	377	2707	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	425	2707	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	448222	2707	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	CHEMBL464859	2707	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	135415429	41050	7	None	2	3	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	8	1	9	4.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(SCc1nc(O)c3sccc3n1)n2CC	nan
	CHEMBL1489478	41050	7	None	2	3	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	8	1	9	4.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(SCc1nc(O)c3sccc3n1)n2CC	nan
	6076	106769	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	CHEMBL1363683	106769	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	CHEMBL316966	106769	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	20923189	19579	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	0	6	2.1	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1	nan
	CHEMBL1301594	19579	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	0	6	2.1	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1	nan
	613860	19998	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	6	2.9	Cc1noc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)c1C	nan
	CHEMBL1305078	19998	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	6	2.9	Cc1noc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)c1C	nan
	2480606	20208	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	2	7	0.6	Cc1cccc(NCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	CHEMBL1306773	20208	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	2	7	0.6	Cc1cccc(NCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	224672	22492	44	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	3	1	3	3.1	O=C(O)CSc1ccnc2cc(Cl)ccc12	nan
	CHEMBL1327484	22492	44	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	3	1	3	3.1	O=C(O)CSc1ccnc2cc(Cl)ccc12	nan
	2384232	22560	27	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	4.2	Cc1sc2ncnc(Sc3ccccc3C(=O)O)c2c1C	nan
	CHEMBL1327902	22560	27	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	4.2	Cc1sc2ncnc(Sc3ccccc3C(=O)O)c2c1C	nan
	1442817	23034	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.6	Cc1nnc(NC(=O)CSc2nc(C(C)C)nc3ccccc23)s1	nan
	CHEMBL1331799	23034	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.6	Cc1nnc(NC(=O)CSc2nc(C(C)C)nc3ccccc23)s1	nan
	6103449	23654	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	0	3	4.0	CCN1/C(=C2\C(=O)N(C)C(=S)N2c2ccccc2)C=Cc2ccccc21	nan
	CHEMBL1336606	23654	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	0	3	4.0	CCN1/C(=C2\C(=O)N(C)C(=S)N2c2ccccc2)C=Cc2ccccc21	nan
	662886	23687	9	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	7	3.5	Brc1ccc(-c2nn3c(-c4ccco4)nnc3s2)o1	nan
	CHEMBL1336927	23687	9	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	7	3.5	Brc1ccc(-c2nn3c(-c4ccco4)nnc3s2)o1	nan
	16011044	26475	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	CCOC(=O)c1ccc(NC(=O)c2ccc3c(c2)NC(=O)c2ccccc2S3)cc1	nan
	CHEMBL1362040	26475	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	CCOC(=O)c1ccc(NC(=O)c2ccc3c(c2)NC(=O)c2ccccc2S3)cc1	nan
	826482	26596	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	250	1	2	6	1.8	CC1(C)Cc2c(sc3ncnc(NN)c23)CO1	nan
	CHEMBL1363060	26596	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	250	1	2	6	1.8	CC1(C)Cc2c(sc3ncnc(NN)c23)CO1	nan
	16024887	27003	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	4.6	CCOc1ccccc1CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1366554	27003	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	4.6	CCOc1ccccc1CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	3207679	28925	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1cccc2cc(C#N)c(SCC(=O)NCc3cccs3)nc12	nan
	CHEMBL1381650	28925	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1cccc2cc(C#N)c(SCC(=O)NCc3cccs3)nc12	nan
	2445448	29416	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	0	7	1.4	COc1ccc(C(C)=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	CHEMBL1386075	29416	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	0	7	1.4	COc1ccc(C(C)=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	15988012	29774	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1388847	29774	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	2917979	29854	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	9	4.0	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)nc1C	nan
	CHEMBL1389475	29854	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	9	4.0	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)nc1C	nan
	686152	30275	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1393131	30275	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1576064	30275	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	15987889	32980	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	8	1	4	5.4	CCN(CC)CC(C)CNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1417926	32980	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	8	1	4	5.4	CCN(CC)CC(C)CNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	20904552	33575	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	8	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	CHEMBL1422972	33575	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	8	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	2375468	34694	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	-0.2	Cn1c(N)c(C(=O)COc2ccc(C#N)cc2)c(=O)n(C)c1=O	nan
	CHEMBL1432350	34694	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	-0.2	Cn1c(N)c(C(=O)COc2ccc(C#N)cc2)c(=O)n(C)c1=O	nan
	16024881	34837	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	4	2.6	CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1433473	34837	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	4	2.6	CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	15991045	34846	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	3	1	3	7.0	Cc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	CHEMBL1433636	34846	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	3	1	3	7.0	Cc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	16015278	34933	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	6	5.3	CC(=O)c1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4)c3C)nc2C)cc1	nan
	CHEMBL1434956	34933	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	6	5.3	CC(=O)c1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4)c3C)nc2C)cc1	nan
	5078950	35290	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1438931	35290	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	5310383	35724	10	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	0.3	O=C(Cn1cnc2c(nnn2-c2ccccc2)c1=O)NCC1CCCO1	nan
	CHEMBL1442757	35724	10	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	0.3	O=C(Cn1cnc2c(nnn2-c2ccccc2)c1=O)NCC1CCCO1	nan
	948433	35737	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	1	4	3.7	COc1ccc(CNC(=O)CSc2cccc3cccnc23)cc1	nan
	CHEMBL1442938	35737	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	1	4	3.7	COc1ccc(CNC(=O)CSc2cccc3cccnc23)cc1	nan
	16019658	35998	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	7	3.2	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1C	nan
	CHEMBL1445403	35998	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	7	3.2	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1C	nan
	3208298	38575	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	3.7	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1nccs1)OCO3	nan
	CHEMBL1466770	38575	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	3.7	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1nccs1)OCO3	nan
	6623284	39227	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	0	7	3.0	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCCC2)s1	nan
	CHEMBL1472373	39227	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	0	7	3.0	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCCC2)s1	nan
	5302642	39355	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	2	4	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2)cc1	nan
	CHEMBL1474011	39355	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	2	4	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2)cc1	nan
	1203028	39380	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	2	8	0.0	CC(=O)Nc1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1474423	39380	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	2	8	0.0	CC(=O)Nc1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	15988309	39711	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	8	2.1	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	CHEMBL1478365	39711	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	8	2.1	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	1387364	40547	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1485560	40547	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1576237	40547	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	4238273	40601	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	6	2.9	Cn1c(SCC(=O)c2ccc3c(c2)NC(=O)CO3)nc2ccccc21	nan
	CHEMBL1485997	40601	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	6	2.9	Cn1c(SCC(=O)c2ccc3c(c2)NC(=O)CO3)nc2ccccc21	nan
	16025632	41498	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	CHEMBL1492743	41498	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	1252362	42267	15	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	5	5.2	COc1ccc(-n2c(-c3cccc(OC)c3)nc(=S)c3c2CCCC3)cc1	nan
	CHEMBL1499911	42267	15	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	5	5.2	COc1ccc(-n2c(-c3cccc(OC)c3)nc(=S)c3c2CCCC3)cc1	nan
	3173852	42359	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	4	3.8	CNC(=S)N(Cc1ccc(OC)cc1)Cc1cc2cc(C)ccc2nc1O	nan
	CHEMBL1500673	42359	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	4	3.8	CNC(=S)N(Cc1ccc(OC)cc1)Cc1cc2cc(C)ccc2nc1O	nan
	16189472	42994	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	2.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)Nc1cccnc1Cl)C(=O)CO2	nan
	CHEMBL1506287	42994	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	2.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)Nc1cccnc1Cl)C(=O)CO2	nan
	20953562	43331	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	7	2.9	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)ncn3n2)cc1	nan
	CHEMBL1509249	43331	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	7	2.9	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)ncn3n2)cc1	nan
	20923188	43498	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	6	2.4	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccccc1	nan
	CHEMBL1510719	43498	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	6	2.4	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccccc1	nan
	16025766	43770	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	4	5.8	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccccc3Cl)CC2)s1	nan
	CHEMBL1514065	43770	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	4	5.8	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccccc3Cl)CC2)s1	nan
	5206706	43780	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.8	CN(C)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)cc1	nan
	CHEMBL1514233	43780	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.8	CN(C)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)cc1	nan
	15988349	43896	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccc(F)cc3)c2n1	nan
	CHEMBL1515965	43896	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccc(F)cc3)c2n1	nan
	4458977	44122	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	11	0.7	CCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1518407	44122	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	11	0.7	CCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	15989681	44220	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	7	1	7	4.1	COc1cc2c(=O)n(Cc3ccccc3Cl)c(=O)n(CC(=O)Nc3ccc(C)c(C)c3)c2cc1OC	nan
	CHEMBL1519224	44220	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	7	1	7	4.1	COc1cc2c(=O)n(Cc3ccccc3Cl)c(=O)n(CC(=O)Nc3ccc(C)c(C)c3)c2cc1OC	nan
	16019398	44928	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	0	9	2.6	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Cl)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1525727	44928	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	0	9	2.6	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Cl)cc4)nnn3c3ccsc23)CC1	nan
	16009804	45277	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	7	4.3	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1C	nan
	CHEMBL1528709	45277	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	7	4.3	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1C	nan
	2808993	45391	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	0	5	3.4	CCc1nc2ccccc2nc1N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1	nan
	CHEMBL1529717	45391	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	0	5	3.4	CCc1nc2ccccc2nc1N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1	nan
	588806	46191	20	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	4	1	4	2.5	Cc1nc(SCCC(=O)O)c2ccccc2n1	nan
	CHEMBL1537195	46191	20	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	4	1	4	2.5	Cc1nc(SCCC(=O)O)c2ccccc2n1	nan
	2810142	46906	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	5	3.6	O=C(Nc1nc2ccsc2c(=O)s1)c1ccc(Cl)cc1	nan
	CHEMBL1543276	46906	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	5	3.6	O=C(Nc1nc2ccsc2c(=O)s1)c1ccc(Cl)cc1	nan
	2158355	47327	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	7	0	7	1.6	COCCN(CCOC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1546597	47327	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	7	0	7	1.6	COCCN(CCOC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	1304353	48006	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	3	5.4	Cc1ccc(-c2sc(C(=O)Nc3ccc(Br)cc3)cc2CC(=O)O)cc1	nan
	CHEMBL1553391	48006	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	3	5.4	Cc1ccc(-c2sc(C(=O)Nc3ccc(Br)cc3)cc2CC(=O)O)cc1	nan
	3725217	48417	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	2	2	6	2.1	CC(C)C1Cc2c(sc3ncnc(NN)c23)CO1	nan
	CHEMBL1557963	48417	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	2	2	6	2.1	CC(C)C1Cc2c(sc3ncnc(NN)c23)CO1	nan
	16017731	49200	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	5	1.5	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)NCCc1ccccc1	nan
	CHEMBL1565042	49200	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	5	1.5	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)NCCc1ccccc1	nan
	7184630	51294	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1ccccc1CNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1583340	51294	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1ccccc1CNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	24856176	51854	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	4	3.3	CN(CC(=O)Nc1ccccc1Cl)C(=O)COC(=O)Cc1c(F)cccc1Cl	nan
	CHEMBL1587934	51854	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	4	3.3	CN(CC(=O)Nc1ccccc1Cl)C(=O)COC(=O)Cc1c(F)cccc1Cl	nan
	16033298	52114	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	5.5	Cc1c(C(=O)NCc2ccc(OC(C)C)cc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1590310	52114	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	5.5	Cc1c(C(=O)NCc2ccc(OC(C)C)cc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16010771	52277	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	6	3.5	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c2cccnc21	nan
	CHEMBL1592455	52277	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	6	3.5	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c2cccnc21	nan
	16029563	52403	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	6	4.2	COc1ccc(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(C)ccc32)cc1Cl	nan
	CHEMBL1594200	52403	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	6	4.2	COc1ccc(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(C)ccc32)cc1Cl	nan
	18553656	52595	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	9	1.0	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(CC(C)(C)C)nc2n(C)c1=O	nan
	CHEMBL1595812	52595	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	9	1.0	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(CC(C)(C)C)nc2n(C)c1=O	nan
	773677	53226	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	1	1	4	3.9	Cc1ccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCC4)cc1	nan
	CHEMBL1601668	53226	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	1	1	4	3.9	Cc1ccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCC4)cc1	nan
	1414561	53594	28	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	5	4.0	C=CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1604975	53594	28	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	5	4.0	C=CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	135693221	54680	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1359119	54680	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1615929	54680	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	6476987	55045	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL1385494	55045	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL1618897	55045	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	135502886	121149	23	None	-2	4	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	221	1	2	4	1.1	NC(=S)c1cc2ccc(O)cc2oc1=O	nan
	CHEMBL358644	121149	23	None	-2	4	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	221	1	2	4	1.1	NC(=S)c1cc2ccc(O)cc2oc1=O	nan
	24360	201644	101	None	-12	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	6	2.1	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL65	201644	101	None	-12	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	6	2.1	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	5359	205965	71	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	4	1	3	3.2	CC(C(=O)O)c1ccc(C(=O)c2cccs2)cc1	nan
	CHEMBL956	205965	71	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	4	1	3	3.2	CC(C(=O)O)c1ccc(C(=O)c2cccs2)cc1	nan
	2647611	52357	11	None	-	1	Human	3.9	pPotency	=	3.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	6	3.0	CC(=O)c1c(C)[nH]c(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)c1C	nan
	CHEMBL1593590	52357	11	None	-	1	Human	3.9	pPotency	=	3.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	6	3.0	CC(=O)c1c(C)[nH]c(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)c1C	nan
	126054	43672	34	None	-	1	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	11	7	12	-0.0	NCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4c3ncn4[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1	nan
	CHEMBL1512545	43672	34	None	-	1	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	11	7	12	-0.0	NCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4c3ncn4[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1	nan
	380	1256	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	657378	1256	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	CHEMBL68738	1256	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	191	13048	53	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	9	-2.0	Nc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	CHEMBL11909	13048	53	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	9	-2.0	Nc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	15988009	19496	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1300978	19496	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	1246444	19543	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	2	8	2.6	COc1cc(OC)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc1OC	nan
	CHEMBL1301318	19543	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	2	8	2.6	COc1cc(OC)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc1OC	nan
	5733367	19581	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	9	1	6	3.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCN3CCOCC3)C2c2ccc(F)cc2)cc1C	nan
	CHEMBL1301612	19581	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	9	1	6	3.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCN3CCOCC3)C2c2ccc(F)cc2)cc1C	nan
	3207945	19621	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	5	2.9	CCOC(=O)CNC(=O)CSc1nc2c(C)cccc2cc1CC	nan
	CHEMBL1302034	19621	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	5	2.9	CCOC(=O)CNC(=O)CSc1nc2c(C)cccc2cc1CC	nan
	2978035	19847	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	4	1.3	O=C(CN1C(=O)c2ccc(Br)cc2C1=O)NCC1CCCO1	nan
	CHEMBL1303768	19847	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	4	1.3	O=C(CN1C(=O)c2ccc(Br)cc2C1=O)NCC1CCCO1	nan
	16194904	21012	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)CC1	nan
	CHEMBL1313100	21012	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)CC1	nan
	127136	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549067	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549068	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549069	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	CHEMBL1314043	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	CHEMBL1556805	21127	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	3151367	21164	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	1.8	CCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1314339	21164	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	1.8	CCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	16009645	21250	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	2	5	5.9	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)cc1OCC	nan
	CHEMBL1315511	21250	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	2	5	5.9	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)cc1OCC	nan
	16009682	21291	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1cccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)c1	nan
	CHEMBL1315996	21291	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1cccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)c1	nan
	16023134	21415	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	6	2.4	CNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)C1	nan
	CHEMBL1317674	21415	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	6	2.4	CNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)C1	nan
	16019581	21450	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	3	0	9	2.7	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1318189	21450	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	3	0	9	2.7	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	16017720	21460	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	0	4	3.1	O=c1c(=O)n(-c2ccccc2)ccn1Cc1cccc(C(F)(F)F)c1	nan
	CHEMBL1318320	21460	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	0	4	3.1	O=c1c(=O)n(-c2ccccc2)ccn1Cc1cccc(C(F)(F)F)c1	nan
	2458272	21483	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3ccc4c(c3)OCCO4)nc2n1	nan
	CHEMBL1318506	21483	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3ccc4c(c3)OCCO4)nc2n1	nan
	15988341	21516	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	2	5	5.3	COc1ccc(-c2cc(C(=O)NCCc3ccccc3)c3c(-c4ccccc4)[nH]nc3n2)cc1OC	nan
	CHEMBL1318769	21516	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	2	5	5.3	COc1ccc(-c2cc(C(=O)NCCc3ccccc3)c3c(-c4ccccc4)[nH]nc3n2)cc1OC	nan
	3245692	21528	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.3	c1ccc(CCNc2nc3ccccc3n3nnnc23)cc1	nan
	CHEMBL1318873	21528	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.3	c1ccc(CCNc2nc3ccccc3n3nnnc23)cc1	nan
	16009520	21907	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3ccc(NC(=O)c4ccccc4F)cc3)cc(=O)n12	nan
	CHEMBL1322132	21907	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3ccc(NC(=O)c4ccccc4F)cc3)cc(=O)n12	nan
	1003845	21939	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)c(F)c4)sc3n2)c1	nan
	CHEMBL1322400	21939	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)c(F)c4)sc3n2)c1	nan
	1021427	22443	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	2	4	4.5	Cn1nc(C(=O)Nc2ccc(Br)cc2)cc1C(=O)Nc1ccc(Br)cc1	nan
	CHEMBL1327019	22443	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	2	4	4.5	Cn1nc(C(=O)Nc2ccc(Br)cc2)cc1C(=O)Nc1ccc(Br)cc1	nan
	1386649	23247	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1386650	23247	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1333441	23247	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	24503354	23393	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	3	2.5	O=C(c1ccc(S(=O)(=O)Nc2ccccc2F)cc1)N1CCC1	nan
	CHEMBL1334480	23393	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	3	2.5	O=C(c1ccc(S(=O)(=O)Nc2ccccc2F)cc1)N1CCC1	nan
	15988003	23482	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)c(F)c3)nnc12	nan
	CHEMBL1335235	23482	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)c(F)c3)nnc12	nan
	135416637	23869	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	2	7	5.8	Cc1ccc(C)c(NC(=O)CSc2nc(O)c3c(C(F)(F)F)cc(-c4cccs4)nc3n2)c1	nan
	CHEMBL1338446	23869	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	2	7	5.8	Cc1ccc(C)c(NC(=O)CSc2nc(O)c3c(C(F)(F)F)cc(-c4cccs4)nc3n2)c1	nan
	1023823	24112	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	4	3.3	NS(=O)(=O)c1c(Sc2ccccc2C(=O)O)ccc2ccccc12	nan
	CHEMBL1340736	24112	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	4	3.3	NS(=O)(=O)c1c(Sc2ccccc2C(=O)O)ccc2ccccc12	nan
	3420063	24263	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	2	7	3.4	COc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)c(OC)c1	nan
	CHEMBL1342030	24263	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	2	7	3.4	COc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)c(OC)c1	nan
	2023917	24839	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	3	4	4.5	O=C(NC(=S)Nc1ccccc1C(=O)O)c1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1346887	24839	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	3	4	4.5	O=C(NC(=S)Nc1ccccc1C(=O)O)c1ccc(-c2ccc(Br)cc2)o1	nan
	6145649	24929	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	7	1	6	2.9	N#Cc1nc(/C=C/c2ccccc2)oc1NCCCN1CCOCC1	nan
	CHEMBL1347564	24929	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	7	1	6	2.9	N#Cc1nc(/C=C/c2ccccc2)oc1NCCCN1CCOCC1	nan
	3099832	24988	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	3.7	Cc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)cc1	nan
	CHEMBL1348101	24988	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	3.7	Cc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)cc1	nan
	16033268	25836	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1cccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	CHEMBL1355268	25836	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1cccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	16004219	25895	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	7	4.6	Brc1ccc(-c2ccc(CNCCSc3nnnn3-c3ccccc3)o2)cc1	nan
	CHEMBL1356105	25895	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	7	4.6	Brc1ccc(-c2ccc(CNCCSc3nnnn3-c3ccccc3)o2)cc1	nan
	16033294	25907	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	6	5.1	CCOc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1356206	25907	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	6	5.1	CCOc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	16018776	25970	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	6	4.8	Cc1cc2c(cc3c(SCC(=O)Nc4cccc(Cl)c4C)nnc(C)n32)o1	nan
	CHEMBL1357046	25970	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	6	4.8	Cc1cc2c(cc3c(SCC(=O)Nc4cccc(Cl)c4C)nnc(C)n32)o1	nan
	16014983	26101	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2cccc(C)c2)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1358814	26101	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2cccc(C)c2)c(C#N)c(-c2ccccc2)n1	nan
	7190674	26470	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1F	nan
	CHEMBL1361981	26470	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1F	nan
	2138626	26554	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1ccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)cc1	nan
	CHEMBL1362650	26554	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1ccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)cc1	nan
	4152428	26808	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1364957	26808	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	15988005	26964	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	2.6	Cc1ccc(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1366276	26964	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	2.6	Cc1ccc(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	15996111	27056	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	4	4.9	CCOCCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1367087	27056	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	4	4.9	CCOCCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	659844	27142	14	None	-11	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	8	3.9	CCCCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OCC)cc2)c1C#N	nan
	CHEMBL1367765	27142	14	None	-11	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	8	3.9	CCCCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OCC)cc2)c1C#N	nan
	5287091	27170	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	2	4.7	Cc1ccc2nc(/C(C#N)=C/c3cccc(Br)c3)[nH]c2c1	nan
	CHEMBL1367954	27170	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	2	4.7	Cc1ccc2nc(/C(C#N)=C/c3cccc(Br)c3)[nH]c2c1	nan
	15991106	27200	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	1	5	6.0	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1C	nan
	CHEMBL1368193	27200	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	1	5	6.0	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1C	nan
	3544515	27230	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	6	1	9	2.2	O=C(O)CCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1368416	27230	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	6	1	9	2.2	O=C(O)CCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	4191572	27299	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	COc1ccccc1Cn1c(=S)[nH]c2ccc(F)cc2c1=O	nan
	CHEMBL1368980	27299	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	COc1ccccc1Cn1c(=S)[nH]c2ccc(F)cc2c1=O	nan
	2743471	28236	20	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	2	1	4	3.7	CSc1cc(-c2ccc(Cl)cc2)nc(O)c1C#N	nan
	CHEMBL1375507	28236	20	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	2	1	4	3.7	CSc1cc(-c2ccc(Cl)cc2)nc(O)c1C#N	nan
	1175821	28240	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	0	10	0.7	CC(C)n1c(SCC(=O)N2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1375543	28240	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	0	10	0.7	CC(C)n1c(SCC(=O)N2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3241220	28278	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	1.4	O=C(Cn1cnc2c(oc3ccccc32)c1=O)NCC1CCCO1	nan
	CHEMBL1375857	28278	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	1.4	O=C(Cn1cnc2c(oc3ccccc32)c1=O)NCC1CCCO1	nan
	5733045	28534	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	5	4.5	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2cccc(Cl)c2)cc1	nan
	CHEMBL1378340	28534	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	5	4.5	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2cccc(Cl)c2)cc1	nan
	3746307	29057	25	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	1	1	5	3.4	Cn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1382865	29057	25	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	1	1	5	3.4	Cn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	2939274	29116	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	7	4.5	CC(C)c1nnc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)s1	nan
	CHEMBL1383461	29116	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	7	4.5	CC(C)c1nnc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)s1	nan
	16194976	29189	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)CC1	nan
	CHEMBL1384046	29189	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)CC1	nan
	15987888	29232	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1384448	29232	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	2944910	29307	10	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	6	4.2	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccnc1)c1cc2ccccc2o1	nan
	CHEMBL1385074	29307	10	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	6	4.2	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccnc1)c1cc2ccccc2o1	nan
	1928929	29558	12	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	3	2	7	5.5	Nc1c(C(=O)Nc2nc3ccccc3s2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1387110	29558	12	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	3	2	7	5.5	Nc1c(C(=O)Nc2nc3ccccc3s2)sc2nc(-c3cccs3)ccc12	nan
	2237376	29580	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	2	8	3.0	CSc1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	CHEMBL1387290	29580	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	2	8	3.0	CSc1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	2779879	29964	28	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	3	4.1	Cc1c(C(=O)c2ccccc2C(=O)O)sc2ccccc12	nan
	CHEMBL1390399	29964	28	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	3	4.1	Cc1c(C(=O)c2ccccc2C(=O)O)sc2ccccc12	nan
	5088202	30461	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cccc(C)c4)sc3n2)cc1	nan
	CHEMBL1394959	30461	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cccc(C)c4)sc3n2)cc1	nan
	16018778	30555	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4ccc(Cl)cc4)nnc(C)n32)o1	nan
	CHEMBL1396136	30555	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4ccc(Cl)cc4)nnc(C)n32)o1	nan
	15987656	30619	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	12	1	6	5.8	CCOc1ccc(CCNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1OCC	nan
	CHEMBL1397047	30619	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	12	1	6	5.8	CCOc1ccc(CCNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1OCC	nan
	16018052	30641	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	4	3.8	Cc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1397347	30641	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	4	3.8	Cc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	15987604	30660	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1ccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)cc1	nan
	CHEMBL1397611	30660	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1ccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)cc1	nan
	866239	30713	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	2.9	Cc1ccc(-n2c(=O)[nH]c3sc4c(c3c2=O)CCCC4)cc1	nan
	CHEMBL1398397	30713	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	2.9	Cc1ccc(-n2c(=O)[nH]c3sc4c(c3c2=O)CCCC4)cc1	nan
	15990870	30870	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	3	5.3	Cc1ccc(C)c(Nc2cc(C(=O)NC3CCCC3)c3ccccc3n2)c1	nan
	CHEMBL1399859	30870	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	3	5.3	Cc1ccc(C)c(Nc2cc(C(=O)NC3CCCC3)c3ccccc3n2)c1	nan
	20904142	30973	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	0	9	1.3	COc1ccc(N2CCN(C(=O)CCc3nnc4ccc(N5CCOCC5)nn34)CC2)cc1	nan
	CHEMBL1400806	30973	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	0	9	1.3	COc1ccc(N2CCN(C(=O)CCc3nnc4ccc(N5CCOCC5)nn34)CC2)cc1	nan
	2859630	31776	19	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	0.9	O=C(CN1C(=O)c2cccc3cccc(c23)C1=O)NCCN1CCOCC1	nan
	CHEMBL1408014	31776	19	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	0.9	O=C(CN1C(=O)c2cccc3cccc(c23)C1=O)NCCN1CCOCC1	nan
	22553366	31825	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	7	1.5	CCOC(=O)C1CCN(C(=O)Cn2c(=O)c3cccn3c3cccnc32)CC1	nan
	CHEMBL1408318	31825	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	7	1.5	CCOC(=O)C1CCN(C(=O)Cn2c(=O)c3cccn3c3cccnc32)CC1	nan
	2911470	32497	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	8	3.8	C=CCOc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1413736	32497	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	8	3.8	C=CCOc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	663378	32522	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	3	0	5	3.4	N#CCCSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1413946	32522	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	3	0	5	3.4	N#CCCSc1ncnc2c1oc1ccccc12	nan
	1175547	32607	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	9	2.6	COc1cc(OC)cc(-n2nnnc2SCC(=O)Nc2ccc(C(C)=O)cc2)c1	nan
	CHEMBL1414657	32607	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	9	2.6	COc1cc(OC)cc(-n2nnnc2SCC(=O)Nc2ccc(C(C)=O)cc2)c1	nan
	2152512	32631	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1ccccc1OC	nan
	CHEMBL1414820	32631	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1ccccc1OC	nan
	16033750	32757	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	3	5.8	CC(C)c1ccc(N2C(=O)N(Cc3ccccc3Cl)c3ccccc3S2(=O)=O)cc1	nan
	CHEMBL1416012	32757	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	3	5.8	CC(C)c1ccc(N2C(=O)N(Cc3ccccc3Cl)c3ccccc3S2(=O)=O)cc1	nan
	1138440	32796	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	10	1.8	CCCn1c(SCC(=O)c2ccc(OC)c(OC)c2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1416338	32796	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	10	1.8	CCCn1c(SCC(=O)c2ccc(OC)c(OC)c2)nc2c1c(=O)n(C)c(=O)n2C	nan
	135445597	32885	21	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	2	1	6	2.5	CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1417116	32885	21	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	2	1	6	2.5	CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	24892379	33045	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	9	1.7	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3Cl)nc2n(C)c1=O	nan
	CHEMBL1418535	33045	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	9	1.7	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3Cl)nc2n(C)c1=O	nan
	24789790	33091	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	0	8	0.8	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3scc(C)n3c2=O)CC1	nan
	CHEMBL1418824	33091	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	0	8	0.8	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3scc(C)n3c2=O)CC1	nan
	5220580	33190	14	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	5	4.0	CC(=O)c1sc(NC(=O)COc2ccc(Cl)cc2Cl)nc1C	nan
	CHEMBL1419730	33190	14	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	5	4.0	CC(=O)c1sc(NC(=O)COc2ccc(Cl)cc2Cl)nc1C	nan
	3699048	33195	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	2	6	3.5	Cc1ccc[n+](C2C(c3cccs3)C(C#N)=C([C-](C#N)C#N)NC2(O)c2ccccc2)c1	nan
	CHEMBL1419826	33195	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	2	6	3.5	Cc1ccc[n+](C2C(c3cccs3)C(C#N)=C([C-](C#N)C#N)NC2(O)c2ccccc2)c1	nan
	5790281	33328	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	10	1	7	3.7	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2cccnc2)cc1	nan
	CHEMBL1420847	33328	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	10	1	7	3.7	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2cccnc2)cc1	nan
	2974740	33336	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	4	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3cccs3)nc12	nan
	CHEMBL1420938	33336	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	4	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3cccs3)nc12	nan
	824727	33367	12	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	2	0	4	2.2	CCOC(=O)c1cc(Br)c(=O)n2ccccc12	nan
	CHEMBL1421240	33367	12	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	2	0	4	2.2	CCOC(=O)c1cc(Br)c(=O)n2ccccc12	nan
	6411582	33470	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	10	2	10	4.3	CCOC(=O)CCCCC(=O)c1[nH]c(O)nc1CSc1nnc2c3cc(Br)ccc3n(C)c2n1	nan
	CHEMBL1422131	33470	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	10	2	10	4.3	CCOC(=O)CCCCC(=O)c1[nH]c(O)nc1CSc1nnc2c3cc(Br)ccc3n(C)c2n1	nan
	4910054	33515	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	9	1.1	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(CCO)CC4)o3)nnc2c2ccccc12	nan
	CHEMBL1422462	33515	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	9	1.1	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(CCO)CC4)o3)nnc2c2ccccc12	nan
	2945586	33646	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.6	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1ccncc1)c1cc2ccccc2o1	nan
	CHEMBL1423531	33646	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.6	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1ccncc1)c1cc2ccccc2o1	nan
	614539	33683	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1cc(Br)cc2c1OCC2	nan
	CHEMBL1423802	33683	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1cc(Br)cc2c1OCC2	nan
	5928009	34002	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	9	-0.1	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CCC(C(N)=O)CC3)nc12	nan
	CHEMBL1426470	34002	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	9	-0.1	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CCC(C(N)=O)CC3)nc12	nan
	20957179	34097	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	9	0.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	CHEMBL1427296	34097	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	9	0.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	2376694	34102	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	8	0.5	Cn1c(N)c(C(=O)CSc2nc3ccccc3[nH]2)c(=O)n(C)c1=O	nan
	CHEMBL1427343	34102	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	8	0.5	Cn1c(N)c(C(=O)CSc2nc3ccccc3[nH]2)c(=O)n(C)c1=O	nan
	20970067	34327	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	9	1	8	2.4	COc1ccc(OC)c(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)c1	nan
	CHEMBL1429318	34327	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	9	1	8	2.4	COc1ccc(OC)c(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)c1	nan
	2950264	34346	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	6	2.6	O=C(CSc1ncnc2sc3c(c12)CCC3)NCC1CCCO1	nan
	CHEMBL1429474	34346	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	6	2.6	O=C(CSc1ncnc2sc3c(c12)CCC3)NCC1CCCO1	nan
	135436945	34841	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	2	4	5.5	Cc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c(C)c1	nan
	CHEMBL1433539	34841	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	2	4	5.5	Cc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c(C)c1	nan
	16030485	34942	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1435046	34942	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	1775325	35001	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	0	6	4.3	COc1ccc(CN2COc3ccc4c(oc(=O)c5ccccc54)c3C2)cc1OC	nan
	CHEMBL1435817	35001	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	0	6	4.3	COc1ccc(CN2COc3ccc4c(oc(=O)c5ccccc54)c3C2)cc1OC	nan
	135433305	35504	1	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	3	8	1.3	CNC(=O)NC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1440872	35504	1	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	3	8	1.3	CNC(=O)NC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	2816654	36143	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	1	6	1.9	CCOC(=O)N1CCc2c(sc3ncnc(O)c23)C1	nan
	CHEMBL1446784	36143	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	1	6	1.9	CCOC(=O)N1CCc2c(sc3ncnc(O)c23)C1	nan
	749058	36207	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	5	4.8	O=c1c2c(-c3cccs3)csc2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1447245	36207	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	5	4.8	O=c1c2c(-c3cccs3)csc2[nH]c(=S)n1-c1ccccc1	nan
	739884	36301	77	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	1	1	2	3.9	O=C(O)c1sc2cc(Cl)ccc2c1Cl	nan
	CHEMBL1448105	36301	77	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	1	1	2	3.9	O=C(O)c1sc2cc(Cl)ccc2c1Cl	nan
	16033236	36482	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2ccccc2Cl)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1449453	36482	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2ccccc2Cl)sc2ncnc(N(C)C3CCCCC3)c12	nan
	2572725	36643	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	6	2.8	Cc1cc(C(=O)OCC(=O)c2ccc(Br)s2)no1	nan
	CHEMBL1450791	36643	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	6	2.8	Cc1cc(C(=O)OCC(=O)c2ccc(Br)s2)no1	nan
	2787753	36862	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	4	3	8	0.6	CC(C)OC(=O)C(C)Nc1nnc(S)nc1O	nan
	CHEMBL1452524	36862	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	4	3	8	0.6	CC(C)OC(=O)C(C)Nc1nnc(S)nc1O	nan
	4984225	37339	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.8	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)Nc2cccnc2Cl)cc1	nan
	CHEMBL1456558	37339	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.8	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)Nc2cccnc2Cl)cc1	nan
	764734	37711	27	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	5	3.6	C=CCn1c(=S)[nH]c2scc(-c3ccco3)c2c1=O	nan
	CHEMBL1459809	37711	27	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	5	3.6	C=CCn1c(=S)[nH]c2scc(-c3ccco3)c2c1=O	nan
	2822524	37811	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	5	3.5	CCOC(=O)c1c(SC)nc2c(Cl)cccc2c1O	nan
	CHEMBL1460605	37811	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	5	3.5	CCOC(=O)c1c(SC)nc2c(Cl)cccc2c1O	nan
	2973900	38130	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	3	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3ccccc3)nc12	nan
	CHEMBL1463377	38130	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	3	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3ccccc3)nc12	nan
	5637963	38210	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	0	5	3.7	CCOC(=O)/C(C#N)=C/c1cc2ccccc2nc1N1CCCCC1	nan
	CHEMBL1464025	38210	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	0	5	3.7	CCOC(=O)/C(C#N)=C/c1cc2ccccc2nc1N1CCCCC1	nan
	1005162	38254	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.9	N#Cc1ccc(-c2ccc(F)cc2)nc1SCC(=O)Nc1sc2c(c1C#N)CCC2	nan
	CHEMBL1464360	38254	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.9	N#Cc1ccc(-c2ccc(F)cc2)nc1SCC(=O)Nc1sc2c(c1C#N)CCC2	nan
	2087618	38268	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	6	2.8	CCOc1cc(C=O)ccc1OCc1cc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1464466	38268	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	6	2.8	CCOc1cc(C=O)ccc1OCc1cc(=O)n2cc(C)ccc2n1	nan
	20904553	38479	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.8	CC(NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12)c1ccccc1	nan
	CHEMBL1466036	38479	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.8	CC(NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12)c1ccccc1	nan
	20923124	38481	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	CHEMBL1466048	38481	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	16681736	38649	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	2	5	3.1	C1COCCO1.O=C(Nc1cccc2ccccc12)C(=O)C1C(=O)Nc2ccccc21	nan
	CHEMBL1467358	38649	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	2	5	3.1	C1COCCO1.O=C(Nc1cccc2ccccc12)C(=O)C1C(=O)Nc2ccccc21	nan
	2788467	38691	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	2	6	3.4	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1467713	38691	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	2	6	3.4	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	4224805	38719	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	2.0	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCCCC3)c(=O)c2c1C	nan
	CHEMBL1468056	38719	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	2.0	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCCCC3)c(=O)c2c1C	nan
	22334123	38866	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1469191	38866	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1OC	nan
	5016620	39321	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	5	3.5	COc1ccc(-c2cc(C(=O)Nc3ccc(C#N)cc3)no2)cc1	nan
	CHEMBL1473482	39321	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	5	3.5	COc1ccc(-c2cc(C(=O)Nc3ccc(C#N)cc3)no2)cc1	nan
	775363	39462	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	7	0.7	Cc1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1C	nan
	CHEMBL1475499	39462	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	7	0.7	Cc1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1C	nan
	16009659	39521	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	7	4.1	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1476377	39521	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	7	4.1	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	5730013	39569	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	4.0	CCC(Sc1nnc2c(n1)[nH]c1ccccc12)C(=O)Nc1nnc(C(C)C)s1	nan
	CHEMBL1476964	39569	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	4.0	CCC(Sc1nnc2c(n1)[nH]c1ccccc12)C(=O)Nc1nnc(C(C)C)s1	nan
	1782877	39628	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	2	6	3.9	COc1ccc(-c2cc3ccc(OCC(=O)NCC4CCC(C(=O)O)CC4)cc3oc2=O)cc1	nan
	CHEMBL1477517	39628	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	2	6	3.9	COc1ccc(-c2cc3ccc(OCC(=O)NCC4CCC(C(=O)O)CC4)cc3oc2=O)cc1	nan
	20957466	39880	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	7	1.7	CC1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	CHEMBL1479770	39880	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	7	1.7	CC1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	5378436	39882	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	6	1.4	Cn1c(=O)[nH]c2nnc(-c3ccc(Cl)c(Cl)c3)nc2c1=O	nan
	CHEMBL1479779	39882	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	6	1.4	Cn1c(=O)[nH]c2nnc(-c3ccc(Cl)c(Cl)c3)nc2c1=O	nan
	7207545	40689	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)cc3F)nn2)s1	nan
	CHEMBL1486756	40689	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)cc3F)nn2)s1	nan
	974443	40909	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	7	0.5	COc1cccc(Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1488414	40909	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	7	0.5	COc1cccc(Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	250222	40948	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	1	3	2.9	O=C1c2ccccc2C(O)(c2ccccc2)N1c1ccncc1	nan
	CHEMBL1488698	40948	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	1	3	2.9	O=C1c2ccccc2C(O)(c2ccccc2)N1c1ccncc1	nan
	2158358	40998	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	2	0	7	1.8	CCOC(=O)N1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1489076	40998	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	2	0	7	1.8	CCOC(=O)N1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	4000951	41132	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	11	1.8	Cn1c(N)c(C(=O)CSc2nn(-c3ccc(F)cc3)c(=S)s2)c(=O)n(C)c1=O	nan
	CHEMBL1490219	41132	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	11	1.8	Cn1c(N)c(C(=O)CSc2nn(-c3ccc(F)cc3)c(=S)s2)c(=O)n(C)c1=O	nan
	5310114	41192	4	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	7	2.1	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)O	nan
	CHEMBL1490578	41192	4	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	7	2.1	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)O	nan
	135436946	41202	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	2	5	5.6	CSc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)cc1	nan
	CHEMBL1490651	41202	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	2	5	5.6	CSc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)cc1	nan
	2857238	41371	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	2	3	4.3	CC(Oc1ccccc1)C(=O)Nc1ccc(NC(=O)c2ccccc2)cc1	nan
	CHEMBL1491753	41371	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	2	3	4.3	CC(Oc1ccccc1)C(=O)Nc1ccc(NC(=O)c2ccccc2)cc1	nan
	3913191	41533	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	2	6	2.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2ccc(O)nc2)c1	nan
	CHEMBL1493081	41533	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	2	6	2.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2ccc(O)nc2)c1	nan
	16009715	41691	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1494680	41691	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	252183	41863	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	3	3	7	-0.3	O=C1NC(=O)C(=NNc2ccc([N+](=O)[O-])cc2)C(=O)N1	nan
	CHEMBL1496411	41863	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	3	3	7	-0.3	O=C1NC(=O)C(=NNc2ccc([N+](=O)[O-])cc2)C(=O)N1	nan
	4023603	42347	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	4921719	42347	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	CHEMBL1500596	42347	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	2100904	42860	4	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	6	3.9	Cc1nn(CCc2nn[nH]n2)c2nc(-c3ccc(Br)cc3)cc(C(F)(F)F)c12	nan
	CHEMBL1505221	42860	4	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	6	3.9	Cc1nn(CCc2nn[nH]n2)c2nc(-c3ccc(Br)cc3)cc(C(F)(F)F)c12	nan
	1103129	43290	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	1	3	4.1	O=C(O)c1cccc(N2C(=O)c3cc4cccc(Br)c4cc3C2=O)c1	nan
	CHEMBL1508887	43290	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	1	3	4.1	O=C(O)c1cccc(N2C(=O)c3cc4cccc(Br)c4cc3C2=O)c1	nan
	15990473	43707	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.6	CCOc1ccccc1NC(=O)c1cn(C2CCCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1513016	43707	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.6	CCOc1ccccc1NC(=O)c1cn(C2CCCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3858365	43727	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	6	5.7	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1513368	43727	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	6	5.7	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	16018934	43752	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	5.9	CCc1nnc(SCc2ccc(F)cc2Cl)c2cc3sc(C)cc3n12	nan
	CHEMBL1513698	43752	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	5.9	CCc1nnc(SCc2ccc(F)cc2Cl)c2cc3sc(C)cc3n12	nan
	16025722	43903	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	6	6.2	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3Cl)s1)C2	nan
	CHEMBL1516031	43903	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	6	6.2	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3Cl)s1)C2	nan
	5110655	44273	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	3.8	Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1519696	44273	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	3.8	Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	2161841	44617	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.5	Cc1nc(SCC(=O)N2CC(=O)Nc3ccccc32)nc(C)c1C	nan
	CHEMBL1522742	44617	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.5	Cc1nc(SCC(=O)N2CC(=O)Nc3ccccc32)nc(C)c1C	nan
	1238361	44749	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	1	5	6.5	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL1523965	44749	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	1	5	6.5	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(C(F)(F)F)c1	nan
	20904542	44884	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	1.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccco3)nnc12	nan
	CHEMBL1525378	44884	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	1.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccco3)nnc12	nan
	2592811	44927	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	4	0	7	2.5	O=[N+]([O-])c1cc2c(c(CSc3ncccn3)c1)OCOC2	nan
	CHEMBL1525704	44927	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	4	0	7	2.5	O=[N+]([O-])c1cc2c(c(CSc3ncccn3)c1)OCOC2	nan
	6078768	44940	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	5	4.9	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(C)cc2)c(C)c1	nan
	CHEMBL1525799	44940	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	5	4.9	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(C)cc2)c(C)c1	nan
	1147569	44948	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	7	3.6	COc1cc(SC)ccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	CHEMBL1525877	44948	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	7	3.6	COc1cc(SC)ccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	4181953	45070	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	1	0	3	3.9	Cn1/c(=N\C(=O)c2ccc(F)cc2)sc2cc(Br)ccc21	nan
	CHEMBL1526825	45070	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	1	0	3	3.9	Cn1/c(=N\C(=O)c2ccc(F)cc2)sc2cc(Br)ccc21	nan
	5380406	45086	77	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	0	1	3	2.7	O=c1oc2cc(O)ccc2c2ccccc12	nan
	CHEMBL1526978	45086	77	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	0	1	3	2.7	O=c1oc2cc(O)ccc2c2ccccc12	nan
	5641185	45297	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	8	0.1	Cc1c(C(=O)NNc2cc(=O)n(C)c(=O)n2C)cccc1[N+](=O)[O-]	nan
	CHEMBL1528897	45297	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	8	0.1	Cc1c(C(=O)NNc2cc(=O)n(C)c(=O)n2C)cccc1[N+](=O)[O-]	nan
	1016791	45350	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	3	5.0	CC(C)c1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1529358	45350	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	3	5.0	CC(C)c1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	7411882	45498	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)cc1	nan
	CHEMBL1530681	45498	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)cc1	nan
	16017598	45617	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)c1	nan
	CHEMBL1531718	45617	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)c1	nan
	16025817	45709	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	1	5	5.3	CCOc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1532579	45709	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	1	5	5.3	CCOc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	20939726	45788	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	0	7	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCOc2ccccc21	nan
	CHEMBL1533261	45788	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	0	7	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCOc2ccccc21	nan
	16033292	45937	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	6	5.4	CSc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1534658	45937	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	6	5.4	CSc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	135521540	46072	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	2	6	4.5	O=C(CCS(=O)(=O)c1ccccc1)Nc1ccc(-c2nc3ccccc3s2)c(O)c1	nan
	CHEMBL1536204	46072	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	2	6	4.5	O=C(CCS(=O)(=O)c1ccccc1)Nc1ccc(-c2nc3ccccc3s2)c(O)c1	nan
	2729862	46653	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	2	8	0.2	Cc1ccc(NCC(O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1541137	46653	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	2	8	0.2	Cc1ccc(NCC(O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	2487501	46699	29	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	2	6	1.3	Oc1nc2ccccc2n2c(S)nnc12	nan
	CHEMBL1541468	46699	29	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	2	6	1.3	Oc1nc2ccccc2n2c(S)nnc12	nan
	16194809	47044	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1nnc2ccc(-c3ccccn3)nn12)NCC1CCCO1	nan
	CHEMBL1544280	47044	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1nnc2ccc(-c3ccccn3)nn12)NCC1CCCO1	nan
	1866349	47164	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	661670	47164	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1406059	47164	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1545185	47164	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	15988305	47961	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	2.5	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1552888	47961	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	2.5	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	1327631	48124	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CCc1ccc(OCC(=O)Nc2ccc3oc(-c4ccc(OC)cc4)nc3c2)cc1	nan
	CHEMBL1555206	48124	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CCc1ccc(OCC(=O)Nc2ccc3oc(-c4ccc(OC)cc4)nc3c2)cc1	nan
	16033300	48137	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	5.3	CCc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1555399	48137	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	5.3	CCc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	20970028	48217	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	5	1.7	CC(C)NS(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1556192	48217	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	5	1.7	CC(C)NS(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	5202629	48435	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	7	2.4	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	CHEMBL1558116	48435	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	7	2.4	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	7411867	48734	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	0	4	4.3	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1560888	48734	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	0	4	4.3	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2)CC1	nan
	20923142	48920	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	1.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC(C)C	nan
	CHEMBL1562552	48920	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	1.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC(C)C	nan
	3505859	48922	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	8	2.3	CCN(CC)S(=O)(=O)c1ccc(C)c(NC(=O)Cn2cnc3cc([N+](=O)[O-])ccc3c2=O)c1	nan
	CHEMBL1562557	48922	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	8	2.3	CCN(CC)S(=O)(=O)c1ccc(C)c(NC(=O)Cn2cnc3cc([N+](=O)[O-])ccc3c2=O)c1	nan
	7524261	49022	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	2.6	CCS(=O)(=O)Nc1cccc(-c2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1563485	49022	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	2.6	CCS(=O)(=O)Nc1cccc(-c2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	5389817	49192	8	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	1	6	3.2	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCOC)C23C(=O)N(C)c2ccccc23)cc1	nan
	CHEMBL1564945	49192	8	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	1	6	3.2	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCOC)C23C(=O)N(C)c2ccccc23)cc1	nan
	1111955	49207	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	4.1	COc1ccc(-n2nc3ccc(NC(=O)COc4ccc(C)c(C)c4)cc3n2)cc1	nan
	CHEMBL1565140	49207	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	4.1	COc1ccc(-n2nc3ccc(NC(=O)COc4ccc(C)c(C)c4)cc3n2)cc1	nan
	15988272	49538	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	0	9	2.0	COC(=O)c1ccc(OC)c(Cn2c(=O)n(-c3ccc(C)cc3)c(=O)c3c2cnn3C)c1	nan
	CHEMBL1567650	49538	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	0	9	2.0	COC(=O)c1ccc(OC)c(Cn2c(=O)n(-c3ccc(C)cc3)c(=O)c3c2cnn3C)c1	nan
	15991345	49733	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	0	5	5.1	CSc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2ccc(C)cn2)cc1	nan
	CHEMBL1569335	49733	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	0	5	5.1	CSc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2ccc(C)cn2)cc1	nan
	15988962	50019	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCN(CCC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1571921	50019	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCN(CCC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	2483422	50522	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	6	1.1	Cn1c(CCC(=O)OCC(=O)NCC(F)(F)F)nc(=O)c2ccccc21	nan
	CHEMBL1576699	50522	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	6	1.1	Cn1c(CCC(=O)OCC(=O)NCC(F)(F)F)nc(=O)c2ccccc21	nan
	5070065	50997	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	1	8	5.1	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(C)=O)s2)c1	nan
	CHEMBL1580853	50997	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	1	8	5.1	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(C)=O)s2)c1	nan
	4295307	51071	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1ccccc1C1C(C(=O)c2cc3ccccc3o2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1581437	51071	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1ccccc1C1C(C(=O)c2cc3ccccc3o2)=C(O)C(=O)N1c1cc(C)on1	nan
	4808157	51263	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	0.5	COc1ccc(OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1583111	51263	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	0.5	COc1ccc(OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	6530035	51771	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	2.6	CCN(CC)S(=O)(=O)c1ccc(C(=O)NCCN2C(=O)S/C(=C\c3cccnc3)C2=O)cc1	nan
	CHEMBL1587266	51771	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	2.6	CCN(CC)S(=O)(=O)c1ccc(C(=O)NCCN2C(=O)S/C(=C\c3cccnc3)C2=O)cc1	nan
	15988968	52174	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)c(OC)c1	nan
	CHEMBL1591154	52174	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)c(OC)c1	nan
	16024517	52191	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	5.0	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C(C)C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1591352	52191	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	5.0	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C(C)C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16018826	52254	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	6	4.2	CCc1cccc(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1592153	52254	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	6	4.2	CCc1cccc(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	16010502	52334	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1593224	52334	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2F)CC1	nan
	1191851	52877	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.0	CCc1ccccc1NC(=O)COc1ccc2oc(-c3ccc(OC)cc3)cc(=O)c2c1	nan
	CHEMBL1598484	52877	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.0	CCc1ccccc1NC(=O)COc1ccc2oc(-c3ccc(OC)cc3)cc(=O)c2c1	nan
	20888741	53067	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	7	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCCC2)s1	nan
	CHEMBL1600180	53067	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	7	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCCC2)s1	nan
	16018860	53273	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	6	4.6	Cc1ccc(NC(=O)CSc2nnc(C)n3c2cc2sccc23)c(C)c1	nan
	CHEMBL1602197	53273	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	6	4.6	Cc1ccc(NC(=O)CSc2nnc(C)n3c2cc2sccc23)c(C)c1	nan
	135460554	53511	7	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	7	2.5	CC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1604187	53511	7	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	7	2.5	CC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	16194880	53590	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	8	2.2	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)OC	nan
	CHEMBL1604935	53590	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	8	2.2	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)OC	nan
	2939815	53863	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2ccccc2n2c(SCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1607085	53863	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2ccccc2n2c(SCC(=O)NCC3CCCO3)nnc12	nan
	16017570	54227	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	6	3.3	CN(Cc1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2cccc(Cl)c2)s1	nan
	CHEMBL1610070	54227	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	6	3.3	CN(Cc1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2cccc(Cl)c2)s1	nan
	7184628	54331	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccccc3)nnc12	nan
	CHEMBL1611000	54331	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccccc3)nnc12	nan
	20957175	54623	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	0	8	1.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)N1CCCCC1	nan
	CHEMBL1613668	54623	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	0	8	1.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)N1CCCCC1	nan
	11077	54736	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	CHEMBL1353221	54736	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	CHEMBL1616414	54736	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	686692	54756	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	CHEMBL1309275	54756	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	CHEMBL1616571	54756	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	694704	55042	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1373811	55042	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1618856	55042	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	3246720	55360	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	CHEMBL1445386	55360	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	CHEMBL1621717	55360	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	135439671	71842	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	2	9	0.1	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/c2c[nH]nc2-c2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1980641	71842	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	2	9	0.1	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/c2c[nH]nc2-c2ccc(F)cc2)n(C)c1=O	nan
	6187702	72413	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	6	2.6	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1ccc(N2CCOCC2)cc1	nan
	CHEMBL1999641	72413	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	6	2.6	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1ccc(N2CCOCC2)cc1	nan
	2058613	107869	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1cccc(OC)c1	nan
	CHEMBL3198223	107869	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1cccc(OC)c1	nan
	2947382	175732	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	1	5	1.8	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)C2CCCO2)c1	nan
	CHEMBL459529	175732	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	1	5	1.8	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)C2CCCO2)c1	nan
	3151452	197893	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	8	1.8	COCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL592554	197893	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	8	1.8	COCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3cccc(C)c3nc21	nan
	3159270	199909	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	0	5	2.6	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCN(C)C)CC2	nan
	CHEMBL605753	199909	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	0	5	2.6	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCN(C)C)CC2	nan
	9687	184743	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1522836	184743	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL485980	184743	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	16682183	25127	1	None	-	1	Human	5.8	pPotency	=	5.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	2	0	5	4.6	CC(C)C(=O)N1CCC2(CC1)Oc1ccc(F)cc1C(=O)C21CC(c2ccc(Cl)cc2)=NO1	nan
	CHEMBL1349353	25127	1	None	-	1	Human	5.8	pPotency	=	5.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	2	0	5	4.6	CC(C)C(=O)N1CCC2(CC1)Oc1ccc(F)cc1C(=O)C21CC(c2ccc(Cl)cc2)=NO1	nan
	123807	856	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	374	856	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	379	856	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	CHEMBL284969	856	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	2099	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	4740	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	7095	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	CHEMBL628	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	DB00806	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	123683	3060	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	422	3060	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	CHEMBL119709	3060	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	DB05511	3060	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	2808307	10272	5	None	-9	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	4	4.2	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)c1ccccc1C(=O)O	nan
	CHEMBL1162415	10272	5	None	-9	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	4	4.2	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)c1ccccc1C(=O)O	nan
	16019490	10882	4	None	-8	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)c1	nan
	CHEMBL1173709	10882	4	None	-8	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)c1	nan
	2729861	20191	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	8	0.0	Cn1c(=O)c2c(ncn2CC(O)CNc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1306604	20191	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	8	0.0	Cn1c(=O)c2c(ncn2CC(O)CNc2ccc(F)cc2)n(C)c1=O	nan
	713572	20294	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	0	2	4	3.0	CC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	CHEMBL1307433	20294	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	0	2	4	3.0	CC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	20884214	20581	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	1.4	CCC(C(=O)NCCN1CCOCC1)n1nc(C)n2c(cc3sccc32)c1=O	nan
	CHEMBL1309746	20581	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	1.4	CCC(C(=O)NCCN1CCOCC1)n1nc(C)n2c(cc3sccc32)c1=O	nan
	1831123	20634	8	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	3	1	7	5.2	Cc1nc2c(sc3nc(N4CCOCC4)c4c(c32)CC(C)(C)OC4)c(-c2ccccc2)c1C(=O)O	nan
	CHEMBL1310276	20634	8	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	3	1	7	5.2	Cc1nc2c(sc3nc(N4CCOCC4)c4c(c32)CC(C)(C)OC4)c(-c2ccccc2)c1C(=O)O	nan
	16194788	20821	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.2	O=C(CSc1nnc2ccc(-c3ccccc3)nn12)NCC1CCCO1	nan
	CHEMBL1311747	20821	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.2	O=C(CSc1nnc2ccc(-c3ccccc3)nn12)NCC1CCCO1	nan
	2820129	20919	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	2	4	2.2	CSc1sc(C(=O)NNC(C)=O)c2c1C=CCC2	nan
	CHEMBL1312452	20919	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	2	4	2.2	CSc1sc(C(=O)NNC(C)=O)c2c1C=CCC2	nan
	622563	20992	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	0	4	3.1	CN1c2ccc(C=O)c3c(C=O)ccc(c23)N(C)C1(C)C	nan
	CHEMBL1312974	20992	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	0	4	3.1	CN1c2ccc(C=O)c3c(C=O)ccc(c23)N(C)C1(C)C	nan
	4584575	21059	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	5	3.7	CC(C)N=C(S)n1cc(C(=O)c2cc(Cl)cc(Cl)c2O)cn1	nan
	CHEMBL1313487	21059	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	5	3.7	CC(C)N=C(S)n1cc(C(=O)c2cc(Cl)cc(Cl)c2O)cn1	nan
	16029652	21288	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	5.0	CCOc1ccc(NC(=O)c2sc3nc(-c4ccc(OC)cc4)cn3c2C)cc1	nan
	CHEMBL1315982	21288	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	5.0	CCOc1ccc(NC(=O)c2sc3nc(-c4ccc(OC)cc4)cn3c2C)cc1	nan
	1116235	21348	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	9	0.7	COc1cc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)cc1Cl	nan
	CHEMBL1316844	21348	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	9	0.7	COc1cc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)cc1Cl	nan
	16030395	21369	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1317102	21369	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16018828	21374	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.1	Cc1ccc(NC(=O)CSc2nncn3c2cc2sccc23)cc1F	nan
	CHEMBL1317182	21374	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.1	Cc1ccc(NC(=O)CSc2nncn3c2cc2sccc23)cc1F	nan
	16018832	21404	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1317561	21404	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	16025821	21441	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	1	5	4.9	CN(C)c1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1318005	21441	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	1	5	4.9	CN(C)c1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	1482206	21518	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	2.1	CS(=O)(=O)c1ccc(-c2cn3cc(C(=O)O)ccc3n2)cc1	nan
	CHEMBL1318777	21518	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	2.1	CS(=O)(=O)c1ccc(-c2cn3cc(C(=O)O)ccc3n2)cc1	nan
	1115262	21539	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	2	4	5.5	O=C(O)c1ccc(Nc2nc(-c3ccccc3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1318956	21539	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	2	4	5.5	O=C(O)c1ccc(Nc2nc(-c3ccccc3)c3cc(Br)ccc3n2)cc1	nan
	16025794	21541	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.2	Cc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1318960	21541	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.2	Cc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	16021547	21555	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	6	2	8	1.8	NS(=O)(=O)c1ccc(CCNC(=O)C2CCN(c3ncnc4c3nc3n4CCCCC3)CC2)cc1	nan
	CHEMBL1319081	21555	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	6	2	8	1.8	NS(=O)(=O)c1ccc(CCNC(=O)C2CCN(c3ncnc4c3nc3n4CCCCC3)CC2)cc1	nan
	6287803	21560	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	6	4.6	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(Br)cc3)ccc2O1	nan
	CHEMBL1319132	21560	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	6	4.6	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(Br)cc3)ccc2O1	nan
	15988299	21583	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	CHEMBL1319322	21583	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	3152547	21769	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	3.2	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1F)c1ccco1	nan
	CHEMBL1320921	21769	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	3.2	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1F)c1ccco1	nan
	829953	21881	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	5	2.4	CCN(CC)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1321896	21881	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	5	2.4	CCN(CC)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	3147388	22047	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	1	4	2.9	Cc1cc(SCC(=O)NCC2CCCO2)nc2ccccc12	nan
	CHEMBL1323473	22047	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	1	4	2.9	Cc1cc(SCC(=O)NCC2CCCO2)nc2ccccc12	nan
	3154196	22148	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	8	-0.1	CN(CC(O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)c1ccccc1	nan
	CHEMBL1324245	22148	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	8	-0.1	CN(CC(O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)c1ccccc1	nan
	16019851	22209	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	11	1	9	1.9	CCOCCCNC(=O)CCc1nnc2ccc(N3CCN(c4cccc(OC)c4)CC3)nn12	nan
	CHEMBL1324764	22209	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	11	1	9	1.9	CCOCCCNC(=O)CCc1nnc2ccc(N3CCN(c4cccc(OC)c4)CC3)nn12	nan
	16018924	22234	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	0	5	5.2	CCc1nnc(SCc2cccc(F)c2)c2cc3sc(C)cc3n12	nan
	CHEMBL1324960	22234	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	0	5	5.2	CCc1nnc(SCc2cccc(F)c2)c2cc3sc(C)cc3n12	nan
	4156222	22293	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	6	2.5	O=C(c1cccc([N+](=O)[O-])c1)N1CCCN(C(=O)c2cccc([N+](=O)[O-])c2)CC1	nan
	CHEMBL1325527	22293	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	6	2.5	O=C(c1cccc([N+](=O)[O-])c1)N1CCCN(C(=O)c2cccc([N+](=O)[O-])c2)CC1	nan
	16012102	22434	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	CHEMBL1326931	22434	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	342695	22626	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	8	0.6	Cn1c([N+](=O)[O-])cnc1N1CCN(c2nncs2)C1=O	nan
	CHEMBL1328402	22626	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	8	0.6	Cn1c([N+](=O)[O-])cnc1N1CCN(c2nncs2)C1=O	nan
	5048043	22651	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1328648	22651	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	16195662	22743	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccncc4)n3n2)CC1	nan
	CHEMBL1329498	22743	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccncc4)n3n2)CC1	nan
	15988282	22780	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.0	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1329775	22780	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.0	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(F)cc3)nnc12	nan
	753118	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1331202	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1532594	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	15989826	23088	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	1	6	3.2	Cc1ccc2nc(NCc3ccccc3Cl)c3nnnn3c2c1	nan
	CHEMBL1332222	23088	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	1	6	3.2	Cc1ccc2nc(NCc3ccccc3Cl)c3nnnn3c2c1	nan
	7120050	23684	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	3.9	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccc(F)cc1	nan
	CHEMBL1336910	23684	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	3.9	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccc(F)cc1	nan
	2997990	23722	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	10	-0.2	Cc1cc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(C)n1C	nan
	CHEMBL1337270	23722	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	10	-0.2	Cc1cc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(C)n1C	nan
	5827230	23801	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	9	3.4	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1338023	23801	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	9	3.4	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	4385163	23982	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	2	4	4.5	COc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1339561	23982	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	2	4	4.5	COc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	8030040	24155	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	2	5	3.2	O=C(NCCNC(=O)c1ccc(-c2ccc(Cl)c(Cl)c2)o1)c1cnccn1	nan
	CHEMBL1341144	24155	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	2	5	3.2	O=C(NCCNC(=O)c1ccc(-c2ccc(Cl)c(Cl)c2)o1)c1cnccn1	nan
	661441	24559	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1344527	24559	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1530959	24559	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	865623	24564	2	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	3	0	5	3.5	CN(C)c1ccc(-c2nnc(-c3cccs3)o2)cc1	nan
	CHEMBL1344555	24564	2	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	3	0	5	3.5	CN(C)c1ccc(-c2nnc(-c3cccs3)o2)cc1	nan
	2937580	24681	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	5	3.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(CC3CCCO3)C2c2ccccc2F)o1	nan
	CHEMBL1345579	24681	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	5	3.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(CC3CCCO3)C2c2ccccc2F)o1	nan
	1375907	24821	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	0	7	1.4	CCOC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	CHEMBL1346739	24821	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	0	7	1.4	CCOC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	5037672	24878	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	8	1.4	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cn2ccccc2n1	nan
	CHEMBL1347181	24878	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	8	1.4	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cn2ccccc2n1	nan
	3748480	24944	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1347701	24944	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	6463240	24966	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	9	0.6	CC(C)n1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1347878	24966	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	9	0.6	CC(C)n1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	4046369	25103	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCCC4)c3)nc2n1	nan
	CHEMBL1349141	25103	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCCC4)c3)nc2n1	nan
	5810234	25138	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1349428	25138	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	664152	25184	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	6	3.1	Cc1nc(SCC(=O)NCC2CCCO2)c2oc3ccccc3c2n1	nan
	CHEMBL1349799	25184	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	6	3.1	Cc1nc(SCC(=O)NCC2CCCO2)c2oc3ccccc3c2n1	nan
	4648816	25226	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	8	2.4	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1350189	25226	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	8	2.4	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	2081076	25257	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	1	5	3.3	O=c1c2c3c(sc2[nH]c(=S)n1Cc1ccco1)CCC3	nan
	CHEMBL1350435	25257	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	1	5	3.3	O=c1c2c3c(sc2[nH]c(=S)n1Cc1ccco1)CCC3	nan
	6618816	25322	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1351035	25322	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	3117452	25327	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	3	1.4	Cc1c2ccccc2cc[n+]1CCCS(=O)(=O)[O-]	nan
	CHEMBL1351071	25327	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	3	1.4	Cc1c2ccccc2cc[n+]1CCCS(=O)(=O)[O-]	nan
	5809890	25451	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	1	6	3.8	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	CHEMBL1352143	25451	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	1	6	3.8	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	24794131	25463	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	0	8	2.7	CSc1ccccc1OCc1cc(C(=O)N2CCN(c3ncccn3)CC2)no1	nan
	CHEMBL1352219	25463	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	0	8	2.7	CSc1ccccc1OCc1cc(C(=O)N2CCN(c3ncccn3)CC2)no1	nan
	20903685	25510	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	0	8	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCC(C)CC4)nn23)CC1	nan
	CHEMBL1352523	25510	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	0	8	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCC(C)CC4)nn23)CC1	nan
	2322442	25549	7	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	5	3.3	Cc1noc(NS(=O)(=O)c2ccc(N3Cc4ccccc4C3=O)cc2)c1C	nan
	CHEMBL1352855	25549	7	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	5	3.3	Cc1noc(NS(=O)(=O)c2ccc(N3Cc4ccccc4C3=O)cc2)c1C	nan
	135490313	25697	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-0.6	Cc1cc(O)nc(SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)n1	nan
	CHEMBL1353870	25697	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-0.6	Cc1cc(O)nc(SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)n1	nan
	20923143	25808	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	6	1.6	CCCNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1354972	25808	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	6	1.6	CCCNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	1116268	25822	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	9	-0.1	COC(=O)c1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1355136	25822	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	9	-0.1	COC(=O)c1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	1003440	25938	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	2	5	5.9	Nc1c(C(=O)Nc2ccc(C(F)(F)F)cc2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1356669	25938	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	2	5	5.9	Nc1c(C(=O)Nc2ccc(C(F)(F)F)cc2)sc2nc(-c3cccs3)ccc12	nan
	16024861	26018	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	4	3.0	CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1357771	26018	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	4	3.0	CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	25162722	26089	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	9	1.4	CCN(CC)c1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nncn1C	nan
	CHEMBL1358718	26089	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	9	1.4	CCN(CC)c1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nncn1C	nan
	4312795	26250	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	4	2.2	CC(Sc1cnc2ccccc2n1)C(=O)O	nan
	CHEMBL1360045	26250	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	4	2.2	CC(Sc1cnc2ccccc2n1)C(=O)O	nan
	3704657	26262	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	6	3.2	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2ncccn2)cc1	nan
	CHEMBL1360163	26262	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	6	3.2	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2ncccn2)cc1	nan
	24000844	26278	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.9	Cn1c2ccccc2c2nnc(SCC(=O)Nc3cccc(C(=O)O)c3)nc21	nan
	CHEMBL1360279	26278	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.9	Cn1c2ccccc2c2nnc(SCC(=O)Nc3cccc(C(=O)O)c3)nc21	nan
	791500	26300	15	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	5	3.4	CCOC(=O)c1c(C)nc(S)c(C#N)c1-c1ccccc1	nan
	CHEMBL1360458	26300	15	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	5	3.4	CCOC(=O)c1c(C)nc(S)c(C#N)c1-c1ccccc1	nan
	3178481	26479	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1362095	26479	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	5309057	26560	2	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	5	3.7	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1362711	26560	2	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	5	3.7	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccn2)CC1	nan
	16022478	26581	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	9	4.3	COc1cccc(NC(=O)c2ccc3c(=O)n4nc(Nc5ccccc5OC)sc4nc3c2)c1	nan
	CHEMBL1362937	26581	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	9	4.3	COc1cccc(NC(=O)c2ccc3c(=O)n4nc(Nc5ccccc5OC)sc4nc3c2)c1	nan
	20917857	26871	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.4	Cc1ccc(CNS(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)o1	nan
	CHEMBL1365432	26871	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.4	Cc1ccc(CNS(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)o1	nan
	2999882	27049	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	7	1	5	2.9	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1ccccc1	nan
	CHEMBL1367025	27049	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	7	1	5	2.9	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1ccccc1	nan
	1914729	27137	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	11	1	3	4.7	CC(=O)c1ccc(CCCCCCCCCC(=O)O)s1	nan
	CHEMBL1367732	27137	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	11	1	3	4.7	CC(=O)c1ccc(CCCCCCCCCC(=O)O)s1	nan
	3820161	27188	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccccc2F)o1	nan
	CHEMBL1368082	27188	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccccc2F)o1	nan
	135419062	27235	6	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	7	4.5	N#Cc1c(O)nc(SCC(=O)c2ccc(Br)cc2)nc1-c1cccs1	nan
	CHEMBL1368444	27235	6	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	7	4.5	N#Cc1c(O)nc(SCC(=O)c2ccc(Br)cc2)nc1-c1cccs1	nan
	3154099	27353	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	4.1	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1369329	27353	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	4.1	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	2443232	27588	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	1	5	6.4	O=C(COC(=O)c1cc(-c2ccccc2Cl)nc2ccccc12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	CHEMBL1370986	27588	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	1	5	6.4	O=C(COC(=O)c1cc(-c2ccccc2Cl)nc2ccccc12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	22548207	27620	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	0.8	CCOC(=O)CNC(=O)Cn1cnc2c(oc3ccccc32)c1=O	nan
	CHEMBL1371227	27620	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	0.8	CCOC(=O)CNC(=O)Cn1cnc2c(oc3ccccc32)c1=O	nan
	663879	28045	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	9	1	7	4.2	Cc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2ccc(OC(C)C)cc2)o1	nan
	CHEMBL1374204	28045	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	9	1	7	4.2	Cc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2ccc(OC(C)C)cc2)o1	nan
	20917681	28050	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	2.0	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)s1	nan
	CHEMBL1374225	28050	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	2.0	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)s1	nan
	4855374	28324	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	0	10	-0.3	CN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1(C#N)CCCCC1	nan
	CHEMBL1376372	28324	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	0	10	-0.3	CN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1(C#N)CCCCC1	nan
	20917816	28760	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	0	5	2.4	CC1CCN(S(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)CC1	nan
	CHEMBL1380363	28760	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	0	5	2.4	CC1CCN(S(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)CC1	nan
	661999	28845	14	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	CHEMBL1380975	28845	14	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	4342649	28958	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	5027943	28958	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	CHEMBL1381980	28958	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	135431552	29026	10	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	6	4.7	N#Cc1c(O)nc(SCc2ccc(Cl)cc2)nc1-c1cccs1	nan
	CHEMBL1382616	29026	10	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	6	4.7	N#Cc1c(O)nc(SCc2ccc(Cl)cc2)nc1-c1cccs1	nan
	921583	29419	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	1	1	3	4.3	Sc1nc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1386089	29419	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	1	1	3	4.3	Sc1nc(-c2ccccc2)nc2ccc(Br)cc12	nan
	5428525	29739	23	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	1	5	1.8	COC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	CHEMBL1388510	29739	23	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	1	5	1.8	COC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	5824610	29787	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	7	1	5	3.1	CN(C)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1388949	29787	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	7	1	5	3.1	CN(C)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	16194879	30135	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c(OC)c1	nan
	CHEMBL1391905	30135	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c(OC)c1	nan
	1256976	30196	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	2	5	3.6	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3cccnc3)nc3ccc(Br)cc23)cc1	nan
	CHEMBL1392432	30196	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	2	5	3.6	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3cccnc3)nc3ccc(Br)cc23)cc1	nan
	7222624	30489	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)c(F)c3)nn2)s1	nan
	CHEMBL1395178	30489	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)c(F)c3)nn2)s1	nan
	16018363	30513	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	6	5.5	COc1ccc(NC(=O)c2ccc3c(c2)sc2nc(-c4ccc(OC)cc4)cn23)cc1	nan
	CHEMBL1395439	30513	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	6	5.5	COc1ccc(NC(=O)c2ccc3c(c2)sc2nc(-c4ccc(OC)cc4)cn23)cc1	nan
	15990211	30664	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	6	3.1	Fc1ccc(CNc2nc3ccc(Cl)cc3n3nnnc23)cc1	nan
	CHEMBL1397707	30664	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	6	3.1	Fc1ccc(CNc2nc3ccc(Cl)cc3n3nnnc23)cc1	nan
	7151328	30725	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	5	3.1	CCS(=O)(=O)Nc1ccc(-c2cn3c(C)csc3n2)cc1	nan
	CHEMBL1398475	30725	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	5	3.1	CCS(=O)(=O)Nc1ccc(-c2cn3c(C)csc3n2)cc1	nan
	20939725	30827	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	0	7	2.9	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)Oc2ccccc21	nan
	CHEMBL1399426	30827	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	0	7	2.9	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)Oc2ccccc21	nan
	16452548	31079	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)c1	nan
	CHEMBL1401713	31079	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)c1	nan
	3709623	31189	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)o1	nan
	CHEMBL1402642	31189	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)o1	nan
	5212778	31217	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	661982	31217	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	CHEMBL1402874	31217	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	3152754	31300	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	5	4.2	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccs1)c1ccco1	nan
	CHEMBL1403767	31300	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	5	4.2	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccs1)c1ccco1	nan
	2816622	31377	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	4.8	COc1ccc(-n2c(=S)[nH]c3sc(-c4ccccc4)cc3c2=O)c(OC)c1	nan
	CHEMBL1404356	31377	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	4.8	COc1ccc(-n2c(=S)[nH]c3sc(-c4ccccc4)cc3c2=O)c(OC)c1	nan
	7245568	31503	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	2.2	COc1ccc(NC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1405733	31503	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	2.2	COc1ccc(NC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4184357	31521	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	6	1	9	4.3	O=C(O)c1ccc(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1405932	31521	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	6	1	9	4.3	O=C(O)c1ccc(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)cc1	nan
	757946	31756	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	2	4.7	Cc1nc2ccc(Br)cc2c(-c2ccccc2)c1C(=O)O	nan
	CHEMBL1407788	31756	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	2	4.7	Cc1nc2ccc(Br)cc2c(-c2ccccc2)c1C(=O)O	nan
	3160259	31829	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	7	2.2	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCC(C)O	nan
	CHEMBL1408356	31829	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	7	2.2	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCC(C)O	nan
	1071246	31902	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	8	0.6	CCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1408937	31902	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	8	0.6	CCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	744304	31937	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	2	4	2.4	COc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	CHEMBL1409203	31937	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	2	4	2.4	COc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	3240452	31939	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	0.4	O=C(Cn1cnc2c(nnn2-c2ccc(F)cc2)c1=O)NCC1CCCO1	nan
	CHEMBL1409223	31939	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	0.4	O=C(Cn1cnc2c(nnn2-c2ccc(F)cc2)c1=O)NCC1CCCO1	nan
	15989908	32045	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1410062	32045	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	20923121	32085	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	2.0	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccco1	nan
	CHEMBL1410345	32085	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	2.0	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccco1	nan
	3998353	32278	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	8	1.0	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCOCC4)c3)nc2n1	nan
	CHEMBL1412011	32278	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	8	1.0	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCOCC4)c3)nc2n1	nan
	16034646	32371	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	3.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1412706	32371	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	3.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(Cl)cc3)nnc12	nan
	1145396	32466	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	5026856	32466	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1413474	32466	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	652152	32609	19	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	2	1	3	2.7	COc1ccc2c(Cl)c(C(N)=O)sc2c1	nan
	CHEMBL1414671	32609	19	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	2	1	3	2.7	COc1ccc2c(Cl)c(C(N)=O)sc2c1	nan
	1004109	32727	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	2	4	5.4	Cc1ccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1F	nan
	CHEMBL1415733	32727	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	2	4	5.4	Cc1ccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1F	nan
	22334931	32787	27	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	4	3.5	O=C(O)CSc1nc2ccccc2nc1Cc1ccccc1F	nan
	CHEMBL1416271	32787	27	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	4	3.5	O=C(O)CSc1nc2ccccc2nc1Cc1ccccc1F	nan
	3953394	32892	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	8	1.5	O=C(CSc1nnc2ccccn12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1417177	32892	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	8	1.5	O=C(CSc1nnc2ccccn12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	24687828	32907	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	0	11	-0.1	COc1ccc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1	nan
	CHEMBL1417257	32907	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	0	11	-0.1	COc1ccc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1	nan
	7184635	33160	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1cccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1419486	33160	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1cccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	4796292	33205	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	6	1.1	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cnccn2)c1	nan
	CHEMBL1419907	33205	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	6	1.1	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cnccn2)c1	nan
	744542	33228	34	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	3	3.4	Cc1cc(SCCC(=O)O)nc2c(C)cccc12	nan
	CHEMBL1420044	33228	34	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	3	3.4	Cc1cc(SCCC(=O)O)nc2c(C)cccc12	nan
	3789487	33298	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	3.0	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(F)cc1)c1ccco1	nan
	CHEMBL1420588	33298	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	3.0	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(F)cc1)c1ccco1	nan
	1473006	33351	13	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	0	2	4.1	COc1cc2cc(Br)cc(Br)c2nc1C	nan
	CHEMBL1421084	33351	13	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	0	2	4.1	COc1cc2cc(Br)cc(Br)c2nc1C	nan
	22421602	33405	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	9	2	8	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1	nan
	CHEMBL1421499	33405	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	9	2	8	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1	nan
	20957484	33412	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	9	1.3	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	CHEMBL1421579	33412	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	9	1.3	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	7190683	33427	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1421703	33427	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	7190642	33569	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1422914	33569	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	741274	33799	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	0	7	0.6	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCC3	nan
	CHEMBL1424800	33799	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	0	7	0.6	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCC3	nan
	3816425	33885	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1425600	33885	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	7299201	33893	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.6	Cc1cccc(C)c1Nc1c(-c2ccc(N3CCOCC3)cc2)nc2cnccn12	nan
	CHEMBL1425693	33893	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.6	Cc1cccc(C)c1Nc1c(-c2ccc(N3CCOCC3)cc2)nc2cnccn12	nan
	5739077	34068	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	8	2.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1427088	34068	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	8	2.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3830309	34201	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	6	4.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1cc2ccccc2o1	nan
	CHEMBL1428271	34201	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	6	4.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1cc2ccccc2o1	nan
	20903609	34452	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	9	1	10	3.0	COc1cc(NC(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)cc(OC)c1	nan
	CHEMBL1430241	34452	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	9	1	10	3.0	COc1cc(NC(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)cc(OC)c1	nan
	990446	34479	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	9	2.1	COc1cccc(-n2nc3c(-n4ncc(C#N)c4N)nnc(C)c3c2C)c1	nan
	CHEMBL1430459	34479	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	9	2.1	COc1cccc(-n2nc3c(-n4ncc(C#N)c4N)nnc(C)c3c2C)c1	nan
	2809114	34627	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	4	4.7	CC(=O)c1sc(-c2ccccc2)cc1NS(=O)(=O)c1ccc(C)cc1	nan
	CHEMBL1431741	34627	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	4	4.7	CC(=O)c1sc(-c2ccccc2)cc1NS(=O)(=O)c1ccc(C)cc1	nan
	4968705	34778	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	0	10	-0.5	CN(C)S(=O)(=O)c1ccc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1433054	34778	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	0	10	-0.5	CN(C)S(=O)(=O)c1ccc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	16019549	34871	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	3	0	9	2.8	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(N1CCOCC1)c1sccc12	nan
	CHEMBL1433993	34871	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	3	0	9	2.8	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(N1CCOCC1)c1sccc12	nan
	20885693	34979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	1	6	2.0	Cc1nn(CCCC(=O)NCCc2ccc(Cl)cc2)c(=O)c2nccn12	nan
	CHEMBL1435443	34979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	1	6	2.0	Cc1nn(CCCC(=O)NCCc2ccc(Cl)cc2)c(=O)c2nccn12	nan
	4380857	34985	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1c(CN(C)C(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cnn1C	nan
	CHEMBL1435516	34985	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1c(CN(C)C(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cnn1C	nan
	5066674	34997	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	2.7	COC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc3c2N(C(C)=O)CC3)cc(C(=O)OC)c1	nan
	CHEMBL1435676	34997	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	2.7	COC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc3c2N(C(C)=O)CC3)cc(C(=O)OC)c1	nan
	3993922	35063	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	7	1.2	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1436555	35063	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	7	1.2	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2ccsc2n1	nan
	16018682	35080	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.1	CCc1ccccc1NC(=O)CSc1nncn2c1cc1oc(C)cc12	nan
	CHEMBL1436824	35080	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.1	CCc1ccccc1NC(=O)CSc1nncn2c1cc1oc(C)cc12	nan
	16026770	35100	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	7	1.7	Cc1csc2nc(COC(=O)CNC(=O)c3ccc(F)cc3)cc(=O)n12	nan
	CHEMBL1437080	35100	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	7	1.7	Cc1csc2nc(COC(=O)CNC(=O)c3ccc(F)cc3)cc(=O)n12	nan
	90660425	35224	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	5	5.1	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccccc2F)cc1C	nan
	CHEMBL1438291	35224	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	5	5.1	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccccc2F)cc1C	nan
	663438	35393	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	6	1.4	O=S(=O)(c1cccc(-c2cn3cccnc3n2)c1)N1CCOCC1	nan
	CHEMBL1439795	35393	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	6	1.4	O=S(=O)(c1cccc(-c2cn3cccnc3n2)c1)N1CCOCC1	nan
	135544645	35402	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	7	3.7	N#Cc1c(O)nc(SCC(=O)Nc2cccc(Cl)c2)nc1-c1ccco1	nan
	CHEMBL1439904	35402	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	7	3.7	N#Cc1c(O)nc(SCC(=O)Nc2cccc(Cl)c2)nc1-c1ccco1	nan
	3363660	35542	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	4976974	35542	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	CHEMBL1441169	35542	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	2854626	35550	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CC(=O)C1=C(C)NC(SCC(=O)c2ccc(Cl)cc2)=C(C#N)C1CC(C)C	nan
	CHEMBL1441242	35550	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CC(=O)C1=C(C)NC(SCC(=O)c2ccc(Cl)cc2)=C(C#N)C1CC(C)C	nan
	20957185	35704	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	8	1.9	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccc(F)cc1	nan
	CHEMBL1442625	35704	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	8	1.9	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccc(F)cc1	nan
	812443	35898	45	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	2	1	4	3.2	C=CCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1444467	35898	45	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	2	1	4	3.2	C=CCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	20923160	35900	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccccc1CNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1444486	35900	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccccc1CNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	16745544	36277	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	1	5	2.5	COc1ccc(C2=CC3=C(Br)C(=O)C(C)(O)C(=O)C3=CO2)cc1	nan
	CHEMBL1447877	36277	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	1	5	2.5	COc1ccc(C2=CC3=C(Br)C(=O)C(C)(O)C(=O)C3=CO2)cc1	nan
	2376086	36341	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	5	2.6	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1448425	36341	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	5	2.6	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	16745680	36491	0	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	0	7	5.7	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1CC(C)C	nan
	CHEMBL1449527	36491	0	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	0	7	5.7	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1CC(C)C	nan
	16018684	36492	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	4.4	Cc1cc(C)c(NC(=O)CSc2nncn3c2cc2oc(C)cc23)c(C)c1	nan
	CHEMBL1449543	36492	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	4.4	Cc1cc(C)c(NC(=O)CSc2nncn3c2cc2oc(C)cc23)c(C)c1	nan
	1094076	36505	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	6	3.0	CC(=O)c1ccc(Nc2nc(=O)c3cccnc3s2)cc1	nan
	CHEMBL1449615	36505	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	6	3.0	CC(=O)c1ccc(Nc2nc(=O)c3cccnc3s2)cc1	nan
	3514089	36649	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1450861	36649	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	6619005	36867	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	5	1	7	4.4	Cc1c(N2C(=O)C(O)=C(C(=O)c3ccc(Br)cc3)C2c2cccnc2)c(=O)n(-c2ccccc2)n1C	nan
	CHEMBL1452549	36867	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	5	1	7	4.4	Cc1c(N2C(=O)C(O)=C(C(=O)c3ccc(Br)cc3)C2c2cccnc2)c(=O)n(-c2ccccc2)n1C	nan
	16194575	37044	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)s1	nan
	CHEMBL1453968	37044	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)s1	nan
	3178522	37108	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	0	9	0.2	CCCCn1c(SCC(=O)N2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1454485	37108	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	0	9	0.2	CCCCn1c(SCC(=O)N2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	2613266	37179	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	0	8	2.8	O=[N+]([O-])c1cc2c(c(CSc3nnc4ccccn34)c1)OCOC2	nan
	CHEMBL1455089	37179	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	0	8	2.8	O=[N+]([O-])c1cc2c(c(CSc3nnc4ccccn34)c1)OCOC2	nan
	1084466	37291	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	6	2.5	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	CHEMBL1456125	37291	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	6	2.5	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	20885676	37343	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	6	1.6	Cc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1456629	37343	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	6	1.6	Cc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	3715206	37352	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	5	3.9	CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1456701	37352	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	5	3.9	CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	3252203	37505	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.2	O=C(CSc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	CHEMBL1457998	37505	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.2	O=C(CSc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	2939635	37608	33	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	247	3	1	3	3.1	Cc1cc(SC(C)C(=O)O)nc2ccccc12	nan
	CHEMBL1458912	37608	33	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	247	3	1	3	3.1	Cc1cc(SC(C)C(=O)O)nc2ccccc12	nan
	1442575	37848	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	6	1	4	3.7	CCCc1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1460883	37848	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	6	1	4	3.7	CCCc1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	4412828	37946	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	9	1	7	2.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)COc2ccc(C#N)cc2)c1	nan
	CHEMBL1461851	37946	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	9	1	7	2.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)COc2ccc(C#N)cc2)c1	nan
	1838049	38011	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	0.4	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1462354	38011	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	0.4	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	15945416	38753	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	3.5	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1468328	38753	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	3.5	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	4905842	38772	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	9	4.4	CSc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(SC)s2)cc1	nan
	CHEMBL1468444	38772	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	9	4.4	CSc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(SC)s2)cc1	nan
	6498441	38881	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	2.7	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NC1CCCC1	nan
	CHEMBL1469364	38881	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	2.7	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NC1CCCC1	nan
	4356276	38984	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	8	4.1	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1470300	38984	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	8	4.1	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	3776625	39039	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Br)c2)no1	nan
	CHEMBL1470725	39039	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Br)c2)no1	nan
	3186626	39060	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	CHEMBL1470851	39060	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	7256722	39383	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	2.4	Cc1ccc2nc(SCC(=O)Nc3ccc(F)cc3F)nc(=O)n2c1	nan
	CHEMBL1474450	39383	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	2.4	Cc1ccc2nc(SCC(=O)Nc3ccc(F)cc3F)nc(=O)n2c1	nan
	15990395	39531	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1cccc(NC(=O)c2nc3ccccc3n(C)c2=O)c1	nan
	CHEMBL1476510	39531	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1cccc(NC(=O)c2nc3ccccc3n(C)c2=O)c1	nan
	1506838	39574	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	4	3.1	Cc1cc(CNC(=O)COc2ccc(C#N)cc2)c2ccccc2n1	nan
	CHEMBL1477044	39574	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	4	3.1	Cc1cc(CNC(=O)COc2ccc(C#N)cc2)c2ccccc2n1	nan
	1471774	39617	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	3.0	CSc1cc(-c2ccccc2)nc(O)c1C#N	nan
	CHEMBL1477426	39617	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	3.0	CSc1cc(-c2ccccc2)nc(O)c1C#N	nan
	20970002	39627	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1	nan
	CHEMBL1477514	39627	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1	nan
	2931382	39921	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	2	5	2.1	COC(=O)c1sccc1NC(=O)C1CC=CCC1C(=O)O	nan
	CHEMBL1480089	39921	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	2	5	2.1	COC(=O)c1sccc1NC(=O)C1CC=CCC1C(=O)O	nan
	7120051	39928	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1480178	39928	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	16018856	39948	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	0	8	5.5	COc1ccc(-c2nc(CSc3nnc(C)n4c3cc3sccc34)c(C)o2)cc1	nan
	CHEMBL1480328	39948	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	0	8	5.5	COc1ccc(-c2nc(CSc3nnc(C)n4c3cc3sccc34)c(C)o2)cc1	nan
	3451317	39961	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	7	0.8	CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2nncn2C)c1	nan
	CHEMBL1480436	39961	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	7	0.8	CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2nncn2C)c1	nan
	3535142	40082	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	9	1	9	3.4	O=C(O)CCCCCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1481365	40082	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	9	1	9	3.4	O=C(O)CCCCCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	3574141	40133	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	0	6	2.1	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	CHEMBL1481920	40133	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	0	6	2.1	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	5736472	40425	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	6	1	7	2.5	O=c1c2ccccc2nc(/C=C/c2ccc([N+](=O)[O-])o2)n1CCCO	nan
	CHEMBL1484332	40425	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	6	1	7	2.5	O=c1c2ccccc2nc(/C=C/c2ccc([N+](=O)[O-])o2)n1CCCO	nan
	5304429	40454	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	1	4	2.4	CC(=O)Nc1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1484671	40454	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	1	4	2.4	CC(=O)Nc1cccc(-c2cn3cccnc3n2)c1	nan
	16012070	40490	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	7	2.9	Cc1cc(=O)n2nc(N3CCC(C(=O)Nc4c(C)cccc4C)CC3)sc2n1	nan
	CHEMBL1484919	40490	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	7	2.9	Cc1cc(=O)n2nc(N3CCC(C(=O)Nc4c(C)cccc4C)CC3)sc2n1	nan
	4399091	40492	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1ccccc1C1C(C(=O)c2ccc(C)o2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1484932	40492	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1ccccc1C1C(C(=O)c2ccc(C)o2)=C(O)C(=O)N1c1cc(C)on1	nan
	1387364	40547	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1485560	40547	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1576237	40547	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	6622721	40818	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	5	3.6	CNc1nc2c(-c3ccc(Cl)cc3)nnn2c2ccccc12	nan
	CHEMBL1487831	40818	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	5	3.6	CNc1nc2c(-c3ccc(Cl)cc3)nnn2c2ccccc12	nan
	1002526	40859	11	None	-2	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	4	4.1	O=C(O)c1cc(-c2ccc3c(c2)OCO3)nc2ccc(Br)cc12	nan
	CHEMBL1488092	40859	11	None	-2	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	4	4.1	O=C(O)c1cc(-c2ccc3c(c2)OCO3)nc2ccc(Br)cc12	nan
	7190684	40917	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1488468	40917	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	5881431	41016	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	1	7	4.2	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1489225	41016	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	1	7	4.2	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2032322	41131	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	7	3.5	CCN(CC)CCCNc1nc(SC)nc2sc3c(c12)CCN(C)C3	nan
	CHEMBL1490215	41131	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	7	3.5	CCN(CC)CCCNc1nc(SC)nc2sc3c(c12)CCN(C)C3	nan
	755499	41238	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	7	1.0	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	CHEMBL1490891	41238	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	7	1.0	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	1283516	41429	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	7	0.9	O=c1[nH]n2cc(-n3cc([N+](=O)[O-])cn3)cnc2c1Br	nan
	CHEMBL1492212	41429	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	7	0.9	O=c1[nH]n2cc(-n3cc([N+](=O)[O-])cn3)cnc2c1Br	nan
	774862	41496	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	0	4	3.1	Cn1c(-c2ccc([N+](=O)[O-])cc2)nc2ccccc21	nan
	CHEMBL1492732	41496	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	0	4	3.1	Cn1c(-c2ccc([N+](=O)[O-])cc2)nc2ccccc21	nan
	3279901	41591	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	4	3.0	CC(=O)NC(CSc1cc(C)nc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1493652	41591	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	4	3.0	CC(=O)NC(CSc1cc(C)nc2ccc(Br)cc12)C(=O)O	nan
	4795978	41594	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	3.8	CN(C)S(=O)(=O)c1cccc(COc2ncnc3c(Cl)cc(Cl)cc23)c1	nan
	CHEMBL1493688	41594	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	3.8	CN(C)S(=O)(=O)c1cccc(COc2ncnc3c(Cl)cc(Cl)cc23)c1	nan
	15988336	41675	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1cccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1494501	41675	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1cccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	664285	41692	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	3	0	5	3.1	CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1494683	41692	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	3	0	5	3.1	CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	748270	41733	41	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	0	4	2.2	Cc1nnc2c3ccccc3c(Cl)nn12	nan
	CHEMBL1495086	41733	41	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	0	4	2.2	Cc1nnc2c3ccccc3c(Cl)nn12	nan
	3186635	41843	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	0	9	-0.8	CCN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1496152	41843	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	0	9	-0.8	CCN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	2561752	42079	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	3.2	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCS3	nan
	CHEMBL1498284	42079	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	3.2	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCS3	nan
	21552	42123	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	7	0.1	Cn1c(=O)c2c(nc(Cc3ccc(N)cc3)n2C)n(C)c1=O	nan
	CHEMBL1498782	42123	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	7	0.1	Cn1c(=O)c2c(nc(Cc3ccc(N)cc3)n2C)n(C)c1=O	nan
	7677140	42176	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	5	2.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1cccnc1	nan
	CHEMBL1499143	42176	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	5	2.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1cccnc1	nan
	2816379	42340	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	2.1	CCOC(=O)c1nnn2c1nc(SCC(C)=O)c1ccccc12	nan
	CHEMBL1500551	42340	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	2.1	CCOC(=O)c1nnn2c1nc(SCC(C)=O)c1ccccc12	nan
	18554434	42377	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	8	1.8	O=C(CSc1ncnc2c1nnn2Cc1ccccc1F)NCC1CCCO1	nan
	CHEMBL1500823	42377	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	8	1.8	O=C(CSc1ncnc2c1nnn2Cc1ccccc1F)NCC1CCCO1	nan
	5077853	42461	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	1	8	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1	nan
	CHEMBL1501692	42461	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	1	8	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1	nan
	7120056	42466	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1501734	42466	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	3884053	42621	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	661074	42621	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	CHEMBL1503060	42621	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	20957430	42658	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	3.2	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(NCc4ccc5c(c4)OCO5)nn23)c1	nan
	CHEMBL1503367	42658	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	3.2	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(NCc4ccc5c(c4)OCO5)nn23)c1	nan
	16452701	42764	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)n1	nan
	CHEMBL1504372	42764	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)n1	nan
	3457991	42894	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	5	1	8	3.2	Cc1ccc(F)cc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	CHEMBL1505540	42894	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	5	1	8	3.2	Cc1ccc(F)cc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	5198374	42908	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	7	2.4	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1505625	42908	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	7	2.4	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	986582	43010	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	3.2	CCc1ccc2oc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)c(C)c2c1	nan
	CHEMBL1506399	43010	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	3.2	CCc1ccc2oc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)c(C)c2c1	nan
	1811810	43043	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	2	3.5	C=CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1506727	43043	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	2	3.5	C=CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	135528107	43565	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	5	3.2	CCN(CC(=O)NC(C)C)Cc1nc(O)c2cc(Br)cc(Br)c2n1	nan
	CHEMBL1511291	43565	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	5	3.2	CCN(CC(=O)NC(C)C)Cc1nc(O)c2cc(Br)cc(Br)c2n1	nan
	16496658	43681	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.1	CC1CCCN(C(=O)COC(=O)CNC(=O)c2sc3ccccc3c2Cl)C1	nan
	CHEMBL1512634	43681	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.1	CC1CCCN(C(=O)COC(=O)CNC(=O)c2sc3ccccc3c2Cl)C1	nan
	15988304	43759	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	0	8	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccccc4)CC3)nnc12	nan
	CHEMBL1513808	43759	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	0	8	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccccc4)CC3)nnc12	nan
	16026221	43874	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	1.2	CCOC(=O)C1CCN(C(=O)Cn2c(=O)cc(C)c3c(C)nn(C)c32)CC1	nan
	CHEMBL1515615	43874	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	1.2	CCOC(=O)C1CCN(C(=O)Cn2c(=O)cc(C)c3c(C)nn(C)c32)CC1	nan
	662069	44027	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	1.8	COC(=O)c1cc(Br)c(=O)n(-c2nccs2)c1	nan
	CHEMBL1517409	44027	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	1.8	COC(=O)c1cc(Br)c(=O)n(-c2nccs2)c1	nan
	3489758	44085	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	2	9	0.9	Cn1c(=O)c2ncn(CC(=O)N=Nc3c(O)[nH]c4ccccc34)c2n(C)c1=O	nan
	CHEMBL1518029	44085	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	2	9	0.9	Cn1c(=O)c2ncn(CC(=O)N=Nc3c(O)[nH]c4ccccc34)c2n(C)c1=O	nan
	16018686	44248	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	6	4.3	Cc1cc2c(cc3c(SCC(=O)Nc4ccc(Cl)cc4F)nncn32)o1	nan
	CHEMBL1519470	44248	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	6	4.3	Cc1cc2c(cc3c(SCC(=O)Nc4ccc(Cl)cc4F)nncn32)o1	nan
	20957225	44266	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	9	1.7	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)nc1	nan
	CHEMBL1519640	44266	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	9	1.7	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)nc1	nan
	2991435	44284	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	6	2.8	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(Br)o2)c1	nan
	CHEMBL1519787	44284	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	6	2.8	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(Br)o2)c1	nan
	5959865	44398	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	6	4.0	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(F)cc3)ccc2O1	nan
	CHEMBL1520789	44398	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	6	4.0	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(F)cc3)ccc2O1	nan
	4197564	44563	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	11	1	8	3.9	COc1cc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	CHEMBL1522190	44563	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	11	1	8	3.9	COc1cc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	5064245	44580	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	5	1	5	1.3	O=C(COc1ncnc2ccccc12)NCC1CCCO1	nan
	CHEMBL1522316	44580	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	5	1	5	1.3	O=C(COc1ncnc2ccccc12)NCC1CCCO1	nan
	3317909	44583	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	3536112	44583	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	CHEMBL1522365	44583	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	20957467	44658	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	9	1	8	1.8	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4)CC3)n2n1	nan
	CHEMBL1523099	44658	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	9	1	8	1.8	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4)CC3)n2n1	nan
	3242118	44671	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	1	5	2.6	Cc1nn(C(C)C(=O)O)c(=O)c2c1sc1ccccc12	nan
	CHEMBL1523214	44671	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	1	5	2.6	Cc1nn(C(C)C(=O)O)c(=O)c2c1sc1ccccc12	nan
	3178468	44729	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	8	0.6	CCn1c(SCC(=O)N2CCCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1523743	44729	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	8	0.6	CCn1c(SCC(=O)N2CCCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	774385	44951	50	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	192	1	1	4	2.3	Cc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1525902	44951	50	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	192	1	1	4	2.3	Cc1ccccc1-c1nnc(S)o1	nan
	6156848	44964	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	6	3.9	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccccc3)ccc2O1	nan
	CHEMBL1525999	44964	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	6	3.9	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccccc3)ccc2O1	nan
	20923115	45223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	0	6	3.1	CCN(c1ccccc1)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1528270	45223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	0	6	3.1	CCN(c1ccccc1)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	1173803	45333	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	0	9	0.3	CCCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1529195	45333	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	0	9	0.3	CCCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1150969	45334	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	2	6	3.2	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	CHEMBL1529199	45334	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	2	6	3.2	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	20957502	45401	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1cccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)c1	nan
	CHEMBL1529803	45401	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1cccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)c1	nan
	3146230	45583	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	6	2.7	Cc1sc2ncnc(SCC(=O)NCC3CCCO3)c2c1C	nan
	CHEMBL1531505	45583	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	6	2.7	Cc1sc2ncnc(SCC(=O)NCC3CCCO3)c2c1C	nan
	20888842	45847	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	9	1.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1533752	45847	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	9	1.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	7677714	45849	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	5	3.2	Cc1ccc(C(=O)NCc2nnc3c(C(F)(F)F)cc(Cl)cn23)o1	nan
	CHEMBL1533761	45849	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	5	3.2	Cc1ccc(C(=O)NCc2nnc3c(C(F)(F)F)cc(Cl)cn23)o1	nan
	16018626	45895	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1ccc(NC(=O)CSc2nncn3c2cc2occc23)c(OC)c1	nan
	CHEMBL1534283	45895	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1ccc(NC(=O)CSc2nncn3c2cc2occc23)c(OC)c1	nan
	2415319	45897	24	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	5	4.0	O=C(O)c1ccccc1Sc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1534296	45897	24	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	5	4.0	O=C(O)c1ccccc1Sc1ncnc2sc3c(c12)CCC3	nan
	15988400	45926	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	7	3.0	CCn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1534534	45926	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	7	3.0	CCn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	3559456	46029	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Br)c2)no1	nan
	CHEMBL1535636	46029	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Br)c2)no1	nan
	752859	46052	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	6	2.6	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccccc2)n1	nan
	CHEMBL1535864	46052	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	6	2.6	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccccc2)n1	nan
	1258096	46087	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	7	3.1	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)c(Cl)c1	nan
	CHEMBL1536340	46087	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	7	3.1	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)c(Cl)c1	nan
	5911396	46111	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	8	3.5	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)OCCO4)C2c2ccc(F)cc2)s1	nan
	CHEMBL1536589	46111	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	8	3.5	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)OCCO4)C2c2ccc(F)cc2)s1	nan
	2968508	46212	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	3.4	O=C(COc1ccccc1)NC(=S)Nc1cccc2cc(O)ccc12	nan
	CHEMBL1537461	46212	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	3.4	O=C(COc1ccccc1)NC(=S)Nc1cccc2cc(O)ccc12	nan
	973903	46372	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	3	7	1.5	O=C(NNc1nc(=O)c2cccnc2s1)c1ccccc1O	nan
	CHEMBL1538711	46372	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	3	7	1.5	O=C(NNc1nc(=O)c2cccnc2s1)c1ccccc1O	nan
	4786350	46425	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	4	0	6	2.6	COC(=O)c1ccc(COc2ncnc3ccccc23)o1	nan
	CHEMBL1539182	46425	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	4	0	6	2.6	COC(=O)c1ccc(COc2ncnc3ccccc23)o1	nan
	4199276	46432	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	10	-0.3	Cn1c(=O)c2nc(NNC(=O)c3ccc([N+](=O)[O-])cc3)cnc2n(C)c1=O	nan
	CHEMBL1539261	46432	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	10	-0.3	Cn1c(=O)c2nc(NNC(=O)c3ccc([N+](=O)[O-])cc3)cnc2n(C)c1=O	nan
	20957177	46457	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	8	2.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccccc1Cl	nan
	CHEMBL1539515	46457	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	8	2.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccccc1Cl	nan
	775376	46741	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	7	-0.1	Cn1c(=O)c2c(ncn2CC(=O)NC2CCCCC2)n(C)c1=O	nan
	CHEMBL1541812	46741	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	7	-0.1	Cn1c(=O)c2c(ncn2CC(=O)NC2CCCCC2)n(C)c1=O	nan
	2027988	46831	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)cc1	nan
	CHEMBL1542663	46831	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)cc1	nan
	7190638	47002	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	7	2.9	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccccc1	nan
	CHEMBL1544038	47002	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	7	2.9	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccccc1	nan
	5291252	47059	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	4	4.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1544399	47059	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	4	4.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	3531704	47119	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	5.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccc(Oc3ccccc3)c2)no1	nan
	CHEMBL1544885	47119	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	5.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccc(Oc3ccccc3)c2)no1	nan
	1254436	47156	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	10	-0.3	Cn1c(=O)c2c(nc(Br)n2Cc2nnc(N)s2)n(C)c1=O	nan
	CHEMBL1545144	47156	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	10	-0.3	Cn1c(=O)c2c(nc(Br)n2Cc2nnc(N)s2)n(C)c1=O	nan
	20923178	47199	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)o1	nan
	CHEMBL1545457	47199	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)o1	nan
	2827527	47212	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	0	2	3.2	Cc1ccc2c(ccc(=S)n2C)c1	nan
	CHEMBL1545583	47212	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	0	2	3.2	Cc1ccc2c(ccc(=S)n2C)c1	nan
	4114707	47264	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2nnc(SCC(=O)NCC3CCCO3)n2c2ccccc12	nan
	CHEMBL1546017	47264	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2nnc(SCC(=O)NCC3CCCO3)n2c2ccccc12	nan
	6620293	47342	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	0	5	3.8	O=C(C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1)N1CCCC1	nan
	CHEMBL1546743	47342	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	0	5	3.8	O=C(C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1)N1CCCC1	nan
	2341870	47352	2	None	-3	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	0	5	4.1	Cc1ccc(C)n1-c1ccc(-c2nnc3n2CCCCC3)s1	nan
	CHEMBL1546820	47352	2	None	-3	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	0	5	4.1	Cc1ccc(C)n1-c1ccc(-c2nnc3n2CCCCC3)s1	nan
	2150404	47595	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	1	1	4	3.8	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1549101	47595	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	1	1	4	3.8	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccccc1	nan
	2482804	47698	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	5	2	8	-0.4	C=CCNC(=O)NC(=O)COC(=O)c1nc2nccc(C)n2n1	nan
	CHEMBL1549963	47698	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	5	2	8	-0.4	C=CCNC(=O)NC(=O)COC(=O)c1nc2nccc(C)n2n1	nan
	7184632	47827	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1550958	47827	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	16030519	47845	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)cc1	nan
	CHEMBL1551209	47845	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)cc1	nan
	1116231	47949	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.4	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(Cl)c2Cl)n(C)c1=O	nan
	CHEMBL1552691	47949	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.4	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(Cl)c2Cl)n(C)c1=O	nan
	16031533	47959	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	6	4.5	CCc1ccccc1NC(=O)CSc1nnc(-c2ccc(OC)cc2)s1	nan
	CHEMBL1552858	47959	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	6	4.5	CCc1ccccc1NC(=O)CSc1nnc(-c2ccc(OC)cc2)s1	nan
	16033232	47969	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2cccc(Cl)c2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1552980	47969	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2cccc(Cl)c2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	2136319	47991	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1553213	47991	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	16018758	48050	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	5	4.5	Cc1cc2c(cc3c(SCc4cccc(F)c4)nnc(C)n32)o1	nan
	CHEMBL1554096	48050	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	5	4.5	Cc1cc2c(cc3c(SCc4cccc(F)c4)nnc(C)n32)o1	nan
	4808155	48228	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	7	0.7	Cn1c(=O)c2c(ncn2CCOc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1556293	48228	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	7	0.7	Cn1c(=O)c2c(ncn2CCOc2ccc(F)cc2)n(C)c1=O	nan
	664905	48367	16	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	3.4	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccco1	nan
	CHEMBL1557499	48367	16	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	3.4	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccco1	nan
	846378	48481	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	5	3.8	CN(C)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	CHEMBL1558527	48481	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	5	3.8	CN(C)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	20970070	48617	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	7	2.8	CCOc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	CHEMBL1559703	48617	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	7	2.8	CCOc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	749967	48817	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	208	2	1	5	2.0	COc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1561641	48817	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	208	2	1	5	2.0	COc1ccccc1-c1nnc(S)o1	nan
	2816163	48988	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	2	0	7	0.8	CCOC(=O)c1nnn2c3ccccc3c(=O)n(C)c12	nan
	CHEMBL1563125	48988	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	2	0	7	0.8	CCOC(=O)c1nnn2c3ccccc3c(=O)n(C)c12	nan
	754624	49082	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	0	6	3.0	O=c1c2c(-c3ccc([N+](=O)[O-])cc3)csc2nc2n1CCC2	nan
	CHEMBL1563900	49082	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	0	6	3.0	O=c1c2c(-c3ccc([N+](=O)[O-])cc3)csc2nc2n1CCC2	nan
	20923125	49223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)cc1	nan
	CHEMBL1565225	49223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)cc1	nan
	5818870	49232	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4cccnc4)C3c3ccccc3F)ccc2O1	nan
	CHEMBL1565288	49232	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4cccnc4)C3c3ccccc3F)ccc2O1	nan
	702333	49714	15	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	0	1	3	2.9	Cn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	CHEMBL1569119	49714	15	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	0	1	3	2.9	Cn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	1072636	50051	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	1.0	CCn1c(SCC(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1572163	50051	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	1.0	CCn1c(SCC(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)nc2c1c(=O)n(C)c(=O)n2C	nan
	4912148	50059	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	8	3.6	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2)s1	nan
	CHEMBL1572210	50059	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	8	3.6	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2)s1	nan
	719137	50080	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	1	1	3	3.4	CCn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	CHEMBL1572461	50080	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	1	1	3	3.4	CCn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	22518619	50285	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	8	3.8	CC(C)OCCCn1c(SCC(=O)Nc2ccccc2C(F)(F)F)nc2nccnc2c1=O	nan
	CHEMBL1574369	50285	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	8	3.8	CC(C)OCCCn1c(SCC(=O)Nc2ccccc2C(F)(F)F)nc2nccnc2c1=O	nan
	3516975	50373	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2sccc2Br)nc(-n2cccc2)n1	nan
	CHEMBL1575467	50373	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2sccc2Br)nc(-n2cccc2)n1	nan
	2109682	50399	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	11	0.2	Cc1ccc(C)c(-n2nnnc2SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1575697	50399	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	11	0.2	Cc1ccc(C)c(-n2nnnc2SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	16189479	50518	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	0	8	-0.2	Cn1c(=O)c(=O)n(C)c2cc(S(=O)(=O)N3CC(=O)N(CCc4ccccc4)C(=O)C3)ccc21	nan
	CHEMBL1576683	50518	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	0	8	-0.2	Cn1c(=O)c(=O)n(C)c2cc(S(=O)(=O)N3CC(=O)N(CCc4ccccc4)C(=O)C3)ccc21	nan
	1173783	50552	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCC(=O)Nc1ccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2CC)cc1	nan
	CHEMBL1577034	50552	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCC(=O)Nc1ccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2CC)cc1	nan
	2960985	50763	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	5740252	50763	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	9587839	50763	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	CHEMBL1578738	50763	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	3221467	50775	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	8	1	6	3.0	CCOC(=O)CNC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1578803	50775	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	8	1	6	3.0	CCOC(=O)CNC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	6409200	50910	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	2	5	3.4	O=C(O)c1ccccc1CSc1n[nH]c2c3ccccc3nc-2n1	nan
	CHEMBL1580121	50910	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	2	5	3.4	O=C(O)c1ccccc1CSc1n[nH]c2c3ccccc3nc-2n1	nan
	20957463	50926	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	10	2	7	2.5	O=C(CCc1nnc2ccc(NCCCN3CCCC3=O)nn12)NCc1ccccc1Cl	nan
	CHEMBL1580225	50926	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	10	2	7	2.5	O=C(CCc1nnc2ccc(NCCCN3CCCC3=O)nn12)NCc1ccccc1Cl	nan
	929935	51009	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	1	2	6	4.2	CC(C)c1nc2sc3c(O)nc(S)nc3c2c2c1CCCC2	nan
	CHEMBL1580962	51009	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	1	2	6	4.2	CC(C)c1nc2sc3c(O)nc(S)nc3c2c2c1CCCC2	nan
	3220371	51017	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	6	2.9	CC(C)C(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1581023	51017	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	6	2.9	CC(C)C(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	2916260	51094	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	10	0.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1581657	51094	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	10	0.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	1324776	51190	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	9	2	8	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2cc(OC)nc(OC)n2)cc1	nan
	CHEMBL1582422	51190	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	9	2	8	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2cc(OC)nc(OC)n2)cc1	nan
	4976300	51362	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	9	4.0	CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(OC)c2)s1	nan
	CHEMBL1583844	51362	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	9	4.0	CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(OC)c2)s1	nan
	5083492	51500	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	13	1	5	5.1	CC[N+](CC)(CCCCS(=O)(=O)[O-])CCNP1(=O)C=C(c2ccccc2)OC(c2ccccc2)=C1	nan
	CHEMBL1585012	51500	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	13	1	5	5.1	CC[N+](CC)(CCCCS(=O)(=O)[O-])CCNP1(=O)C=C(c2ccccc2)OC(c2ccccc2)=C1	nan
	6624747	51731	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	2.6	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccccc3)nnc12	nan
	CHEMBL1586923	51731	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	2.6	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccccc3)nnc12	nan
	2384712	52038	21	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	3	4.8	Brc1ccc(-c2nc3ccccc3s2)s1	nan
	CHEMBL1589567	52038	21	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	3	4.8	Brc1ccc(-c2nc3ccccc3s2)s1	nan
	16030403	52113	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	4	4.8	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCC(C)C)cc1	nan
	CHEMBL1590296	52113	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	4	4.8	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCC(C)C)cc1	nan
	16022890	52164	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	2	6	5.2	COc1cc2cc(CNc3ccccc3)c(=O)n(CC(=O)Nc3cccc(Cl)c3C)c2cc1OC	nan
	CHEMBL1590948	52164	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	2	6	5.2	COc1cc2cc(CNc3ccccc3)c(=O)n(CC(=O)Nc3cccc(Cl)c3C)c2cc1OC	nan
	16029271	52249	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	4	0	8	1.5	CCOC(=O)c1noc2ncn(Cc3cccc(C#N)c3)c(=O)c12	nan
	CHEMBL1592100	52249	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	4	0	8	1.5	CCOC(=O)c1noc2ncn(Cc3cccc(C#N)c3)c(=O)c12	nan
	3431356	52270	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	9	2	4	5.8	CCc1ccc(Nc2cc(C(=O)NCCCN(C)c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1592367	52270	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	9	2	4	5.8	CCc1ccc(Nc2cc(C(=O)NCCCN(C)c3ccccc3)c3ccccc3n2)cc1	nan
	16331440	52295	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	0	6	1.9	CC(C(=O)OCC(=O)N(C)C1(C#N)CCCCC1)N1C(=O)c2ccccc2C1=O	nan
	CHEMBL1592707	52295	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	0	6	1.9	CC(C(=O)OCC(=O)N(C)C1(C#N)CCCCC1)N1C(=O)c2ccccc2C1=O	nan
	22518595	52426	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.0	COc1ccccc1NC(=O)CSc1nc2nccnc2c(=O)n1Cc1cccs1	nan
	CHEMBL1594419	52426	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.0	COc1ccccc1NC(=O)CSc1nc2nccnc2c(=O)n1Cc1cccs1	nan
	3630300	52438	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	5	4.9	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(Cl)cc2)n1	nan
	CHEMBL1594498	52438	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	5	4.9	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(Cl)cc2)n1	nan
	16018788	52559	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	CCc1cccc(C)c1NC(=O)CSc1nnc(CC)n2c1cc1occc12	nan
	CHEMBL1595485	52559	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	CCc1cccc(C)c1NC(=O)CSc1nnc(CC)n2c1cc1occc12	nan
	135454734	52638	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	3	9	1.2	Nc1cc(O)nc(SCC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)n1	nan
	CHEMBL1596208	52638	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	3	9	1.2	Nc1cc(O)nc(SCC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)n1	nan
	3151377	52655	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCCC1	nan
	CHEMBL1596336	52655	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCCC1	nan
	2743162	52753	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)cc(Cl)c2)n1	nan
	CHEMBL1597261	52753	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)cc(Cl)c2)n1	nan
	5175738	52799	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	3	2	5	6.0	Nc1c(C(=O)Nc2ccc(F)cc2)sc2nc(-c3cccs3)cc(C(F)(F)F)c12	nan
	CHEMBL1597711	52799	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	3	2	5	6.0	Nc1c(C(=O)Nc2ccc(F)cc2)sc2nc(-c3cccs3)cc(C(F)(F)F)c12	nan
	16018618	52812	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)cc(NC(=O)CSc2nncn3c2cc2occc23)c1	nan
	CHEMBL1597835	52812	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)cc(NC(=O)CSc2nncn3c2cc2occc23)c1	nan
	2931308	52915	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	2.4	COC(=O)c1cc(C)sc1NC(=O)C1CC=CCC1C(=O)O	nan
	CHEMBL1598795	52915	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	2.4	COC(=O)c1cc(C)sc1NC(=O)C1CC=CCC1C(=O)O	nan
	16033260	52931	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1598947	52931	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	7202413	53099	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	8	1.2	Cc1nnc2sc(SCC(=O)N3CCC(C)CC3)nn2c1=O	nan
	CHEMBL1600469	53099	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	8	1.2	Cc1nnc2sc(SCC(=O)N3CCC(C)CC3)nn2c1=O	nan
	893043	53123	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	3	2.4	O=c1[nH]c(=S)c2c(n1-c1ccccc1)CCC2	nan
	CHEMBL1600661	53123	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	3	2.4	O=c1[nH]c(=S)c2c(n1-c1ccccc1)CCC2	nan
	15988297	53284	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.1	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1F	nan
	CHEMBL1602305	53284	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.1	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1F	nan
	20923199	53317	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N(C)Cc1ccco1	nan
	CHEMBL1602602	53317	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N(C)Cc1ccco1	nan
	2138501	53321	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	7	1.0	COc1ccc(C=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	CHEMBL1602628	53321	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	7	1.0	COc1ccc(C=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	16301839	53323	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	11	1.2	Cn1c(N)c(C(=O)CSc2nnc(NC3CCCCC3)s2)c(=O)n(C)c1=O	nan
	CHEMBL1602634	53323	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	11	1.2	Cn1c(N)c(C(=O)CSc2nnc(NC3CCCCC3)s2)c(=O)n(C)c1=O	nan
	2960993	53533	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	5740253	53533	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	9587840	53533	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	CHEMBL1604402	53533	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	5925277	53550	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	8	1.2	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCCOC)CC1	nan
	CHEMBL1604541	53550	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	8	1.2	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCCOC)CC1	nan
	2928283	53598	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCC4)c3nc12	nan
	CHEMBL1605019	53598	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCC4)c3nc12	nan
	6460757	54183	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	6	2.4	Cc1cc2c(SCC(=O)NCC3CCCO3)ncnc2s1	nan
	CHEMBL1609708	54183	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	6	2.4	Cc1cc2c(SCC(=O)NCC3CCCO3)ncnc2s1	nan
	15991073	54314	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	CHEMBL1610897	54314	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	7889635	54372	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	7	1.5	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3)cc(=O)n12	nan
	CHEMBL1611331	54372	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	7	1.5	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3)cc(=O)n12	nan
	778300	54547	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	2	1	10	-1.1	Cn1c(=O)c2c(ncn2Cc2nnc(N)s2)n(C)c1=O	nan
	CHEMBL1612871	54547	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	2	1	10	-1.1	Cn1c(=O)c2c(ncn2Cc2nnc(N)s2)n(C)c1=O	nan
	705485	54943	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	CHEMBL1321656	54943	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	CHEMBL1617945	54943	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	20279	55055	95	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	CHEMBL1619	55055	95	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	1187262	55327	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	CHEMBL1462585	55327	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	CHEMBL1621394	55327	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	44143728	59916	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	CHEMBL1553539	59916	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	CHEMBL1741041	59916	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	135641876	71806	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	10	-0.7	COc1cc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1O	nan
	CHEMBL1979668	71806	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	10	-0.7	COc1cc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1O	nan
	135475570	72298	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	7	2.3	CCN(CC)S(=O)(=O)c1cccc(N/N=C2/C(=O)Oc3ccccc3C2=O)c1	nan
	CHEMBL1995496	72298	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	7	2.3	CCN(CC)S(=O)(=O)c1cccc(N/N=C2/C(=O)Oc3ccccc3C2=O)c1	nan
	9632269	72561	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2cccnc2)n(C)c1=O	nan
	CHEMBL2004582	72561	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2cccnc2)n(C)c1=O	nan
	9553490	107498	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	9	-0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C/c2ccco2)n(C)c1=O	nan
	CHEMBL3194107	107498	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	9	-0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C/c2ccco2)n(C)c1=O	nan
	6905987	107840	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.5	Sc1nnc(-c2ccccn2)n1/N=C/c1ccc(-c2ccccc2Br)o1	nan
	CHEMBL3198000	107840	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.5	Sc1nnc(-c2ccccn2)n1/N=C/c1ccc(-c2ccccc2Br)o1	nan
	540540	107921	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	7	1.1	CC(=O)/N=c1\sc2nc3ccccc3nc2n1N(C(C)=O)C(C)=O	nan
	CHEMBL3198706	107921	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	7	1.1	CC(=O)/N=c1\sc2nc3ccccc3nc2n1N(C(C)=O)C(C)=O	nan
	5339637	108010	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	7	2	5	1.4	O=C(COc1ccccc1)NCC(=O)N/N=C/c1cccs1	nan
	CHEMBL3199816	108010	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	7	2	5	1.4	O=C(COc1ccccc1)NCC(=O)N/N=C/c1cccs1	nan
	9553411	108402	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	-0.0	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccccc2)n(C)c1=O	nan
	CHEMBL3210887	108402	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	-0.0	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccccc2)n(C)c1=O	nan
	9634938	108412	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccncc2)n(C)c1=O	nan
	CHEMBL3211064	108412	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccncc2)n(C)c1=O	nan
	1116825	183671	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	2.4	Cc1ccnc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	CHEMBL483773	183671	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	2.4	Cc1ccnc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	7190719	199251	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1ccc(CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL601822	199251	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1ccc(CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	3259	23142	46	None	-	1	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	836	0	2	5	6.1	O=C1OC2(c3ccccc31)c1cc(I)c(O)c(I)c1Oc1c2cc(I)c(O)c1I	nan
	CHEMBL1332616	23142	46	None	-	1	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	836	0	2	5	6.1	O=C1OC2(c3ccccc31)c1cc(I)c(O)c(I)c1Oc1c2cc(I)c(O)c1I	nan
	3228920	29510	5	None	-31	2	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	2	5	5.9	O=C(CSc1nc(-c2ccccc2F)nc2nc[nH]c12)Nc1c(Cl)cc(Cl)cc1Cl	nan
	CHEMBL1386739	29510	5	None	-31	2	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	2	5	5.9	O=C(CSc1nc(-c2ccccc2F)nc2nc[nH]c12)Nc1c(Cl)cc(Cl)cc1Cl	nan
	2099	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	4740	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	7095	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	CHEMBL628	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	DB00806	2985	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	3220395	19412	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	6	2.7	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1300380	19412	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	6	2.7	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	16452711	19534	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	8	2.9	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)c1C	nan
	CHEMBL1301248	19534	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	8	2.9	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)c1C	nan
	4134237	19812	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	4	3.0	CC1CCCN(C(=O)CSc2cnc3ccccc3n2)C1	nan
	CHEMBL1303471	19812	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	4	3.0	CC1CCCN(C(=O)CSc2cnc3ccccc3n2)C1	nan
	2816749	20021	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	0	6	1.5	CCOC(=O)N1CCc2c(sc3ncn(C)c(=O)c23)C1	nan
	CHEMBL1305245	20021	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	0	6	1.5	CCOC(=O)N1CCc2c(sc3ncn(C)c(=O)c23)C1	nan
	225068	20124	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	2	6	0.5	CC(=O)Nc1ccc(Cc2nc3c(=O)n(C)c(=O)n(C)c3[nH]2)cc1	nan
	CHEMBL1306052	20124	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	2	6	0.5	CC(=O)Nc1ccc(Cc2nc3c(=O)n(C)c(=O)n(C)c3[nH]2)cc1	nan
	2377168	20462	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	6	1.7	NS(=O)(=O)c1ccc(CCNC(=O)CSc2ncnc3ccccc23)cc1	nan
	CHEMBL1308771	20462	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	6	1.7	NS(=O)(=O)c1ccc(CCNC(=O)CSc2ncnc3ccccc23)cc1	nan
	6311448	20681	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	2	6	2.6	CNc1ccc(/C=C(\C#N)C(=O)Nc2ccccn2)cc1[N+](=O)[O-]	nan
	CHEMBL1310631	20681	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	2	6	2.6	CNc1ccc(/C=C(\C#N)C(=O)Nc2ccccn2)cc1[N+](=O)[O-]	nan
	4454085	20887	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	8	1.1	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1312229	20887	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	8	1.1	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	3269960	20949	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	9	3.7	O=C(O)CCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1312645	20949	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	9	3.7	O=C(O)CCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	5811072	20982	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	7	3.8	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	CHEMBL1312900	20982	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	7	3.8	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	3719872	21063	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	3.8	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)no1	nan
	CHEMBL1313510	21063	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	3.8	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)no1	nan
	7151338	21142	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	2.8	CCS(=O)(=O)Nc1ccc(-c2cn3ccsc3n2)cc1	nan
	CHEMBL1314161	21142	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	2.8	CCS(=O)(=O)Nc1ccc(-c2cn3ccsc3n2)cc1	nan
	16010497	21184	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.0	COc1ccc(CCNC(=O)c2cnc3ccc(C)cn3c2=O)cc1OC	nan
	CHEMBL1314605	21184	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.0	COc1ccc(CCNC(=O)c2cnc3ccc(C)cn3c2=O)cc1OC	nan
	4119285	21266	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	CHEMBL1315733	21266	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	16020283	21304	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	5	4.1	CCOc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)cc1	nan
	CHEMBL1316147	21304	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	5	4.1	CCOc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)cc1	nan
	2645859	21337	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	6	2.6	Cc1cnc(C(=O)OCC(=O)c2ccc(Br)s2)cn1	nan
	CHEMBL1316688	21337	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	6	2.6	Cc1cnc(C(=O)OCC(=O)c2ccc(Br)s2)cn1	nan
	16019079	21411	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.2	CCc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1317634	21411	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.2	CCc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	16025698	21439	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	6.1	CC(NC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1)c1ccccc1	nan
	CHEMBL1317991	21439	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	6.1	CC(NC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1)c1ccccc1	nan
	16018836	21496	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	1	6	4.6	O=C(CSc1nncn2c1cc1sccc12)Nc1ccc(Br)cc1F	nan
	CHEMBL1318579	21496	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	1	6	4.6	O=C(CSc1nncn2c1cc1sccc12)Nc1ccc(Br)cc1F	nan
	658390	21919	21	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	2.7	CSc1sc(C(=O)O)c2c1C(=O)CCC2	nan
	CHEMBL132222	21919	21	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	2.7	CSc1sc(C(=O)O)c2c1C(=O)CCC2	nan
	4302597	22153	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	6	3.1	Cc1c(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)nn1C	nan
	CHEMBL1324305	22153	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	6	3.1	Cc1c(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)nn1C	nan
	16825458	22408	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1OC	nan
	CHEMBL1326698	22408	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1OC	nan
	961104	22713	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	5	2	5	1.8	CCOC(=O)c1[nH]cnc1C(=O)Nc1ccccc1OC	nan
	CHEMBL1329229	22713	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	5	2	5	1.8	CCOC(=O)c1[nH]cnc1C(=O)Nc1ccccc1OC	nan
	753118	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1331202	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1532594	22962	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	5302178	23434	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	CHEMBL1334923	23434	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	4213677	23535	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	2	9	2.3	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc5c(c4)OCO5)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1335629	23535	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	2	9	2.3	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc5c(c4)OCO5)c(=N)n(CC4CCCO4)c3nc12	nan
	2410320	23770	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	6	2.5	Cc1ccc(S(=O)(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	CHEMBL1337652	23770	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	6	2.5	Cc1ccc(S(=O)(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	6624813	24088	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	7	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCCCC3)nnc12	nan
	CHEMBL1340556	24088	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	7	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCCCC3)nnc12	nan
	16189291	24240	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	0	8	2.6	CCOC(=O)C(CC)Sc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1341871	24240	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	0	8	2.6	CCOC(=O)C(CC)Sc1ccc2nnc(-c3cccnc3)n2n1	nan
	2835302	24426	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	1	2	4	3.4	CCC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	CHEMBL1343308	24426	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	1	2	4	3.4	CCC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	9115295	24460	23	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	4	4.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1C(F)(F)F	nan
	CHEMBL1343609	24460	23	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	4	4.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1C(F)(F)F	nan
	874496	24520	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	4	2	2	4.0	CC(C)C(=O)Nc1ccc(Nc2ccccc2)cc1	nan
	CHEMBL1344171	24520	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	4	2	2	4.0	CC(C)C(=O)Nc1ccc(Nc2ccccc2)cc1	nan
	5040775	24540	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	5	1.5	CC1CCCCC1NC(=O)Cn1nnc2ccccc2c1=O	nan
	CHEMBL1344340	24540	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	5	1.5	CC1CCCCC1NC(=O)Cn1nnc2ccccc2c1=O	nan
	7190697	24609	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	9	1.0	CCOC(=O)CNC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1344913	24609	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	9	1.0	CCOC(=O)CNC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	1279973	24654	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	10	0.8	COCc1cc(C)nc(Sc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1C#N	nan
	CHEMBL1345308	24654	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	10	0.8	COCc1cc(C)nc(Sc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1C#N	nan
	16187878	24734	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	8	3.6	CCOC(=O)CC(NC(=O)CCc1c(C)nc2nc(C)nn2c1C)c1ccc(OC(C)C)cc1	nan
	CHEMBL1346041	24734	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	8	3.6	CCOC(=O)CC(NC(=O)CCc1c(C)nc2nc(C)nn2c1C)c1ccc(OC(C)C)cc1	nan
	4911180	24736	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	8	4.3	C=CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1346060	24736	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	8	4.3	C=CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	6626039	24818	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	7	1	8	2.2	CCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	CHEMBL1346717	24818	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	7	1	8	2.2	CCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	4884017	24841	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	0	6	2.9	CCN1c2ccc(S(=O)(=O)N3CCOCC3)cc2N(Cc2ccc(OC)cc2)C1C	nan
	CHEMBL1346905	24841	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	0	6	2.9	CCN1c2ccc(S(=O)(=O)N3CCOCC3)cc2N(Cc2ccc(OC)cc2)C1C	nan
	5916900	25135	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1349404	25135	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2421577	25228	5	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	0	5	3.2	COC(=O)CCc1c(C)c(C(=O)c2ccco2)c2ccccn12	nan
	CHEMBL1350197	25228	5	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	0	5	3.2	COC(=O)CCc1c(C)c(C(=O)c2ccco2)c2ccccn12	nan
	2429966	25284	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	0	7	2.8	COc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1OC	nan
	CHEMBL1350669	25284	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	0	7	2.8	COc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1OC	nan
	5921143	25473	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	10	1.5	CCCN1C(=O)/C(=C/c2c(N3CCNC(=O)C3CC(=O)OC)nc3c(C)cccn3c2=O)SC1=S	nan
	CHEMBL1352285	25473	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	10	1.5	CCCN1C(=O)/C(=C/c2c(N3CCNC(=O)C3CC(=O)OC)nc3c(C)cccn3c2=O)SC1=S	nan
	2926991	25504	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	4.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)n1	nan
	CHEMBL1352465	25504	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	4.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)n1	nan
	16015204	25768	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	4.5	COC(=O)c1c(-c2cccs2)csc1NC(=O)c1ccc(OC)c(OC)c1	nan
	CHEMBL1354415	25768	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	4.5	COC(=O)c1c(-c2cccs2)csc1NC(=O)c1ccc(OC)c(OC)c1	nan
	16030461	25820	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	4	4.2	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1355113	25820	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	4	4.2	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	23602530	25902	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	5	2.2	Cc1ccc(Cn2c(CCC(=O)O)nc3ncccc3c2=O)cc1	nan
	CHEMBL1356159	25902	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	5	2.2	Cc1ccc(Cn2c(CCC(=O)O)nc3ncccc3c2=O)cc1	nan
	16018072	25955	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	7	1	4	3.8	Cc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1356862	25955	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	7	1	4	3.8	Cc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	1077055	25997	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	8	0.3	CC(=O)c1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1357427	25997	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	8	0.3	CC(=O)c1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	16021425	26010	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)c1	nan
	CHEMBL1357639	26010	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)c1	nan
	16030521	26024	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)c1	nan
	CHEMBL1357883	26024	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)c1	nan
	16030369	26049	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	4.9	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(C)cc2)c1	nan
	CHEMBL1358199	26049	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	4.9	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(C)cc2)c1	nan
	15987639	26075	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	4	5.5	Cc1ccc(NC(=O)CSc2nc3ccccc3nc2Cc2ccccc2F)cc1F	nan
	CHEMBL1358546	26075	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	4	5.5	Cc1ccc(NC(=O)CSc2nc3ccccc3nc2Cc2ccccc2F)cc1F	nan
	881482	26603	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	3	3.7	O=S(=O)(Nc1ccccn1)c1ccc(Cl)c2ccccc12	nan
	CHEMBL1363117	26603	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	3	3.7	O=S(=O)(Nc1ccccn1)c1ccc(Cl)c2ccccc12	nan
	3193431	26650	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	7	0	8	4.3	COc1ccc(Cn2nnnc2C(c2ccc3ncccc3c2)N2CCN(C3CCCCC3)CC2)cc1	nan
	CHEMBL1363552	26650	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	7	0	8	4.3	COc1ccc(Cn2nnnc2C(c2ccc3ncccc3c2)N2CCN(C3CCCCC3)CC2)cc1	nan
	1261960	26654	9	None	-7	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	5	3.5	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)cc1	nan
	CHEMBL1363571	26654	9	None	-7	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	5	3.5	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)cc1	nan
	7190718	26766	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1cccc(CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1364582	26766	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1cccc(CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	20884309	26773	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	8	1.1	CCc1nn(CC(=O)NCCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	CHEMBL1364643	26773	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	8	1.1	CCc1nn(CC(=O)NCCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	4152428	26808	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1364957	26808	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	5109926	26841	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	2	8	2.6	COc1ccc(CCn2c(=N)c(C(=O)NCC3CCCO3)cc3c(=O)n4cccc(C)c4nc32)cc1	nan
	CHEMBL1365247	26841	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	2	8	2.6	COc1ccc(CCn2c(=N)c(C(=O)NCC3CCCO3)cc3c(=O)n4cccc(C)c4nc32)cc1	nan
	2959558	26844	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	3.3	CCOC(=O)N1CCN(C(=O)COc2ccc3ccccc3c2Br)CC1	nan
	CHEMBL1365264	26844	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	3.3	CCOC(=O)N1CCN(C(=O)COc2ccc3ccccc3c2Br)CC1	nan
	15988059	26900	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	1	10	2.6	COC(=O)c1cccc(Nc2nn3c(=O)c4cc5c(cc4nc3s2)OCO5)c1	nan
	CHEMBL1365674	26900	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	1	10	2.6	COC(=O)c1cccc(Nc2nn3c(=O)c4cc5c(cc4nc3s2)OCO5)c1	nan
	16015914	26906	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	2	0	4	6.1	Cc1c(C(=O)N2CCC(c3nc4ccccc4s3)CC2)oc2cc(Br)ccc12	nan
	CHEMBL1365703	26906	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	2	0	4	6.1	Cc1c(C(=O)N2CCC(c3nc4ccccc4s3)CC2)oc2cc(Br)ccc12	nan
	912209	26919	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	3	5	1.9	NC(S)=Nc1cccc(-c2nnc(S)o2)c1	nan
	CHEMBL1365893	26919	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	3	5	1.9	NC(S)=Nc1cccc(-c2nnc(S)o2)c1	nan
	3719648	27494	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	4.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc3ccccc23)s1	nan
	CHEMBL1370349	27494	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	4.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc3ccccc23)s1	nan
	1775727	27772	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	0	5	4.3	COc1ccccc1CN1COc2ccc3c(oc(=O)c4ccccc43)c2C1	nan
	CHEMBL1372393	27772	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	0	5	4.3	COc1ccccc1CN1COc2ccc3c(oc(=O)c4ccccc43)c2C1	nan
	16193912	28211	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	6	4.8	CCCCN(CC)CCCNC(=O)C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1	nan
	CHEMBL1375345	28211	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	6	4.8	CCCCN(CC)CCCNC(=O)C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1	nan
	2818996	28357	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.9	COc1ccc(-c2c(C#N)c(N)nc(Sc3ccc(Cl)cc3)c2C#N)cc1	nan
	CHEMBL1376612	28357	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.9	COc1ccc(-c2c(C#N)c(N)nc(Sc3ccc(Cl)cc3)c2C#N)cc1	nan
	20876288	28964	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	5	3.5	Cc1ccc(CN2CCSc3ccc(C(=O)NCCCN4CCN(C)CC4)cc32)cc1	nan
	CHEMBL1382060	28964	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	5	3.5	Cc1ccc(CN2CCSc3ccc(C(=O)NCCCN4CCN(C)CC4)cc32)cc1	nan
	4902824	29036	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1382669	29036	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	408543	29389	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	3	1	3	2.4	O=C(O)CSc1ccc2ccccc2n1	nan
	CHEMBL1385852	29389	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	3	1	3	2.4	O=C(O)CSc1ccc2ccccc2n1	nan
	16452903	29414	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1ccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)cc1	nan
	CHEMBL1386060	29414	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1ccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)cc1	nan
	5866058	29439	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)c1	nan
	CHEMBL1386260	29439	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)c1	nan
	2219052	29915	10	None	-3	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	6	4.2	CCCCn1nnc(NC(=O)c2sc3cc(Cl)ccc3c2Cl)n1	nan
	CHEMBL1389959	29915	10	None	-3	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	6	4.2	CCCCn1nnc(NC(=O)c2sc3cc(Cl)ccc3c2Cl)n1	nan
	974402	30043	14	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	2	2	3.4	CC(C)NC(=S)NC(=O)c1ccc(-c2ccccc2)cc1	nan
	CHEMBL1391097	30043	14	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	2	2	3.4	CC(C)NC(=S)NC(=O)c1ccc(-c2ccccc2)cc1	nan
	4385170	30187	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	4	4.9	CCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1392345	30187	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	4	4.9	CCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	2492440	30220	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	3.4	Cc1ccccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1392606	30220	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	3.4	Cc1ccccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	7207181	30267	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.9	O=C(CSc1ccc(-c2ccco2)nn1)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1393087	30267	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.9	O=C(CSc1ccc(-c2ccco2)nn1)NCc1ccc2c(c1)OCO2	nan
	16025764	30478	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	0	3	4.6	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCCCC2)s1	nan
	CHEMBL1395096	30478	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	0	3	4.6	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCCCC2)s1	nan
	5839687	30621	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	1.7	COCCNC(=O)/C(C#N)=C/c1c(N2CCCCCC2)nc2ccccn2c1=O	nan
	CHEMBL1397071	30621	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	1.7	COCCNC(=O)/C(C#N)=C/c1c(N2CCCCCC2)nc2ccccn2c1=O	nan
	5789902	30683	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	5	4.0	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1397920	30683	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	5	4.0	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	3288231	30704	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	4	5.7	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	CHEMBL1398189	30704	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	4	5.7	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	15991174	30734	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	3	3	7	1.6	Cc1cc(Nc2ccc(C(=O)O)c(O)c2)n2ncnc2n1	nan
	CHEMBL1398548	30734	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	3	3	7	1.6	Cc1cc(Nc2ccc(C(=O)O)c(O)c2)n2ncnc2n1	nan
	16025760	30866	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1399794	30866	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	135444909	30927	10	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	8	3	10	3.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)cc2)n1	nan
	CHEMBL1400344	30927	10	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	8	3	10	3.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)cc2)n1	nan
	16023027	30954	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1400601	30954	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	2005962	30960	8	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	7	3.5	CC(C)OCCCN1CN(S(=O)(=O)c2cccs2)c2nc3ccccc3nc21	nan
	CHEMBL1400661	30960	8	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	7	3.5	CC(C)OCCCN1CN(S(=O)(=O)c2cccs2)c2nc3ccccc3nc21	nan
	4176332	30997	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	3	1	5	3.6	CN1CCN(NC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)CC1	nan
	CHEMBL1401042	30997	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	3	1	5	3.6	CN1CCN(NC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)CC1	nan
	7693269	31037	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	1	1	4.1	O=C(c1cc2cc(Br)ccc2[nH]1)N1CCc2ccccc21	nan
	CHEMBL1401345	31037	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	1	1	4.1	O=C(c1cc2cc(Br)ccc2[nH]1)N1CCc2ccccc21	nan
	1842681	32385	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	0	8	1.2	CCOC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1412841	32385	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	0	8	1.2	CCOC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	3159273	32570	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	5	3.0	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCCN(C)C)CC2	nan
	CHEMBL1414335	32570	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	5	3.0	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCCN(C)C)CC2	nan
	773430	32686	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	O=C(O)c1ccc2nc3c(nc2c1)-c1ccccc1C3=O	nan
	CHEMBL1415344	32686	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	O=C(O)c1ccc2nc3c(nc2c1)-c1ccccc1C3=O	nan
	1172271	32983	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	0	9	0.1	CCCn1c(SCC(=O)N2CCN(CC)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1417950	32983	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	0	9	0.1	CCCn1c(SCC(=O)N2CCN(CC)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	20957513	33152	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	12	2	8	2.6	CSc1ccc(CCNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1419386	33152	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	12	2	8	2.6	CSc1ccc(CCNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	656126	34100	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	4.1	CCOC(=O)c1c(NC(=O)CSc2nc(C)cc(C)c2C#N)sc(C(C)=O)c1C	nan
	CHEMBL1427319	34100	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	4.1	CCOC(=O)c1c(NC(=O)CSc2nc(C)cc(C)c2C#N)sc(C(C)=O)c1C	nan
	24792443	34176	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	5	3.1	CCc1nc(SCC(=O)NNC(=O)c2ccc(C)cc2)c2ccccc2n1	nan
	CHEMBL1428040	34176	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	5	3.1	CCc1nc(SCC(=O)NNC(=O)c2ccc(C)cc2)c2ccccc2n1	nan
	5295519	34874	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	10	0.1	COC(=O)c1cc(OC)c(OC)c(OC)c1NC(=O)c1cc(=O)n(C)c(=O)n1C	nan
	CHEMBL1434105	34874	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	10	0.1	COC(=O)c1cc(OC)c(OC)c(OC)c1NC(=O)c1cc(=O)n(C)c(=O)n1C	nan
	16959503	34958	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	9	2.5	CC(C)Oc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	CHEMBL1435220	34958	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	9	2.5	CC(C)Oc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	2448286	34981	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	11	1.6	Cn1c(N)c(C(=O)CSc2nn(-c3ccccc3)c(=S)s2)c(=O)n(C)c1=O	nan
	CHEMBL1435449	34981	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	11	1.6	Cn1c(N)c(C(=O)CSc2nn(-c3ccccc3)c(=S)s2)c(=O)n(C)c1=O	nan
	16018790	35105	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.6	CCc1nnc(SCC(=O)Nc2ccc(Cl)cc2F)c2cc3occc3n12	nan
	CHEMBL1437127	35105	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.6	CCc1nnc(SCC(=O)Nc2ccc(Cl)cc2F)c2cc3occc3n12	nan
	135401612	35366	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	3	7	1.5	Nc1cc(O)nc(SCC(=O)Nc2cccnc2Cl)n1	nan
	CHEMBL1439558	35366	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	3	7	1.5	Nc1cc(O)nc(SCC(=O)Nc2cccnc2Cl)n1	nan
	15990899	35476	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	9	1	10	5.2	COc1cc2nc(SCC(=O)Nc3cccc(C)c3)n3nc(CCn4c(C)nc5ccccc54)nc3c2cc1OC	nan
	CHEMBL1440596	35476	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	9	1	10	5.2	COc1cc2nc(SCC(=O)Nc3cccc(C)c3)n3nc(CCn4c(C)nc5ccccc54)nc3c2cc1OC	nan
	16034663	35501	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3)nnc12	nan
	CHEMBL1440811	35501	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3)nnc12	nan
	5898351	35671	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	6	4.2	Cc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	CHEMBL1442346	35671	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	6	4.2	Cc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	986518	35730	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	4	3.3	Cc1c(C(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2ccc(Cl)cc12	nan
	CHEMBL1442810	35730	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	4	3.3	Cc1c(C(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2ccc(Cl)cc12	nan
	16009462	35739	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.6	CC(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1442959	35739	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.6	CC(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	7245567	35763	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1ccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1443187	35763	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1ccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4920871	36151	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	7	1.9	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NCC1CCCO1	nan
	CHEMBL1446831	36151	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	7	1.9	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NCC1CCCO1	nan
	139030	36174	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	196	0	1	2	2.9	O=C1C=C(O)c2cccc3cccc1c23	nan
	CHEMBL1446983	36174	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	196	0	1	2	2.9	O=C1C=C(O)c2cccc3cccc1c23	nan
	771978	36185	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	6	1.2	O=C(Nc1ncccn1)c1ccc([N+](=O)[O-])o1	nan
	CHEMBL1447058	36185	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	6	1.2	O=C(Nc1ncccn1)c1ccc([N+](=O)[O-])o1	nan
	1511203	36263	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	2	7	2.6	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NC(C)(C)CO	nan
	CHEMBL1447724	36263	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	2	7	2.6	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NC(C)(C)CO	nan
	5310565	36662	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	8	1.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)N1CCOCC1	nan
	CHEMBL1450965	36662	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	8	1.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)N1CCOCC1	nan
	16457956	36779	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	4	8	1.1	CCN(CC)S(=O)(=O)c1cccc(C(=O)NNC(=O)c2ccc3nc(O)c(O)nc3c2)c1	nan
	CHEMBL1451892	36779	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	4	8	1.1	CCN(CC)S(=O)(=O)c1cccc(C(=O)NNC(=O)c2ccc3nc(O)c(O)nc3c2)c1	nan
	2173828	37369	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	3	5.6	CCN(CC)c1nc(-c2ccccc2Cl)c2cc(Br)ccc2n1	nan
	CHEMBL1456908	37369	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	3	5.6	CCN(CC)c1nc(-c2ccccc2Cl)c2cc(Br)ccc2n1	nan
	20904573	37676	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	1	8	2.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCN(Cc4ccccc4)CC3)nnc12	nan
	CHEMBL1459467	37676	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	1	8	2.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCN(Cc4ccccc4)CC3)nnc12	nan
	734076	37705	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	4	1	4	2.4	CCCC(=O)Nc1nc(C)c(C(C)=O)s1	nan
	CHEMBL1459745	37705	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	4	1	4	2.4	CCCC(=O)Nc1nc(C)c(C(C)=O)s1	nan
	1511643	37706	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	8	1.3	Cc1cc([N+](=O)[O-])nn1CC(=O)Nc1cccc2nonc12	nan
	CHEMBL1459750	37706	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	8	1.3	Cc1cc([N+](=O)[O-])nn1CC(=O)Nc1cccc2nonc12	nan
	1838806	37836	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	7	3.6	CCOc1cccc(Nc2cc3n(c(=O)n2)CCc2cc(OC)c(OC)cc2-3)c1	nan
	CHEMBL1460751	37836	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	7	3.6	CCOc1cccc(Nc2cc3n(c(=O)n2)CCc2cc(OC)c(OC)cc2-3)c1	nan
	16188836	38059	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	0	4	4.0	CC1=NOC(=O)/C1=C\c1ccc(-c2ccccc2Br)o1	nan
	CHEMBL1462764	38059	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	0	4	4.0	CC1=NOC(=O)/C1=C\c1ccc(-c2ccccc2Br)o1	nan
	3332154	38398	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	8	3.2	Cc1nc(N)sc1N=Nc1c(C)n(C)n(-c2ccccc2)c1=O	nan
	CHEMBL1465412	38398	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	8	3.2	Cc1nc(N)sc1N=Nc1c(C)n(C)n(-c2ccccc2)c1=O	nan
	20957223	38505	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	8	2.0	Cc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1466244	38505	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	8	2.0	Cc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	2350819	38511	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.3	Cc1cc(Br)ccc1SCC(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	CHEMBL1466307	38511	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.3	Cc1cc(Br)ccc1SCC(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	7190691	38851	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	8	3.1	CC(=O)c1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1469069	38851	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	8	3.1	CC(=O)c1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	1179824	39031	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	2	7	3.6	CCOC(=O)c1sc2ncnc(Nc3cccc(C(=O)O)c3)c2c1C	nan
	CHEMBL1470707	39031	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	2	7	3.6	CCOC(=O)c1sc2ncnc(Nc3cccc(C(=O)O)c3)c2c1C	nan
	7207497	39046	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	5	4.2	Cc1c(Cl)cccc1NC(=O)CSc1ccc(-c2cccnc2)nn1	nan
	CHEMBL1470773	39046	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	5	4.2	Cc1c(Cl)cccc1NC(=O)CSc1ccc(-c2cccnc2)nn1	nan
	16012892	39260	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	7	2.9	CCNC(=O)c1c(NC(=O)c2nc(S(=O)(=O)CC)ncc2Cl)sc2c1CCCC2	nan
	CHEMBL1472696	39260	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	7	2.9	CCNC(=O)c1c(NC(=O)c2nc(S(=O)(=O)CC)ncc2Cl)sc2c1CCCC2	nan
	16030433	39402	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	1	6	5.0	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)c1OC	nan
	CHEMBL1474670	39402	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	1	6	5.0	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)c1OC	nan
	4547893	39576	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	6	3.3	COc1ccccc1C(=O)Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1	nan
	CHEMBL1477066	39576	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	6	3.3	COc1ccccc1C(=O)Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1	nan
	1313916	39841	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1479446	39841	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	16021977	40208	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	6	4.5	CCOC(=O)c1ccc(NC(=O)c2c(C)nn(-c3ccc(F)cc3)c2-n2cccc2)cc1	nan
	CHEMBL1482573	40208	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	6	4.5	CCOC(=O)c1ccc(NC(=O)c2c(C)nn(-c3ccc(F)cc3)c2-n2cccc2)cc1	nan
	16025700	40427	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1cccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	CHEMBL1484349	40427	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1cccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	4969640	40458	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	1.5	COc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)CSc1nncs1	nan
	CHEMBL1484709	40458	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	1.5	COc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)CSc1nncs1	nan
	2267309	40963	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.8	Cc1cc(N)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	CHEMBL1488814	40963	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.8	Cc1cc(N)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	3157588	41233	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	3.7	CC(=O)C1=C(O)C(=O)N(CCc2c[nH]c3ccccc23)C1c1ccccc1	nan
	CHEMBL1490855	41233	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	3.7	CC(=O)C1=C(O)C(=O)N(CCc2c[nH]c3ccccc23)C1c1ccccc1	nan
	3755909	41814	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2ccc(Br)s2)nc(-n2cccc2)n1	nan
	CHEMBL1495948	41814	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2ccc(Br)s2)nc(-n2cccc2)n1	nan
	6501461	42433	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	9	2.7	CCC(Sc1nnc(-c2ccco2)n1C)C(=O)Nc1nnc(C)s1	nan
	CHEMBL1501425	42433	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	9	2.7	CCC(Sc1nnc(-c2ccco2)n1C)C(=O)Nc1nnc(C)s1	nan
	20968950	42483	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	0.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCC(C(N)=O)CC1)C(=O)CO2	nan
	CHEMBL1501847	42483	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	0.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCC(C(N)=O)CC1)C(=O)CO2	nan
	7692847	42623	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	6	3.1	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc2c(c1)OCO2	nan
	CHEMBL1503072	42623	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	6	3.1	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc2c(c1)OCO2	nan
	1243282	42741	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	2	1	5	4.6	Fc1ccc(-n2c(S)nnc2-c2ccc3ccccc3n2)cc1Cl	nan
	CHEMBL1504174	42741	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	2	1	5	4.6	Fc1ccc(-n2c(S)nnc2-c2ccc3ccccc3n2)cc1Cl	nan
	20888797	42962	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	9	1.5	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1506053	42962	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	9	1.5	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCN(CCO)CC2)s1	nan
	3965652	42984	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	5	3.6	Oc1nc(S)ncc1Oc1ccc(Cl)cc1Cl	nan
	CHEMBL1506226	42984	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	5	3.6	Oc1nc(S)ncc1Oc1ccc(Cl)cc1Cl	nan
	664243	43223	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.7	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)no1	nan
	CHEMBL1508235	43223	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.7	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)no1	nan
	1564171	43304	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	8	3.9	C=CCn1c(SCC(=O)Nc2sccc2C#N)nc2sc(C)c(C)c2c1=O	nan
	CHEMBL1509018	43304	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	8	3.9	C=CCn1c(SCC(=O)Nc2sccc2C#N)nc2sc(C)c(C)c2c1=O	nan
	660816	43468	49	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	5	3.2	COc1ccccc1-c1nnc(S)n1-c1ccccc1	nan
	CHEMBL1510509	43468	49	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	5	3.2	COc1ccccc1-c1nnc(S)n1-c1ccccc1	nan
	4736989	43626	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	7	1.4	O=C(O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1511802	43626	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	7	1.4	O=C(O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	16407031	43642	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	9	1	9	3.2	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCCN4CCOCC4)cc3c3ccnc2c31	nan
	CHEMBL1512174	43642	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	9	1	9	3.2	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCCN4CCOCC4)cc3c3ccnc2c31	nan
	16021393	43649	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	4	6.6	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(C(F)(F)F)c4)cc(C)c3c2)c1	nan
	CHEMBL1512269	43649	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	4	6.6	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(C(F)(F)F)c4)cc(C)c3c2)c1	nan
	16018932	43794	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	0	7	6.7	CCc1nnc(SCc2nc(-c3cccc(Cl)c3)oc2C)c2cc3sc(C)cc3n12	nan
	CHEMBL1514500	43794	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	0	7	6.7	CCc1nnc(SCc2nc(-c3cccc(Cl)c3)oc2C)c2cc3sc(C)cc3n12	nan
	20885685	43861	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccccc1CNC(=O)CCCn1nc(C)n2ccnc2c1=O	nan
	CHEMBL1515364	43861	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccccc1CNC(=O)CCCn1nc(C)n2ccnc2c1=O	nan
	16018754	43887	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	8	3.8	COc1cc(NC(=O)CSc2nnc(C)n3c2cc2oc(C)cc23)cc(OC)c1	nan
	CHEMBL1515810	43887	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	8	3.8	COc1cc(NC(=O)CSc2nnc(C)n3c2cc2oc(C)cc23)cc(OC)c1	nan
	4350514	44941	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	1.9	Cc1nc2ccccc2c(=O)n1NC(=O)Cc1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1525803	44941	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	1.9	Cc1nc2ccccc2c(=O)n1NC(=O)Cc1ccc([N+](=O)[O-])cc1	nan
	135455188	45250	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	9	3.3	N#Cc1c(O)nc(SCC(=O)Nc2nnc(C(F)(F)F)s2)nc1-c1ccccc1	nan
	CHEMBL1528492	45250	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	9	3.3	N#Cc1c(O)nc(SCC(=O)Nc2nnc(C(F)(F)F)s2)nc1-c1ccccc1	nan
	3535143	45414	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	9	3.6	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4ccccc4n3)nc3ccsc3c2=O)CC1	nan
	CHEMBL1529863	45414	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	9	3.6	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4ccccc4n3)nc3ccsc3c2=O)CC1	nan
	16030435	45437	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	4	5.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccccc2Cl)cc1	nan
	CHEMBL1530187	45437	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	4	5.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccccc2Cl)cc1	nan
	54677747	45701	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	1	2	7	4.6	O=c1oc2ccccc2c(O)c1[C@H]1c2ccc(O)cc2Oc2c1c(=O)oc1ccccc21	nan
	CHEMBL1532491	45701	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	1	2	7	4.6	O=c1oc2ccccc2c(O)c1[C@H]1c2ccc(O)cc2Oc2c1c(=O)oc1ccccc21	nan
	6498569	45735	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	7	2	5	1.0	Cc1ccc(OCC(=O)NCCNC(=O)c2cnccn2)cc1C	nan
	CHEMBL1532759	45735	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	7	2	5	1.0	Cc1ccc(OCC(=O)NCCNC(=O)c2cnccn2)cc1C	nan
	6060971	45739	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	8	1	6	3.4	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(CCN3CCOCC3)C2c2ccccc2)cc1	nan
	CHEMBL1532782	45739	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	8	1	6	3.4	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(CCN3CCOCC3)C2c2ccccc2)cc1	nan
	3262927	46058	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	1.3	O=C(OCN1C(=O)c2ccccc2C1=O)c1cc(S(=O)(=O)N2CCOCC2)ccc1F	nan
	CHEMBL1535967	46058	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	1.3	O=C(OCN1C(=O)c2ccccc2C1=O)c1cc(S(=O)(=O)N2CCOCC2)ccc1F	nan
	6018171	46060	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	6	3.9	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1	nan
	CHEMBL1535987	46060	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	6	3.9	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1	nan
	7120055	46121	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	4.4	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1C	nan
	CHEMBL1536665	46121	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	4.4	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1C	nan
	2086676	46190	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	8	1.3	Cn1c(=O)c(C(=O)COc2ccc(C#N)cc2)c(N)n(Cc2ccccc2)c1=O	nan
	CHEMBL1537193	46190	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	8	1.3	Cn1c(=O)c(C(=O)COc2ccc(C#N)cc2)c(N)n(Cc2ccccc2)c1=O	nan
	20888841	46222	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	0	8	2.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CC)CC2)s1	nan
	CHEMBL1537517	46222	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	0	8	2.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CC)CC2)s1	nan
	22334156	46441	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	6	1	9	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1539318	46441	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	6	1	9	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1OC	nan
	3151316	46444	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1539382	46444	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CC4CCCO4)c3nc12	nan
	17581317	46662	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	1	5	3.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc(Br)o1	nan
	CHEMBL1541200	46662	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	1	5	3.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc(Br)o1	nan
	6228228	46775	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	7	4.0	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2)s1	nan
	CHEMBL1542130	46775	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	7	4.0	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2)s1	nan
	2359872	46804	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	4	2.8	O=C(CSc1cnc2ccccc2n1)NC1CCCC1	nan
	CHEMBL1542457	46804	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	4	2.8	O=C(CSc1cnc2ccccc2n1)NC1CCCC1	nan
	2346972	46823	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	10	-1.0	CN(C)S(=O)(=O)c1cccc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1542615	46823	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	10	-1.0	CN(C)S(=O)(=O)c1cccc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	135420430	46828	11	None	-4	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	8	3.5	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1cc(C)on1	nan
	CHEMBL1542646	46828	11	None	-4	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	8	3.5	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1cc(C)on1	nan
	1866349	47164	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	661670	47164	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1406059	47164	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1545185	47164	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	4876432	47189	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	2	6	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	CHEMBL1545378	47189	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	2	6	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	2595072	47190	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	6	1	4	3.1	O=C(CSc1ncnc2ccccc12)NCCc1ccccc1	nan
	CHEMBL1545386	47190	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	6	1	4	3.1	O=C(CSc1ncnc2ccccc12)NCCc1ccccc1	nan
	2115012	47257	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	10	0.2	CCCn1c(N)c(C(=O)COC(=O)c2c(C)noc2C)c(=O)n(C)c1=O	nan
	CHEMBL1545973	47257	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	10	0.2	CCCn1c(N)c(C(=O)COC(=O)c2c(C)noc2C)c(=O)n(C)c1=O	nan
	241512	47560	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	1	2	2	3.2	c1ccc(-c2ccc3c(c2)NCCN3)cc1	nan
	CHEMBL1548782	47560	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	1	2	2	3.2	c1ccc(-c2ccc3c(c2)NCCN3)cc1	nan
	16189384	47779	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	573	10	2	9	1.4	CSCCC(NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C)C(=O)NC1CCN(Cc2ccccc2)CC1	nan
	CHEMBL1550614	47779	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	573	10	2	9	1.4	CSCCC(NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C)C(=O)NC1CCN(Cc2ccccc2)CC1	nan
	16019521	47851	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	9	2.5	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCN(C)CC2)c2sccc23)c1	nan
	CHEMBL1551283	47851	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	9	2.5	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCN(C)CC2)c2sccc23)c1	nan
	6414933	47883	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	4.2	CCOC(=O)c1ccc(NC(=O)C(CC)Sc2nnc3c4ccccc4n(C)c3n2)cc1	nan
	CHEMBL1551836	47883	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	4.2	CCOC(=O)c1ccc(NC(=O)C(CC)Sc2nnc3c4ccccc4n(C)c3n2)cc1	nan
	16018808	47895	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	8	1	7	2.7	CCc1nnc(SC(CC)C(=O)NCCOC)c2cc3occc3n12	nan
	CHEMBL1551969	47895	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	8	1	7	2.7	CCc1nnc(SC(CC)C(=O)NCCOC)c2cc3occc3n12	nan
	5301786	47919	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	1	8	1.0	Cc1ccc(-c2c(C)n3c4c(=O)n(C)c(=O)n(C)c4nc3n2CCO)cc1	nan
	CHEMBL1552221	47919	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	1	8	1.0	Cc1ccc(-c2c(C)n3c4c(=O)n(C)c(=O)n(C)c4nc3n2CCO)cc1	nan
	1622536	47982	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	4.7	CCCCOC(=O)c1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2N)cc1	nan
	CHEMBL1553105	47982	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	4.7	CCCCOC(=O)c1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2N)cc1	nan
	16020969	48018	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	5.0	Cc1oc(-c2cccc(Br)c2)nc1CSc1nc2cccnc2[nH]1	nan
	CHEMBL1553552	48018	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	5.0	Cc1oc(-c2cccc(Br)c2)nc1CSc1nc2cccnc2[nH]1	nan
	4291583	48053	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	14	4	8	2.2	CSCCC(NS(=O)(=O)c1ccc2c(c1)Cc1cc(S(=O)(=O)NC(CCSC)C(=O)O)ccc1-2)C(=O)O	nan
	CHEMBL1554139	48053	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	14	4	8	2.2	CSCCC(NS(=O)(=O)c1ccc2c(c1)Cc1cc(S(=O)(=O)NC(CCSC)C(=O)O)ccc1-2)C(=O)O	nan
	20877874	48092	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	0	4	3.5	CCCN1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1554696	48092	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	0	4	3.5	CCCN1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	16011310	48159	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	5	5.5	CCc1nnc(SCc2cccc(Cl)c2)c2cc3sccc3n12	nan
	CHEMBL1555647	48159	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	5	5.5	CCc1nnc(SCc2cccc(Cl)c2)c2cc3sccc3n12	nan
	16030467	48686	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	4	5.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)NCc1ccccc1Cl	nan
	CHEMBL1560326	48686	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	4	5.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)NCc1ccccc1Cl	nan
	2415608	48738	22	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	2	7	2.8	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3cc4c(cc3nc2Cl)OCCO4)cc1	nan
	CHEMBL1560923	48738	22	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	2	7	2.8	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3cc4c(cc3nc2Cl)OCCO4)cc1	nan
	15988392	48964	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.8	CCn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	CHEMBL1562908	48964	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.8	CCn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	3805026	49077	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Cl)cc2)no1	nan
	CHEMBL1563863	49077	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Cl)cc2)no1	nan
	6228410	49140	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	7	4.1	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2F)s1	nan
	CHEMBL1564525	49140	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	7	4.1	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2F)s1	nan
	4802105	49308	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	2.8	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCCC2)ccc1Cl	nan
	CHEMBL1565823	49308	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	2.8	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCCC2)ccc1Cl	nan
	225436	49551	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	198	0	1	3	1.2	O=C1c2ccccc2C(=O)c2[nH]cnc21	nan
	CHEMBL1567800	49551	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	198	0	1	3	1.2	O=C1c2ccccc2C(=O)c2[nH]cnc21	nan
	2054020	49661	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	7	4.7	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nc2ccccc2s1	nan
	CHEMBL1568611	49661	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	7	4.7	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nc2ccccc2s1	nan
	2883018	49824	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	0	1	5	1.6	N#Cc1c2n(c3c(N)ncnc13)CCCCC2	nan
	CHEMBL1570092	49824	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	0	1	5	1.6	N#Cc1c2n(c3c(N)ncnc13)CCCCC2	nan
	16018256	49958	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	CCOc1ccc(CCNC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)cc1OCC	nan
	CHEMBL1571269	49958	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	CCOc1ccc(CCNC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)cc1OCC	nan
	25163648	50091	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	4	4.3	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)N(C)Cc1c(F)cccc1Cl	nan
	CHEMBL1572593	50091	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	4	4.3	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)N(C)Cc1c(F)cccc1Cl	nan
	20957176	50169	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	0	9	0.2	CN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	CHEMBL1573164	50169	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	0	9	0.2	CN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	4200979	50494	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	7	1.0	COC(=O)CCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1576536	50494	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	7	1.0	COC(=O)CCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	1132498	50705	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	5	5.1	Cc1ccc2nsnc2c1NC(=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1578314	50705	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	5	5.1	Cc1ccc2nsnc2c1NC(=O)c1sc2ccccc2c1Cl	nan
	3220367	50960	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	1	6	2.4	COCCNC(=O)C(OC(=O)c1nsc(Cl)c1Cl)C(C)C	nan
	CHEMBL1580567	50960	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	1	6	2.4	COCCNC(=O)C(OC(=O)c1nsc(Cl)c1Cl)C(C)C	nan
	4343313	51159	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.2	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)n1	nan
	CHEMBL1582134	51159	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.2	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)n1	nan
	3338549	51175	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1582307	51175	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	20917770	51330	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	7	2.4	CN(Cc1ccco1)S(=O)(=O)c1ccc(CN2C(=O)c3cccnc3C2=O)s1	nan
	CHEMBL1583626	51330	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	7	2.4	CN(Cc1ccco1)S(=O)(=O)c1ccc(CN2C(=O)c3cccnc3C2=O)s1	nan
	18562929	51478	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	9	1.1	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCOCC4)nn23)cc1	nan
	CHEMBL1584882	51478	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	9	1.1	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCOCC4)nn23)cc1	nan
	2427540	51899	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	10	1.4	Cn1c(N)c(C(=O)CSc2nc3ccccc3c(=O)n2Cc2ccccc2)c(=O)n(C)c1=O	nan
	CHEMBL1588321	51899	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	10	1.4	Cn1c(N)c(C(=O)CSc2nc3ccccc3c(=O)n2Cc2ccccc2)c(=O)n(C)c1=O	nan
	20923114	51924	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	9	0	6	2.7	CCCN(CCC)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1588547	51924	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	9	0	6	2.7	CCCN(CCC)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	20885679	52128	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	1.9	Cc1nn(CCCC(=O)NCc2ccccc2Cl)c(=O)c2nccn12	nan
	CHEMBL1590561	52128	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	1.9	Cc1nn(CCCC(=O)NCc2ccccc2Cl)c(=O)c2nccn12	nan
	16023172	52152	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	3.4	CCCCNC(=O)CSc1nnc(C)c2c(C)n(-c3ccccc3)nc12	nan
	CHEMBL1590852	52152	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	3.4	CCCCNC(=O)CSc1nnc(C)c2c(C)n(-c3ccccc3)nc12	nan
	16016417	52193	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	3.4	Cc1cc(O)c(CN2CCN(c3ccccc3)CC2)c2oc(=O)cc(C)c12	nan
	CHEMBL1591358	52193	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	3.4	Cc1cc(O)c(CN2CCN(c3ccccc3)CC2)c2oc(=O)cc(C)c12	nan
	16009611	52350	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1cccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c1)c1ccc(F)cc1	nan
	CHEMBL1593455	52350	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1cccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c1)c1ccc(F)cc1	nan
	16453157	52808	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	8	2.7	O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1nn(-c2ccccc2)ccc1=O	nan
	CHEMBL1597782	52808	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	8	2.7	O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1nn(-c2ccccc2)ccc1=O	nan
	15990388	53014	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.4	Cc1c(NC(=O)c2nc3ccccc3n(C)c2=O)cccc1[N+](=O)[O-]	nan
	CHEMBL1599627	53014	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.4	Cc1c(NC(=O)c2nc3ccccc3n(C)c2=O)cccc1[N+](=O)[O-]	nan
	20917744	53093	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	7	2.3	Cc1ccc(CNS(=O)(=O)c2ccc(CN3C(=O)c4cccnc4C3=O)s2)o1	nan
	CHEMBL1600418	53093	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	7	2.3	Cc1ccc(CNS(=O)(=O)c2ccc(CN3C(=O)c4cccnc4C3=O)s2)o1	nan
	3252667	53109	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	4.8	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1600566	53109	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	4.8	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	5389427	53189	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	1	7	4.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3cc(C)on3)C2c2ccccc2OC)cc1	nan
	CHEMBL1601252	53189	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	1	7	4.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3cc(C)on3)C2c2ccccc2OC)cc1	nan
	723168	53513	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	4	1	4	4.2	O=C(O)Cc1sc(-c2ccccc2)nc1-c1cccs1	nan
	CHEMBL1604196	53513	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	4	1	4	4.2	O=C(O)Cc1sc(-c2ccccc2)nc1-c1cccs1	nan
	2235547	53651	30	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	3	1	5	2.4	CCOc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1605444	53651	30	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	3	1	5	2.4	CCOc1ccccc1-c1nnc(S)o1	nan
	2927721	53800	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	2	7	2.6	CCOCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1606632	53800	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	2	7	2.6	CCOCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	3417563	53890	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3983329	53890	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1607267	53890	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3146573	54115	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	7	3.5	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1609156	54115	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	7	3.5	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	1941998	54148	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4F)sc3n2)c1	nan
	CHEMBL1609358	54148	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4F)sc3n2)c1	nan
	5389862	54280	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	6	3.5	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	CHEMBL1610515	54280	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	6	3.5	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	9550945	54443	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	2	0	5	3.2	CCOC(=O)N1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1611989	54443	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	2	0	5	3.2	CCOC(=O)N1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	2120111	55399	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	CHEMBL1484562	55399	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	CHEMBL1622008	55399	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	1724830	55544	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	CHEMBL1520781	55544	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	CHEMBL1623209	55544	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	9619025	71610	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	10	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1OC	nan
	CHEMBL1973418	71610	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	10	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1OC	nan
	5065598	72226	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	0	8	2.9	CCOC(=O)Cn1/c(=N/C(=O)c2cccs2)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1992834	72226	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	0	8	2.9	CCOC(=O)Cn1/c(=N/C(=O)c2cccs2)sc2cc(C(=O)OC)ccc21	nan
	5286961	72477	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	9915251	72477	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL2001904	72477	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	95028	93362	28	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	2	0	6	0.5	Cn1c(=O)c2c(ncn2Cc2ccccc2)n(C)c1=O	nan
	CHEMBL24759	93362	28	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	2	0	6	0.5	Cn1c(=O)c2c(ncn2Cc2ccccc2)n(C)c1=O	nan
	135723776	107085	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	2	5	2.6	Cc1cc(O)nc(N/N=C/c2c(F)c(F)c(F)c(F)c2F)n1	nan
	CHEMBL3189383	107085	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	2	5	2.6	Cc1cc(O)nc(N/N=C/c2c(F)c(F)c(F)c(F)c2F)n1	nan
	5342833	107095	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	3	9	-2.3	Cn1c(=O)c2nc(N/N=C(/C#N)C(N)=O)[nH]c2n(C)c1=O	nan
	CHEMBL3189560	107095	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	3	9	-2.3	Cn1c(=O)c2nc(N/N=C(/C#N)C(N)=O)[nH]c2n(C)c1=O	nan
	4564145	107348	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(Br)cc2)n(C)c1C	nan
	CHEMBL3192424	107348	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(Br)cc2)n(C)c1C	nan
	135526880	107768	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	135643494	107768	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	137199718	107768	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	CHEMBL3197292	107768	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	9660607	107794	5	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	3	3.8	Cc1ccc(N2C(=O)CS/C2=N\C(=S)Nc2ccccc2)cc1	nan
	CHEMBL3197507	107794	5	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	3	3.8	Cc1ccc(N2C(=O)CS/C2=N\C(=S)Nc2ccccc2)cc1	nan
	9583775	108394	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	2	7	2.1	Nc1c(C(=O)N/N=C/c2ccc([N+](=O)[O-])cc2)cnn1-c1ccccc1	nan
	CHEMBL3210811	108394	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	2	7	2.1	Nc1c(C(=O)N/N=C/c2ccc([N+](=O)[O-])cc2)cnn1-c1ccccc1	nan
	3669734	197034	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	2.6	CCOC(=O)N1CCN(C(=O)CCCCn2c(=S)[nH]c3ccsc3c2=O)CC1	nan
	CHEMBL582737	197034	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	2.6	CCOC(=O)N1CCN(C(=O)CCCCn2c(=S)[nH]c3ccsc3c2=O)CC1	nan
	3324	204702	112	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	7	1	9	0.5	CC(=O)OCC(CCn1cnc2cnc(N)nc21)COC(C)=O	nan
	CHEMBL880	204702	112	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	7	1	9	0.5	CC(=O)OCC(CCn1cnc2cnc(N)nc21)COC(C)=O	nan
	1028	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	139148732	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	479	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	5816	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	CHEMBL679	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	DB00668	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	3289443	6972	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	5	5.0	Nc1c(C(=O)Nc2cccc(F)c2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1084955	6972	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	5	5.0	Nc1c(C(=O)Nc2cccc(F)c2)sc2nc(-c3cccs3)ccc12	nan
	4112670	10365	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	3	4	5.5	O=C(NCCc1ccc(Cl)cc1)C1CCC(CNc2nc(=S)[nH]c3ccccc23)CC1	nan
	CHEMBL1165197	10365	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	3	4	5.5	O=C(NCCc1ccc(Cl)cc1)C1CCC(CNc2nc(=S)[nH]c3ccccc23)CC1	nan
	1003890	18162	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)c1	nan
	CHEMBL1271075	18162	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)c1	nan
	790786	19554	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	1	4.5	CCc1c(C)nc2ccc(Br)cc2c1Cl	nan
	CHEMBL1301385	19554	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	1	4.5	CCc1c(C)nc2ccc(Br)cc2c1Cl	nan
	6621843	19643	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	1	5	2.4	CCCNc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1302226	19643	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	1	5	2.4	CCCNc1nc2ccccc2n2c(C)nnc12	nan
	926200	19867	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	4	4.0	Fc1cnc(N2CCc3ccccc32)nc1N1CCc2ccccc21	nan
	CHEMBL1303908	19867	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	4	4.0	Fc1cnc(N2CCc3ccccc32)nc1N1CCc2ccccc21	nan
	20881176	20155	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	1	7	2.3	CC(C)CCn1c(=O)c2ccccc2n2c(CCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1306246	20155	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	1	7	2.3	CC(C)CCn1c(=O)c2ccccc2n2c(CCC(=O)NCC3CCCO3)nnc12	nan
	2220688	20306	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	0	6	4.3	Cc1ccc(-c2cc(C(=O)N3CCN(c4ncccn4)CC3)c3cc(Br)ccc3n2)o1	nan
	CHEMBL1307526	20306	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	0	6	4.3	Cc1ccc(-c2cc(C(=O)N3CCN(c4ncccn4)CC3)c3cc(Br)ccc3n2)o1	nan
	2962628	20397	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	5	5.0	CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2C(=O)c2ccccc2)c(Br)cc1OCC(=O)O	nan
	CHEMBL1308267	20397	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	5	5.0	CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2C(=O)c2ccccc2)c(Br)cc1OCC(=O)O	nan
	3774396	20615	2	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	1	3	6	1.7	CSc1nc(S)c2[nH]c(S)nc2n1	nan
	CHEMBL1310138	20615	2	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	1	3	6	1.7	CSc1nc(S)c2[nH]c(S)nc2n1	nan
	6247103	20928	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	4.4	COc1cc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc(OC)c1OC	nan
	CHEMBL1312514	20928	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	4.4	COc1cc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc(OC)c1OC	nan
	2927414	21285	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	8	1.9	CCOCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1315953	21285	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	8	1.9	CCOCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	16187669	21633	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	11	2	7	3.0	CCC1CCCCN1CCCNC(=O)CCCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1319736	21633	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	11	2	7	3.0	CCC1CCCCN1CCCNC(=O)CCCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	1473386	21741	23	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	7	0.7	CCOC(=O)CSc1nc(=O)n2ccccc2n1	nan
	CHEMBL1320637	21741	23	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	7	0.7	CCOC(=O)CSc1nc(=O)n2ccccc2n1	nan
	2363935	21782	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	1	8	0.0	Cn1c(N)c(C(=O)COC(=O)CCc2ccccc2)c(=O)n(C)c1=O	nan
	CHEMBL1321001	21782	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	1	8	0.0	Cn1c(N)c(C(=O)COC(=O)CCc2ccccc2)c(=O)n(C)c1=O	nan
	1485315	21799	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	5	1.6	CS(=O)(=O)NNC(=O)c1cc2cc3ccccc3nc2s1	nan
	CHEMBL1321144	21799	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	5	1.6	CS(=O)(=O)NNC(=O)c1cc2cc3ccccc3nc2s1	nan
	20903731	21818	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	9	1	7	2.2	CC1CCN(c2ccc3nnc(CCC(=O)NCCCOC(C)C)n3n2)CC1	nan
	CHEMBL1321331	21818	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	9	1	7	2.2	CC1CCN(c2ccc3nnc(CCC(=O)NCCCOC(C)C)n3n2)CC1	nan
	16014625	21850	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.3	CC(=O)Nc1ccc(NC(=O)C2CCN(c3cnccn3)CC2)cc1	nan
	CHEMBL1321666	21850	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.3	CC(=O)Nc1ccc(NC(=O)C2CCN(c3cnccn3)CC2)cc1	nan
	16031994	22025	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	6	5.3	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Cl)c(Cl)c3)nn2)s1	nan
	CHEMBL1323264	22025	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	6	5.3	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Cl)c(Cl)c3)nn2)s1	nan
	857564	22082	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cccc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1323763	22082	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cccc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	1955570	22183	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccccc4C)sc3n2)c1	nan
	CHEMBL1324540	22183	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccccc4C)sc3n2)c1	nan
	16019112	22207	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	1	8	3.6	Cc1ccccc1NC(=O)Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	CHEMBL1324746	22207	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	1	8	3.6	Cc1ccccc1NC(=O)Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	20957487	22285	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4F)CC3)n2n1	nan
	CHEMBL1325415	22285	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4F)CC3)n2n1	nan
	654648	22316	13	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.4	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	CHEMBL1325819	22316	13	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.4	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	16411657	22470	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	4	0.9	CC1=NN(c2ccccc2)C(=O)C1/C=C1/NC(=S)NC1=O	nan
	CHEMBL1327209	22470	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	4	0.9	CC1=NN(c2ccccc2)C(=O)C1/C=C1/NC(=S)NC1=O	nan
	3725176	22692	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3cccc(C)c3)n2)cc1	nan
	CHEMBL1329088	22692	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3cccc(C)c3)n2)cc1	nan
	2965680	23593	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	4	4.4	CC(NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12)C1CCCO1	nan
	CHEMBL1336138	23593	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	4	4.4	CC(NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12)C1CCCO1	nan
	2928436	23622	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	2	8	1.7	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1Cc1ccco1	nan
	CHEMBL1336360	23622	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	2	8	1.7	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1Cc1ccco1	nan
	16023198	23847	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.0	Cc1nnc(SCC(=O)NCc2cccc(F)c2)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1338308	23847	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.0	Cc1nnc(SCC(=O)NCc2cccc(F)c2)c2nn(-c3ccccc3)c(C)c12	nan
	4907461	23965	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	5	3.7	CCCCNc1ncnc2sc3c(c12)CCN(CCC)C3	nan
	CHEMBL1339392	23965	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	5	3.7	CCCCNc1ncnc2sc3c(c12)CCN(CCC)C3	nan
	4173573	24410	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	2	8	0.8	Cc1cccn2c(=O)c3cc(C(N)=S)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1343182	24410	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	2	8	0.8	Cc1cccn2c(=O)c3cc(C(N)=S)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	2439152	24423	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	0	5	2.2	Cc1ccc2nc(Cn3cc(C(F)(F)F)ccc3=O)cc(=O)n2c1	nan
	CHEMBL1343295	24423	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	0	5	2.2	Cc1ccc2nc(Cn3cc(C(F)(F)F)ccc3=O)cc(=O)n2c1	nan
	4918386	24773	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	2.5	Cc1cc(CNC(=O)C(C)n2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	CHEMBL1346435	24773	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	2.5	Cc1cc(CNC(=O)C(C)n2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	20904584	24789	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	9	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccccn4)CC3)nnc12	nan
	CHEMBL1346578	24789	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	9	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccccn4)CC3)nnc12	nan
	6112144	24804	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	9	1	7	3.5	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1346652	24804	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	9	1	7	3.5	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	5181544	25122	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	8	3.5	COC(=O)c1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1349309	25122	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	8	3.5	COC(=O)c1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	663780	25200	13	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	2	8	2.2	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CCCOC(C)C)c(=O)n2c1	nan
	CHEMBL1349978	25200	13	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	2	8	2.2	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CCCOC(C)C)c(=O)n2c1	nan
	860395	25209	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	3	3.8	O=C(O)c1cc(-c2cccs2)nc2ccc(F)cc12	nan
	CHEMBL1350037	25209	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	3	3.8	O=C(O)c1cc(-c2cccs2)nc2ccc(F)cc12	nan
	1013700	25400	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	0	3	3.6	O=C(COc1ccc2cc(Br)ccc2c1Br)N1CCOCC1	nan
	CHEMBL1351652	25400	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	0	3	3.6	O=C(COc1ccc2cc(Br)ccc2c1Br)N1CCOCC1	nan
	4137672	25544	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	4	4.1	O=C(O)c1ccccc1SCc1cn2cc(Br)ccc2n1	nan
	CHEMBL1352828	25544	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	4	4.1	O=C(O)c1ccccc1SCc1cn2cc(Br)ccc2n1	nan
	15991076	25840	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	6.6	COc1cc2ccccc2cc1C(=O)Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1	nan
	CHEMBL1355303	25840	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	6.6	COc1cc2ccccc2cc1C(=O)Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1	nan
	16019626	25924	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	8	3.2	Cc1ccc(-n2nnc(-c3nc(-c4cccs4)no3)c2N)c(C)c1	nan
	CHEMBL1356419	25924	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	8	3.2	Cc1ccc(-n2nnc(-c3nc(-c4cccs4)no3)c2N)c(C)c1	nan
	16033238	25976	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	5	5.6	Cc1cccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1C	nan
	CHEMBL1357134	25976	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	5	5.6	Cc1cccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1C	nan
	4084525	26293	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	0	6	3.9	CCOC(=O)c1sc2nc(C)nc(N3CCCCC3C)c2c1C	nan
	CHEMBL1360386	26293	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	0	6	3.9	CCOC(=O)c1sc2nc(C)nc(N3CCCCC3C)c2c1C	nan
	1130278	26323	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	4.0	Cc1ccc(NC(=O)CSc2nnc(COc3ccccc3C)o2)cc1	nan
	CHEMBL1360712	26323	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	4.0	Cc1ccc(NC(=O)CSc2nnc(COc3ccccc3C)o2)cc1	nan
	2112396	26764	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	7	4.0	CNS(=O)(=O)c1cccc(C(=O)OCC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1	nan
	CHEMBL1364577	26764	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	7	4.0	CNS(=O)(=O)c1cccc(C(=O)OCC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1	nan
	3244890	27547	13	None	-5	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.7	O=C(O)CCc1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1370669	27547	13	None	-5	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.7	O=C(O)CCc1ccc(-c2ccc(Br)cc2)o1	nan
	135443907	27890	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	2	9	4.5	CCOc1ccc2nc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)sc2c1	nan
	CHEMBL1373145	27890	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	2	9	4.5	CCOc1ccc2nc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)sc2c1	nan
	16018180	27892	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(OC)c(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)c1	nan
	CHEMBL1373157	27892	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(OC)c(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)c1	nan
	2727621	27993	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	7	3.3	CSc1c(C#N)c(N)nc2sc(C(=O)c3ccccc3)c(N)c12	nan
	CHEMBL1373780	27993	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	7	3.3	CSc1c(C#N)c(N)nc2sc(C(=O)c3ccccc3)c(N)c12	nan
	16019289	28234	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	5	4.9	Cc1ccc(NC(=O)CSc2ccc(-c3cccs3)nn2)cc1Cl	nan
	CHEMBL1375486	28234	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	5	4.9	Cc1ccc(NC(=O)CSc2ccc(-c3cccs3)nn2)cc1Cl	nan
	2361888	28395	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc(O)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	CHEMBL1377052	28395	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc(O)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	887924	28479	9	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	4	4.8	Cc1ccc2c(Cl)c(C(=O)Nc3ccc4c(c3)OCO4)sc2c1	nan
	CHEMBL1377850	28479	9	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	4	4.8	Cc1ccc2c(Cl)c(C(=O)Nc3ccc4c(c3)OCO4)sc2c1	nan
	135527311	28967	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	8	3.7	COC(=O)CSc1nc(O)c2c(C(F)(F)F)cc(-c3cccs3)nc2n1	nan
	CHEMBL1382080	28967	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	8	3.7	COC(=O)CSc1nc(O)c2c(C(F)(F)F)cc(-c3cccs3)nc2n1	nan
	15987888	29232	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1384448	29232	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	54710218	29529	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	4	3.7	Cc1ccc(Sc2c(O)c3ccccc3n(C)c2=O)cc1	nan
	CHEMBL1386873	29529	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	4	3.7	Cc1ccc(Sc2c(O)c3ccccc3n(C)c2=O)cc1	nan
	4047539	29727	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	8	0.8	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1388441	29727	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	8	0.8	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	733870	29843	34	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	1	4	3.6	CC(=O)c1sc(NC(=O)c2ccc(Cl)cc2)nc1C	nan
	CHEMBL1389324	29843	34	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	1	4	3.6	CC(=O)c1sc(NC(=O)c2ccc(Cl)cc2)nc1C	nan
	829950	29957	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	5	1.6	CN(C)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1390362	29957	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	5	1.6	CN(C)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	5027542	30001	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	7	1.5	O=C(CN1C(=O)C2CC=CCC2C1=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1390760	30001	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	7	1.5	O=C(CN1C(=O)C2CC=CCC2C1=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	3634961	30115	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	4315628	30115	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	CHEMBL1391748	30115	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	5898126	30147	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	4.1	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccs2)cc1	nan
	CHEMBL1392030	30147	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	4.1	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccs2)cc1	nan
	4531942	30184	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	11	0.0	CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1392325	30184	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	11	0.0	CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	1102249	30244	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	2	4	4.5	O=C(Nc1ccc(Br)cn1)c1cccc(C(=O)Nc2ccc(Br)cn2)c1	nan
	CHEMBL1392808	30244	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	2	4	4.5	O=C(Nc1ccc(Br)cn1)c1cccc(C(=O)Nc2ccc(Br)cn2)c1	nan
	16018254	30743	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	4	1.1	CNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	CHEMBL1398599	30743	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	4	1.1	CNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	16873489	30874	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	8	2.5	O=[N+]([O-])c1ccccc1S(=O)(=O)Nc1cccc(-c2ccc3nncn3n2)c1	nan
	CHEMBL1399932	30874	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	8	2.5	O=[N+]([O-])c1ccccc1S(=O)(=O)Nc1cccc(-c2ccc3nncn3n2)c1	nan
	20957244	31030	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	0	9	2.5	CCOc1ccc(N(C)C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1401299	31030	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	0	9	2.5	CCOc1ccc(N(C)C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	5053439	31045	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	6	1.2	COC(CNC(=O)c1ccc2nc3ccccc3c(=O)n2c1)OC	nan
	CHEMBL1401405	31045	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	6	1.2	COC(CNC(=O)c1ccc2nc3ccccc3c(=O)n2c1)OC	nan
	5734701	31242	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1	nan
	CHEMBL1403145	31242	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1	nan
	5302177	31328	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	0	5	2.0	O=c1nc2ccccn2c2ccc(S(=O)(=O)N3CCCCC3)cc12	nan
	CHEMBL1404020	31328	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	0	5	2.0	O=c1nc2ccccn2c2ccc(S(=O)(=O)N3CCCCC3)cc12	nan
	1504305	31530	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	5	0	7	1.7	Cc1cc(C)n(C(=O)CCCn2cc([N+](=O)[O-])cn2)n1	nan
	CHEMBL1405977	31530	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	5	0	7	1.7	Cc1cc(C)n(C(=O)CCCn2cc([N+](=O)[O-])cn2)n1	nan
	5221227	31760	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	10	-0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCN4CCOCC4)c3nc12	nan
	CHEMBL1407863	31760	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	10	-0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCN4CCOCC4)c3nc12	nan
	975666	31897	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	7	1.6	Cc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	CHEMBL1408899	31897	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	7	1.6	Cc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	3152548	31913	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1)c1ccco1	nan
	CHEMBL1409014	31913	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1)c1ccco1	nan
	3147984	31994	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	2.5	CCN(CC)C(=O)CSc1nnc2c3ccccc3n(C)c2n1	nan
	CHEMBL1409671	31994	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	2.5	CCN(CC)C(=O)CSc1nnc2c3ccccc3n(C)c2n1	nan
	2740105	32063	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	0	4	3.3	N#Cc1c(N2CCCC2)nsc1-c1ccccc1	nan
	CHEMBL1410151	32063	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	0	4	3.3	N#Cc1c(N2CCCC2)nsc1-c1ccccc1	nan
	2965406	32068	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	5	4.1	O=C(NCCCn1ccnc1)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1410223	32068	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	5	4.1	O=C(NCCCn1ccnc1)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	609181	32252	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	1	3	4.1	CC1(C(=O)Nc2nc3ccccc3s2)CC1(Br)Br	nan
	CHEMBL1411818	32252	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	1	3	4.1	CC1(C(=O)Nc2nc3ccccc3s2)CC1(Br)Br	nan
	2328662	32373	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	7	2.6	CCOC(=O)Cc1csc(-n2sc3ccccc3c2=O)n1	nan
	CHEMBL1412731	32373	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	7	2.6	CCOC(=O)Cc1csc(-n2sc3ccccc3c2=O)n1	nan
	716956	32611	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.5	COc1cc(-c2oc3ccc(C)cc3c(=O)c2O)cc(OC)c1OC	nan
	CHEMBL1414686	32611	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.5	COc1cc(-c2oc3ccc(C)cc3c(=O)c2O)cc(OC)c1OC	nan
	16019291	32954	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	4	5.2	Clc1cccc(CSc2ccc(-c3cccs3)nn2)c1	nan
	CHEMBL1417757	32954	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	4	5.2	Clc1cccc(CSc2ccc(-c3cccs3)nn2)c1	nan
	17581531	32976	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.5	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCCS3	nan
	CHEMBL1417902	32976	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.5	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCCS3	nan
	1505908	33177	11	None	-21	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	1.5	Cc1c(F)cccc1NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C	nan
	CHEMBL1419634	33177	11	None	-21	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	1.5	Cc1c(F)cccc1NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C	nan
	2138543	33461	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	CHEMBL1422079	33461	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	3937026	34023	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.5	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCC1	nan
	CHEMBL1426645	34023	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.5	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCC1	nan
	5909825	34665	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	1	9	2.5	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1432124	34665	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	1	9	2.5	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	16011119	34943	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.2	Cc1ccc(CNC(=O)C(C)n2nc(C)n3c(cc4sccc43)c2=O)cc1	nan
	CHEMBL1435058	34943	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.2	Cc1ccc(CNC(=O)C(C)n2nc(C)n3c(cc4sccc43)c2=O)cc1	nan
	16018536	35069	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	5	5.2	O=C(NCc1cccs1)c1ccc2c(c1)sc1nc(-c3ccccc3)cn12	nan
	CHEMBL1436706	35069	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	5	5.2	O=C(NCc1cccs1)c1ccc2c(c1)sc1nc(-c3ccccc3)cn12	nan
	16011654	35075	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1ccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)cc1	nan
	CHEMBL1436776	35075	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1ccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)cc1	nan
	790330	35298	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2nc(C)cc(S)c2c1	nan
	CHEMBL1439016	35298	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2nc(C)cc(S)c2c1	nan
	22333977	35319	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)c(OC)c1	nan
	CHEMBL1439223	35319	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)c(OC)c1	nan
	974773	35484	7	None	-19	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	1	2	2	2.9	O=C(O)c1ccc2cccc(Cl)c2c1O	nan
	CHEMBL1440675	35484	7	None	-19	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	1	2	2	2.9	O=C(O)c1ccc2cccc(Cl)c2c1O	nan
	1048151	35980	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	3.8	COc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1445229	35980	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	3.8	COc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	16407102	35986	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	8	1	9	2.8	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCN4CCOCC4)cc3c3ccnc2c31	nan
	CHEMBL1445287	35986	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	8	1	9	2.8	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCN4CCOCC4)cc3c3ccnc2c31	nan
	3244615	36394	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	8	1.2	O=C(Cn1cnc2sc3c(c2c1=O)CCCC3)NCCC(=O)N1CCC2(CC1)OCCO2	nan
	CHEMBL1448799	36394	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	8	1.2	O=C(Cn1cnc2sc3c(c2c1=O)CCCC3)NCCC(=O)N1CCC2(CC1)OCCO2	nan
	5333438	36495	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	3	5	0.9	O=C(O)/C=C\C(=O)Nc1cc(O)ccc1[N+](=O)[O-]	nan
	CHEMBL1449557	36495	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	3	5	0.9	O=C(O)/C=C\C(=O)Nc1cc(O)ccc1[N+](=O)[O-]	nan
	946874	36909	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	8	2.2	COC(=O)CSc1nc2ccccc2nc1SCC(=O)OC	nan
	CHEMBL1452913	36909	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	8	2.2	COC(=O)CSc1nc2ccccc2nc1SCC(=O)OC	nan
	15990397	36975	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	7	2.2	COc1cc(NC(=O)c2nc3ccccc3n(C)c2=O)cc(OC)c1OC	nan
	CHEMBL1453389	36975	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	7	2.2	COc1cc(NC(=O)c2nc3ccccc3n(C)c2=O)cc(OC)c1OC	nan
	2072948	37119	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	4	3.4	Brc1ccc2ncnc(NCc3cccnc3)c2c1	nan
	CHEMBL1454562	37119	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	4	3.4	Brc1ccc2ncnc(NCc3cccnc3)c2c1	nan
	20957239	37466	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	5	1	8	2.5	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1F	nan
	CHEMBL1457707	37466	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	5	1	8	2.5	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1F	nan
	8031083	37662	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	7	2.1	CCOC(=O)CCc1c(C)c2ccc3c(c2oc1=O)CN(CCCO)CO3	nan
	CHEMBL1459326	37662	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	7	2.1	CCOC(=O)CCc1c(C)c2ccc3c(c2oc1=O)CN(CCCO)CO3	nan
	1947745	38074	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	1947746	38074	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	CHEMBL1462881	38074	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	3593326	38096	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	8	1.1	CCOC(=O)C1=NN(c2ccc([N+](=O)[O-])cc2)CC1C(=O)OC	nan
	CHEMBL1463045	38096	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	8	1.1	CCOC(=O)C1=NN(c2ccc([N+](=O)[O-])cc2)CC1C(=O)OC	nan
	3889908	38179	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	663903	38179	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	CHEMBL1463781	38179	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	4834173	38401	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	6	2.7	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cccc(C#N)c2)c1	nan
	CHEMBL1465419	38401	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	6	2.7	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cccc(C#N)c2)c1	nan
	2124679	38491	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.7	O=C(COc1ncnc2ccc(Br)cc12)NCc1ccco1	nan
	CHEMBL1466120	38491	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.7	O=C(COc1ncnc2ccc(Br)cc12)NCc1ccco1	nan
	5840379	38627	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	4	1	9	0.8	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CC(C)OC(C)C3)nc12	nan
	CHEMBL1467214	38627	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	4	1	9	0.8	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CC(C)OC(C)C3)nc12	nan
	2824481	38779	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	5	3.9	N#Cc1c(N2CCSCC2)nsc1-c1ccccc1Cl	nan
	CHEMBL1468502	38779	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	5	3.9	N#Cc1c(N2CCSCC2)nsc1-c1ccccc1Cl	nan
	5911323	38902	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.0	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(C)cc2)cc1	nan
	CHEMBL1469507	38902	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.0	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(C)cc2)cc1	nan
	3186594	39083	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1471097	39083	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	5302637	39291	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	4	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2)cc1	nan
	CHEMBL1473111	39291	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	4	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2)cc1	nan
	16009440	39356	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	7	4.0	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1C	nan
	CHEMBL1474025	39356	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	7	4.0	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1C	nan
	16018838	39359	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	0	5	4.9	Clc1cccc(CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1474070	39359	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	0	5	4.9	Clc1cccc(CSc2nncn3c2cc2sccc23)c1	nan
	16033266	39481	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.3	Cc1c(C(=O)NC(C)c2ccccc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1475712	39481	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.3	Cc1c(C(=O)NC(C)c2ccccc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16030277	39485	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccc(F)cc3)CC2)cc1	nan
	CHEMBL1475778	39485	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccc(F)cc3)CC2)cc1	nan
	16018142	39508	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	6	1	2	4.0	Cn1cc(CCCC(=O)NCc2ccc(F)cc2)c2ccccc21	nan
	CHEMBL1476187	39508	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	6	1	2	4.0	Cn1cc(CCCC(=O)NCc2ccc(F)cc2)c2ccccc21	nan
	16018630	39516	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	4.0	O=C(CSc1nncn2c1cc1occc12)Nc1ccc(F)c(Cl)c1	nan
	CHEMBL1476304	39516	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	4.0	O=C(CSc1nncn2c1cc1occc12)Nc1ccc(F)c(Cl)c1	nan
	16018040	39529	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	6	3.1	COc1ccc(OC)c(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1476501	39529	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	6	3.1	COc1ccc(OC)c(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	135407487	39542	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(CNC(=O)CSc2nc3[nH]nc(C)c3c(=N)n2-c2ccccc2Cl)cc1	nan
	CHEMBL1476621	39542	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(CNC(=O)CSc2nc3[nH]nc(C)c3c(=N)n2-c2ccccc2Cl)cc1	nan
	676907	39640	46	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	205	1	1	3	2.8	COc1ccc2c(C)cc(S)nc2c1	nan
	CHEMBL1477596	39640	46	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	205	1	1	3	2.8	COc1ccc2c(C)cc(S)nc2c1	nan
	16018964	39878	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.2	CCC(C)NC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1479750	39878	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.2	CCC(C)NC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16018270	40373	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	5	5.5	CC(=O)Nc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	CHEMBL1484019	40373	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	5	5.5	CC(=O)Nc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	4613858	40769	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	1	2	7	0.9	COC(=O)c1sc2[nH]c(=S)n(N)c(=O)c2c1C	nan
	CHEMBL1487438	40769	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	1	2	7	0.9	COC(=O)c1sc2[nH]c(=S)n(N)c(=O)c2c1C	nan
	1173795	40918	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	1.9	CCCn1c(SCC(=O)Nc2ccc(NC(=O)CC)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1488482	40918	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	1.9	CCCn1c(SCC(=O)Nc2ccc(NC(=O)CC)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3152454	40950	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	3	8	0.4	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1CCCO	nan
	CHEMBL1488709	40950	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	3	8	0.4	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1CCCO	nan
	1294912	41389	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	2	8	3.8	COc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	CHEMBL1491898	41389	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	2	8	3.8	COc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	3944710	41396	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	8	2.1	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cc(O)nc2ccccc12	nan
	CHEMBL1491951	41396	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	8	2.1	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cc(O)nc2ccccc12	nan
	2958357	41719	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	6	2.9	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCC3	nan
	CHEMBL1494894	41719	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	6	2.9	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCC3	nan
	3601528	41752	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	2	7	5.3	COc1ccc(C(=O)Nc2nc3n(n2)C(c2ccc(Cl)cc2)C=C(c2ccccc2)N3)cc1OC	nan
	CHEMBL1495241	41752	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	2	7	5.3	COc1ccc(C(=O)Nc2nc3n(n2)C(c2ccc(Cl)cc2)C=C(c2ccccc2)N3)cc1OC	nan
	3120647	41759	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	3	1	4	6.9	O=C(Nc1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1)c1cc2ccccc2o1	nan
	CHEMBL1495306	41759	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	3	1	4	6.9	O=C(Nc1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1)c1cc2ccccc2o1	nan
	3296097	41856	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	5	1	9	4.1	CCc1ccc(-n2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3nncc-3c2O)cc1	nan
	CHEMBL1496299	41856	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	5	1	9	4.1	CCc1ccc(-n2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3nncc-3c2O)cc1	nan
	2175955	42342	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3cccnc3)cc2)c1C	nan
	CHEMBL1500554	42342	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3cccnc3)cc2)c1C	nan
	2868511	42370	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	4	3.5	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(C)cc2)cc1	nan
	CHEMBL1500746	42370	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	4	3.5	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(C)cc2)cc1	nan
	3146565	42604	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	4.0	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1502935	42604	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	4.0	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	2998667	42776	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	9	-1.9	CC(=O)OCCNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1504458	42776	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	9	-1.9	CC(=O)OCCNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	2497236	42974	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	6	4.6	CCOc1ccc(-c2nc(-c3cccs3)c(CC(=O)O)s2)cc1OC	nan
	CHEMBL1506154	42974	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	6	4.6	CCOc1ccc(-c2nc(-c3cccs3)c(CC(=O)O)s2)cc1OC	nan
	1442564	43380	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	3.5	COC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1509687	43380	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	3.5	COC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	6305743	43391	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	7	1	5	3.2	COCCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1509795	43391	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	7	1	5	3.2	COCCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	15988981	43671	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	8	2	7	4.1	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccccc3Cl)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1512541	43671	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	8	2	7	4.1	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccccc3Cl)c(=O)c3sccc32)c(C)c1	nan
	1116224	43789	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.1	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(C(F)(F)F)c2)n(C)c1=O	nan
	CHEMBL1514415	43789	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.1	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(C(F)(F)F)c2)n(C)c1=O	nan
	16018038	43863	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	5	3.8	CSc1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1515402	43863	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	5	3.8	CSc1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	16016056	43892	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	7	5.0	COc1ccccc1-c1noc(-c2ccc(NCCc3ccccc3)c([N+](=O)[O-])c2)n1	nan
	CHEMBL1515947	43892	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	7	5.0	COc1ccccc1-c1noc(-c2ccc(NCCc3ccccc3)c([N+](=O)[O-])c2)n1	nan
	5069160	43966	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	CHEMBL1516839	43966	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	5389765	44180	9	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	8	1	6	3.1	COCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	CHEMBL1518887	44180	9	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	8	1	6	3.1	COCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	1238913	44323	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	0	9	-1.1	Cn1c(=O)c2c(nc(SCC(=O)N3CCOCC3)n2C)n(C)c1=O	nan
	CHEMBL1520162	44323	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	0	9	-1.1	Cn1c(=O)c2c(nc(SCC(=O)N3CCOCC3)n2C)n(C)c1=O	nan
	2165182	44448	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	5	2.9	Cc1ccc(-c2cc(C(=O)NCCN3CCOCC3)c3ccccc3n2)o1	nan
	CHEMBL1521212	44448	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	5	2.9	Cc1ccc(-c2cc(C(=O)NCCN3CCOCC3)c3ccccc3n2)o1	nan
	3111808	44499	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1	nan
	CHEMBL1521616	44499	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1	nan
	20957509	44620	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1522776	44620	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	4126696	44635	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	5	5.9	COc1ccc(-n2cc(-c3ccccc3)nc2SCC(=O)Nc2ccccc2)cc1Cl	nan
	CHEMBL1522905	44635	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	5	5.9	COc1ccc(-n2cc(-c3ccccc3)nc2SCC(=O)Nc2ccccc2)cc1Cl	nan
	2561590	44993	7	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	0	8	4.1	Cc1cc(C(=O)CSc2nc3ccccc3c(=O)n2C)c(C)n1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1526230	44993	7	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	0	8	4.1	Cc1cc(C(=O)CSc2nc3ccccc3c(=O)n2C)c(C)n1Cc1ccc2c(c1)OCO2	nan
	15991183	45143	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	1	4	6.8	O=C(Nc1cccc(-c2nc3ccccc3o2)c1)c1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1527553	45143	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	1	4	6.8	O=C(Nc1cccc(-c2nc3ccccc3o2)c1)c1ccc(-c2ccc(Br)cc2)o1	nan
	16014288	45494	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	2	8	3.8	Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3nc(SC(C)C)ncc3Cl)cc2)n1	nan
	CHEMBL1530646	45494	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	2	8	3.8	Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3nc(SC(C)C)ncc3Cl)cc2)n1	nan
	6078364	45503	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)cc1	nan
	CHEMBL1530717	45503	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)cc1	nan
	950608	45886	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	1.5	N#C/C(=C\c1c(N2CCCCCC2)nc2ccccn2c1=O)C(N)=O	nan
	CHEMBL1534139	45886	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	1.5	N#C/C(=C\c1c(N2CCCCCC2)nc2ccccn2c1=O)C(N)=O	nan
	5310696	45899	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	10	1	6	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OCC(C)C)cc2C)C1c1cccnc1	nan
	CHEMBL1534309	45899	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	10	1	6	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OCC(C)C)cc2C)C1c1cccnc1	nan
	1856407	46134	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	1.1	CCOC(=O)N1CCN(c2nc3c(C)cccn3c(=O)c2C=O)CC1	nan
	CHEMBL1536792	46134	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	1.1	CCOC(=O)N1CCN(c2nc3c(C)cccn3c(=O)c2C=O)CC1	nan
	1442728	46188	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	4	4.3	CC(C)c1nc(SCC(=O)NC2CCCCC2)c2ccccc2n1	nan
	CHEMBL1537182	46188	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	4	4.3	CC(C)c1nc(SCC(=O)NC2CCCCC2)c2ccccc2n1	nan
	6165328	46433	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	6	4.3	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Cl)cc2)cc1	nan
	CHEMBL1539268	46433	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	6	4.3	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Cl)cc2)cc1	nan
	2944889	46629	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	10	1	7	5.1	CCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccco2)cc1OCC	nan
	CHEMBL1540923	46629	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	10	1	7	5.1	CCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccco2)cc1OCC	nan
	1867273	47106	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	CHEMBL1544770	47106	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	3600899	47137	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	9	4.3	O=c1cc(CSc2nc3nncc-3c(O)n2-c2ccc(Br)cc2)nc2ccc(Br)cn12	nan
	CHEMBL1545051	47137	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	9	4.3	O=c1cc(CSc2nc3nncc-3c(O)n2-c2ccc(Br)cc2)nc2ccc(Br)cn12	nan
	135514845	47336	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	8	2.7	CN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	CHEMBL1546713	47336	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	8	2.7	CN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	1442627	47543	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	2	6	3.1	CCCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	CHEMBL1548632	47543	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	2	6	3.1	CCCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	16016034	47923	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	1	7	4.1	COc1ccccc1-c1noc(-c2ccc(NC(C)C)c([N+](=O)[O-])c2)n1	nan
	CHEMBL1552261	47923	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	1	7	4.1	COc1ccccc1-c1noc(-c2ccc(NC(C)C)c([N+](=O)[O-])c2)n1	nan
	16017890	47940	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	1.5	COCCCNC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	CHEMBL1552564	47940	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	1.5	COCCCNC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	16023050	47941	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	3.1	CCNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)C1	nan
	CHEMBL1552569	47941	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	3.1	CCNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)C1	nan
	3260331	47998	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	3	4.6	O=C(Cn1cc(C(=O)C2CC2)c2ccccc21)Nc1ccc(Br)cc1	nan
	CHEMBL1553312	47998	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	3	4.6	O=C(Cn1cc(C(=O)C2CC2)c2ccccc21)Nc1ccc(Br)cc1	nan
	16030436	48073	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	2.9	CC(C)C(=O)Nc1ccccc1OCc1cc(=O)n2ccccc2n1	nan
	CHEMBL1554451	48073	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	2.9	CC(C)C(=O)Nc1ccccc1OCc1cc(=O)n2ccccc2n1	nan
	16016784	48131	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	5.4	CCOC(=O)C1CCCN(C(=O)c2[nH]c3ccccc3c2Sc2ccc(Cl)cc2)C1	nan
	CHEMBL1555295	48131	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	5.4	CCOC(=O)C1CCCN(C(=O)c2[nH]c3ccccc3c2Sc2ccc(Cl)cc2)C1	nan
	16196698	48154	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	7	1.9	Cc1cc2nnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)n2c2ccccc12	nan
	CHEMBL1555603	48154	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	7	1.9	Cc1cc2nnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)n2c2ccccc12	nan
	2869543	48323	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	3.9	CCOC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	CHEMBL1557161	48323	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	3.9	CCOC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	1272771	48363	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	6	5.4	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)cc4C)sc3n2)cc1OC	nan
	CHEMBL1557478	48363	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	6	5.4	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)cc4C)sc3n2)cc1OC	nan
	3239737	48500	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	7	1.4	Cc1nn(C(C)C(=O)NCC2CCCO2)c(=O)c2cc3occc3n12	nan
	CHEMBL1558668	48500	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	7	1.4	Cc1nn(C(C)C(=O)NCC2CCCO2)c(=O)c2cc3occc3n12	nan
	1503106	48690	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	5	3.1	Cc1cc(CNC(=O)COc2ccc([N+](=O)[O-])cc2)c2ccccc2n1	nan
	CHEMBL1560348	48690	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	5	3.1	Cc1cc(CNC(=O)COc2ccc([N+](=O)[O-])cc2)c2ccccc2n1	nan
	2456723	48975	7	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	2	8	3.7	CCOC(=O)c1cc(-c2ccccc2)sc1NC(=O)COC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1	nan
	CHEMBL1562996	48975	7	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	2	8	3.7	CCOC(=O)c1cc(-c2ccccc2)sc1NC(=O)COC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1	nan
	3221518	49084	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	8	1	5	3.8	CCCNC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1563919	49084	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	8	1	5	3.8	CCCNC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	2952819	49149	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.3	O=C(Cn1nc(-c2cccc([N+](=O)[O-])c2)c2ccccc2c1=O)NCC1CCCO1	nan
	CHEMBL1564585	49149	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.3	O=C(Cn1nc(-c2cccc([N+](=O)[O-])c2)c2ccccc2c1=O)NCC1CCCO1	nan
	2869470	49344	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	0	5	3.6	Cc1nnc(Oc2ccc([N+](=O)[O-])cc2)c2ccccc12	nan
	CHEMBL1566109	49344	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	0	5	3.6	Cc1nnc(Oc2ccc([N+](=O)[O-])cc2)c2ccccc12	nan
	16008434	49433	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	5	4.7	O=C(c1ccc(Cl)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCCO3	nan
	CHEMBL1566810	49433	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	5	4.7	O=C(c1ccc(Cl)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCCO3	nan
	1017457	49540	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	11	0.2	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC3CCCCC3)n2C)n(C)c1=O	nan
	CHEMBL1567667	49540	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	11	0.2	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC3CCCCC3)n2C)n(C)c1=O	nan
	2912191	49629	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	4.4	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)cc2)o1	nan
	CHEMBL1568384	49629	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	4.4	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)cc2)o1	nan
	665555	49926	8	None	-1	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	5	4.9	Cc1nc(SCC(=O)Nc2ccc(C)c(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1570874	49926	8	None	-1	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	5	4.9	Cc1nc(SCC(=O)Nc2ccc(C)c(F)c2)c2oc3ccccc3c2n1	nan
	4333346	50124	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	4	4.3	COc1ccc(CCNC(=O)CSc2ccc3ccccc3c2)cc1OC	nan
	CHEMBL1572841	50124	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	4	4.3	COc1ccc(CCNC(=O)CSc2ccc3ccccc3c2)cc1OC	nan
	20957497	50330	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	10	2	7	2.1	Cc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1574892	50330	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	10	2	7	2.1	Cc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	1938572	50545	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	6	3.6	O=C(COc1ccccc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1576963	50545	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	6	3.6	O=C(COc1ccccc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	1632391	50698	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	3	4	2.0	O=C(O)CCC(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	CHEMBL1578274	50698	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	3	4	2.0	O=C(O)CCC(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	3504887	50750	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	7	1.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC1	nan
	CHEMBL1578618	50750	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	7	1.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC1	nan
	20903631	50756	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	0	9	1.2	COc1cccc(N2CCN(c3ccc4nnc(CCC(=O)N5CCN(C)CC5)n4n3)CC2)c1	nan
	CHEMBL1578662	50756	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	0	9	1.2	COc1cccc(N2CCN(c3ccc4nnc(CCC(=O)N5CCN(C)CC5)n4n3)CC2)c1	nan
	16475	51395	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	4	4	1.9	Nc1ccc(-c2ccc(N)c(C(=O)O)c2)cc1C(=O)O	nan
	CHEMBL1584156	51395	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	4	4	1.9	Nc1ccc(-c2ccc(N)c(C(=O)O)c2)cc1C(=O)O	nan
	1997175	51442	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	0	7	0.9	CN1CCN(c2nc3ccccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	CHEMBL1584587	51442	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	0	7	0.9	CN1CCN(c2nc3ccccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	20881207	51686	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	10	1	8	2.5	CC(C)OCCCn1c(=O)c2ccccc2n2c(CCC(=O)NCc3ccccn3)nnc12	nan
	CHEMBL1586569	51686	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	10	1	8	2.5	CC(C)OCCCn1c(=O)c2ccccc2n2c(CCC(=O)NCc3ccccn3)nnc12	nan
	3186634	51687	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	0	9	-1.2	CN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1586576	51687	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	0	9	-1.2	CN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	658021	51959	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	0	5	3.0	CSC1=NP(=S)(SC)N(C)c2nc3n(c21)CCC3	nan
	CHEMBL1588879	51959	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	0	5	3.0	CSC1=NP(=S)(SC)N(C)c2nc3n(c21)CCC3	nan
	7190667	52069	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1cccc(F)c1	nan
	CHEMBL1589799	52069	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1cccc(F)c1	nan
	16030609	52112	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	0	5	5.7	CCN(C(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1)c1cccc(C)c1	nan
	CHEMBL1590288	52112	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	0	5	5.7	CCN(C(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1)c1cccc(C)c1	nan
	6221827	52142	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.0	COc1ccc(CNC(=O)Cc2c(C)c3c(O)cc(C)cc3oc2=O)cc1	nan
	CHEMBL1590750	52142	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.0	COc1ccc(CNC(=O)Cc2c(C)c3c(O)cc(C)cc3oc2=O)cc1	nan
	16030275	52223	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	0	4	4.9	CCCCN(C)C(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1591718	52223	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	0	4	4.9	CCCCN(C)C(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16031876	52275	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	5	5.0	CCC1CCCCN1Cc1cn2c(-c3ccc(Br)cc3)nnc2s1	nan
	CHEMBL1592401	52275	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	5	5.0	CCC1CCCCN1Cc1cn2c(-c3ccc(Br)cc3)nnc2s1	nan
	5768121	52487	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	6	4.6	Cc1cc(OCC(C)C)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	CHEMBL1594882	52487	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	6	4.6	Cc1cc(OCC(C)C)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	4968658	52597	7	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3ccc(Cl)cc3)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1595841	52597	7	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3ccc(Cl)cc3)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	4875333	53221	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	4	3.5	CCn1c2ccccc2c2nc3cc(C(=O)O)ccc3nc21	nan
	CHEMBL1601617	53221	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	4	3.5	CCn1c2ccccc2c2nc3cc(C(=O)O)ccc3nc21	nan
	15988911	53536	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	7	4.2	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3c(C)cc(C)cc3C)c2=O)c1	nan
	CHEMBL1604412	53536	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	7	4.2	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3c(C)cc(C)cc3C)c2=O)c1	nan
	824096	53628	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	220	0	2	5	1.2	N=c1c2c3c(sc2ncn1N)CCCC3	nan
	CHEMBL1605294	53628	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	220	0	2	5	1.2	N=c1c2c3c(sc2ncn1N)CCCC3	nan
	16020886	53714	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1ccc(CSc2nc3cccnc3n2Cc2ccc(C(=O)NC3CCCCC3)cc2)cc1	nan
	CHEMBL1605955	53714	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1ccc(CSc2nc3cccnc3n2Cc2ccc(C(=O)NC3CCCCC3)cc2)cc1	nan
	3973561	54087	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	7	4.1	COc1ccc2cc(C(=O)COC(=O)COc3ccc4c(C)cc(=O)oc4c3)ccc2c1	nan
	CHEMBL1608925	54087	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	7	4.1	COc1ccc2cc(C(=O)COC(=O)COc3ccc4c(C)cc(=O)oc4c3)ccc2c1	nan
	4916122	54206	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.7	Cc1cccc(NC(=O)C(C)n2cc([N+](=O)[O-])cn2)n1	nan
	CHEMBL1609905	54206	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.7	Cc1cccc(NC(=O)C(C)n2cc([N+](=O)[O-])cn2)n1	nan
	3151454	54391	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	2	8	1.4	COCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1611459	54391	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	2	8	1.4	COCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	2810155	54582	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	5	3.6	Cc1ccccc1C(=O)Nc1nc2c(C)csc2c(=O)s1	nan
	CHEMBL1613272	54582	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	5	3.6	Cc1ccccc1C(=O)Nc1nc2c(C)csc2c(=O)s1	nan
	6489921	55048	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1384004	55048	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1618913	55048	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	135415554	55477	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	CHEMBL1494334	55477	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	CHEMBL1622628	55477	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	24792259	55536	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1517470	55536	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1623157	55536	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	4323731	107198	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	3	3	4	5.9	Oc1c(Br)cc(/C=N/c2ccc3[nH]c(-c4ccccc4)nc3c2)c(O)c1Br	nan
	CHEMBL3190756	107198	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	3	3	4	5.9	Oc1c(Br)cc(/C=N/c2ccc3[nH]c(-c4ccccc4)nc3c2)c(O)c1Br	nan
	4073001	108214	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	8	2.6	COC(=O)Cn1/c(=N/C(=O)c2ccc(OC)c(OC)c2)sc2cc(OC)ccc21	nan
	CHEMBL3208346	108214	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	8	2.6	COC(=O)Cn1/c(=N/C(=O)c2ccc(OC)c(OC)c2)sc2cc(OC)ccc21	nan
	6870745	108596	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	0	7	2.1	Cc1nc2ccccc2c(=O)n1/N=C/c1ccc([N+](=O)[O-])o1	nan
	CHEMBL3213340	108596	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	0	7	2.1	Cc1nc2ccccc2c(=O)n1/N=C/c1ccc([N+](=O)[O-])o1	nan
	2941245	146304	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.8	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccccc3)C2c2cccnc2)o1	nan
	CHEMBL392515	146304	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.8	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccccc3)C2c2cccnc2)o1	nan
	1016096	191189	21	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	CHEMBL519824	191189	21	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	726062	195353	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	CHEMBL1583656	195353	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	CHEMBL567206	195353	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	2998030	31288	6	None	-	1	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	3	6	0.5	COCCNC(=O)NC(=O)COC(=O)C12CC3CC(CC(NC(C)=O)(C3)C1)C2	nan
	CHEMBL1403647	31288	6	None	-	1	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	3	6	0.5	COCCNC(=O)NC(=O)COC(=O)C12CC3CC(CC(NC(C)=O)(C3)C1)C2	nan
	975392	42211	9	None	-1	2	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	1	2	4.3	Cc1cc(Br)c2nc3c(c(C(=O)O)c2c1)CCCCC3	nan
	CHEMBL1499411	42211	9	None	-1	2	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	1	2	4.3	Cc1cc(Br)c2nc3c(c(C(=O)O)c2c1)CCCCC3	nan
	16019550	10592	14	None	-131	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.3	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	CHEMBL1170886	10592	14	None	-131	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.3	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	4204374	19358	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	6	2	6	3.4	COc1cc2nc(S)nc(NCCC(C)C)c2cc1OC	nan
	CHEMBL1299978	19358	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	6	2	6	3.4	COc1cc2nc(S)nc(NCCC(C)C)c2cc1OC	nan
	2421557	19507	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	0	7	3.6	COC(=O)CCc1c(C)c(C(=O)c2cc(OC)c(OC)c(OC)c2)c2ccccn12	nan
	CHEMBL1301080	19507	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	0	7	3.6	COC(=O)CCc1c(C)c(C(=O)c2cc(OC)c(OC)c(OC)c2)c2ccccn12	nan
	22548258	20078	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CO4)CC2)cc1	nan
	CHEMBL1305765	20078	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CO4)CC2)cc1	nan
	16194269	20267	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	7	1	8	2.4	O=C(CSC1=Nc2ccccc2C2=NC(CC(=O)N3CCN(c4ccccc4)CC3)C(=O)N12)NCC1CCCO1	nan
	CHEMBL1307199	20267	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	7	1	8	2.4	O=C(CSC1=Nc2ccccc2C2=NC(CC(=O)N3CCN(c4ccccc4)CC3)C(=O)N12)NCC1CCCO1	nan
	3740686	20895	14	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)no1	nan
	CHEMBL1312274	20895	14	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)no1	nan
	4465171	21043	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCCC2)c1	nan
	CHEMBL1313361	21043	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCCC2)c1	nan
	2197541	21094	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.3	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCC3)c2C#N)cc1	nan
	CHEMBL1313695	21094	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.3	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCC3)c2C#N)cc1	nan
	2679228	21149	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	7	4.0	COc1ccc2oc(C(=O)Nc3nc4ccc(S(C)(=O)=O)cc4s3)c(C)c2c1	nan
	CHEMBL1314240	21149	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	7	4.0	COc1ccc2oc(C(=O)Nc3nc4ccc(S(C)(=O)=O)cc4s3)c(C)c2c1	nan
	16034516	21181	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.6	Cc1nnc(SCC(=O)NCc2ccccc2F)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1314574	21181	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.6	Cc1nnc(SCC(=O)NCc2ccccc2F)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	135419125	21212	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	3	5.7	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2ccccc2)C1	nan
	CHEMBL1315137	21212	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	3	5.7	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2ccccc2)C1	nan
	16012610	21219	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	4	0	10	4.0	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(Cl)cc5)s4)c3nc12	nan
	CHEMBL1315199	21219	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	4	0	10	4.0	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(Cl)cc5)s4)c3nc12	nan
	4119285	21266	11	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	CHEMBL1315733	21266	11	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	24892214	21282	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	8	2.2	COc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1315929	21282	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	8	2.2	COc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	7599144	21290	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	5	3.1	Cc1cc(NC(=O)c2cccn(Cc3cccc(Cl)c3)c2=O)no1	nan
	CHEMBL1315995	21290	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	5	3.1	Cc1cc(NC(=O)c2cccn(Cc3cccc(Cl)c3)c2=O)no1	nan
	16018244	21454	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3ccccc3Cl)cc1CC2	nan
	CHEMBL1318247	21454	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3ccccc3Cl)cc1CC2	nan
	15944876	21575	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1319259	21575	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16010992	21659	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	2.6	CCc1cc2c(cc3c(=O)n(CC(=O)NCCc4ccc(OC)c(OC)c4)ncn32)s1	nan
	CHEMBL1319991	21659	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	2.6	CCc1cc2c(cc3c(=O)n(CC(=O)NCCc4ccc(OC)c(OC)c4)ncn32)s1	nan
	4164390	21746	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	5	6.1	CC(C)OC(=O)c1c(NC(=O)C2c3ccccc3Oc3ccccc32)sc2c1CCCC2	nan
	CHEMBL1320657	21746	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	5	6.1	CC(C)OC(=O)c1c(NC(=O)C2c3ccccc3Oc3ccccc32)sc2c1CCCC2	nan
	25102515	21768	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	4	4.1	Cc1cc(=O)oc2cc(NC(=O)COc3cccc(C(F)(F)F)c3)ccc12	nan
	CHEMBL1320916	21768	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	4	4.1	Cc1cc(=O)oc2cc(NC(=O)COc3cccc(C(F)(F)F)c3)ccc12	nan
	794839	21823	34	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	4	2.8	Sc1nnc(-c2cccc(Br)c2)o1	nan
	CHEMBL1321356	21823	34	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	4	2.8	Sc1nnc(-c2cccc(Br)c2)o1	nan
	16018780	21825	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4cccc(Cl)c4)nnc(C)n32)o1	nan
	CHEMBL1321426	21825	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4cccc(Cl)c4)nnc(C)n32)o1	nan
	3996443	21875	7	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	10	-0.7	Cn1c(N)c(C(=O)COC(=O)COc2ccccc2C#N)c(=O)n(C)c1=O	nan
	CHEMBL1321877	21875	7	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	10	-0.7	Cn1c(N)c(C(=O)COC(=O)COc2ccccc2C#N)c(=O)n(C)c1=O	nan
	16009867	22117	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.5	CCOc1ccccc1NC(=O)Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1324000	22117	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.5	CCOc1ccccc1NC(=O)Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21	nan
	1442375	22223	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	4.1	CC(C)(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1324849	22223	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	4.1	CC(C)(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	22517548	22338	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	1.6	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Br	nan
	CHEMBL1326013	22338	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	1.6	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Br	nan
	20927538	22451	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	0	7	1.3	CN(Cc1ccco1)C(=O)Cn1cc(S(=O)(=O)N2CCCC2)c(S(=O)(=O)N2CCCC2)c1	nan
	CHEMBL1327078	22451	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	0	7	1.3	CN(Cc1ccco1)C(=O)Cn1cc(S(=O)(=O)N2CCCC2)c(S(=O)(=O)N2CCCC2)c1	nan
	2645777	22546	15	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	3	4.4	N#Cc1c(S)nc(-c2ccccc2Cl)c2c1CCCC2	nan
	CHEMBL1327817	22546	15	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	3	4.4	N#Cc1c(S)nc(-c2ccccc2Cl)c2c1CCCC2	nan
	2816375	22773	26	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	1	7	1.7	CCOC(=O)c1nnn2c1nc(S)c1ccccc12	nan
	CHEMBL1329724	22773	26	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	1	7	1.7	CCOC(=O)c1nnn2c1nc(S)c1ccccc12	nan
	3151322	22782	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.0	N=c1c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1329807	22782	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.0	N=c1c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	16030826	22931	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	2	5	2.9	NC(=O)C1CCN(C(=O)c2ccccc2NC(=O)c2nsc3ccccc23)CC1	nan
	CHEMBL1330985	22931	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	2	5	2.9	NC(=O)C1CCN(C(=O)c2ccccc2NC(=O)c2nsc3ccccc23)CC1	nan
	2815453	23169	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	0	5	0.3	Cn1c2c(c(=O)n3ncnc13)CCCC2	nan
	CHEMBL1332830	23169	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	0	5	0.3	Cn1c2c(c(=O)n3ncnc13)CCCC2	nan
	16019110	23178	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	3.3	O=C(Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21)Nc1ccccc1	nan
	CHEMBL1332893	23178	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	3.3	O=C(Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21)Nc1ccccc1	nan
	16018748	23181	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	0	5	4.7	Cc1nnc(SCc2ccc(Cl)cc2)c2cc3occc3n12	nan
	CHEMBL1332908	23181	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	0	5	4.7	Cc1nnc(SCc2ccc(Cl)cc2)c2cc3occc3n12	nan
	876371	23245	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	4	2.2	Cc1cc(/C=C2/C(=O)NC(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	CHEMBL1333432	23245	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	4	2.2	Cc1cc(/C=C2/C(=O)NC(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	16031513	23650	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.0	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(C(F)(F)F)c3)s2)cc1	nan
	CHEMBL1336578	23650	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.0	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(C(F)(F)F)c3)s2)cc1	nan
	16011266	23832	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	3.5	Cc1cccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)c1	nan
	CHEMBL1338231	23832	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	3.5	Cc1cccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)c1	nan
	16009346	23906	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	4	5.1	CCc1ccc2c(c1)c(=O)c(C(=O)c1ccc(C)cc1)cn2CC(=O)Nc1ccccc1C	nan
	CHEMBL1338819	23906	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	4	5.1	CCc1ccc2c(c1)c(=O)c(C(=O)c1ccc(C)cc1)cn2CC(=O)Nc1ccccc1C	nan
	1451340	24025	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	7	1	7	4.2	Cc1nonc1NC(=O)CSc1nc(CCC2CCCC2)nc2ccccc12	nan
	CHEMBL1339937	24025	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	7	1	7	4.2	Cc1nonc1NC(=O)CSc1nc(CCC2CCCC2)nc2ccccc12	nan
	1173483	24235	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	7	4.1	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1nc(C)c(C)s1)OCO3	nan
	CHEMBL1341833	24235	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	7	4.1	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1nc(C)c(C)s1)OCO3	nan
	3208214	24505	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2cc(C)cc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1344061	24505	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2cc(C)cc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	1442646	24693	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	CCCc1nc(SCC(=O)N2CCc3ccccc3C2)c2ccccc2n1	nan
	CHEMBL1345722	24693	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	CCCc1nc(SCC(=O)N2CCc3ccccc3C2)c2ccccc2n1	nan
	2322587	24713	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	9	1	6	1.7	CCN(CC)S(=O)(=O)c1ccc(C(=O)OCCNC(=O)c2cccnc2)cc1	nan
	CHEMBL1345885	24713	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	9	1	6	1.7	CCN(CC)S(=O)(=O)c1ccc(C(=O)OCCNC(=O)c2cccnc2)cc1	nan
	3475758	24733	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc(OC)c1OC	nan
	CHEMBL1346015	24733	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc(OC)c1OC	nan
	911360	24776	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	0	1	4	1.3	Cn1c(O)nc2c(Cl)nccc21	nan
	CHEMBL1346457	24776	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	0	1	4	1.3	Cn1c(O)nc2c(Cl)nccc21	nan
	745324	24830	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	5	4.4	Cc1ccc(NC(S)=Nc2cccc(-c3nnc(S)o3)c2)cc1	nan
	CHEMBL1346824	24830	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	5	4.4	Cc1ccc(NC(S)=Nc2cccc(-c3nnc(S)o3)c2)cc1	nan
	664458	24871	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	4	0	6	4.4	O=C(CSc1ncnc2c1oc1ccccc12)c1cccs1	nan
	CHEMBL1347130	24871	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	4	0	6	4.4	O=C(CSc1ncnc2c1oc1ccccc12)c1cccs1	nan
	866600	24907	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	0	6	1.7	CCN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1347433	24907	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	0	6	1.7	CCN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	2158422	25072	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	7	2.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)CC1	nan
	CHEMBL1348934	25072	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	7	2.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)CC1	nan
	7711373	25108	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	2.9	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccco1	nan
	CHEMBL1349179	25108	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	2.9	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccco1	nan
	20920345	25455	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1352171	25455	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	3742858	25666	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Br)cc2)no1	nan
	CHEMBL1353643	25666	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Br)cc2)no1	nan
	16009768	25794	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	9	2	6	5.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)COc2cccc(OC)c2)cc1	nan
	CHEMBL1354836	25794	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	9	2	6	5.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)COc2cccc(OC)c2)cc1	nan
	16022445	25801	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	1	3	4.8	CC1Cn2c(C(=O)NCc3cccc(Br)c3)cc3cccc(c32)S1	nan
	CHEMBL1354873	25801	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	1	3	4.8	CC1Cn2c(C(=O)NCc3cccc(Br)c3)cc3cccc(c32)S1	nan
	16024821	25875	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccc(Cl)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1355809	25875	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccc(Cl)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	5292880	25885	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	4	6.5	COc1cc(/C=C(\C#N)c2nc3ccccc3[nH]2)cc(Cl)c1OCc1ccccc1Cl	nan
	CHEMBL1355927	25885	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	4	6.5	COc1cc(/C=C(\C#N)c2nc3ccccc3[nH]2)cc(Cl)c1OCc1ccccc1Cl	nan
	7878585	25889	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.9	O=C(CNC(=O)c1ccc(Cl)cc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1356005	25889	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.9	O=C(CNC(=O)c1ccc(Cl)cc1)OCc1cc(=O)n2ccsc2n1	nan
	6200344	25961	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	7	1	6	2.7	COc1cccc(/C=C/c2nc(C#N)c(NCCN(C)C)o2)c1	nan
	CHEMBL1356982	25961	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	7	1	6	2.7	COc1cccc(/C=C/c2nc(C#N)c(NCCN(C)C)o2)c1	nan
	1004107	26149	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	2	5	5.3	CCOc1cccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)c1	nan
	CHEMBL1359199	26149	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	2	5	5.3	CCOc1cccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)c1	nan
	16009637	26451	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	6	4.5	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1ccccc1	nan
	CHEMBL1361843	26451	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	6	4.5	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1ccccc1	nan
	4114478	26802	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.1	COc1cccc(NC(=O)Cn2cc(C(=O)C3CCCCC3)c3ccccc32)c1	nan
	CHEMBL1364874	26802	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.1	COc1cccc(NC(=O)Cn2cc(C(=O)C3CCCCC3)c3ccccc32)c1	nan
	22641	27050	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	7	0.8	CC(=O)OCCn1c2nc(=O)[nH]c(=O)c-2nc2cc(C)c(C)cc21	nan
	CHEMBL1367036	27050	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	7	0.8	CC(=O)OCCn1c2nc(=O)[nH]c(=O)c-2nc2cc(C)c(C)cc21	nan
	2378240	27155	24	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	2	1	4	2.7	Fc1ccccc1-c1nnc(S)n1C1CC1	nan
	CHEMBL1367871	27155	24	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	2	1	4	2.7	Fc1ccccc1-c1nnc(S)n1C1CC1	nan
	12006141	27482	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	4	4.8	Cc1ccc(CSc2ccc(-c3cccs3)nn2)cc1	nan
	CHEMBL1370265	27482	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	4	4.8	Cc1ccc(CSc2ccc(-c3cccs3)nn2)cc1	nan
	16455091	27594	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	2	8	3.0	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccc(F)cc4)ccc3=O)cc2)c1C	nan
	CHEMBL1371016	27594	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	2	8	3.0	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccc(F)cc4)ccc3=O)cc2)c1C	nan
	135406328	27792	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	1	7	1.3	Cc1cc(C)c2c(O)nc(SCC(=O)N3CCOCC3)nc2n1	nan
	CHEMBL1372508	27792	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	1	7	1.3	Cc1cc(C)c2c(O)nc(SCC(=O)N3CCOCC3)nc2n1	nan
	2138011	28171	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3ccccc3c2=O)cc1	nan
	CHEMBL1375055	28171	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3ccccc3c2=O)cc1	nan
	3571741	28176	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	4.6	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1375116	28176	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	4.6	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3)c3cc(Br)ccc3n2)cc1	nan
	16025702	28207	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	5.9	CCOc1ccccc1CNC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1	nan
	CHEMBL1375311	28207	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	5.9	CCOc1ccccc1CNC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1	nan
	2874807	28696	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	7	4.6	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccc(C)cc3c2=O)C2=C(O)CCCC2=N1	nan
	CHEMBL1379763	28696	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	7	4.6	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccc(C)cc3c2=O)C2=C(O)CCCC2=N1	nan
	1564382	28876	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	7	1	7	5.8	CCCCn1c(NC(=O)c2ccc(Br)o2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	CHEMBL1381243	28876	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	7	1	7	5.8	CCCCn1c(NC(=O)c2ccc(Br)o2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	666048	29080	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	9	2.0	c1cncc(-c2nn3c(Cn4nnc5ccccc54)nnc3s2)c1	nan
	CHEMBL1383055	29080	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	9	2.0	c1cncc(-c2nn3c(Cn4nnc5ccccc54)nnc3s2)c1	nan
	220464	29082	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	0	2	2.9	Cn1ccc(=S)c2ccccc21	nan
	CHEMBL1383064	29082	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	0	2	2.9	Cn1ccc(=S)c2ccccc21	nan
	4805097	29095	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	2	0	7	0.4	CC1Cc2ccccc2N1C(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1383239	29095	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	2	0	7	0.4	CC1Cc2ccccc2N1C(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1186390	29316	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	1	0	3	4.7	O=C(Oc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	CHEMBL1385192	29316	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	1	0	3	4.7	O=C(Oc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	4877595	29519	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	5	3.8	O=C(CSc1nnc(-c2ccc(F)cc2)c2ccccc12)NCC1CCCO1	nan
	CHEMBL1386797	29519	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	5	3.8	O=C(CSc1nnc(-c2ccc(F)cc2)c2ccccc12)NCC1CCCO1	nan
	865072	29775	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	4.0	CCOC(=O)CSc1nc(-c2ccccc2)nc2ccccc12	nan
	CHEMBL1388860	29775	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	4.0	CCOC(=O)CSc1nc(-c2ccccc2)nc2ccccc12	nan
	2406693	29798	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	8	2.5	COC(=O)c1sc2nc(C)nc(SCC(=O)N3CCC(C(=O)O)CC3)c2c1C	nan
	CHEMBL1389013	29798	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	8	2.5	COC(=O)c1sc2nc(C)nc(SCC(=O)N3CCC(C(=O)O)CC3)c2c1C	nan
	1261479	29945	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	2	5	3.5	Cc1cc(C)c2nc(-c3ccccn3)cc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c2c1	nan
	CHEMBL1390223	29945	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	2	5	3.5	Cc1cc(C)c2nc(-c3ccccn3)cc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c2c1	nan
	16033258	30393	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1c(C(=O)Nc2ccccc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1394084	30393	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1c(C(=O)Nc2ccccc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16019740	30395	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	8	2.9	CCn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	CHEMBL1394098	30395	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	8	2.9	CCn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	16019075	30423	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	4.4	CC(C)Oc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1394443	30423	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	4.4	CC(C)Oc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	1179391	30584	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(=O)(=O)N4CCCC4)cc3s2)cc1	nan
	CHEMBL1396599	30584	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(=O)(=O)N4CCCC4)cc3s2)cc1	nan
	16031181	30650	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.3	COc1cc(NC(=O)c2cc3cc4cc(OC)ccc4nc3o2)cc(OC)c1	nan
	CHEMBL1397472	30650	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.3	COc1cc(NC(=O)c2cc3cc4cc(OC)ccc4nc3o2)cc(OC)c1	nan
	16028170	30688	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	2	3	4.2	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(Cl)c3)cc21	nan
	CHEMBL1397995	30688	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	2	3	4.2	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(Cl)c3)cc21	nan
	729756	30711	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	1	3	3.9	Cc1ccc(/C=C(\C#N)C(=O)Nc2ccc(Br)cc2)o1	nan
	CHEMBL1398350	30711	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	1	3	3.9	Cc1ccc(/C=C(\C#N)C(=O)Nc2ccc(Br)cc2)o1	nan
	16031340	30718	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	3	4.7	CCc1ccc(CNC(=O)c2cnc(N3CCCCC3)c3ccccc23)cc1	nan
	CHEMBL1398430	30718	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	3	4.7	CCc1ccc(CNC(=O)c2cnc(N3CCCCC3)c3ccccc23)cc1	nan
	15989002	30719	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2cccc(F)c2)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1398440	30719	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2cccc(F)c2)c1=O)NCc1ccc2c(c1)OCO2	nan
	16026774	30722	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	2.2	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3Cl)cc(=O)n12	nan
	CHEMBL1398452	30722	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	2.2	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3Cl)cc(=O)n12	nan
	24790947	31013	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccc(F)cc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1401193	31013	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccc(F)cc4)CC3)ccc2c1)N1CCCCC1	nan
	16017881	31293	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	2.3	CCOc1ccc(NC(=O)Cn2ccn(-c3ccc(F)c(F)c3)c(=O)c2=O)cc1	nan
	CHEMBL1403689	31293	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	2.3	CCOc1ccc(NC(=O)Cn2ccn(-c3ccc(F)c(F)c3)c(=O)c2=O)cc1	nan
	654955	31558	5	None	-4	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	4.7	CS(=O)(=O)c1sc2nc(-c3cccs3)cc(-c3ccccc3)c2c1N	nan
	CHEMBL1406204	31558	5	None	-4	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	4.7	CS(=O)(=O)c1sc2nc(-c3cccs3)cc(-c3ccccc3)c2c1N	nan
	135416200	31560	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	45369539	31560	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	CHEMBL1406220	31560	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	16025790	31610	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	4	4.5	CCC(C)NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1406711	31610	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	4	4.5	CCC(C)NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	1257542	31678	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.4	Cc1cccnc1NC(=O)Cn1nc([N+](=O)[O-])cc1C	nan
	CHEMBL1407331	31678	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.4	Cc1cccnc1NC(=O)Cn1nc([N+](=O)[O-])cc1C	nan
	5834534	31734	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	5	5.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(Cl)cc2)c(C)c1	nan
	CHEMBL1407665	31734	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	5	5.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(Cl)cc2)c(C)c1	nan
	1509257	31755	12	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	2	1	5	3.5	CCN1CCc2nc3sc(C(=O)N4CCc5ccccc5C4)c(N)c3cc2C1	nan
	CHEMBL1407777	31755	12	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	2	1	5	3.5	CCN1CCc2nc3sc(C(=O)N4CCc5ccccc5C4)c(N)c3cc2C1	nan
	981045	31947	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	0	9	-0.1	CCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1409260	31947	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	0	9	-0.1	CCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	2649456	32056	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	2	0	5	2.7	O=c1ccc(C(F)(F)F)cn1Cc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1410109	32056	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	2	0	5	2.7	O=c1ccc(C(F)(F)F)cn1Cc1cc(=O)n2cc(Br)ccc2n1	nan
	1191742	32079	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	4.3	O=C(O)CSc1ncnc2scc(-c3ccc(Br)cc3)c12	nan
	CHEMBL1410306	32079	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	4.3	O=C(O)CSc1ncnc2scc(-c3ccc(Br)cc3)c12	nan
	15990415	32293	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	5	5.5	COc1ccc(Cl)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1412135	32293	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	5	5.5	COc1ccc(Cl)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3151320	32327	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.4	N=c1c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1412407	32327	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.4	N=c1c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	1484210	32332	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	0	5	3.6	CCSc1nnc(-c2ccccc2SC)o1	nan
	CHEMBL1412417	32332	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	0	5	3.6	CCSc1nnc(-c2ccccc2SC)o1	nan
	4433827	32835	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	2.8	CSc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CN(C)CC3	nan
	CHEMBL1416667	32835	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	2.8	CSc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CN(C)CC3	nan
	3245881	33379	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	9	2.6	COc1cc2nc(S)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	CHEMBL1421316	33379	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	9	2.6	COc1cc2nc(S)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	5102370	33674	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	9	1	5	1.7	CCN(CC)S(=O)(=O)c1cccc(C(=O)NCCCn2ccnc2)c1	nan
	CHEMBL1423739	33674	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	9	1	5	1.7	CCN(CC)S(=O)(=O)c1cccc(C(=O)NCCCn2ccnc2)c1	nan
	4872167	33901	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	7	5.2	CCCCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1425797	33901	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	7	5.2	CCCCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	2968003	33956	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	5	3.3	COc1ccc(-c2cc3ccc(OC(C)C(=O)O)cc3oc2=O)cc1	nan
	CHEMBL1426170	33956	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	5	3.3	COc1ccc(-c2cc3ccc(OC(C)C(=O)O)cc3oc2=O)cc1	nan
	5933014	34566	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	10	2	6	2.7	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccccc2)cc1	nan
	CHEMBL1431128	34566	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	10	2	6	2.7	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccccc2)cc1	nan
	2365417	34587	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	1	6	5.2	Cc1ccc2nc(-c3ccc(NC(=O)COC(=O)c4cncc(Br)c4)cc3)sc2c1	nan
	CHEMBL1431340	34587	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	1	6	5.2	Cc1ccc2nc(-c3ccc(NC(=O)COC(=O)c4cncc(Br)c4)cc3)sc2c1	nan
	2317063	34781	8	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	2	5	5.6	CCCCOc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2)cc1	nan
	CHEMBL1433074	34781	8	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	2	5	5.6	CCCCOc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2)cc1	nan
	16016637	34834	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	1	5	5.0	CCOc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2-n2cccc2)cc1	nan
	CHEMBL1433449	34834	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	1	5	5.0	CCOc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2-n2cccc2)cc1	nan
	16012551	34881	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	5	5.5	CCOc1ccc(-c2cc(NC(=O)c3cccc(Cl)c3)c(C(=O)OC)s2)cc1	nan
	CHEMBL1434218	34881	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	5	5.5	CCOc1ccc(-c2cc(NC(=O)c3cccc(Cl)c3)c(C(=O)OC)s2)cc1	nan
	16033555	34930	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	0	4	4.8	Cc1nc(Oc2ccccc2C)c2oc3ccccc3c2n1	nan
	CHEMBL1434916	34930	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	0	4	4.8	Cc1nc(Oc2ccccc2C)c2oc3ccccc3c2n1	nan
	16025666	35053	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	7	4.3	Cc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1	nan
	CHEMBL1436433	35053	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	7	4.3	Cc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1	nan
	16015798	35074	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	4	5.6	Cc1ccc(-c2nc3cc(Cl)ccc3o2)cc1NC(=O)COc1ccc(F)cc1	nan
	CHEMBL1436774	35074	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	4	5.6	Cc1ccc(-c2nc3cc(Cl)ccc3o2)cc1NC(=O)COc1ccc(F)cc1	nan
	16018841	35122	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	4	5.0	Cc1c(C(=O)Nc2ccc(F)cc2F)oc2ccc3c(c12)C(=O)CC(C)(C)O3	nan
	CHEMBL1437356	35122	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	4	5.0	Cc1c(C(=O)Nc2ccc(F)cc2F)oc2ccc3c(c12)C(=O)CC(C)(C)O3	nan
	1004026	35152	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	6	5.2	CCOc1ccccc1NC(=O)c1sc2nc(-c3ccc(OC)cc3)ccc2c1N	nan
	CHEMBL1437726	35152	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	6	5.2	CCOc1ccccc1NC(=O)c1sc2nc(-c3ccc(OC)cc3)ccc2c1N	nan
	16022287	35252	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	1	4	3.3	CCCCNC(=O)c1cccc(-n2c(C)nc3cccnc32)c1	nan
	CHEMBL1438563	35252	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	1	4	3.3	CCCCNC(=O)c1cccc(-n2c(C)nc3cccnc32)c1	nan
	5809896	35313	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	4.0	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1439160	35313	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	4.0	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	15988173	35333	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	4	2.9	Cc1ccc(CNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	CHEMBL1439335	35333	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	4	2.9	Cc1ccc(CNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	1454908	35823	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	1	4	3.5	Sc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1443793	35823	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	1	4	3.5	Sc1nc(COc2ccccc2)nc2ccccc12	nan
	1234247	36066	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	5	2.7	Cc1nnc(S)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1446078	36066	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	5	2.7	Cc1nnc(S)c2nn(-c3ccccc3)c(C)c12	nan
	16026772	36123	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	1.8	Cc1ccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	CHEMBL1446594	36123	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	1.8	Cc1ccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	2957415	36490	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	2.5	CC(=O)c1nc(N2C(=O)C3CC=C(C)CC3C2=O)sc1C	nan
	CHEMBL1449518	36490	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	2.5	CC(=O)c1nc(N2C(=O)C3CC=C(C)CC3C2=O)sc1C	nan
	2334194	36540	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	8	3.6	CCOC(=O)c1c(NS(=O)(=O)c2ccccc2)n(CCCOC)c2nc3ccccc3nc12	nan
	CHEMBL1449923	36540	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	8	3.6	CCOC(=O)c1c(NS(=O)(=O)c2ccccc2)n(CCCOC)c2nc3ccccc3nc12	nan
	4977513	36577	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(OC(C)C)cc2)no1	nan
	CHEMBL1450219	36577	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(OC(C)C)cc2)no1	nan
	2945668	36752	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	1.8	CCc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	CHEMBL1451692	36752	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	1.8	CCc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	24792337	36830	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	7	1.6	Cc1cc2nnc(SCC(=O)NC3CCCCC3)n2c(N)n1	nan
	CHEMBL1452223	36830	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	7	1.6	Cc1cc2nnc(SCC(=O)NC3CCCCC3)n2c(N)n1	nan
	15988498	36870	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	11	2	9	2.9	CCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	CHEMBL1452564	36870	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	11	2	9	2.9	CCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	2298970	36876	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3ccncc3)cc2)c1C	nan
	CHEMBL1452655	36876	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3ccncc3)cc2)c1C	nan
	24790128	37166	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	5	3.2	COc1ccc(-c2[nH]ncc2CN2CCN(C(=O)c3cccs3)CC2)c(F)c1	nan
	CHEMBL1454939	37166	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	5	3.2	COc1ccc(-c2[nH]ncc2CN2CCN(C(=O)c3cccs3)CC2)c(F)c1	nan
	16030361	37226	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	9	1	5	4.7	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)c1	nan
	CHEMBL1455531	37226	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	9	1	5	4.7	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)c1	nan
	16025668	37425	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	8	4.6	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1Cl	nan
	CHEMBL1457411	37425	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	8	4.6	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1Cl	nan
	1355891	37541	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	11	1	7	3.2	COc1ccc(OC)c(N(CC(=O)NCc2ccccc2)S(=O)(=O)c2ccc(OC)c(OC)c2)c1	nan
	CHEMBL1458278	37541	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	11	1	7	3.2	COc1ccc(OC)c(N(CC(=O)NCc2ccccc2)S(=O)(=O)c2ccc(OC)c(OC)c2)c1	nan
	2949787	37639	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.4	COc1ccccc1C1C(C(=O)c2ccco2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1459163	37639	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.4	COc1ccccc1C1C(C(=O)c2ccco2)=C(O)C(=O)N1c1cc(C)on1	nan
	1445336	37643	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	8	3.9	COc1ccccc1N1CCN(C(=O)CSc2ncnc3c2cnn3-c2ccc(C)c(C)c2)CC1	nan
	CHEMBL1459184	37643	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	8	3.9	COc1ccccc1N1CCN(C(=O)CSc2ncnc3c2cnn3-c2ccc(C)c(C)c2)CC1	nan
	6033330	37783	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	11	1	8	3.9	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1460387	37783	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	11	1	8	3.9	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	5160710	37823	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	2	2	4.5	CCCOc1ccc(NC(=O)c2cc3cc(C)ccc3[nH]2)cc1	nan
	CHEMBL1460665	37823	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	2	2	4.5	CCCOc1ccc(NC(=O)c2cc3cc(C)ccc3[nH]2)cc1	nan
	3502512	37908	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	8	1.0	N#Cc1c(N2CCOCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	CHEMBL1461443	37908	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	8	1.0	N#Cc1c(N2CCOCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	2810150	37991	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	4.1	Cc1csc2c(=O)sc(NC(=O)c3ccc(F)cc3Cl)nc12	nan
	CHEMBL1462227	37991	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	4.1	Cc1csc2c(=O)sc(NC(=O)c3ccc(F)cc3Cl)nc12	nan
	4524521	38026	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	7	0.2	Cn1c(C(=O)NCCN2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1462442	38026	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	7	0.2	Cn1c(C(=O)NCCN2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	1491130	38082	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	5	1	5	3.3	O=C(O)COc1ccc(-c2nccc(-c3cccs3)n2)cc1	nan
	CHEMBL1462936	38082	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	5	1	5	3.3	O=C(O)COc1ccc(-c2nccc(-c3cccs3)n2)cc1	nan
	135464100	38194	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	2	6	3.3	N#Cc1c(O)nc(SCC(=O)NC2CCCCC2)nc1-c1ccccc1	nan
	CHEMBL1463888	38194	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	2	6	3.3	N#Cc1c(O)nc(SCC(=O)NC2CCCCC2)nc1-c1ccccc1	nan
	2808819	38445	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	4.1	Cc1csc2ncnc(NC3CCN(Cc4ccccc4)CC3)c12	nan
	CHEMBL1465720	38445	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	4.1	Cc1csc2ncnc(NC3CCN(Cc4ccccc4)CC3)c12	nan
	1100812	38486	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	6	4.4	CCOC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	CHEMBL1466098	38486	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	6	4.4	CCOC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	665758	38506	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	7	4.3	COc1cc(OC)cc(-c2nc(-c3cc4cc(C)ccc4nc3OC)no2)c1	nan
	CHEMBL1466279	38506	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	7	4.3	COc1cc(OC)cc(-c2nc(-c3cc4cc(C)ccc4nc3OC)no2)c1	nan
	20953708	38808	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.2	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)nc(C)n3n2)cc1	nan
	CHEMBL1468743	38808	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.2	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)nc(C)n3n2)cc1	nan
	2913184	38904	15	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	7	3.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	CHEMBL1469528	38904	15	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	7	3.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	1226649	38928	14	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	2	4	4.1	CC(=O)NC(=S)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1	nan
	CHEMBL1469733	38928	14	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	2	4	4.1	CC(=O)NC(=S)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1	nan
	794237	39055	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	5	3.5	COc1ccc(C(=O)Nc2nnc(-c3ccccc3)s2)cc1	nan
	CHEMBL1470825	39055	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	5	3.5	COc1ccc(C(=O)Nc2nnc(-c3ccccc3)s2)cc1	nan
	1025062	39239	9	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	7	1	5	5.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c(C#N)c(C)c1CC(=O)c1ccc(Br)cc1	nan
	CHEMBL1472426	39239	9	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	7	1	5	5.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c(C#N)c(C)c1CC(=O)c1ccc(Br)cc1	nan
	16025800	39360	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	5	3.7	COCCCNC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1474073	39360	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	5	3.7	COCCCNC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	16017955	39377	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	5	3.3	Cc1ccc(NC(=O)c2nc(-c3ccncc3)no2)c(Cl)c1	nan
	CHEMBL1474407	39377	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	5	3.3	Cc1ccc(NC(=O)c2nc(-c3ccncc3)no2)c(Cl)c1	nan
	923699	39558	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	1	4	4.8	Cc1cc(C)cc(C(=O)Nc2ccc(-c3nc4ncccc4o3)cc2)c1	nan
	CHEMBL1476840	39558	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	1	4	4.8	Cc1cc(C)cc(C(=O)Nc2ccc(-c3nc4ncccc4o3)cc2)c1	nan
	16030273	39598	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccccc3F)CC2)cc1	nan
	CHEMBL1477298	39598	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccccc3F)CC2)cc1	nan
	3492613	39846	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	4.6	COc1ccc(-n2cc(-c3ccc(Br)cc3)nc2S)cc1	nan
	CHEMBL1479477	39846	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	4.6	COc1ccc(-n2cc(-c3ccc(Br)cc3)nc2S)cc1	nan
	1077503	39874	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	7	1.9	CCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1479731	39874	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	7	1.9	CCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	2059287	40154	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	5	3.5	CCCCN(CC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1482087	40154	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	5	3.5	CCCCN(CC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	2490618	40173	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	9	0.0	CCc1ccc(OCC(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)cc1	nan
	CHEMBL1482290	40173	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	9	0.0	CCc1ccc(OCC(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)cc1	nan
	16020212	40624	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	7	2	8	3.8	Cc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	CHEMBL1486218	40624	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	7	2	8	3.8	Cc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	5835099	41089	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	1	6	5.0	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1C	nan
	CHEMBL1489865	41089	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	1	6	5.0	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1C	nan
	24791694	41186	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	4	4.0	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cccnc4)C3)ccc2c1	nan
	CHEMBL1490547	41186	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	4	4.0	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cccnc4)C3)ccc2c1	nan
	135438626	41451	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	3	9	0.8	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nc(N)cc(O)n1	nan
	CHEMBL1492401	41451	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	3	9	0.8	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nc(N)cc(O)n1	nan
	16018070	41487	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	4	3.5	O=C(CCCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1	nan
	CHEMBL1492679	41487	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	4	3.5	O=C(CCCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1	nan
	1327115	41577	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	1	5	4.8	COc1cccc(-c2cc3c(=O)n(-c4ccccc4)c(=S)[nH]c3s2)c1	nan
	CHEMBL1493481	41577	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	1	5	4.8	COc1cccc(-c2cc3c(=O)n(-c4ccccc4)c(=S)[nH]c3s2)c1	nan
	3034554	41685	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	7	1.5	Cn1c(=S)c2nc(SCCN3CCCC3)[nH]c2n(C)c1=O	nan
	CHEMBL1494615	41685	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	7	1.5	Cn1c(=S)c2nc(SCCN3CCCC3)[nH]c2n(C)c1=O	nan
	976285	42081	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	0	5	2.1	Cc1csc2nc(=O)c(-c3ccccc3)nn12	nan
	CHEMBL1498297	42081	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	0	5	2.1	Cc1csc2nc(=O)c(-c3ccccc3)nn12	nan
	3127165	42351	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	0.5	CC(C(O)c1ccccc1)N(C)CCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1500612	42351	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	0.5	CC(C(O)c1ccccc1)N(C)CCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	135413586	42431	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	2	10	3.0	CCOC(=O)Cc1csc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)n1	nan
	CHEMBL1501394	42431	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	2	10	3.0	CCOC(=O)Cc1csc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)n1	nan
	5903312	42569	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	8	0.1	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2ccccn2c1=O	nan
	CHEMBL1502541	42569	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	8	0.1	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2ccccn2c1=O	nan
	790333	43003	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1cc(S)c2cccc(C)c2n1	nan
	CHEMBL1506363	43003	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1cc(S)c2cccc(C)c2n1	nan
	2146623	43334	17	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	4	5.0	CC(=O)c1ccc(NC(=O)c2ccc(CSc3ccccc3)o2)cc1	nan
	CHEMBL1509267	43334	17	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	4	5.0	CC(=O)c1ccc(NC(=O)c2ccc(CSc3ccccc3)o2)cc1	nan
	4617873	43647	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	2	3	4.4	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccccc3Br)cc2)cc1	nan
	CHEMBL1512241	43647	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	2	3	4.4	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccccc3Br)cc2)cc1	nan
	7877577	43747	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	7	1.4	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1513627	43747	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	7	1.4	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2ccsc2n1	nan
	7598873	43785	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	3	3.9	CCc1ccccc1NC(=O)c1cccn(Cc2ccccc2F)c1=O	nan
	CHEMBL1514321	43785	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	3	3.9	CCc1ccccc1NC(=O)c1cccn(Cc2ccccc2F)c1=O	nan
	16030561	43798	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	6	0	5	5.5	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1514538	43798	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	6	0	5	5.5	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCN(c2ccccc2F)CC1	nan
	16009347	43801	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cc(C)cc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	CHEMBL1514567	43801	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cc(C)cc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	16018206	43811	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1cc(NC(=O)c2oc3c(c2C)-c2nn(Cc4cccc(Cl)c4)cc2CC3)cc(OC)c1	nan
	CHEMBL1514692	43811	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1cc(NC(=O)c2oc3c(c2C)-c2nn(Cc4cccc(Cl)c4)cc2CC3)cc(OC)c1	nan
	3207800	44059	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2nc(SCC(=O)Nc3cc(C)on3)c(C#N)cc2c1	nan
	CHEMBL1517790	44059	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2nc(SCC(=O)Nc3cc(C)on3)c(C#N)cc2c1	nan
	2091511	44111	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	0	8	2.5	Cc1ccc2nc(CSc3nnc(-c4ccncc4)n3C)cc(=O)n2c1	nan
	CHEMBL1518274	44111	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	0	8	2.5	Cc1ccc2nc(CSc3nnc(-c4ccncc4)n3C)cc(=O)n2c1	nan
	24818303	44113	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	1	3	4.4	CN(C)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	CHEMBL1518303	44113	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	1	3	4.4	CN(C)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	5151092	44116	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	1	2	3.2	CNC(=O)c1c2c(nc3ccc(Br)cc13)CCCC2	nan
	CHEMBL1518360	44116	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	1	2	3.2	CNC(=O)c1c2c(nc3ccc(Br)cc13)CCCC2	nan
	16019804	44280	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	9	1	8	1.6	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCCOC)nnc12	nan
	CHEMBL1519737	44280	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	9	1	8	1.6	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCCOC)nnc12	nan
	4917226	44345	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	2	4	5.8	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(OC2CCCC2)cc1	nan
	CHEMBL1520355	44345	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	2	4	5.8	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(OC2CCCC2)cc1	nan
	24677542	44422	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	8	4	5	3.0	CCCCCNC(=O)c1ccc(NS(=O)(=O)c2ccc3[nH]c(O)nc3c2)cc1	nan
	CHEMBL1520946	44422	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	8	4	5	3.0	CCCCCNC(=O)c1ccc(NS(=O)(=O)c2ccc3[nH]c(O)nc3c2)cc1	nan
	902803	44586	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	5	1	2	4.5	O=C(Nc1ccccc1)c1ccc(COc2ccccc2)cc1	nan
	CHEMBL1522424	44586	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	5	1	2	4.5	O=C(Nc1ccccc1)c1ccc(COc2ccccc2)cc1	nan
	15988611	44793	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	8	3.9	CC(=O)c1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1524392	44793	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	8	3.9	CC(=O)c1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1	nan
	3239863	44952	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	0	8	2.4	CCOC(=O)CC(=O)CSc1ccc2nnc(-c3ccccc3)n2n1	nan
	CHEMBL1525909	44952	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	0	8	2.4	CCOC(=O)CC(=O)CSc1ccc2nnc(-c3ccccc3)n2n1	nan
	2930800	45032	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	7	2.5	COC(=O)c1sc(NC(=O)C2CCCCC2C(=O)O)c(C(=O)OC)c1C	nan
	CHEMBL1526492	45032	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	7	2.5	COC(=O)c1sc(NC(=O)C2CCCCC2C(=O)O)c(C(=O)OC)c1C	nan
	2349018	45213	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	2	1	4	3.4	CCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1528175	45213	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	2	1	4	3.4	CCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	1355435	45227	11	None	-22	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	3.3	Cc1cn(S(=O)(=O)c2ccc(Br)c3ccccc23)cn1	nan
	CHEMBL1528299	45227	11	None	-22	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	3.3	Cc1cn(S(=O)(=O)c2ccc(Br)c3ccccc23)cn1	nan
	5073065	45325	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	6	-0.6	O=C(Cn1cnc2ccccc2c1=O)NCC(=O)N1CCOCC1	nan
	CHEMBL1529152	45325	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	6	-0.6	O=C(Cn1cnc2ccccc2c1=O)NCC(=O)N1CCOCC1	nan
	3240741	45418	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	9	1	8	4.6	COc1ccc(CC(=O)Nc2ccc(-c3noc(-c4cc(OC)c(OC)c(OC)c4)n3)cc2)cc1	nan
	CHEMBL1529936	45418	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	9	1	8	4.6	COc1ccc(CC(=O)Nc2ccc(-c3noc(-c4cc(OC)c(OC)c(OC)c4)n3)cc2)cc1	nan
	3212225	45443	2	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1530244	45443	2	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	16024952	45445	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.0	CCOC(=O)c1cccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)c1	nan
	CHEMBL1530263	45445	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.0	CCOC(=O)c1cccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)c1	nan
	16017576	45456	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	7	2.2	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1530393	45456	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	7	2.2	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	4907979	45464	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	6	3.0	OCCCNc1ncnc2sc3c(c12)CCN(Cc1ccccc1)C3	nan
	CHEMBL1530465	45464	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	6	3.0	OCCCNc1ncnc2sc3c(c12)CCN(Cc1ccccc1)C3	nan
	1161207	45544	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	8	2	7	3.1	COc1ccccc1OCC(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1531098	45544	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	8	2	7	3.1	COc1ccccc1OCC(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	1355556	45607	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	1	3	3.8	O=S(=O)(Nc1cccnc1)c1ccc(Br)c2ccccc12	nan
	CHEMBL1531651	45607	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	1	3	3.8	O=S(=O)(Nc1cccnc1)c1ccc(Br)c2ccccc12	nan
	16025786	45827	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	4	5.3	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)s1	nan
	CHEMBL1533608	45827	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	4	5.3	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)s1	nan
	3151323	45912	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.3	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1534442	45912	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.3	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CC4CCCO4)c3nc12	nan
	3238163	46152	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	8	0.6	Cc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	CHEMBL1536880	46152	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	8	0.6	Cc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	2989967	46234	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	3.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)no1	nan
	CHEMBL1537625	46234	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	3.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)no1	nan
	767265	46489	31	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	5	3.5	Sc1nnc(-c2ccco2)n1-c1ccc(Cl)cc1	nan
	CHEMBL1539766	46489	31	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	5	3.5	Sc1nnc(-c2ccco2)n1-c1ccc(Cl)cc1	nan
	891408	46924	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	4	0	6	1.7	O=C(OCc1cccc([N+](=O)[O-])c1)c1cnccn1	nan
	CHEMBL1543385	46924	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	4	0	6	1.7	O=C(OCc1cccc([N+](=O)[O-])c1)c1cnccn1	nan
	4634206	47016	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	10	-0.9	CCOc1ccccc1OCC(=O)NNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1544116	47016	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	10	-0.9	CCOc1ccccc1OCC(=O)NNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1487485	47020	19	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	3	3.1	Cc1ccc(-n2ncc(Br)c(Br)c2=O)cc1	nan
	CHEMBL1544131	47020	19	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	3	3.1	Cc1ccc(-n2ncc(Br)c(Br)c2=O)cc1	nan
	1867273	47106	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	CHEMBL1544770	47106	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	3781367	47158	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	2	8	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	CHEMBL1545158	47158	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	2	8	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	28358049	47405	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	5398465	47405	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	CHEMBL1547311	47405	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	7080334	47416	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	3.6	Cc1c(-c2cccc(NC(=O)c3ccco3)c2)nc2ncccn12	nan
	CHEMBL1547414	47416	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	3.6	Cc1c(-c2cccc(NC(=O)c3ccco3)c2)nc2ncccn12	nan
	1476696	47443	23	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	0	4	4.8	CSc1cc(-c2ccc(Cl)cc2)n(Cc2ccccc2)c(=O)c1C#N	nan
	CHEMBL1547693	47443	23	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	0	4	4.8	CSc1cc(-c2ccc(Cl)cc2)n(Cc2ccccc2)c(=O)c1C#N	nan
	3830390	47537	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	2	8	-1.2	CN(N)N=Nc1nc2c(=O)n(C)c(=O)n(C)c2[nH]1	nan
	CHEMBL1548599	47537	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	2	8	-1.2	CN(N)N=Nc1nc2c(=O)n(C)c(=O)n(C)c2[nH]1	nan
	20885691	47838	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	7	1	6	1.9	CCc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1551091	47838	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	7	1	6	1.9	CCc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	2053967	47857	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	0	5	4.3	CCCCN(CCCC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1551348	47857	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	0	5	4.3	CCCCN(CCCC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	7151074	47914	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.1	O=C(CSc1nccn1Cc1ccc(Cl)cc1)Nc1ccc2c(c1)OCCO2	nan
	CHEMBL1552167	47914	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.1	O=C(CSc1nccn1Cc1ccc(Cl)cc1)Nc1ccc2c(c1)OCCO2	nan
	16025798	48106	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	4	5.0	O=C(NCc1ccc(F)cc1)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1554965	48106	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	4	5.0	O=C(NCc1ccc(F)cc1)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	16019077	48164	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1555692	48164	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2913061	48270	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	6	3.8	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1556761	48270	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	6	3.8	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	4158621	48316	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(F)cc1Cl	nan
	CHEMBL1557087	48316	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(F)cc1Cl	nan
	2448835	48702	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	9	1.4	CCCn1c(N)c(C(=O)CSc2nc3cc(Cl)c[nH]c-3n2)c(=O)n(C)c1=O	nan
	CHEMBL1560544	48702	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	9	1.4	CCCn1c(N)c(C(=O)CSc2nc3cc(Cl)c[nH]c-3n2)c(=O)n(C)c1=O	nan
	20921616	48749	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	2.6	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccccc3)s2)cc1OC	nan
	CHEMBL1561011	48749	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	2.6	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccccc3)s2)cc1OC	nan
	7190686	48924	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccccc1NC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1562578	48924	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccccc1NC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	3152540	48934	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.0	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1)c1ccco1	nan
	CHEMBL1562668	48934	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.0	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1)c1ccco1	nan
	4367682	49342	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	1	3	2.6	Cc1nc2ccc(Br)cc2c2c1CC(CO)O2	nan
	CHEMBL1566103	49342	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	1	3	2.6	Cc1nc2ccc(Br)cc2c2c1CC(CO)O2	nan
	1569279	49415	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	3.3	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCCN1CCOCC1	nan
	CHEMBL1566690	49415	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	3.3	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCCN1CCOCC1	nan
	7881996	49423	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	1	8	1.2	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1566736	49423	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	1	8	1.2	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	3146574	49488	15	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	8	3.2	COc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1567207	49488	15	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	8	3.2	COc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	1226038	49658	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	3	0	3	5.3	CC(C)c1ccc(-c2cc(C(=O)N3CCOCC3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1568600	49658	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	3	0	3	5.3	CC(C)c1ccc(-c2cc(C(=O)N3CCOCC3)c3cc(Br)ccc3n2)cc1	nan
	20904702	49749	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	8	2.1	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1569451	49749	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	8	2.1	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	16017333	49801	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	7	1.6	COc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCCC3)s2)c1	nan
	CHEMBL1569922	49801	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	7	1.6	COc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCCC3)s2)c1	nan
	1840878	49812	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	2	7	1.8	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NC1CCCCC1	nan
	CHEMBL1570011	49812	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	2	7	1.8	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NC1CCCCC1	nan
	2134950	49929	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3sccc32)c1	nan
	CHEMBL1570886	49929	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3sccc32)c1	nan
	16017067	50257	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.8	CCC(C(=O)NCc1ccccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1574126	50257	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.8	CCC(C(=O)NCc1ccccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	860331	50364	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc2ccccc2nc1SCC(=O)NC1CCCC1	nan
	CHEMBL1575355	50364	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc2ccccc2nc1SCC(=O)NC1CCCC1	nan
	3771682	50454	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	5	5.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(C(C)C)cc2)n1	nan
	CHEMBL1576217	50454	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	5	5.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(C(C)C)cc2)n1	nan
	20957197	50521	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	9	2.0	COc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1576697	50521	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	9	2.0	COc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	5738492	50709	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	7	1	6	3.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc3c(c2)CC(C)O3)C1c1cccnc1	nan
	CHEMBL1578334	50709	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	7	1	6	3.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc3c(c2)CC(C)O3)C1c1cccnc1	nan
	2503775	50762	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	1	5	2.3	O=C(CSc1nnc2ccccn12)NCCc1ccc(F)cc1	nan
	CHEMBL1578723	50762	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	1	5	2.3	O=C(CSc1nnc2ccccn12)NCCc1ccc(F)cc1	nan
	4605879	50784	10	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.3	C=CCSc1nc(O)c2c(n1)OC(N)=C(C#N)C2C(C)C	nan
	CHEMBL1578918	50784	10	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.3	C=CCSc1nc(O)c2c(n1)OC(N)=C(C#N)C2C(C)C	nan
	2366506	50953	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc2c(c1)OCCO2	nan
	CHEMBL1580473	50953	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc2c(c1)OCCO2	nan
	135433335	51166	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	1426566	51166	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	CHEMBL1582229	51166	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	5310097	51187	1	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.7	Cc1ccc(-c2nnc3ccc(SC(C)C(=O)O)nn23)cc1	nan
	CHEMBL1582406	51187	1	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.7	Cc1ccc(-c2nnc3ccc(SC(C)C(=O)O)nn23)cc1	nan
	4099137	51253	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccccc1Cl	nan
	CHEMBL1583052	51253	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccccc1Cl	nan
	661828	51828	14	None	-14	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(OC)c(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1587683	51828	14	None	-14	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(OC)c(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2004544	51963	16	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1F	nan
	CHEMBL1588950	51963	16	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1F	nan
	1003437	52169	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	3	2	5	5.3	Cc1cc(F)ccc1NC(=O)c1sc2nc(-c3cccs3)ccc2c1N	nan
	CHEMBL1591017	52169	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	3	2	5	5.3	Cc1cc(F)ccc1NC(=O)c1sc2nc(-c3cccs3)ccc2c1N	nan
	16019053	52178	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	6	4.0	CCCSCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1591213	52178	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	6	4.0	CCCSCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16015858	52182	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.3	O=C(COc1ccccc1Cl)Nc1ccc2oc(-c3ccccc3F)nc2c1	nan
	CHEMBL1591250	52182	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.3	O=C(COc1ccccc1Cl)Nc1ccc2oc(-c3ccccc3F)nc2c1	nan
	16027414	52240	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	3.6	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1ccccc1	nan
	CHEMBL1591957	52240	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	3.6	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1ccccc1	nan
	16029938	52286	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	6	2.8	Cc1ccn2c(=O)c(NC(=O)c3cccc([N+](=O)[O-])c3C)c(C)nc2c1	nan
	CHEMBL1592574	52286	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	6	2.8	Cc1ccn2c(=O)c(NC(=O)c3cccc([N+](=O)[O-])c3C)c(C)nc2c1	nan
	15990931	52306	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	2	3	6.1	CC(C)c1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1592841	52306	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	2	3	6.1	CC(C)c1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)cc1	nan
	801483	52423	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	2	4	5.2	Oc1cccc(-c2nc(-c3cccs3)c(-c3cccs3)[nH]2)c1	nan
	CHEMBL1594404	52423	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	2	4	5.2	Oc1cccc(-c2nc(-c3cccs3)c(-c3cccs3)[nH]2)c1	nan
	7189836	52617	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	7	3.3	COc1ccc(C(=O)Nc2nc3cc4c(cc3s2)OCO4)c(OC)c1	nan
	CHEMBL1596046	52617	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	7	3.3	COc1ccc(C(=O)Nc2nc3cc4c(cc3s2)OCO4)c(OC)c1	nan
	4137685	52663	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	5.8	COc1cccc(C(=O)c2sc3nc(-c4ccccc4)cc(C(F)(F)F)c3c2N)c1	nan
	CHEMBL1596431	52663	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	5.8	COc1cccc(C(=O)c2sc3nc(-c4ccccc4)cc(C(F)(F)F)c3c2N)c1	nan
	3916490	52786	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.7	CCN(CC)S(=O)(=O)c1cccc(NC(=O)COc2ncnc3sccc23)c1	nan
	CHEMBL1597614	52786	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.7	CCN(CC)S(=O)(=O)c1cccc(NC(=O)COc2ncnc3sccc23)c1	nan
	16195124	52980	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	2.4	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC)cc2)C12C(=O)N(C)c1ccccc12	nan
	CHEMBL1599313	52980	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	2.4	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC)cc2)C12C(=O)N(C)c1ccccc12	nan
	135419123	53121	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	1	3	5.5	Cc1ccc(C2=Nc3ccccc3N=C(c3ccc(F)cc3)C2)c(O)c1	nan
	CHEMBL1600651	53121	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	1	3	5.5	Cc1ccc(C2=Nc3ccccc3N=C(c3ccc(F)cc3)C2)c(O)c1	nan
	16018987	53132	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	3.7	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1OC	nan
	CHEMBL1600729	53132	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	3.7	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1OC	nan
	16009272	53380	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	3.2	COc1ccc(CNC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)cc1	nan
	CHEMBL1603189	53380	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	3.2	COc1ccc(CNC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)cc1	nan
	2816428	53497	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	2	0	5	2.8	C=CCn1c2ccccc2c2nn(C)c(=S)nc21	nan
	CHEMBL1604034	53497	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	2	0	5	2.8	C=CCn1c2ccccc2c2nn(C)c(=S)nc21	nan
	3765596	53669	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1605561	53669	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	4524651	54159	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	5	2.5	CC1CCCCC1NC(=O)c1cc2c(=O)n3ccccc3nc2n1C	nan
	CHEMBL1609461	54159	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	5	2.5	CC1CCCCC1NC(=O)c1cc2c(=O)n3ccccc3nc2n1C	nan
	901441	54170	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	1	1	3	3.3	Cc1cc2sc(C(=O)O)c(C)c2s1	nan
	CHEMBL1609556	54170	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	1	1	3	3.3	Cc1cc2sc(C(=O)O)c(C)c2s1	nan
	6498451	54251	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	9	1.8	COc1cc2c3nc4n(c(=O)c3n(CC(=O)NCC3CCCO3)c2cc1OC)CCS4	nan
	CHEMBL1610295	54251	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	9	1.8	COc1cc2c3nc4n(c(=O)c3n(CC(=O)NCC3CCCO3)c2cc1OC)CCS4	nan
	16022543	54309	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	2	8	4.1	CCN(CC)CCNC(=O)c1ccc2c(=O)n3nc(Nc4cccc(Cl)c4C)sc3nc2c1	nan
	CHEMBL1610849	54309	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	2	8	4.1	CCN(CC)CCNC(=O)c1ccc2c(=O)n3nc(Nc4cccc(Cl)c4C)sc3nc2c1	nan
	16013346	54432	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	1	5	4.2	Cc1cc2oc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCCC4)cc3)cc(=O)c2cc1C	nan
	CHEMBL1611855	54432	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	1	5	4.2	Cc1cc2oc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCCC4)cc3)cc(=O)c2cc1C	nan
	2816611	54496	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	2	7	2.8	CCOC(=O)N1CCc2c(sc3nc(S)nc(S)c23)C1	nan
	CHEMBL1612443	54496	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	2	7	2.8	CCOC(=O)N1CCc2c(sc3nc(S)nc(S)c23)C1	nan
	2967714	54530	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	4.5	COc1ccc(C(=O)Nc2ccc(C(=O)Nc3cccc(C)c3)cc2)cc1	nan
	CHEMBL1612735	54530	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	4.5	COc1ccc(C(=O)Nc2ccc(C(=O)Nc3cccc(C)c3)cc2)cc1	nan
	16019073	54568	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	1	6	4.1	CCOc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1613149	54568	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	1	6	4.1	CCOc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	4723782	54969	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	CHEMBL1342613	54969	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	CHEMBL1618192	54969	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	20279	55055	95	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	CHEMBL1619	55055	95	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	1712157	55279	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	CHEMBL1455081	55279	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	CHEMBL1620984	55279	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	616262	55417	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	CHEMBL1505364	55417	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	CHEMBL1622190	55417	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	1554378	55849	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1577432	55849	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1625977	55849	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	3098134	71729	5	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.6	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\c1cccc(O)c1	nan
	CHEMBL1977502	71729	5	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.6	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\c1cccc(O)c1	nan
	9687993	107304	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	6	2.7	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1cccc([N+](=O)[O-])c1	nan
	CHEMBL3191955	107304	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	6	2.7	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1cccc([N+](=O)[O-])c1	nan
	3095208	107493	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	4	2.6	O=C1C=C(Nc2ccccc2C(=O)O)c2ccccc2C1=O	nan
	CHEMBL3194086	107493	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	4	2.6	O=C1C=C(Nc2ccccc2C(=O)O)c2ccccc2C1=O	nan
	9638310	107673	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	6	1.5	C/C(=N\NC(=O)c1cnccn1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3196238	107673	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	6	1.5	C/C(=N\NC(=O)c1cnccn1)c1ccc([N+](=O)[O-])cc1	nan
	102175	140728	66	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	4	9	-1.5	CNc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	nan
	CHEMBL383144	140728	66	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	4	9	-1.5	CNc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	nan
	6083	203097	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	CHEMBL1315633	203097	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	CHEMBL752	203097	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	4324298	28400	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	0.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccc(=O)n(C)n2)c1	nan
	CHEMBL1377104	28400	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	0.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccc(=O)n(C)n2)c1	nan
	15988970	43792	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	3	6.2	CCc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	CHEMBL1514445	43792	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	3	6.2	CCc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	15988960	48245	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	3	5.5	CC(C)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1556439	48245	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	3	5.5	CC(C)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	3119935	52410	19	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	2	6	3.7	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1594298	52410	19	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	2	6	3.7	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	735254	10344	77	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	178	1	1	3	2.4	S=c1[nH]nc(-c2ccccc2)o1	nan
	CHEMBL1164316	10344	77	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	178	1	1	3	2.4	S=c1[nH]nc(-c2ccccc2)o1	nan
	5904441	11231	12	None	-6	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	3.1	N#C/C(=C\c1ccc([N+](=O)[O-])o1)c1nc2ccccc2[nH]1	nan
	CHEMBL117966	11231	12	None	-6	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	3.1	N#C/C(=C\c1ccc([N+](=O)[O-])o1)c1nc2ccccc2[nH]1	nan
	1004068	18163	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)cc1	nan
	CHEMBL1271076	18163	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)cc1	nan
	3626929	19327	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.7	CC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCCCC3)c3ccccc23)cc1	nan
	CHEMBL1299573	19327	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.7	CC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCCCC3)c3ccccc23)cc1	nan
	5852174	19417	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	4.0	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1300425	19417	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	4.0	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	15988009	19496	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1300978	19496	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	3688325	19587	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	6	2.9	CC(=O)Nc1cccc(C2=CC(c3ccco3)n3ncnc3N2)c1	nan
	CHEMBL1301688	19587	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	6	2.9	CC(=O)Nc1cccc(C2=CC(c3ccco3)n3ncnc3N2)c1	nan
	20957233	19627	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	2.3	CC(CNC(=O)CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)c1ccccc1	nan
	CHEMBL1302111	19627	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	2.3	CC(CNC(=O)CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)c1ccccc1	nan
	17584169	19740	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	5	3.3	O=C(COc1cc2oc(=O)c3c(c2cc1Cl)CCC3)Nc1ccccn1	nan
	CHEMBL1302915	19740	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	5	3.3	O=C(COc1cc2oc(=O)c3c(c2cc1Cl)CCC3)Nc1ccccn1	nan
	852288	19903	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	5	0.9	Cn1c(C(=O)O)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1304220	19903	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	5	0.9	Cn1c(C(=O)O)cc2c(=O)n3ccccc3nc21	nan
	4145244	19912	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	0.6	Cn1cnnc1SCC(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1304271	19912	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	0.6	Cn1cnnc1SCC(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	2429052	20012	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	5	5.8	O=C(COC(=O)CSc1cccc2cccc(Cl)c12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	CHEMBL1305188	20012	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	5	5.8	O=C(COC(=O)CSc1cccc2cccc(Cl)c12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	353380	20182	2	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	2	2	2	5.7	O=C(Nc1ccc(Br)c2ccccc12)c1ccc2ccccc2c1O	nan
	CHEMBL1306524	20182	2	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	2	2	2	5.7	O=C(Nc1ccc(Br)c2ccccc12)c1ccc2ccccc2c1O	nan
	4300736	20310	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	3	2	7	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4c(c3)OCCO4)sc2c1	nan
	CHEMBL1307550	20310	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	3	2	7	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4c(c3)OCCO4)sc2c1	nan
	16194293	20342	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	1	8	3.4	CCc1nnc(NC(=O)CSc2ccc(-c3cccs3)nn2)s1	nan
	CHEMBL1307806	20342	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	1	8	3.4	CCc1nnc(NC(=O)CSc2ccc(-c3cccs3)nn2)s1	nan
	24819826	20367	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	6	2	3	4.1	O=C(NCCCSc1ccccc1)c1cc(Br)ccc1O	nan
	CHEMBL1307980	20367	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	6	2	3	4.1	O=C(NCCCSc1ccccc1)c1cc(Br)ccc1O	nan
	713805	20423	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	0	9	0.6	COc1nc(N2CCCC2)nc(-n2nnc(C(C)=O)c2C)n1	nan
	CHEMBL1308437	20423	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	0	9	0.6	COc1nc(N2CCCC2)nc(-n2nnc(C(C)=O)c2C)n1	nan
	935829	20441	17	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	0	4	3.3	Cc1nc2ccccc2nc1SCC(=O)N1CCC(C)CC1	nan
	CHEMBL1308605	20441	17	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	0	4	3.3	Cc1nc2ccccc2nc1SCC(=O)N1CCC(C)CC1	nan
	2815890	20486	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	5	10	-1.9	CNc1nc2c(N)ncnc2n1[C@H]1O[C@@H](CO)[C@H](O)[C@@H]1O	nan
	CHEMBL1308946	20486	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	5	10	-1.9	CNc1nc2c(N)ncnc2n1[C@H]1O[C@@H](CO)[C@H](O)[C@@H]1O	nan
	4619601	20493	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	0	7	2.2	CCN(C(=O)CSC1=Nc2ccccc2C2CC=NN12)C1CCS(=O)(=O)C1	nan
	CHEMBL1309010	20493	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	0	7	2.2	CCN(C(=O)CSC1=Nc2ccccc2C2CC=NN12)C1CCS(=O)(=O)C1	nan
	4038913	20586	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.9	CCN(C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12)C1CCS(=O)(=O)C1	nan
	CHEMBL1309767	20586	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.9	CCN(C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12)C1CCS(=O)(=O)C1	nan
	20923170	20683	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1C	nan
	CHEMBL1310648	20683	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1C	nan
	3163618	20720	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.6	Cc1ccc(NC(=O)CSc2nnc(-c3ccncc3)s2)cc1	nan
	CHEMBL1310953	20720	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.6	Cc1ccc(NC(=O)CSc2nnc(-c3ccncc3)s2)cc1	nan
	1504615	20769	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	6	2.0	Cc1cc(CNC(=O)Cn2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	CHEMBL1311384	20769	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	6	2.0	Cc1cc(CNC(=O)Cn2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	652682	20828	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	8	1	6	4.3	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1311808	20828	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	8	1	6	4.3	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	24892134	20845	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	2.7	Cn1c(=O)c2c(SCC(=O)Nc3ccccc3F)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1311956	20845	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	2.7	Cn1c(=O)c2c(SCC(=O)Nc3ccccc3F)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	2769005	21018	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	4	0	7	1.1	CCOC(=O)CSc1nc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1313156	21018	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	4	0	7	1.1	CCOC(=O)CSc1nc(=O)n2cc(C)ccc2n1	nan
	20914264	21021	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.9	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)cc1	nan
	CHEMBL1313185	21021	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.9	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)cc1	nan
	4002385	21044	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	662194	21044	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1313374	21044	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	16033288	21169	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	5.3	Cc1ccc(C)c(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	CHEMBL1314411	21169	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	5.3	Cc1ccc(C)c(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	1046209	21237	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	2	1	8	2.8	Cn1c(=O)c2c(nc3n(-c4ccc(O)cc4)c(-c4ccc(Br)cc4)cn23)n(C)c1=O	nan
	CHEMBL1315398	21237	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	2	1	8	2.8	Cn1c(=O)c2c(nc3n(-c4ccc(O)cc4)c(-c4ccc(Br)cc4)cn23)n(C)c1=O	nan
	16014663	21248	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	6	3.8	COc1ccc(-c2nsc(NC(=O)COc3ccc(C)c(C)c3)n2)cc1	nan
	CHEMBL1315498	21248	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	6	3.8	COc1ccc(-c2nsc(NC(=O)COc3ccc(C)c(C)c3)n2)cc1	nan
	16017636	21296	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	5	2	8	4.3	COc1ccc(NC(=O)c2sc3nc(-c4cc5ccc(OC)cc5oc4=O)[nH]c(=O)c3c2C)cc1	nan
	CHEMBL1316057	21296	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	5	2	8	4.3	COc1ccc(NC(=O)c2sc3nc(-c4cc5ccc(OC)cc5oc4=O)[nH]c(=O)c3c2C)cc1	nan
	16018724	21302	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	7	4.2	COc1ccc(Cl)cc1NC(=O)CSc1nnc(C)n2c1cc1occc12	nan
	CHEMBL1316127	21302	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	7	4.2	COc1ccc(Cl)cc1NC(=O)CSc1nnc(C)n2c1cc1occc12	nan
	16009825	21355	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc(OC)c1	nan
	CHEMBL1316937	21355	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc(OC)c1	nan
	24980344	21358	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	5	3.0	Cc1ccc(C(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	CHEMBL1316966	21358	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	5	3.0	Cc1ccc(C(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	7159295	21377	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	6	1	9	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccccc2)c1=O	nan
	CHEMBL1317213	21377	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	6	1	9	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccccc2)c1=O	nan
	17757011	21382	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	2	1	4	5.3	O=C1COc2ccc(-c3cc(-c4ccccc4)c4c(n3)-c3ccccc3OC4)cc2N1	nan
	CHEMBL1317304	21382	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	2	1	4	5.3	O=C1COc2ccc(-c3cc(-c4ccccc4)c4c(n3)-c3ccccc3OC4)cc2N1	nan
	1215486	21383	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	5.6	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1317307	21383	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	5.6	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(F)cc1	nan
	4318326	21536	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	1	6	3.1	COc1ccc2nc(C)cc(SCC(NC(C)=O)C(=O)OC(C)C)c2c1	nan
	CHEMBL1318910	21536	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	1	6	3.1	COc1ccc2nc(C)cc(SCC(NC(C)=O)C(=O)OC(C)C)c2c1	nan
	621902	21540	10	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	5	0	5	3.5	CCSc1cnn(-c2ccccc2)c(=O)c1SCC	nan
	CHEMBL1318957	21540	10	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	5	0	5	3.5	CCSc1cnn(-c2ccccc2)c(=O)c1SCC	nan
	3152777	21666	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3cccc(O)c3)sc2c1	nan
	CHEMBL1320029	21666	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3cccc(O)c3)sc2c1	nan
	15990516	21786	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.1	COc1ccc2nc3sc(C(=O)NCCc4ccc(Cl)cc4)cc3cc2c1	nan
	CHEMBL1321040	21786	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.1	COc1ccc2nc3sc(C(=O)NCCc4ccc(Cl)cc4)cc3cc2c1	nan
	2158383	22015	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1323129	22015	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	864393	22075	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.1	Cc1cc(SCC(=O)NC2CCCCC2)nc2ccccc12	nan
	CHEMBL1323679	22075	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.1	Cc1cc(SCC(=O)NC2CCCCC2)nc2ccccc12	nan
	2138908	22103	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	5.0	CCOC(=O)c1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1323878	22103	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	5.0	CCOC(=O)c1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	716947	22158	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	3.9	CCOc1ccc(-c2oc3ccc(C)cc3c(=O)c2O)cc1	nan
	CHEMBL1324368	22158	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	3.9	CCOc1ccc(-c2oc3ccc(C)cc3c(=O)c2O)cc1	nan
	2929091	22167	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.2	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCC1	nan
	CHEMBL1324435	22167	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.2	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCC1	nan
	16017079	22189	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	4	1	5	6.2	CCC(C(=O)Nc1cc(C(F)(F)F)ccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1324580	22189	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	4	1	5	6.2	CCC(C(=O)Nc1cc(C(F)(F)F)ccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	6619868	22222	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	2	5	3.4	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc3c(c2)N(Cc2ccccc2)CCS3)cc1	nan
	CHEMBL1324841	22222	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	2	5	3.4	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc3c(c2)N(Cc2ccccc2)CCS3)cc1	nan
	135415532	22296	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	7	2.6	Cc1cc(O)nc(SCc2nc3ncccn3c2Br)n1	nan
	CHEMBL1325556	22296	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	7	2.6	Cc1cc(O)nc(SCc2nc3ncccn3c2Br)n1	nan
	1086445	22419	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	6	3.7	COc1ccc(-c2ccc3c(N)c(C(=O)NC(C)C)sc3n2)cc1OC	nan
	CHEMBL1326816	22419	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	6	3.7	COc1ccc(-c2ccc3c(N)c(C(=O)NC(C)C)sc3n2)cc1OC	nan
	5739163	22477	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1327274	22477	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCO2	nan
	2128134	22500	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	0	5	2.3	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cccnc2Cl)c1	nan
	CHEMBL1327541	22500	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	0	5	2.3	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cccnc2Cl)c1	nan
	5899385	22557	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	1	7	3.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3cccnc3)ccc2O1	nan
	CHEMBL1327895	22557	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	1	7	3.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3cccnc3)ccc2O1	nan
	3464558	22591	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	5	3.3	COc1ccc(S(=O)(=O)N2CCN(CC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1	nan
	CHEMBL1328124	22591	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	5	3.3	COc1ccc(S(=O)(=O)N2CCN(CC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1	nan
	1779937	22756	11	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	1	4	4.3	COc1ccc2sc3c(O)nc4ccccc4c3c2c1	nan
	CHEMBL1329604	22756	11	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	1	4	4.3	COc1ccc2sc3c(O)nc4ccccc4c3c2c1	nan
	16013718	22878	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	3.7	CCc1nonc1NC(=O)c1oc2ccc(Br)cc2c1C	nan
	CHEMBL1330644	22878	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	3.7	CCc1nonc1NC(=O)c1oc2ccc(Br)cc2c1C	nan
	2991043	23084	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	0.4	Cn1c(=O)c2c(nc(CN3CCc4ccccc4C3)n2CCCO)n(C)c1=O	nan
	CHEMBL1332170	23084	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	0.4	Cn1c(=O)c2c(nc(CN3CCc4ccccc4C3)n2CCCO)n(C)c1=O	nan
	1861856	23157	13	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	2	6	2.5	COc1cc2[nH]c(=S)n(NC(=O)c3ccccc3)c(=O)c2cc1OC	nan
	CHEMBL1332727	23157	13	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	2	6	2.5	COc1cc2[nH]c(=S)n(NC(=O)c3ccccc3)c(=O)c2cc1OC	nan
	5302228	23527	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	0	6	3.3	COc1ccc(N(C)S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccc(Cl)cn23)cc1	nan
	CHEMBL1335569	23527	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	0	6	3.3	COc1ccc(N(C)S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccc(Cl)cn23)cc1	nan
	16018981	23606	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	4.3	O=C(NCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1336206	23606	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	4.3	O=C(NCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2807849	23628	64	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	2	1	3	3.2	CC(=O)c1sc(-c2ccccc2)cc1N	nan
	CHEMBL1336437	23628	64	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	2	1	3	3.2	CC(=O)c1sc(-c2ccccc2)cc1N	nan
	2222525	23648	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	7	3.0	CC(=O)c1sc2nc(SCC(=O)N3CCCCC3)nc(O)c2c1C	nan
	CHEMBL1336564	23648	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	7	3.0	CC(=O)c1sc2nc(SCC(=O)N3CCCCC3)nc(O)c2c1C	nan
	2844395	23707	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	4	2	3	1.3	CC(C)NC(=O)CC(=O)NN=C1CCCCC1	nan
	CHEMBL1337153	23707	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	4	2	3	1.3	CC(C)NC(=O)CC(=O)NN=C1CCCCC1	nan
	1480701	23819	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	2.0	COC(=O)c1nc2ccc(N3CCOCC3)cc2c(C)c1C(=O)OC	nan
	CHEMBL1338156	23819	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	2.0	COC(=O)c1nc2ccc(N3CCOCC3)cc2c(C)c1C(=O)OC	nan
	861738	23857	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc(SCC(=O)NC2CCCC2)nc2ccccc12	nan
	CHEMBL1338383	23857	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc(SCC(=O)NC2CCCC2)nc2ccccc12	nan
	4677074	24223	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	1	3	2.8	Sc1nc2ccccc2n2cccc12	nan
	CHEMBL1341748	24223	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	1	3	2.8	Sc1nc2ccccc2n2cccc12	nan
	2334933	24293	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	4	3.5	O=C(COC(=O)CSc1ccc2ccccc2c1Br)NC1CC1	nan
	CHEMBL1342297	24293	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	4	3.5	O=C(COC(=O)CSc1ccc2ccccc2c1Br)NC1CC1	nan
	650550	24358	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	0	6	3.4	COc1ccc(-c2nsc3c(N4CCCC4)ncnc23)cc1	nan
	CHEMBL1342739	24358	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	0	6	3.4	COc1ccc(-c2nsc3c(N4CCCC4)ncnc23)cc1	nan
	16445815	24519	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	CHEMBL1344160	24519	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	7190688	24545	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1344377	24545	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	3106500	24570	8	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	7	1.5	CC1=NN(C(N)=S)C(=O)C1N=Nc1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1344603	24570	8	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	7	1.5	CC1=NN(C(N)=S)C(=O)C1N=Nc1ccc([N+](=O)[O-])cc1	nan
	20907339	24629	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	5	2.6	CCOCCCNC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	CHEMBL1345074	24629	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	5	2.6	CCOCCCNC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	6103434	24769	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	7	3.7	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1346374	24769	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	7	3.7	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	2122298	24904	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	1	5	2.7	CC(=O)c1sc(NC(=O)COc2ccccc2)nc1C	nan
	CHEMBL1347404	24904	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	1	5	2.7	CC(=O)c1sc(NC(=O)COc2ccccc2)nc1C	nan
	899068	24952	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	1	6	3.6	CSc1nc(S)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1347767	24952	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	1	6	3.6	CSc1nc(S)c2c3c(sc2n1)COC(C)(C)C3	nan
	1481616	25018	18	None	-15	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	0	4	4.3	COc1cccc(CSc2nc3ccccc3cc2C=O)c1	nan
	CHEMBL1348389	25018	18	None	-15	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	0	4	4.3	COc1cccc(CSc2nc3ccccc3cc2C=O)c1	nan
	1378026	25038	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.2	COc1ccc(NC(=O)c2ccc(C(=O)c3cc(OC)ccc3OC)cc2)cc1	nan
	CHEMBL1348606	25038	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.2	COc1ccc(NC(=O)c2ccc(C(=O)c3cc(OC)ccc3OC)cc2)cc1	nan
	2205361	25041	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	4	3	9	2.3	COC(=O)c1sc(N=C(S)NNC(=O)c2c(Br)c(C)nn2C)c(C(=O)OC)c1C	nan
	CHEMBL1348642	25041	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	4	3	9	2.3	COC(=O)c1sc(N=C(S)NNC(=O)c2c(Br)c(C)nn2C)c(C(=O)OC)c1C	nan
	2084877	25055	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	1	5	3.8	COCCNC(=O)CSc1cc(-c2ccccc2)c2ccc(OC)cc2n1	nan
	CHEMBL1348812	25055	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	1	5	3.8	COCCNC(=O)CSc1cc(-c2ccccc2)c2ccc(OC)cc2n1	nan
	1256964	25061	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	1	4	5.1	O=C(NCc1cccs1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	CHEMBL1348841	25061	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	1	4	5.1	O=C(NCc1cccs1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	3783556	25141	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.0	C=CCN1C(=O)NC(=O)/C(=C\Nc2c(C)n(C)n(-c3ccccc3)c2=O)C1=O	nan
	CHEMBL1349443	25141	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.0	C=CCN1C(=O)NC(=O)/C(=C\Nc2c(C)n(C)n(-c3ccccc3)c2=O)C1=O	nan
	24746879	25154	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.5	COC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1349543	25154	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.5	COC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	4831863	25234	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	0.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)Cn1nnc2ccccc2c1=O	nan
	CHEMBL1350232	25234	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	0.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)Cn1nnc2ccccc2c1=O	nan
	663661	25270	16	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	5	4.5	c1ccc2[nH]c(CSc3ncnc4c3oc3ccccc34)nc2c1	nan
	CHEMBL1350581	25270	16	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	5	4.5	c1ccc2[nH]c(CSc3ncnc4c3oc3ccccc34)nc2c1	nan
	2881707	25399	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	3.2	Cc1nnc(Nc2ccc(C(=O)N3CCOCC3)cc2)c2ccccc12	nan
	CHEMBL1351647	25399	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	3.2	Cc1nnc(Nc2ccc(C(=O)N3CCOCC3)cc2)c2ccccc12	nan
	5308898	25416	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	1	3	2.4	CCc1cc(=O)oc2cc(C)cc(O)c12	nan
	CHEMBL1351746	25416	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	1	3	2.4	CCc1cc(=O)oc2cc(C)cc(O)c12	nan
	2802516	25471	41	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.2	Sc1nc(-c2ccccc2)n(-c2ccccc2)n1	nan
	CHEMBL1352266	25471	41	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.2	Sc1nc(-c2ccccc2)n(-c2ccccc2)n1	nan
	1435022	25561	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	6	4.3	CCc1nc(SCC(=O)Nc2nc3c(s2)CCCC3)c2ccccc2n1	nan
	CHEMBL1352936	25561	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	6	4.3	CCc1nc(SCC(=O)Nc2nc3c(s2)CCCC3)c2ccccc2n1	nan
	7285290	25595	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	2	3.5	Cc1nc(-c2ccc(Br)cc2)ccc1C(=O)O	nan
	CHEMBL1353200	25595	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	2	3.5	Cc1nc(-c2ccc(Br)cc2)ccc1C(=O)O	nan
	15989677	25757	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc(OC)c1	nan
	CHEMBL1354335	25757	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc(OC)c1	nan
	16030401	25793	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	8	1	4	5.0	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)cc1	nan
	CHEMBL1354835	25793	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	8	1	4	5.0	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)cc1	nan
	16010860	25796	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	2.8	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1	nan
	CHEMBL1354858	25796	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	2.8	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1	nan
	15988167	25859	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.9	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3ccccc32)c1	nan
	CHEMBL1355668	25859	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.9	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3ccccc32)c1	nan
	16024817	25959	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1356900	25959	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	1165987	26065	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	6	4.0	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCC(C)C)n2)cc1OC	nan
	CHEMBL1358322	26065	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	6	4.0	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCC(C)C)n2)cc1OC	nan
	1003453	26080	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	2	5	5.6	Nc1c(C(=O)Nc2ccccc2Br)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1358598	26080	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	2	5	5.6	Nc1c(C(=O)Nc2ccccc2Br)sc2nc(-c3cccs3)ccc12	nan
	663400	26127	13	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.8	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(Cl)c1	nan
	CHEMBL1359009	26127	13	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.8	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(Cl)c1	nan
	5104589	26208	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	3	6.6	O=C(Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1)c1ccc2ccccc2c1	nan
	CHEMBL1359625	26208	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	3	6.6	O=C(Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1)c1ccc2ccccc2c1	nan
	4438847	26335	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	1.1	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1cccc[n+]1[O-]	nan
	CHEMBL1360781	26335	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	1.1	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1cccc[n+]1[O-]	nan
	15989315	26337	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	10	1	7	4.6	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4ccccc4n(Cc4cccc(C)c4)c3=O)cc2)cc1OC	nan
	CHEMBL1360796	26337	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	10	1	7	4.6	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4ccccc4n(Cc4cccc(C)c4)c3=O)cc2)cc1OC	nan
	15991495	26373	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	3	5	3.9	O=C(O)Cc1sc(Nc2ccc(C(=O)O)cc2)nc1-c1ccccc1	nan
	CHEMBL1361126	26373	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	3	5	3.9	O=C(O)Cc1sc(Nc2ccc(C(=O)O)cc2)nc1-c1ccccc1	nan
	2816171	26421	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	8	1.3	CCOC(=O)c1nnn2c1nc(N1CCOCC1)c1ccccc12	nan
	CHEMBL1361598	26421	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	8	1.3	CCOC(=O)c1nnn2c1nc(N1CCOCC1)c1ccccc12	nan
	6238059	26492	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	2	6	2.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1362160	26492	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	2	6	2.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccc(F)cc2)cc1	nan
	15988824	26508	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	7	4.2	COc1ccc(-c2cc(C(=O)Nc3ccn(Cc4ccc(C)cc4)n3)no2)cc1OC	nan
	CHEMBL1362337	26508	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	7	4.2	COc1ccc(-c2cc(C(=O)Nc3ccn(Cc4ccc(C)cc4)n3)no2)cc1OC	nan
	6625370	26826	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	7	2.2	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(F)c3)sc2n1	nan
	CHEMBL1365096	26826	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	7	2.2	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(F)c3)sc2n1	nan
	1315619	26859	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	3	5	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1C(=O)NCc1ccco1)c1ccco1	nan
	CHEMBL1365331	26859	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	3	5	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1C(=O)NCc1ccco1)c1ccco1	nan
	2138525	26878	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	7	4.6	Cc1ccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)cc1	nan
	CHEMBL1365483	26878	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	7	4.6	Cc1ccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)cc1	nan
	5068934	26927	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	3	3.0	O=C(CCS(=O)(=O)Cc1cccc(Cl)c1)NCCc1ccccc1	nan
	CHEMBL1365953	26927	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	3	3.0	O=C(CCS(=O)(=O)Cc1cccc(Cl)c1)NCCc1ccccc1	nan
	7190319	26929	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	3	0	6	3.0	CCSc1ccc2nnc(-c3cccs3)n2n1	nan
	CHEMBL1365969	26929	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	3	0	6	3.0	CCSc1ccc2nnc(-c3cccs3)n2n1	nan
	16194607	27107	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	10	1	7	1.7	CCN(CC)CCCNC(=O)Cn1cnc2ccc(S(=O)(=O)N3CCC(C)CC3)cc2c1=O	nan
	CHEMBL1367480	27107	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	10	1	7	1.7	CCN(CC)CCCNC(=O)Cn1cnc2ccc(S(=O)(=O)N3CCC(C)CC3)cc2c1=O	nan
	16033554	27238	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	4	1.7	CC(=O)Nc1ccc(NC(=O)CN2C(=O)CN(C)C(=O)c3ccccc32)cc1	nan
	CHEMBL1368494	27238	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	4	1.7	CC(=O)Nc1ccc(NC(=O)CN2C(=O)CN(C)C(=O)c3ccccc32)cc1	nan
	16009410	27329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	5.2	CCC(CC)c1nn2c(=O)cc(COc3ccc(NC(=O)c4ccccc4C)cc3)nc2s1	nan
	CHEMBL1369161	27329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	5.2	CCC(CC)c1nn2c(=O)cc(COc3ccc(NC(=O)c4ccccc4C)cc3)nc2s1	nan
	20880788	27488	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	3.4	CC1CCCC(C)N1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	CHEMBL1370306	27488	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	3.4	CC1CCCC(C)N1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	2622707	27558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	0	6	2.9	O=[N+]([O-])c1cccc(CSc2nnc3ccccn23)c1	nan
	CHEMBL1370729	27558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	0	6	2.9	O=[N+]([O-])c1cccc(CSc2nnc3ccccn23)c1	nan
	3178485	27611	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCn1c(SCC(=O)N2CCCCC2C)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1371157	27611	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCn1c(SCC(=O)N2CCCCC2C)nc2c1c(=O)n(C)c(=O)n2C	nan
	2155682	27801	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	4	0	5	3.1	CC1CCN(C(=O)CSc2nnc(-c3ccccc3)o2)CC1	nan
	CHEMBL1372587	27801	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	4	0	5	3.1	CC1CCN(C(=O)CSc2nnc(-c3ccccc3)o2)CC1	nan
	2965534	27823	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	5	5.1	CCOc1ccc(-c2cc(C(=O)NCCCn3ccnc3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1372738	27823	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	5	5.1	CCOc1ccc(-c2cc(C(=O)NCCCn3ccnc3)c3cc(Br)ccc3n2)cc1	nan
	2562079	27997	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	1	5	2.6	O=C(O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1373813	27997	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	1	5	2.6	O=C(O)CSc1ncnc2c1oc1ccccc12	nan
	2478421	28151	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	1	7	0.8	CC1(C)NC(=O)N(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)C1=O	nan
	CHEMBL1374872	28151	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	1	7	0.8	CC1(C)NC(=O)N(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)C1=O	nan
	3122786	28220	18	None	-10	4	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	4	5.1	COc1ccc(C2CC(c3cccs3)=NN2c2ccccc2)cc1	nan
	CHEMBL1375375	28220	18	None	-10	4	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	4	5.1	COc1ccc(C2CC(c3cccs3)=NN2c2ccccc2)cc1	nan
	4077805	28302	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	5	3.9	C=CCn1c(=S)[nH]c2scc(-c3ccc(C)o3)c2c1=O	nan
	CHEMBL1376201	28302	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	5	3.9	C=CCn1c(=S)[nH]c2scc(-c3ccc(C)o3)c2c1=O	nan
	2815476	28385	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	4	4.6	O=S(=O)(Nc1ccccc1C(F)(F)F)c1ccc(-c2ccccn2)s1	nan
	CHEMBL1376936	28385	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	4	4.6	O=S(=O)(Nc1ccccc1C(F)(F)F)c1ccc(-c2ccccn2)s1	nan
	16016416	28421	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	5	3.6	Cc1cc(O)c(CN2CCN(c3ccc(F)cc3)CC2)c2oc(=O)cc(C)c12	nan
	CHEMBL1377283	28421	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	5	3.6	Cc1cc(O)c(CN2CCN(c3ccc(F)cc3)CC2)c2oc(=O)cc(C)c12	nan
	2400757	28455	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	2.1	O=C(CNC(=O)c1cccc(F)c1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1377678	28455	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	2.1	O=C(CNC(=O)c1cccc(F)c1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	2864532	28507	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	3	4.2	CC(C)(C)C(=O)C1=C(O)C(=O)N(c2ccccc2)C1c1ccccc1	nan
	CHEMBL1378083	28507	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	3	4.2	CC(C)(C)C(=O)C1=C(O)C(=O)N(c2ccccc2)C1c1ccccc1	nan
	3522811	28563	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	8	0.8	Cc1nc(SCC(=O)NCCc2ccccc2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1378692	28563	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	8	0.8	Cc1nc(SCC(=O)NCCc2ccccc2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	4647380	28638	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	12	1	9	0.8	COCCN(CCOC)S(=O)(=O)c1ccc(C(=O)Nc2nnc(COC)o2)cc1	nan
	CHEMBL1379293	28638	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	12	1	9	0.8	COCCN(CCOC)S(=O)(=O)c1ccc(C(=O)Nc2nnc(COC)o2)cc1	nan
	5904589	28740	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	2	6	3.9	O=C(C1=C(O)C(=O)N(Cc2ccccc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1380259	28740	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	2	6	3.9	O=C(C1=C(O)C(=O)N(Cc2ccccc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	2768996	28789	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	6	2.2	O=c1c2ccccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	CHEMBL1380557	28789	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	6	2.2	O=c1c2ccccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	2815634	28805	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	4	5.8	O=C(Nc1ccc(F)cc1)Nc1sccc1-c1nc2ccccc2s1	nan
	CHEMBL1380666	28805	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	4	5.8	O=C(Nc1ccc(F)cc1)Nc1sccc1-c1nc2ccccc2s1	nan
	3604840	28815	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	CHEMBL1380782	28815	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	723113	28835	22	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	2	4	4	3.9	Nc1ccc2[nH]c(-c3ccc(-c4nc5cc(N)ccc5[nH]4)cc3)nc2c1	nan
	CHEMBL1380889	28835	22	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	2	4	4	3.9	Nc1ccc2[nH]c(-c3ccc(-c4nc5cc(N)ccc5[nH]4)cc3)nc2c1	nan
	866607	28888	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1381324	28888	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	1247739	29068	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	6	4.6	Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1nnc(C(F)(F)F)s1	nan
	CHEMBL1382928	29068	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	6	4.6	Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1nnc(C(F)(F)F)s1	nan
	4908738	29090	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	1	8	4.6	CCCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1383134	29090	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	1	8	4.6	CCCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	4196061	29256	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	10	2	5	3.4	CCCCCNC(=O)c1ccc2c(=O)n(CCCOCC)c(=S)[nH]c2c1	nan
	CHEMBL1384631	29256	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	10	2	5	3.4	CCCCCNC(=O)c1ccc2c(=O)n(CCCOCC)c(=S)[nH]c2c1	nan
	1392125	29343	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	6	2.0	O=C1NC(=S)N(Cc2ccc(F)cc2)C(=O)/C1=C/NCc1ccc2c(c1)OCO2	nan
	CHEMBL1385415	29343	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	6	2.0	O=C1NC(=S)N(Cc2ccc(F)cc2)C(=O)/C1=C/NCc1ccc2c(c1)OCO2	nan
	20876328	29440	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	5	3.3	CN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(F)cc2)CCS3)CC1	nan
	CHEMBL1386262	29440	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	5	3.3	CN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(F)cc2)CCS3)CC1	nan
	17584980	29482	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	1	7	2.2	Cc1cc(O)c2c(C)c(CC(=O)N3CCN(C(=O)C4COc5ccccc5O4)CC3)c(=O)oc2c1	nan
	CHEMBL1386530	29482	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	1	7	2.2	Cc1cc(O)c2c(C)c(CC(=O)N3CCN(C(=O)C4COc5ccccc5O4)CC3)c(=O)oc2c1	nan
	3254139	29516	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.8	CSc1nc(SC(C)C(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1386773	29516	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.8	CSc1nc(SC(C)C(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	3220391	29566	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	7	1	6	2.1	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCCOC	nan
	CHEMBL1387168	29566	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	7	1	6	2.1	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCCOC	nan
	16189864	29599	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	0	5	4.4	O=C(c1ccc(C(F)(F)F)cc1)C1CCCN(Cc2cccn2-c2ncccn2)C1	nan
	CHEMBL1387467	29599	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	0	5	4.4	O=C(c1ccc(C(F)(F)F)cc1)C1CCCN(Cc2cccn2-c2ncccn2)C1	nan
	899135	29642	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	3	3.2	NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1387789	29642	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	3	3.2	NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	2360761	29643	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	1	5	2.5	COc1ccc2c(C)cc3nnc(S)n3c2c1	nan
	CHEMBL1387791	29643	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	1	5	2.5	COc1ccc2c(C)cc3nnc(S)n3c2c1	nan
	2377721	29686	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	0	6	3.9	Cc1cc(C)nc(Sc2ncnc3c2oc2ccccc23)n1	nan
	CHEMBL1388175	29686	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	0	6	3.9	Cc1cc(C)nc(Sc2ncnc3c2oc2ccccc23)n1	nan
	3303130	29850	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	6.0	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Oc3ccccc3)c2)n1	nan
	CHEMBL1389429	29850	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	6.0	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Oc3ccccc3)c2)n1	nan
	5047557	29896	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	5	2.7	COC(=O)c1cc(C)sc1NC(=O)C1C2C=CC(CC2)C1C(=O)O	nan
	CHEMBL1389758	29896	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	5	2.7	COC(=O)c1cc(C)sc1NC(=O)C1C2C=CC(CC2)C1C(=O)O	nan
	671729	29959	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	4	3.8	O=C(Nc1ccc2c(c1)C(=O)N(c1ccccc1)C2=O)c1cccs1	nan
	CHEMBL1390374	29959	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	4	3.8	O=C(Nc1ccc2c(c1)C(=O)N(c1ccccc1)C2=O)c1cccs1	nan
	576025	29980	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	0	0	4	1.6	O=c1c2ccccc2c(=O)n2n1Cc1ccccc1C2	nan
	CHEMBL1390537	29980	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	0	0	4	1.6	O=c1c2ccccc2c(=O)n2n1Cc1ccccc1C2	nan
	1245900	30033	11	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	6	3.8	CCSc1nnc(NC(=O)c2cc3c(s2)CCCC3)s1	nan
	CHEMBL1391017	30033	11	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	6	3.8	CCSc1nnc(NC(=O)c2cc3c(s2)CCCC3)s1	nan
	5260648	30057	33	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	1	1	3	2.1	Cc1cc(Br)cn2cc(C(=O)O)nc12	nan
	CHEMBL1391195	30057	33	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	1	1	3	2.1	Cc1cc(Br)cn2cc(C(=O)O)nc12	nan
	6619983	30143	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	0	7	2.4	COC(=O)C(C)Sc1ccc2nnc(-c3ccccc3)n2n1	nan
	CHEMBL1391987	30143	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	0	7	2.4	COC(=O)C(C)Sc1ccc2nnc(-c3ccccc3)n2n1	nan
	3236381	30242	3	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	8	2.5	CCOC(=O)c1sc2ncnc(N3CCN(C(=O)OCC)CC3)c2c1C	nan
	CHEMBL1392800	30242	3	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	8	2.5	CCOC(=O)c1sc2ncnc(N3CCN(C(=O)OCC)CC3)c2c1C	nan
	135414599	30339	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	4	0.2	O=C1CC2C(=O)NCCN2C(NC(=O)c2ccc(Cl)cc2)=N1	nan
	CHEMBL1393609	30339	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	4	0.2	O=C1CC2C(=O)NCCN2C(NC(=O)c2ccc(Cl)cc2)=N1	nan
	950424	30437	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	0	7	1.6	CCN1CCN(c2nc3c(C)cccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	CHEMBL1394651	30437	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	0	7	1.6	CCN1CCN(c2nc3c(C)cccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	1689018	30451	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.2	CCOC(=O)c1sc2ncn(CC(=O)Nc3cc(C)cc(C)c3)c(=O)c2c1C	nan
	CHEMBL1394885	30451	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.2	CCOC(=O)c1sc2ncn(CC(=O)Nc3cc(C)cc(C)c3)c(=O)c2c1C	nan
	8087252	30514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	0	5	4.3	COc1cccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)c1	nan
	CHEMBL1395507	30514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	0	5	4.3	COc1cccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)c1	nan
	16009438	30523	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1	nan
	CHEMBL1395616	30523	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1	nan
	16017578	30558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)cc1	nan
	CHEMBL1396189	30558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)cc1	nan
	24819156	30575	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	0	6	6.1	COc1ccc(-c2oc3ccc(N4CCOCC4)cc3c2/C=C/c2ccc(OC)c(OC)c2)cc1	nan
	CHEMBL1396464	30575	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	0	6	6.1	COc1ccc(-c2oc3ccc(N4CCOCC4)cc3c2/C=C/c2ccc(OC)c(OC)c2)cc1	nan
	16022449	30612	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	4	4.9	CC(C)Oc1ccc(CNC(=O)c2cc3cccc4c3n2CC(C)S4)cc1	nan
	CHEMBL1396952	30612	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	4	4.9	CC(C)Oc1ccc(CNC(=O)c2cc3cccc4c3n2CC(C)S4)cc1	nan
	2017205	30632	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	2	6	5.8	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C(F)(F)F)cc4)sc3n2)cc1OC	nan
	CHEMBL1397215	30632	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	2	6	5.8	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C(F)(F)F)cc4)sc3n2)cc1OC	nan
	16019456	30701	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	2.5	COc1cc(NS(=O)(=O)c2c(C)nc3sc(C)c(C)n3c2=O)cc(OC)c1	nan
	CHEMBL1398166	30701	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	2.5	COc1cc(NS(=O)(=O)c2c(C)nc3sc(C)c(C)n3c2=O)cc(OC)c1	nan
	2964735	30742	11	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cccc(C2C(C(=O)c3cc4cccc(OC)c4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	CHEMBL1398596	30742	11	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cccc(C2C(C(=O)c3cc4cccc(OC)c4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	16012160	30760	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	2.0	Cc1cc(=O)n2nc(N(C)CC(=O)NCc3cccc(Br)c3)sc2n1	nan
	CHEMBL1398785	30760	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	2.0	Cc1cc(=O)n2nc(N(C)CC(=O)NCc3cccc(Br)c3)sc2n1	nan
	20888752	30857	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	9	1.2	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1399722	30857	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	9	1.2	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	7997207	30899	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	5	3.3	Cc1ccc(NC(=O)COC(=O)c2ccc(-n3cccn3)cc2)cc1C	nan
	CHEMBL1400115	30899	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	5	3.3	Cc1ccc(NC(=O)COC(=O)c2ccc(-n3cccn3)cc2)cc1C	nan
	2874407	30923	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.0	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CC(C)(C)CC2=N1	nan
	CHEMBL1400295	30923	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.0	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CC(C)(C)CC2=N1	nan
	2157035	31008	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	5.0	Cc1ccc(-c2nc(S(=O)(=O)c3ccccc3)c(SCC(=O)NC3CCCCC3)o2)cc1	nan
	CHEMBL1401131	31008	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	5.0	Cc1ccc(-c2nc(S(=O)(=O)c3ccccc3)c(SCC(=O)NC3CCCCC3)o2)cc1	nan
	5389771	31011	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	6	2.9	C=CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOC)C2c2cccnc2)cc1	nan
	CHEMBL1401159	31011	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	6	2.9	C=CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOC)C2c2cccnc2)cc1	nan
	20876293	31201	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	5	3.9	CCN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(C)cc2)CCS3)CC1	nan
	CHEMBL1402721	31201	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	5	3.9	CCN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(C)cc2)CCS3)CC1	nan
	16025411	31204	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	7	3.3	COC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	CHEMBL1402769	31204	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	7	3.3	COC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	1091654	31311	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	2	5	4.5	COc1ccc(NC(=O)c2ccco2)cc1NC(=O)COc1ccc(Cl)cc1C	nan
	CHEMBL1403849	31311	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	2	5	4.5	COc1ccc(NC(=O)c2ccco2)cc1NC(=O)COc1ccc(Cl)cc1C	nan
	2405342	31447	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2cc3c(cc2nc1Cl)OCCO3)c1ccccc1	nan
	CHEMBL1405208	31447	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2cc3c(cc2nc1Cl)OCCO3)c1ccccc1	nan
	16018264	31482	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.7	CCOC(=O)c1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	CHEMBL1405564	31482	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.7	CCOC(=O)c1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	3258366	31590	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	2	6	3.5	CCC1(C)Cc2c(sc3nc(S)nc(S)c23)CO1	nan
	CHEMBL1406514	31590	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	2	6	3.5	CCC1(C)Cc2c(sc3nc(S)nc(S)c23)CO1	nan
	5739089	31638	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.7	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(F)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1407014	31638	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.7	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(F)c1)c1ccc2c(c1)OCO2	nan
	20877853	31851	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	0	5	3.7	CCOC(=O)C1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1408512	31851	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	0	5	3.7	CCOC(=O)C1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	704023	32004	39	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	4	3.6	Sc1ncnc2sc(-c3ccccc3)cc12	nan
	CHEMBL1409776	32004	39	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	4	3.6	Sc1ncnc2sc(-c3ccccc3)cc12	nan
	4197372	32023	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.5	O=C(Nc1nc(-c2cccs2)c(C(=O)C(F)(F)F)s1)c1ccco1	nan
	CHEMBL1409901	32023	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.5	O=C(Nc1nc(-c2cccs2)c(C(=O)C(F)(F)F)s1)c1ccco1	nan
	1348850	32036	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cc(-c3nc4ccccc4s3)ccc2C)cc1	nan
	CHEMBL1409994	32036	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cc(-c3nc4ccccc4s3)ccc2C)cc1	nan
	6472686	32065	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	1.5	COc1cccc2cc(C(=O)NCCN3CCOCC3)oc12	nan
	CHEMBL1410184	32065	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	1.5	COc1cccc2cc(C(=O)NCCN3CCOCC3)oc12	nan
	16019689	32141	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	1	8	2.9	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1410849	32141	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	1	8	2.9	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	16025704	32228	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.5	COc1ccc(OC)c(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	CHEMBL1411590	32228	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.5	COc1ccc(OC)c(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	15988174	32329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	2	4	3.0	Cc1ccc(CCNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	CHEMBL1412411	32329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	2	4	3.0	Cc1ccc(CCNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	972224	32382	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	5	3.8	CCc1c(C)sc(N=C(S)Nc2cccnc2)c1C(=O)OC	nan
	CHEMBL1412818	32382	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	5	3.8	CCc1c(C)sc(N=C(S)Nc2cccnc2)c1C(=O)OC	nan
	16018140	32392	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	2	4.5	Cn1cc(CCCC(=O)NCc2ccccc2Cl)c2ccccc21	nan
	CHEMBL1412876	32392	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	2	4.5	Cn1cc(CCCC(=O)NCc2ccccc2Cl)c2ccccc21	nan
	646994	32426	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.4	Cc1ccc(S(=O)(=O)N(Cc2cc3cc4c(cc3nc2O)OCCO4)CC2CCCO2)cc1	nan
	CHEMBL1413144	32426	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.4	Cc1ccc(S(=O)(=O)N(Cc2cc3cc4c(cc3nc2O)OCCO4)CC2CCCO2)cc1	nan
	16018722	32463	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	4.1	Cc1ccc(C)c(NC(=O)CSc2nnc(C)n3c2cc2occc23)c1	nan
	CHEMBL1413449	32463	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	4.1	Cc1ccc(C)c(NC(=O)CSc2nnc(C)n3c2cc2occc23)c1	nan
	4149556	32499	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	3	4.3	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1F	nan
	CHEMBL1413747	32499	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	3	4.3	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1F	nan
	16018046	32618	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	4	3.8	O=C(CCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1Cl	nan
	CHEMBL1414743	32618	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	4	3.8	O=C(CCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1Cl	nan
	16187993	32675	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)NCc1ccccn1)C(=O)CO2	nan
	CHEMBL1415247	32675	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)NCc1ccccn1)C(=O)CO2	nan
	2910208	32840	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.3	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(F)cc1)c1ccco1	nan
	CHEMBL1416738	32840	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.3	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(F)cc1)c1ccco1	nan
	5014048	32884	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	3	5.9	Cc1ccc(CCNC(=O)c2cc(Nc3ccc(C)c(C)c3)nc3ccccc23)cc1	nan
	CHEMBL1417106	32884	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	3	5.9	Cc1ccc(CCNC(=O)c2cc(Nc3ccc(C)c(C)c3)nc3ccccc23)cc1	nan
	8901980	32915	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	5	4.1	CCOC(=O)Nc1ccc2c(CN(C)Cc3ccc(F)cc3)cc(=O)oc2c1	nan
	CHEMBL1417351	32915	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	5	4.1	CCOC(=O)Nc1ccc2c(CN(C)Cc3ccc(F)cc3)cc(=O)oc2c1	nan
	2911345	33028	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	3999653	33028	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	CHEMBL1418370	33028	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	1388232	33100	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	1	1	4	5.2	Cc1cccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCc2ccccc2-4)c1	nan
	CHEMBL1418971	33100	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	1	1	4	5.2	Cc1cccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCc2ccccc2-4)c1	nan
	2077572	33146	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	1	6	1.9	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1419336	33146	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	1	6	1.9	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	2370216	33480	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	0	3	4.2	O=C(COc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	CHEMBL1422190	33480	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	0	3	4.2	O=C(COc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	2035062	33503	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	2.6	CC(=O)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1422374	33503	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	2.6	CC(=O)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	16187581	33506	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	8	0	7	2.8	C=CCN(Cc1nc(-c2cc(OC)ccc2OC)oc1C)C1CCS(=O)(=O)C1	nan
	CHEMBL1422392	33506	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	8	0	7	2.8	C=CCN(Cc1nc(-c2cc(OC)ccc2OC)oc1C)C1CCS(=O)(=O)C1	nan
	5931057	33562	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	7	4.0	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1422871	33562	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	7	4.0	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	1609403	33661	6	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	0	5	4.7	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Br)cc2)c1	nan
	CHEMBL1423632	33661	6	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	0	5	4.7	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Br)cc2)c1	nan
	2308387	33696	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	0	8	2.6	Cc1c(CCOC(=O)c2cc([N+](=O)[O-])ccc2Cl)sc[n+]1CCCCS(=O)(=O)[O-]	nan
	CHEMBL1423887	33696	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	0	8	2.6	Cc1c(CCOC(=O)c2cc([N+](=O)[O-])ccc2Cl)sc[n+]1CCCCS(=O)(=O)[O-]	nan
	3546539	33761	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	1.2	O=C1NC(=S)N(C2CC2)C(=O)/C1=C/NCc1ccc(F)cc1	nan
	CHEMBL1424530	33761	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	1.2	O=C1NC(=S)N(C2CC2)C(=O)/C1=C/NCc1ccc(F)cc1	nan
	16192280	33907	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	4	4.2	CSc1ccc(C(=O)C2CCCN(C(=O)c3ccsc3)C2)cc1	nan
	CHEMBL1425858	33907	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	4	4.2	CSc1ccc(C(=O)C2CCCN(C(=O)c3ccsc3)C2)cc1	nan
	1229909	34182	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	6	2.7	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)n1	nan
	CHEMBL1428119	34182	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	6	2.7	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)n1	nan
	20903654	34333	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	0	9	1.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	CHEMBL1429390	34333	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	0	9	1.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	3259805	34338	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	7	1.9	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)COC(=O)c1cccnc1Cl	nan
	CHEMBL1429423	34338	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	7	1.9	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)COC(=O)c1cccnc1Cl	nan
	18562990	34385	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	2.0	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccc(F)cc1	nan
	CHEMBL1429771	34385	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	2.0	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccc(F)cc1	nan
	11834440	34404	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	4030418	34404	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	CHEMBL1429883	34404	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	3402414	34425	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-2.3	Cn1c(N)c(C(=O)COC(=O)C2=NNC(=O)CC2)c(=O)n(C)c1=O	nan
	CHEMBL1430091	34425	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-2.3	Cn1c(N)c(C(=O)COC(=O)C2=NNC(=O)CC2)c(=O)n(C)c1=O	nan
	2578265	34429	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	6	1.8	CC1CCC2(CC1)NC(=O)N(Cc1cc(=O)n3ccsc3n1)C2=O	nan
	CHEMBL1430109	34429	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	6	1.8	CC1CCC2(CC1)NC(=O)N(Cc1cc(=O)n3ccsc3n1)C2=O	nan
	4987698	34699	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(O)c1)c1cc2ccccc2o1	nan
	CHEMBL1432401	34699	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(O)c1)c1cc2ccccc2o1	nan
	657881	34710	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	2	1	5	1.9	CCOC(=O)c1c(C)nsc1S	nan
	CHEMBL1432472	34710	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	2	1	5	1.9	CCOC(=O)c1c(C)nsc1S	nan
	5123174	34730	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	3.3	COCCCn1c(=S)[nH]c2c(sc3ccccc32)c1=O	nan
	CHEMBL1432655	34730	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	3.3	COCCCn1c(=S)[nH]c2c(sc3ccccc32)c1=O	nan
	16019017	34877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	3.9	Cc1cccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c1	nan
	CHEMBL1434147	34877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	3.9	Cc1cccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c1	nan
	3566323	34925	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	9	1	9	4.0	CCOC(=O)CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c1ccc(OCC)c(OC)c1	nan
	CHEMBL1434864	34925	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	9	1	9	4.0	CCOC(=O)CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c1ccc(OCC)c(OC)c1	nan
	16015297	35030	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.3	CCn1c(CN2CCC(C)CC2)nc2cc(NC(=O)COc3ccc(Cl)c(C)c3)ccc21	nan
	CHEMBL1436095	35030	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.3	CCn1c(CN2CCC(C)CC2)nc2cc(NC(=O)COc3ccc(Cl)c(C)c3)ccc21	nan
	7526401	35043	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	4	2.2	N#Cc1ccccc1NS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2	nan
	CHEMBL1436243	35043	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	4	2.2	N#Cc1ccccc1NS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2	nan
	16019444	35045	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.9	Cc1nc2sc(C)c(C)n2c(=O)c1S(=O)(=O)NCCc1ccc(Cl)cc1	nan
	CHEMBL1436274	35045	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.9	Cc1nc2sc(C)c(C)n2c(=O)c1S(=O)(=O)NCCc1ccc(Cl)cc1	nan
	1743255	35047	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	3	1	5	3.4	N#CCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccccc3)nc2c1Br	nan
	CHEMBL1436298	35047	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	3	1	5	3.4	N#CCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccccc3)nc2c1Br	nan
	1004082	35093	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	5	4.8	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(C)cc4)sc3n2)cc1	nan
	CHEMBL1437042	35093	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	5	4.8	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(C)cc4)sc3n2)cc1	nan
	16030497	35123	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.8	CCc1cccc(C)c1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1437361	35123	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.8	CCc1cccc(C)c1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	5297283	35157	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	5	2.5	COc1ccc(C2CC(=O)Nc3c2c(=O)nc2c(C)cccn32)cc1	nan
	CHEMBL1437774	35157	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	5	2.5	COc1ccc(C2CC(=O)Nc3c2c(=O)nc2c(C)cccn32)cc1	nan
	2980985	35245	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	2	3	3.2	CC(C)(C)C(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	CHEMBL1438501	35245	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	2	3	3.2	CC(C)(C)C(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	16027383	35278	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	CHEMBL1438820	35278	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	16030423	35417	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.2	Cc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1	nan
	CHEMBL1440057	35417	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.2	Cc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1	nan
	24816825	35427	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	3	3.4	O=C(c1ccc(S(=O)(=O)Nc2cccc(C(F)(F)F)c2)cc1)N1CCC1	nan
	CHEMBL1440121	35427	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	3	3.4	O=C(c1ccc(S(=O)(=O)Nc2cccc(C(F)(F)F)c2)cc1)N1CCC1	nan
	22583638	35547	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	7	3.9	C=CCn1c(SCC(=O)N2CCN(c3ccccc3)CC2)nc2c3ccccc3nc-2c1O	nan
	CHEMBL1441228	35547	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	7	3.9	C=CCn1c(SCC(=O)N2CCN(c3ccccc3)CC2)nc2c3ccccc3nc-2c1O	nan
	4066521	35559	11	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	6	2.4	CC(=O)c1sc(NC(=O)C2COc3ccccc3O2)nc1C	nan
	CHEMBL1441350	35559	11	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	6	2.4	CC(=O)c1sc(NC(=O)C2COc3ccccc3O2)nc1C	nan
	2965654	35628	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	5	5.1	O=C(Nc1ccc([N+](=O)[O-])cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	CHEMBL1441978	35628	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	5	5.1	O=C(Nc1ccc([N+](=O)[O-])cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	16008702	35753	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	10	1	8	3.3	CCOC(=O)CC(NC(=O)CCc1c(C)nc2ncnn2c1C)c1ccc(OC(C)C)cc1	nan
	CHEMBL1443046	35753	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	10	1	8	3.3	CCOC(=O)CC(NC(=O)CCc1c(C)nc2ncnn2c1C)c1ccc(OC(C)C)cc1	nan
	2854033	35836	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	3	5.2	Fc1ccc(N2N=C(c3cccs3)CC2c2ccccc2)cc1	nan
	CHEMBL1443903	35836	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	3	5.2	Fc1ccc(N2N=C(c3cccs3)CC2c2ccccc2)cc1	nan
	5904887	35854	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	CHEMBL1444052	35854	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	16249191	36015	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	2	10	0.0	CC(C)[C@H](NS(=O)(=O)c1ccc(Cl)cc1)C(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	CHEMBL1445550	36015	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	2	10	0.0	CC(C)[C@H](NS(=O)(=O)c1ccc(Cl)cc1)C(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	6236858	36136	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccncc4)C3c3ccccc3F)ccc2O1	nan
	CHEMBL1446709	36136	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccncc4)C3c3ccccc3F)ccc2O1	nan
	2946413	36235	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	4	4.9	OC(COc1ccc2ccccc2c1Br)Cn1cnc(-c2ccccc2)c1	nan
	CHEMBL1447526	36235	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	4	4.9	OC(COc1ccc2ccccc2c1Br)Cn1cnc(-c2ccccc2)c1	nan
	5168521	36253	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	3.7	Cc1cc(C)c(NC(=O)Cn2cnc3c(oc4ccccc43)c2=O)c(C)c1	nan
	CHEMBL1447670	36253	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	3.7	Cc1cc(C)c(NC(=O)Cn2cnc3c(oc4ccccc43)c2=O)c(C)c1	nan
	975514	36403	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	2	3.7	COc1ccc2cc(Br)ccc2c1CC(=O)NC(C)C	nan
	CHEMBL1448872	36403	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	2	3.7	COc1ccc2cc(Br)ccc2c1CC(=O)NC(C)C	nan
	5003875	36731	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1Cl)c1cc(-c2ccc(Cl)cc2)on1	nan
	CHEMBL1451527	36731	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1Cl)c1cc(-c2ccc(Cl)cc2)on1	nan
	16009656	36794	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	6	4.8	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)cc2)c1	nan
	CHEMBL1451944	36794	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	6	4.8	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)cc2)c1	nan
	8087990	36810	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	0	8	1.3	Cc1nc2scc(C)n2c(=O)c1S(=O)(=O)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1452085	36810	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	0	8	1.3	Cc1nc2scc(C)n2c(=O)c1S(=O)(=O)N1CCN(c2ccccn2)CC1	nan
	2172625	36819	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	2	6	2.6	Cc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)c(C)s1	nan
	CHEMBL1452137	36819	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	2	6	2.6	Cc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)c(C)s1	nan
	2874437	36878	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	0	10	-0.3	Cn1c(=O)c2c(ncn2CC(=O)N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)n(C)c1=O	nan
	CHEMBL1452667	36878	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	0	10	-0.3	Cn1c(=O)c2c(ncn2CC(=O)N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)n(C)c1=O	nan
	3242606	36977	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	9	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc4c(c3)OCO4)nnc12	nan
	CHEMBL1453430	36977	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	9	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc4c(c3)OCO4)nnc12	nan
	5924128	37024	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1453845	37024	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	16025308	37034	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	3.1	O=C(Cn1c2ncccc2c(=O)n1-c1ccccc1)Nc1ccc(F)c(F)c1	nan
	CHEMBL1453921	37034	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	3.1	O=C(Cn1c2ncccc2c(=O)n1-c1ccccc1)Nc1ccc(F)c(F)c1	nan
	16009318	37077	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	5	3.3	Cc1cc(C)cc(OCc2cc(=O)n3cc(C)sc3n2)c1	nan
	CHEMBL1454181	37077	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	5	3.3	Cc1cc(C)cc(OCc2cc(=O)n3cc(C)sc3n2)c1	nan
	16015117	37097	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccccc1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	CHEMBL1454422	37097	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccccc1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	20920416	37165	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1454925	37165	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	35802	37167	98	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	3	2	4	3.1	COC(=O)Nc1nc2cc(C(=O)c3ccc(F)cc3)ccc2[nH]1	nan
	CHEMBL1454946	37167	98	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	3	2	4	3.1	COC(=O)Nc1nc2cc(C(=O)c3ccc(F)cc3)ccc2[nH]1	nan
	5739327	37221	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1455509	37221	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCO2	nan
	20923165	37318	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	1	6	2.4	CCC(C)(C)NS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1456385	37318	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	1	6	2.4	CCC(C)(C)NS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	3356561	37396	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.9	CCC1(C)Cc2c(sc3nc(SC)nc(S)c23)CO1	nan
	CHEMBL1457175	37396	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.9	CCC1(C)Cc2c(sc3nc(SC)nc(S)c23)CO1	nan
	16018620	37407	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.2	O=C(CSc1nncn2c1cc1occc12)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1457242	37407	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.2	O=C(CSc1nncn2c1cc1occc12)Nc1ccccc1C(F)(F)F	nan
	24686163	37498	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	3	5.1	CCN(CC)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	CHEMBL1457962	37498	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	3	5.1	CCN(CC)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	3927980	37535	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	6	3.1	CCCN1C(=O)C2(C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCCOC)c2ccccc21	nan
	CHEMBL1458233	37535	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	6	3.1	CCCN1C(=O)C2(C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCCOC)c2ccccc21	nan
	4962629	37569	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	4	3.5	Cc1cc(F)ccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1458588	37569	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	4	3.5	Cc1cc(F)ccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	6460246	37570	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	5	3.1	Cc1nnc2c(SC(C)C)nc3ccccc3n12	nan
	CHEMBL1458589	37570	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	5	3.1	Cc1nnc2c(SC(C)C)nc3ccccc3n12	nan
	7475827	37649	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	0	9	0.2	CC(C)Cc1nc(SCC(=O)N2CCOCC2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1459222	37649	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	0	9	0.2	CC(C)Cc1nc(SCC(=O)N2CCOCC2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	3239559	37758	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	2	0	3	3.4	CCn1c(=S)ccc2ccc(OC)cc21	nan
	CHEMBL1460186	37758	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	2	0	3	3.4	CCn1c(=S)ccc2ccc(OC)cc21	nan
	4091063	37864	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	7	2.1	COC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	CHEMBL1461057	37864	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	7	2.1	COC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	135413805	37972	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	3	9	1.2	N#Cc1cc(Nc2c(N)ncnc2O)c([N+](=O)[O-])cc1C#N	nan
	CHEMBL1462053	37972	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	3	9	1.2	N#Cc1cc(Nc2c(N)ncnc2O)c([N+](=O)[O-])cc1C#N	nan
	4636986	38054	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	2	10	0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1462720	38054	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	2	10	0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	993137	38091	17	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	3.4	CC(=O)c1sc(NC(=O)COc2ccc(Br)cc2)nc1C	nan
	CHEMBL1463012	38091	17	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	3.4	CC(=O)c1sc(NC(=O)COc2ccc(Br)cc2)nc1C	nan
	2225463	38145	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	3	3.3	O=C(NCCCN1CCCC1=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1463545	38145	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	3	3.3	O=C(NCCCN1CCCC1=O)c1sc2ccccc2c1Cl	nan
	6184422	38216	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	10	1	8	3.5	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1464067	38216	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	10	1	8	3.5	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	135449395	38223	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	3.1	CCN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	CHEMBL1464106	38223	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	3.1	CCN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	5778449	38311	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCOC)CC1	nan
	CHEMBL1464778	38311	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCOC)CC1	nan
	2457314	38322	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	10	0.1	COc1ccc(OC)c(/C=C/C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1464838	38322	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	10	0.1	COc1ccc(OC)c(/C=C/C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	3791918	38333	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)ccc2Cl)n1	nan
	CHEMBL1464872	38333	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)ccc2Cl)n1	nan
	985269	38378	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	0	5	4.7	c1ccc(-c2cc3c(N4CCN(c5ccccc5)CC4)ncnc3s2)cc1	nan
	CHEMBL1465210	38378	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	0	5	4.7	c1ccc(-c2cc3c(N4CCN(c5ccccc5)CC4)ncnc3s2)cc1	nan
	1435001	38454	4	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	2	6	2.8	CCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	CHEMBL1465814	38454	4	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	2	6	2.8	CCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	1479844	38492	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	4	5.2	CSc1nc(Sc2ccccc2Cl)c2ccccc2n1	nan
	CHEMBL1466134	38492	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	4	5.2	CSc1nc(Sc2ccccc2Cl)c2ccccc2n1	nan
	1836205	38495	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1466152	38495	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	2982726	38530	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	7	1.1	CCOC(=O)C1=C(CN2CCOCC2)NC(=O)NC1c1cccc([N+](=O)[O-])c1	nan
	CHEMBL1466461	38530	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	7	1.1	CCOC(=O)C1=C(CN2CCOCC2)NC(=O)NC1c1cccc([N+](=O)[O-])c1	nan
	5831389	38595	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	6	3.9	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1466919	38595	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	6	3.9	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	2161641	38651	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	2	7	3.0	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccs2)cc1	nan
	CHEMBL1467371	38651	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	2	7	3.0	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccs2)cc1	nan
	2146410	38653	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	2	3.3	CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1467397	38653	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	2	3.3	CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	5028075	38689	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.9	COc1ccc(NC(=O)COC(=O)c2cc(SC)ccc2Cl)c(OC)c1	nan
	CHEMBL1467702	38689	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.9	COc1ccc(NC(=O)COC(=O)c2cc(SC)ccc2Cl)c(OC)c1	nan
	5786830	38700	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	3.4	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1467854	38700	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	3.4	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)cc1	nan
	652110	38788	4	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	4	0	5	3.0	COC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	CHEMBL1468599	38788	4	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	4	0	5	3.0	COC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	20904121	38862	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCOCC4)nn23)c1	nan
	CHEMBL1469174	38862	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCOCC4)nn23)c1	nan
	5726945	38876	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	4	3.5	CC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	CHEMBL1469326	38876	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	4	3.5	CC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	3812545	38982	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(OC)c(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1470290	38982	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(OC)c(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2964736	38998	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(c4cc(C)on4)C3c3cccs3)oc12	nan
	CHEMBL1470378	38998	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(c4cc(C)on4)C3c3cccs3)oc12	nan
	15988466	39255	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.3	COc1ccc(NC(=O)Cn2c(=O)c3cc(Cl)ccc3n3nncc23)cc1	nan
	CHEMBL1472605	39255	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.3	COc1ccc(NC(=O)Cn2c(=O)c3cc(Cl)ccc3n3nncc23)cc1	nan
	16011470	39271	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(CCNC(=O)c2ccc(Cn3c(SCc4ccccc4)nc4cccnc43)cc2)cc1	nan
	CHEMBL1472792	39271	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(CCNC(=O)c2ccc(Cn3c(SCc4ccccc4)nc4cccnc43)cc2)cc1	nan
	6229347	39351	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	3.0	COc1ccccc1CCNC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	CHEMBL1473886	39351	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	3.0	COc1ccccc1CCNC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	20886471	39363	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	4	4.3	CCCOc1ccc(CNC(=O)c2ccc3c(c2)N(CC)CCS3)cc1	nan
	CHEMBL1474147	39363	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	4	4.3	CCCOc1ccc(CNC(=O)c2ccc3c(c2)N(CC)CCS3)cc1	nan
	15988056	39424	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	2	4	3.5	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(Cl)cc3)ccc2c1=O	nan
	CHEMBL1475000	39424	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	2	4	3.5	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(Cl)cc3)ccc2c1=O	nan
	5297460	39435	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	1	5	4.0	CCOc1ccc(-c2oc3ccccc3c(=O)c2O)cc1OCC	nan
	CHEMBL1475143	39435	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	1	5	4.0	CCOc1ccc(-c2oc3ccccc3c(=O)c2O)cc1OCC	nan
	16018222	39444	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	3.0	COc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1475268	39444	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	3.0	COc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	135410479	39454	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	2	4	5.5	Cc1ccc(NC(=O)c2cnn3c2NC(c2ccccc2)=CC3c2ccccc2)cc1	nan
	CHEMBL1475406	39454	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	2	4	5.5	Cc1ccc(NC(=O)c2cnn3c2NC(c2ccccc2)=CC3c2ccccc2)cc1	nan
	16031507	39455	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(F)c3)s2)cc1	nan
	CHEMBL1475415	39455	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(F)c3)s2)cc1	nan
	16015334	39518	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	6	5.7	COc1ccc(Cc2c(C)nn(-c3nc(C)c(C(=O)Nc4ccc(C)cc4C)s3)c2C)cc1	nan
	CHEMBL1476342	39518	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	6	5.7	COc1ccc(Cc2c(C)nn(-c3nc(C)c(C(=O)Nc4ccc(C)cc4C)s3)c2C)cc1	nan
	2033254	39564	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	7	2.8	CSc1nc(NCCCN(C)C)c2c3c(sc2n1)CN(C)CC3	nan
	CHEMBL1476899	39564	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	7	2.8	CSc1nc(NCCCN(C)C)c2c3c(sc2n1)CN(C)CC3	nan
	1138445	39662	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1477799	39662	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1442565	39705	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	5	3.9	CCOC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1478306	39705	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	5	3.9	CCOC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	1005239	39799	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	2	1	5	5.8	N#Cc1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	CHEMBL1479144	39799	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	2	1	5	5.8	N#Cc1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	16018188	39827	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	1	5	3.8	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccccc32)cc1	nan
	CHEMBL1479369	39827	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	1	5	3.8	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccccc32)cc1	nan
	5914213	40317	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1483546	40317	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	796660	40401	4	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	5	2.9	COc1cc2oc(=O)c(Br)c(C)c2c(OC)c1OC	nan
	CHEMBL1484186	40401	4	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	5	2.9	COc1cc2oc(=O)c(Br)c(C)c2c(OC)c1OC	nan
	16025365	40475	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	7	1	7	5.4	CC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1484843	40475	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	7	1	7	5.4	CC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	2881633	40501	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	5	2.3	Cc1nnc(Nc2ccc(S(N)(=O)=O)cc2)c2ccccc12	nan
	CHEMBL1485038	40501	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	5	2.3	Cc1nnc(Nc2ccc(S(N)(=O)=O)cc2)c2ccccc12	nan
	16020293	40533	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	8	2	7	4.3	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(C)cc3)c2=O)cc1	nan
	CHEMBL1485379	40533	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	8	2	7	4.3	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(C)cc3)c2=O)cc1	nan
	866572	40581	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	6	1.3	CN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1485808	40581	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	6	1.3	CN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	15991110	40600	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1c(F)cccc1F	nan
	CHEMBL1485996	40600	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1c(F)cccc1F	nan
	20869704	40604	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2cccc(OC)c2)c1=O	nan
	CHEMBL1486007	40604	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2cccc(OC)c2)c1=O	nan
	2951279	40605	13	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	7	4.2	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccco4)C3c3cccnc3)oc12	nan
	CHEMBL1486010	40605	13	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	7	4.2	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccco4)C3c3cccnc3)oc12	nan
	3647805	40692	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	2	4	3.1	CCCCC(CC)CNC(=O)CC1N=C2c3ccccc3NC(=S)N2C1=O	nan
	CHEMBL1486794	40692	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	2	4	3.1	CCCCC(CC)CNC(=O)CC1N=C2c3ccccc3NC(=S)N2C1=O	nan
	3149629	40743	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	1	5	2.4	O=C(O)CSc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1487236	40743	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	1	5	2.4	O=C(O)CSc1ncnc2sc3c(c12)CCC3	nan
	6296199	40754	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	8	2.9	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1487315	40754	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	8	2.9	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3494131	40947	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccs2)no1	nan
	CHEMBL1488696	40947	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccs2)no1	nan
	16016559	41001	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	1	4	3.7	Cc1ccc(-c2nonc2NC(=O)c2ccc(F)cc2)cc1C	nan
	CHEMBL1489095	41001	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	1	4	3.7	Cc1ccc(-c2nonc2NC(=O)c2ccc(F)cc2)cc1C	nan
	4604410	41167	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1c(Cl)cccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1490398	41167	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1c(Cl)cccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	15992220	41176	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	3862718	41176	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	5941821	41176	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	CHEMBL1490493	41176	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	5307465	41309	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	0	6	2.5	Cc1sc2nc3ccc(N4CCCC4)nn3c(=O)c2c1C	nan
	CHEMBL1491386	41309	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	0	6	2.5	Cc1sc2nc3ccc(N4CCCC4)nn3c(=O)c2c1C	nan
	648659	41376	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	8	1.5	CCCn1c(SCC(=O)N2CCc3ccccc3C2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1491811	41376	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	8	1.5	CCCn1c(SCC(=O)N2CCc3ccccc3C2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3240716	41391	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	11	2	7	3.9	CCOc1cc2[nH]c(=S)n(CCCCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	CHEMBL1491907	41391	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	11	2	7	3.9	CCOc1cc2[nH]c(=S)n(CCCCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	20917809	41415	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.1	O=C1c2cccnc2C(=O)N1Cc1ccc(F)cc1S(=O)(=O)NCc1ccco1	nan
	CHEMBL1492082	41415	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.1	O=C1c2cccnc2C(=O)N1Cc1ccc(F)cc1S(=O)(=O)NCc1ccco1	nan
	6533452	41428	16	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.4	COc1ccc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc1OC	nan
	CHEMBL1492209	41428	16	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.4	COc1ccc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc1OC	nan
	135414697	41441	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	3.7	N#Cc1c(O)nc(SCc2ccc(F)cc2)nc1-c1ccco1	nan
	CHEMBL1492324	41441	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	3.7	N#Cc1c(O)nc(SCc2ccc(F)cc2)nc1-c1ccco1	nan
	3151464	41478	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.1	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1492596	41478	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.1	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	3241814	41484	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	6	1.1	Cn1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1492641	41484	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	6	1.1	Cn1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	4118355	41571	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	4	4.7	Cc1ccc(C(C)(C)C)cc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1493417	41571	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	4	4.7	Cc1ccc(C(C)(C)C)cc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	7899292	41578	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	8	1.5	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)c1	nan
	CHEMBL1493482	41578	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	8	1.5	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)c1	nan
	16014523	41639	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	4.8	Cc1cc(Nc2ccc(C)c(Cl)c2)n2nc(-c3ccccc3)nc2n1	nan
	CHEMBL1494140	41639	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	4.8	Cc1cc(Nc2ccc(C)c(Cl)c2)n2nc(-c3ccccc3)nc2n1	nan
	4578483	41667	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	6	6.0	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(Cl)c4Cl)cc3n2)cc1OC	nan
	CHEMBL1494437	41667	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	6	6.0	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(Cl)c4Cl)cc3n2)cc1OC	nan
	2740372	41682	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	5	3.8	CCOC(=O)c1csc(-c2sccc2Br)n1	nan
	CHEMBL1494595	41682	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	5	3.8	CCOC(=O)c1csc(-c2sccc2Br)n1	nan
	6245779	41707	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	6	5.1	Cc1cc(OCc2ccccc2)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	CHEMBL1494772	41707	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	6	5.1	Cc1cc(OCc2ccccc2)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	2961508	41756	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	5740308	41756	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	9587859	41756	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	CHEMBL1495283	41756	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	7743649	41861	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	4	4.3	Cc1cc(SCC(=O)NC2(C#N)CCCCC2)nc2c(C)cccc12	nan
	CHEMBL1496365	41861	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	4	4.3	Cc1cc(SCC(=O)NC2(C#N)CCCCC2)nc2c(C)cccc12	nan
	7709279	41918	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	3.1	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCS3	nan
	CHEMBL1496847	41918	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	3.1	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCS3	nan
	5760983	41919	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	4	1	4	5.4	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(Br)cc1)c1ccc(Br)cc1	nan
	CHEMBL1496850	41919	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	4	1	4	5.4	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(Br)cc1)c1ccc(Br)cc1	nan
	16195573	41952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	2	7	3.2	CCOc1cc2[nH]c(=S)n(CCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	CHEMBL1497122	41952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	2	7	3.2	CCOc1cc2[nH]c(=S)n(CCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	265605	42117	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	236	1	0	6	0.1	CC(C)c1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1498670	42117	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	236	1	0	6	0.1	CC(C)c1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	20875207	42296	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	3	4.2	O=C(Nc1ccccc1F)c1oc2ccccc2c1NC(=O)C1CC1	nan
	CHEMBL1500175	42296	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	3	4.2	O=C(Nc1ccccc1F)c1oc2ccccc2c1NC(=O)C1CC1	nan
	17583267	42367	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	3.8	COc1cc(NC(=O)COc2cc(C)cc3oc(=O)c(C)c(C)c23)cc(OC)c1OC	nan
	CHEMBL1500728	42367	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	3.8	COc1cc(NC(=O)COc2cc(C)cc3oc(=O)c(C)c(C)c23)cc(OC)c1OC	nan
	2768366	42564	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	3	2	4	2.2	COc1ccc(-c2ccc(C(=O)O)c(O)n2)cc1	nan
	CHEMBL1502516	42564	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	3	2	4	2.2	COc1ccc(-c2ccc(C(=O)O)c(O)n2)cc1	nan
	859554	42616	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	7	3.3	Cc1cc(NC(=O)CSc2ncnc3sc(C)c(C)c23)no1	nan
	CHEMBL1503032	42616	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	7	3.3	Cc1cc(NC(=O)CSc2ncnc3sc(C)c(C)c23)no1	nan
	5294012	42696	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	7	4.0	CC(C)n1c2ccccc2c2nnc(SCC(=O)Nc3ccccc3C(=O)O)nc21	nan
	CHEMBL1503589	42696	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	7	4.0	CC(C)n1c2ccccc2c2nnc(SCC(=O)Nc3ccccc3C(=O)O)nc21	nan
	20956972	42877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	1.9	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)cc1F	nan
	CHEMBL1505377	42877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	1.9	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)cc1F	nan
	4157311	42887	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	5	0	9	4.0	O=c1c2sccc2nc(SCc2cc(=O)n3cc(Br)ccc3n2)n1Cc1ccccn1	nan
	CHEMBL1505478	42887	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	5	0	9	4.0	O=c1c2sccc2nc(SCc2cc(=O)n3cc(Br)ccc3n2)n1Cc1ccccn1	nan
	5936247	42888	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccccc1C1C(C(=O)c2ccc3c(c2)OCCO3)=C(O)C(=O)N1Cc1cccnc1	nan
	CHEMBL1505481	42888	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccccc1C1C(C(=O)c2ccc3c(c2)OCCO3)=C(O)C(=O)N1Cc1cccnc1	nan
	3152549	43117	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1Cl)c1ccco1	nan
	CHEMBL1507420	43117	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1Cl)c1ccco1	nan
	2905772	43134	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	11	-0.4	CCOC(=O)Cc1csc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)n1	nan
	CHEMBL1507551	43134	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	11	-0.4	CCOC(=O)Cc1csc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)n1	nan
	20888750	43146	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	8	1.8	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	CHEMBL1507635	43146	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	8	1.8	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	664007	43244	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	5	5.5	Cc1cc(NC(=O)c2ccc3nc(-c4ccccc4)c(-c4ccccc4)nc3c2)no1	nan
	CHEMBL1508441	43244	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	5	5.5	Cc1cc(NC(=O)c2ccc3nc(-c4ccccc4)c(-c4ccccc4)nc3c2)no1	nan
	1862355	43273	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1ccc(-c2cc(-c3cccnc3)c(C#N)c(N)n2)cc1	nan
	CHEMBL1508668	43273	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1ccc(-c2cc(-c3cccnc3)c(C#N)c(N)n2)cc1	nan
	6224737	43342	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	8	4.0	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1509331	43342	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	8	4.0	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	22514400	43420	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	7	0.6	CCOC(=O)C1CCN(C(=O)Cn2nc(C)n3cccc3c2=O)CC1	nan
	CHEMBL1510088	43420	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	7	0.6	CCOC(=O)C1CCN(C(=O)Cn2nc(C)n3cccc3c2=O)CC1	nan
	4547589	43444	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	3	4.9	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1Cl	nan
	CHEMBL1510328	43444	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	3	4.9	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1Cl	nan
	24792485	43465	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1cc2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2cc1OC	nan
	CHEMBL1510493	43465	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1cc2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2cc1OC	nan
	6042599	43588	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)cc1	nan
	CHEMBL1511435	43588	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)cc1	nan
	16027534	43638	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)cc1	nan
	CHEMBL1512013	43638	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)cc1	nan
	16024951	43656	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	2	6	4.8	CCOc1ccc(Nc2nc(N)c(C(=O)c3ccccc3Cl)s2)cc1	nan
	CHEMBL1512414	43656	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	2	6	4.8	CCOc1ccc(Nc2nc(N)c(C(=O)c3ccccc3Cl)s2)cc1	nan
	4395410	43768	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	0	4	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCc1ccc(F)cc1	nan
	CHEMBL1514024	43768	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	0	4	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCc1ccc(F)cc1	nan
	16018164	43797	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	5	3.4	COc1ccccc1CNC(=O)CCCn1c(=O)c2cccn2c2ccccc21	nan
	CHEMBL1514529	43797	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	5	3.4	COc1ccccc1CNC(=O)CCCn1c(=O)c2cccn2c2ccccc21	nan
	4081154	43877	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	3	5.1	O=C(Nc1c(C(=O)c2ccccc2)oc2ccccc12)c1ccc(F)cc1	nan
	CHEMBL1515694	43877	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	3	5.1	O=C(Nc1c(C(=O)c2ccccc2)oc2ccccc12)c1ccc(F)cc1	nan
	135546812	43894	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	5	3.6	CCc1ccc(NC(=O)CSc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)cc1	nan
	CHEMBL1515954	43894	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	5	3.6	CCc1ccc(NC(=O)CSc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)cc1	nan
	16022285	43953	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	2	6	2.3	Cc1nc2cccnc2n1-c1cccc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1	nan
	CHEMBL1516713	43953	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	2	6	2.3	Cc1nc2cccnc2n1-c1cccc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1	nan
	1466061	43964	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	5	3.8	CCOc1ccc2nc(O)c(CN(CCc3ccccc3)C(=O)N3CCOCC3)cc2c1	nan
	CHEMBL1516817	43964	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	5	3.8	CCOc1ccc2nc(O)c(CN(CCc3ccccc3)C(=O)N3CCOCC3)cc2c1	nan
	3433386	44052	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	CHEMBL1517698	44052	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	16018535	44193	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	1	4	4.2	CC(=O)N1CCOc2cc(S(=O)(=O)Nc3cc(C(F)(F)F)ccc3Cl)c(C)cc21	nan
	CHEMBL1518991	44193	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	1	4	4.2	CC(=O)N1CCOc2cc(S(=O)(=O)Nc3cc(C(F)(F)F)ccc3Cl)c(C)cc21	nan
	2135572	44208	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1519131	44208	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	16025796	44263	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.4	CC(NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1)c1ccccc1	nan
	CHEMBL1519614	44263	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.4	CC(NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1)c1ccccc1	nan
	16030429	44405	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(F)cc2)cc1	nan
	CHEMBL1520828	44405	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(F)cc2)cc1	nan
	15988916	44416	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	8	2	8	4.4	Cc1cc(C)c(NC(=O)Cn2c(=O)n(Cc3ccc(C(=O)NCc4ccco4)cc3)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1520905	44416	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	8	2	8	4.4	Cc1cc(C)c(NC(=O)Cn2c(=O)n(Cc3ccc(C(=O)NCc4ccco4)cc3)c(=O)c3sccc32)c(C)c1	nan
	289464	44464	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	1	4.5	O=C(O)c1cc2ccccc2c2cc(Br)ccc12	nan
	CHEMBL1521339	44464	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	1	4.5	O=C(O)c1cc2ccccc2c2cc(Br)ccc12	nan
	2745168	44523	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	1	6	1.2	COCc1nc(S)c(C#N)cc1C(=O)OC	nan
	CHEMBL1521853	44523	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	1	6	1.2	COCc1nc(S)c(C#N)cc1C(=O)OC	nan
	689389	44569	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	6	1	5	3.4	CCN(CC)CCNc1cc(C)c(C#N)c2nc3ccccc3n12	nan
	CHEMBL1522224	44569	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	6	1	5	3.4	CCN(CC)CCNc1cc(C)c(C#N)c2nc3ccccc3n12	nan
	1167955	44702	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	5	5.0	O=C(CSc1nc(-c2ccc(F)cc2)nc2ccc(F)cc12)Nc1cccc(C(=O)O)c1	nan
	CHEMBL1523483	44702	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	5	5.0	O=C(CSc1nc(-c2ccc(F)cc2)nc2ccc(F)cc12)Nc1cccc(C(=O)O)c1	nan
	17201681	44764	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	2	2.4	O=C(C1CC(=O)N(c2ccc(Br)cc2)C1)N1CCCC1	nan
	CHEMBL1524084	44764	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	2	2.4	O=C(C1CC(=O)N(c2ccc(Br)cc2)C1)N1CCCC1	nan
	16018239	44808	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	3	3.5	CCOc1ccc(NC(=O)N2CCOc3ccccc32)cc1	nan
	CHEMBL1524566	44808	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	3	3.5	CCOc1ccc(NC(=O)N2CCOc3ccccc32)cc1	nan
	818605	44833	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	0	4	2.3	COc1ccc(C=O)cc1CN1C(=O)c2ccccc2C1=O	nan
	CHEMBL1524802	44833	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	0	4	2.3	COc1ccc(C=O)cc1CN1C(=O)c2ccccc2C1=O	nan
	16015121	44852	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	CHEMBL1525000	44852	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	4624396	44878	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.1	CCOc1ccc(-c2csc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)n2)cc1	nan
	CHEMBL1525327	44878	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.1	CCOc1ccc(-c2csc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)n2)cc1	nan
	551547	44895	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	3	4.6	O=C(NCC1CCCO1)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1525441	44895	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	3	4.6	O=C(NCC1CCCO1)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	2904040	44922	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	2	3	3.0	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc(-c3ccccc3)cc2)cc1	nan
	CHEMBL1525655	44922	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	2	3	3.0	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc(-c3ccccc3)cc2)cc1	nan
	2868184	44943	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Cl)cc1	nan
	CHEMBL1525829	44943	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Cl)cc1	nan
	16018537	44980	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	1.6	CCOC(=O)C1CCCN(C(=O)CCS(=O)(=O)c2cc3c(cc2Cl)NC(=O)CO3)C1	nan
	CHEMBL1526153	44980	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	1.6	CCOC(=O)C1CCCN(C(=O)CCS(=O)(=O)c2cc3c(cc2Cl)NC(=O)CO3)C1	nan
	3151412	45113	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	8	0.7	COCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1527265	45113	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	8	0.7	COCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	3772745	45157	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	4	4.9	COc1cccc(-c2cc(C(=O)NCC3CCCO3)c3cc(Br)cc(C)c3n2)c1	nan
	CHEMBL1527660	45157	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	4	4.9	COc1cccc(-c2cc(C(=O)NCC3CCCO3)c3cc(Br)cc(C)c3n2)c1	nan
	1253448	45171	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1527795	45171	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	661360	45178	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	7	1.5	COc1ccc(-n2ncc3c(N4CCC(C(N)=O)CC4)ncnc32)cc1	nan
	CHEMBL1527862	45178	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	7	1.5	COc1ccc(-n2ncc3c(N4CCC(C(N)=O)CC4)ncnc32)cc1	nan
	1077518	45269	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	6	2.5	CCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1528629	45269	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	6	2.5	CCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	16813521	45313	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	1.8	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCC4)nn23)cc1	nan
	CHEMBL1529059	45313	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	1.8	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCC4)nn23)cc1	nan
	54694033	45338	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	2	5	2.6	CCCn1c(=O)c(C(=O)NCc2ccco2)c(O)c2ccccc21	nan
	CHEMBL1529241	45338	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	2	5	2.6	CCCn1c(=O)c(C(=O)NCc2ccco2)c(O)c2ccccc21	nan
	625773	45504	50	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	3	4.3	O=C(O)c1cc(-c2ccc(Cl)s2)nc2ccccc12	nan
	CHEMBL153072	45504	50	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	3	4.3	O=C(O)c1cc(-c2ccc(Cl)s2)nc2ccccc12	nan
	3151486	45522	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	2	8	1.8	CCOCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1530888	45522	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	2	8	1.8	CCOCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cccc(C)c3nc21	nan
	4216259	45560	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	2.0	CCCCn1c(=O)[nH]c(=O)c2c1nc(Cn1ncc(Cl)c(Cl)c1=O)n2CCC	nan
	CHEMBL1531245	45560	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	2.0	CCCCn1c(=O)[nH]c(=O)c2c1nc(Cn1ncc(Cl)c(Cl)c1=O)n2CCC	nan
	2737056	45647	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	191	1	0	4	1.4	O=C1CC(=O)c2c1cccc2[N+](=O)[O-]	nan
	CHEMBL1532031	45647	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	191	1	0	4	1.4	O=C1CC(=O)c2c1cccc2[N+](=O)[O-]	nan
	2085635	45698	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	2	0	5	2.9	Cc1ccc2nc(Cn3cc(C(F)(F)F)cc(Cl)c3=O)cc(=O)n2c1	nan
	CHEMBL1532467	45698	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	2	0	5	2.9	Cc1ccc2nc(Cn3cc(C(F)(F)F)cc(Cl)c3=O)cc(=O)n2c1	nan
	3721626	45729	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	5	3.9	COc1ccc2c(c1)c1ncnc(N(C)C3CCCCC3)c1n2C	nan
	CHEMBL1532723	45729	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	5	3.9	COc1ccc2c(c1)c1ncnc(N(C)C3CCCCC3)c1n2C	nan
	3312243	45970	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4ccc(F)cc4)c3nc12	nan
	CHEMBL1535016	45970	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4ccc(F)cc4)c3nc12	nan
	135403580	46070	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	7	4.6	N#Cc1c(O)nc(SCC(=O)Nc2ccc(OC(F)(F)Cl)cc2)nc1-c1ccccc1	nan
	CHEMBL1536174	46070	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	7	4.6	N#Cc1c(O)nc(SCC(=O)Nc2ccc(OC(F)(F)Cl)cc2)nc1-c1ccccc1	nan
	5310128	46086	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1ccc2nnc(-c3ccncc3)n2n1)NCC1CCCO1	nan
	CHEMBL1536319	46086	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1ccc2nnc(-c3ccncc3)n2n1)NCC1CCCO1	nan
	20878456	46119	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	8	2.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2ccccc23)cc1	nan
	CHEMBL1536657	46119	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	8	2.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2ccccc23)cc1	nan
	5059230	46130	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	2.5	N#CC1=C([C-](C#N)C#N)NC(O)(C2CC2)C([n+]2ccccc2)C1c1ccccc1F	nan
	CHEMBL1536738	46130	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	2.5	N#CC1=C([C-](C#N)C#N)NC(O)(C2CC2)C([n+]2ccccc2)C1c1ccccc1F	nan
	5235682	46198	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(Cl)c2)no1	nan
	CHEMBL1537295	46198	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(Cl)c2)no1	nan
	7190492	46369	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1538682	46369	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	3220383	46443	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	3.3	CC(C)CC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1539378	46443	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	3.3	CC(C)CC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	6133031	46471	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	7	2.4	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1539594	46471	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	7	2.4	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	1567287	46576	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	6	-1.0	CN1C(=O)C(=CNCCN2CCOCC2)C(=O)N(C)C1=S	nan
	CHEMBL1540479	46576	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	6	-1.0	CN1C(=O)C(=CNCCN2CCOCC2)C(=O)N(C)C1=S	nan
	2983027	46593	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	1.8	O=C(NCc1cccnc1)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	CHEMBL1540590	46593	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	1.8	O=C(NCc1cccnc1)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	2431987	46618	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	1	5	3.0	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1540855	46618	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	1	5	3.0	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	3833515	46643	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	7	5.1	C=CCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1541029	46643	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	7	5.1	C=CCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	6273159	46729	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1541682	46729	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	659524	46916	7	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	1	0	3	4.1	Brc1cc(Br)c2ncnc(N3CCCCC3)c2c1	nan
	CHEMBL1543331	46916	7	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	1	0	3	4.1	Brc1cc(Br)c2ncnc(N3CCCCC3)c2c1	nan
	16194876	47162	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(OC)c(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1545182	47162	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(OC)c(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	2997987	47193	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.0	Cc1sc2ncnc(OCC(=O)NCC3CCCO3)c2c1C	nan
	CHEMBL1545423	47193	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.0	Cc1sc2ncnc(OCC(=O)NCC3CCCO3)c2c1C	nan
	16188698	47283	0	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	2	4.2	Cc1ccccc1CC1(CO)CCCN(C(=O)c2cc(Cl)ccc2F)C1	nan
	CHEMBL1546168	47283	0	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	2	4.2	Cc1ccccc1CC1(CO)CCCN(C(=O)c2cc(Cl)ccc2F)C1	nan
	5389436	47404	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	3.8	COc1cccc(C2C(C(=O)c3ccc(OC)c(OC)c3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1547272	47404	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	3.8	COc1cccc(C2C(C(=O)c3ccc(OC)c(OC)c3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	16437942	47732	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	9	2.2	CCCS(=O)(=O)c1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)n1	nan
	CHEMBL1550174	47732	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	9	2.2	CCCS(=O)(=O)c1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)n1	nan
	3579665	47777	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	7	2.3	COC(=O)c1c(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c1CCN(C(C)=O)C2	nan
	CHEMBL1550602	47777	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	7	2.3	COC(=O)c1c(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c1CCN(C(C)=O)C2	nan
	5308895	47832	1	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	0	5	4.0	N#CC1=C2SCN(Cc3ccccc3)CN2C(=O)CC1c1cccs1	nan
	CHEMBL1551015	47832	1	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	0	5	4.0	N#CC1=C2SCN(Cc3ccccc3)CN2C(=O)CC1c1cccs1	nan
	16031535	47872	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)s2)cc1	nan
	CHEMBL1551622	47872	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)s2)cc1	nan
	16015115	47881	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.3	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	CHEMBL1551830	47881	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.3	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	15989679	47937	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1OC	nan
	CHEMBL1552471	47937	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1OC	nan
	16030838	47956	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	53229832	47956	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	CHEMBL1552774	47956	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	1004132	47990	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	2	4	4.9	Cc1ccc(CNC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1	nan
	CHEMBL1553209	47990	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	2	4	4.9	Cc1ccc(CNC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1	nan
	15988065	47993	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	2	1	8	3.6	O=c1c2cc3c(cc2nc2sc(Nc4ccc(F)c(Cl)c4)nn12)OCO3	nan
	CHEMBL1553232	47993	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	2	1	8	3.6	O=c1c2cc3c(cc2nc2sc(Nc4ccc(F)c(Cl)c4)nn12)OCO3	nan
	16008431	48000	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	5	4.1	O=C(c1ccc(F)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCO3	nan
	CHEMBL1553329	48000	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	5	4.1	O=C(c1ccc(F)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCO3	nan
	16018243	48003	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	1	1	2	4.1	Cc1c(Cl)cccc1NC(=O)N1CCOc2ccccc21	nan
	CHEMBL1553372	48003	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	1	1	2	4.1	Cc1c(Cl)cccc1NC(=O)N1CCOc2ccccc21	nan
	1364295	48033	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	2	5	5.3	O=C(COc1ccc(Cl)cc1)Nc1ccc(O)c(-c2nc3ccccc3s2)c1	nan
	CHEMBL1553843	48033	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	2	5	5.3	O=C(COc1ccc(Cl)cc1)Nc1ccc(O)c(-c2nc3ccccc3s2)c1	nan
	5302298	48043	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	2	2	5	5.5	Nc1c(C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)sc2nc3c(cc12)N1CCC3CC1	nan
	CHEMBL1554006	48043	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	2	2	5	5.5	Nc1c(C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)sc2nc3c(cc12)N1CCC3CC1	nan
	16018784	48057	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	1	8	3.8	CCc1nnc(SCC(=O)Nc2ccc(OC)c(OC)c2)c2cc3occc3n12	nan
	CHEMBL1554189	48057	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	1	8	3.8	CCc1nnc(SCC(=O)Nc2ccc(OC)c(OC)c2)c2cc3occc3n12	nan
	16018201	48098	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	3	3.8	Cc1ccc2c(c1)N(C(=O)N1CCC(C(=O)NCCc3ccccc3)CC1)CC(C)O2	nan
	CHEMBL1554848	48098	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	3	3.8	Cc1ccc2c(c1)N(C(=O)N1CCC(C(=O)NCCc3ccccc3)CC1)CC(C)O2	nan
	3151378	48174	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	2	7	2.9	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCCC4)c3nc12	nan
	CHEMBL1555780	48174	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	2	7	2.9	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCCC4)c3nc12	nan
	16019891	48376	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	0	9	5.1	CCC(=O)Oc1cc(C(C)(C)C)cc2cc(-c3nc(-c4ccc(OC)cc4OC)no3)c(=O)oc12	nan
	CHEMBL1557596	48376	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	0	9	5.1	CCC(=O)Oc1cc(C(C)(C)C)cc2cc(-c3nc(-c4ccc(OC)cc4OC)no3)c(=O)oc12	nan
	3239255	48466	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	3.8	COc1ccc(-c2nn(C)c3sc(C(=O)NCc4ccco4)cc23)cc1OC	nan
	CHEMBL1558431	48466	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	3.8	COc1ccc(-c2nn(C)c3sc(C(=O)NCc4ccco4)cc23)cc1OC	nan
	662047	48629	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	7	3.8	COc1cccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1559829	48629	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	7	3.8	COc1cccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2612492	48781	6	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	7	3.9	Cc1nc(SCC(=O)Nc2cc(C)on2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1561287	48781	6	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	7	3.9	Cc1nc(SCC(=O)Nc2cc(C)on2)c2c3c(sc2n1)CCCC3	nan
	670483	48791	35	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	2	1	4	3.4	Fc1cccc(-c2nnc(S)n2-c2ccccc2)c1	nan
	CHEMBL1561393	48791	35	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	2	1	4	3.4	Fc1cccc(-c2nnc(S)n2-c2ccccc2)c1	nan
	16025728	48898	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	6	5.8	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3C)s1)C2	nan
	CHEMBL1562331	48898	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	6	5.8	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3C)s1)C2	nan
	135788252	48945	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	8	3.1	COC(=O)c1cc(-c2ccc(OC)cc2F)nc2nc(SC)nc(O)c12	nan
	CHEMBL1562765	48945	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	8	3.1	COC(=O)c1cc(-c2ccc(OC)cc2F)nc2nc(SC)nc(O)c12	nan
	20956964	48946	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	9	0.6	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)CC1	nan
	CHEMBL1562772	48946	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	9	0.6	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)CC1	nan
	15988783	48991	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	7	1	10	2.8	Cc1sc2ncn(CC(=O)Nc3ccc(C(C)C)cc3)c(=O)c2c1S(=O)(=O)N1CCN(c2ncccn2)CC1	nan
	CHEMBL1563146	48991	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	7	1	10	2.8	Cc1sc2ncn(CC(=O)Nc3ccc(C(C)C)cc3)c(=O)c2c1S(=O)(=O)N1CCN(c2ncccn2)CC1	nan
	20923169	49048	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	0	6	2.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)CC(C)C1	nan
	CHEMBL1563711	49048	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	0	6	2.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)CC(C)C1	nan
	16009570	49184	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cn2c(=O)cc(COc3cccc(NC(=O)c4ccccc4C)c3)nc2s1	nan
	CHEMBL1564898	49184	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cn2c(=O)cc(COc3cccc(NC(=O)c4ccccc4C)c3)nc2s1	nan
	22517528	49196	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	3.0	CC1CCN(S(=O)(=O)c2nnc(NC(=O)c3ccccc3Br)s2)CC1	nan
	CHEMBL1564984	49196	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	3.0	CC1CCN(S(=O)(=O)c2nnc(NC(=O)c3ccccc3Br)s2)CC1	nan
	16001900	49633	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	8	2	8	3.6	COc1ccc(CCNc2nc(S)nc3cc(OC)c(OC)cc23)cc1OC	nan
	CHEMBL1568426	49633	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	8	2	8	3.6	COc1ccc(CCNc2nc(S)nc3cc(OC)c(OC)cc23)cc1OC	nan
	2952518	49702	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	571	9	3	9	6.0	CCOc1ccccc1NC(=O)CSC1=C(C#N)C(c2ccco2)C(C(=O)Nc2nc3ccccc3s2)=C(C)N1	nan
	CHEMBL1569028	49702	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	571	9	3	9	6.0	CCOc1ccccc1NC(=O)CSC1=C(C#N)C(c2ccco2)C(C(=O)Nc2nc3ccccc3s2)=C(C)N1	nan
	18562928	49716	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	8	1	8	2.2	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCCC4)nn23)cc1	nan
	CHEMBL1569159	49716	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	8	1	8	2.2	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCCC4)nn23)cc1	nan
	3152775	49941	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3ccc(O)cc3)sc2c1	nan
	CHEMBL1571071	49941	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3ccc(O)cc3)sc2c1	nan
	3564285	50233	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	5036767	50233	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	CHEMBL1573867	50233	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	1325969	50245	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	0	7	5.3	COc1cc(-c2nnc(COc3ccc4cc(Br)ccc4c3)o2)cc(OC)c1OC	nan
	CHEMBL1574014	50245	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	0	7	5.3	COc1cc(-c2nnc(COc3ccc4cc(Br)ccc4c3)o2)cc(OC)c1OC	nan
	3613213	50409	11	None	-1000	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	2	3	4.6	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(F)cc1	nan
	CHEMBL1575774	50409	11	None	-1000	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	2	3	4.6	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(F)cc1	nan
	2352763	50437	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	1	4	2.6	NC(=O)COC(=O)CSc1cccc2cccc(Cl)c12	nan
	CHEMBL1576037	50437	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	1	4	2.6	NC(=O)COC(=O)CSc1cccc2cccc(Cl)c12	nan
	135433192	50728	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	4	3.8	Oc1nc(SCc2ccccc2F)nc2ccccc12	nan
	CHEMBL1578484	50728	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	4	3.8	Oc1nc(SCc2ccccc2F)nc2ccccc12	nan
	18107118	50746	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	5	2.9	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccccn1	nan
	CHEMBL1578588	50746	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	5	2.9	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccccn1	nan
	1838209	50792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	2	8	1.2	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NCc1ccco1	nan
	CHEMBL1578976	50792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	2	8	1.2	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NCc1ccco1	nan
	3802907	50859	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	4542697	50859	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	CHEMBL1579576	50859	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	16196197	50871	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	3610394	50871	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	CHEMBL1579745	50871	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	2357568	50889	7	None	-5	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	6	4.7	O=C(CSc1nnc(-c2cccs2)n1-c1ccccc1)Nc1ccccc1	nan
	CHEMBL1579942	50889	7	None	-5	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	6	4.7	O=C(CSc1nnc(-c2cccs2)n1-c1ccccc1)Nc1ccccc1	nan
	4831734	50918	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	7	1	6	3.8	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2c3c(nc4ccccc24)CCC3)c1	nan
	CHEMBL1580173	50918	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	7	1	6	3.8	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2c3c(nc4ccccc24)CCC3)c1	nan
	1476967	50950	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	0	6	2.0	c1cn(-c2ccc(-c3ccnc4ncnn34)cc2)cn1	nan
	CHEMBL1580435	50950	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	0	6	2.0	c1cn(-c2ccc(-c3ccnc4ncnn34)cc2)cn1	nan
	7190795	50963	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	0	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)c1ccccc1	nan
	CHEMBL1580576	50963	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	0	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)c1ccccc1	nan
	16194926	51037	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	2.5	Cc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1581174	51037	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	2.5	Cc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	3357076	51114	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	5	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccncc2)c1	nan
	CHEMBL1581844	51114	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	5	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccncc2)c1	nan
	3151315	51267	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.9	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1583158	51267	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.9	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CC4CCCO4)c3nc12	nan
	3721854	51384	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	2	1	7	2.1	Nc1c(C(=O)N2CCOCC2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1584034	51384	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	2	1	7	2.1	Nc1c(C(=O)N2CCOCC2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	3911608	51492	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.5	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	CHEMBL1584955	51492	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.5	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	7207569	51671	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	1	7	1.8	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccccc1	nan
	CHEMBL1586420	51671	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	1	7	1.8	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccccc1	nan
	7190486	51767	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1587249	51767	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	5225306	51803	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.9	CC1CCCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1587533	51803	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.9	CC1CCCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	4975167	51816	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	7	1	5	3.1	CCCc1cc(=O)oc2c(C)c(OCC(=O)NCc3ccccn3)ccc12	nan
	CHEMBL1587597	51816	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	7	1	5	3.1	CCCc1cc(=O)oc2c(C)c(OCC(=O)NCc3ccccn3)ccc12	nan
	5236958	51997	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	2.7	CCN(CC)S(=O)(=O)c1ccc(Cl)c(NC(=O)CSc2cccc[n+]2[O-])c1	nan
	CHEMBL1589189	51997	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	2.7	CCN(CC)S(=O)(=O)c1ccc(Cl)c(NC(=O)CSc2cccc[n+]2[O-])c1	nan
	16022898	52082	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	7	1	6	2.7	CCOCCCNc1nc2ccccc2n2c(CC)nnc12	nan
	CHEMBL1589922	52082	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	7	1	6	2.7	CCOCCCNc1nc2ccccc2n2c(CC)nnc12	nan
	16009827	52093	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1OC	nan
	CHEMBL1590063	52093	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1OC	nan
	1391194	52163	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	1391195	52163	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	CHEMBL1590944	52163	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	18572144	52186	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	2	6	2.6	Cn1c(SCC(=O)NCCc2ccccc2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	CHEMBL1591283	52186	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	2	6	2.6	Cn1c(SCC(=O)NCCc2ccccc2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	20903635	52209	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	0	9	1.9	CCCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	CHEMBL1591509	52209	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	0	9	1.9	CCCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	16012276	52232	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	2.3	Cc1cc(C)n2nc(CNC(=O)c3ccc(Cl)cc3)nc2n1	nan
	CHEMBL1591819	52232	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	2.3	Cc1cc(C)n2nc(CNC(=O)c3ccc(Cl)cc3)nc2n1	nan
	5303336	52266	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	4.2	CCOc1ccc(-c2oc3cc(Cl)ccc3c(=O)c2O)cc1OC	nan
	CHEMBL1592283	52266	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	4.2	CCOc1ccc(-c2oc3cc(Cl)ccc3c(=O)c2O)cc1OC	nan
	2790635	52376	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	2	4	4.1	Cc1ccc(OCCCC(=O)Nc2sc3c(c2C(N)=O)CCC(C)C3)cc1	nan
	CHEMBL1593935	52376	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	2	4	4.1	Cc1ccc(OCCCC(=O)Nc2sc3c(c2C(N)=O)CCC(C)C3)cc1	nan
	3476583	52560	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1595488	52560	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	1958370	52578	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	2.5	COCCNS(=O)(=O)c1cc(-c2nn3c(C)nnc3c3ccccc23)ccc1C	nan
	CHEMBL1595653	52578	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	2.5	COCCNS(=O)(=O)c1cc(-c2nn3c(C)nnc3c3ccccc23)ccc1C	nan
	4601439	52752	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	2	7	3.9	COc1cccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)c1	nan
	CHEMBL1597228	52752	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	2	7	3.9	COc1cccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)c1	nan
	4151069	52964	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	10	0.6	COC(=O)c1cc(NS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc(C(=O)OC)c1	nan
	CHEMBL1599214	52964	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	10	0.6	COC(=O)c1cc(NS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc(C(=O)OC)c1	nan
	2890665	53036	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	3	1	3	3.6	CC(=O)C1=C(O)C(=O)N(c2ccc(F)cc2)C1c1ccc(C)cc1	nan
	CHEMBL1599834	53036	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	3	1	3	3.6	CC(=O)C1=C(O)C(=O)N(c2ccc(F)cc2)C1c1ccc(C)cc1	nan
	16020305	53353	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	12	1	6	4.3	CCCN(CCC)C(=O)Cn1c(=O)n(-c2ccc(CC)cc2)c(=O)c2ccc(C(=O)NCCc3ccccc3)cc21	nan
	CHEMBL1602912	53353	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	12	1	6	4.3	CCCN(CCC)C(=O)Cn1c(=O)n(-c2ccc(CC)cc2)c(=O)c2ccc(C(=O)NCCc3ccccc3)cc21	nan
	910705	53440	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	2	0	4	2.4	O=[N+]([O-])c1ccc(-c2cn3c(n2)CCC3)cc1	nan
	CHEMBL1603668	53440	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	2	0	4	2.4	O=[N+]([O-])c1ccc(-c2cn3c(n2)CCC3)cc1	nan
	1146176	53588	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	0	4	4.7	CC1CCN(C(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)n2)CC1	nan
	CHEMBL1604923	53588	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	0	4	4.7	CC1CCN(C(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)n2)CC1	nan
	16019480	53677	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	0	9	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCN(CC)CC2)c2sccc23)cc1	nan
	CHEMBL1605620	53677	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	0	9	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCN(CC)CC2)c2sccc23)cc1	nan
	1410148	53791	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.5	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccnc4)nc3c2)cc1	nan
	CHEMBL1606536	53791	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.5	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccnc4)nc3c2)cc1	nan
	2918495	53823	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	8	2.5	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1OC	nan
	CHEMBL1606762	53823	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	8	2.5	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1OC	nan
	5730347	53873	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	4	0	4	3.9	CCC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	CHEMBL1607132	53873	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	4	0	4	3.9	CCC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	4426797	53957	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	10	-0.6	Cn1c(=O)c2c(nc(CN3CCN(C(=O)c4ccco4)CC3)n2CCCO)n(C)c1=O	nan
	CHEMBL1607800	53957	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	10	-0.6	Cn1c(=O)c2c(nc(CN3CCN(C(=O)c4ccco4)CC3)n2CCCO)n(C)c1=O	nan
	1325691	53990	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	1	1	7	3.2	Sc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1608119	53990	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	1	1	7	3.2	Sc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CCCC3	nan
	2966904	53994	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	7	2	7	3.4	CC(=O)c1sc2nc(SCC(=O)NCCc3ccccc3)nc(O)c2c1C	nan
	CHEMBL1608140	53994	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	7	2	7	3.4	CC(=O)c1sc2nc(SCC(=O)NCCc3ccccc3)nc(O)c2c1C	nan
	16406841	54000	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	6	3.1	Cc1c(Br)c(=O)oc2cc(OCC(=O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)ccc12	nan
	CHEMBL1608190	54000	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	6	3.1	Cc1c(Br)c(=O)oc2cc(OCC(=O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)ccc12	nan
	54686430	54065	29	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	2	4	1.8	CCCNC(=O)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	CHEMBL1608771	54065	29	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	2	4	1.8	CCCNC(=O)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	6107794	54123	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	7	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c(OC)c1	nan
	CHEMBL1609202	54123	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	7	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c(OC)c1	nan
	2576098	54155	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	2.7	Cc1sc2ncnc(NCCCN3CCCC3=O)c2c1C	nan
	CHEMBL1609414	54155	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	2.7	Cc1sc2ncnc(NCCCN3CCCC3=O)c2c1C	nan
	3641030	54211	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	3	5.1	CC(=O)c1ccc(NC(=O)c2ccc(-c3ccc(Cl)cc3)o2)cc1	nan
	CHEMBL1609950	54211	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	3	5.1	CC(=O)c1ccc(NC(=O)c2ccc(-c3ccc(Cl)cc3)o2)cc1	nan
	2868074	54229	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccc(Br)cc1	nan
	CHEMBL1610073	54229	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccc(Br)cc1	nan
	2790804	54340	14	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	6	3.8	O=[N+]([O-])c1ccc(-c2nc(NCC3CCCO3)c3ccccc3n2)cc1	nan
	CHEMBL1611050	54340	14	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	6	3.8	O=[N+]([O-])c1ccc(-c2nc(NCC3CCCO3)c3ccccc3n2)cc1	nan
	2934073	54591	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccc(Cl)c1)c1ccco1	nan
	CHEMBL1613356	54591	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccc(Cl)c1)c1ccco1	nan
	4581262	55025	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	CHEMBL1377318	55025	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	CHEMBL1618739	55025	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	1099157	55051	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	CHEMBL1389219	55051	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	CHEMBL1618947	55051	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	4055296	55177	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	CHEMBL1420869	55177	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	CHEMBL1620041	55177	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	655842	55324	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1466356	55324	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1621365	55324	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	3848238	55698	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	CHEMBL1548688	55698	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	CHEMBL1624498	55698	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	3589783	55711	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	CHEMBL1566042	55711	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	CHEMBL1624662	55711	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	9560158	71839	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1980603	71839	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	9624156	71913	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	4.4	N#CCC(=O)N/N=C/c1ccc(N2N=C(c3ccccc3)CC2c2ccccc2)cc1	nan
	CHEMBL1982521	71913	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	4.4	N#CCC(=O)N/N=C/c1ccc(N2N=C(c3ccccc3)CC2c2ccccc2)cc1	nan
	1995859	72443	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	7	1.3	COCCCn1/c(=N/C(C)=O)c(C#N)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL2000901	72443	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	7	1.3	COCCCn1/c(=N/C(C)=O)c(C#N)cc2c(=O)n3cccc(C)c3nc21	nan
	65599	104930	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL311948	104930	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	2864416	106390	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	1.6	Cc1[nH]n(-c2ccc([N+](=O)[O-])cc2)c(=O)c1/C=N/CCN1CCN(C(=O)C(C)C)CC1	nan
	CHEMBL3145301	106390	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	1.6	Cc1[nH]n(-c2ccc([N+](=O)[O-])cc2)c(=O)c1/C=N/CCN1CCN(C(=O)C(C)C)CC1	nan
	5935610	107108	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	1	1	3	3.9	CCn1c2c(c3cc(Br)ccc31)CCC/C2=N\O	nan
	CHEMBL3189713	107108	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	1	1	3	3.9	CCn1c2c(c3cc(Br)ccc31)CCC/C2=N\O	nan
	6279969	107385	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	0	6	2.1	CN(C)/C=N/c1nc2nccc(-c3cccs3)n2n1	nan
	CHEMBL3192852	107385	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	0	6	2.1	CN(C)/C=N/c1nc2nccc(-c3cccs3)n2n1	nan
	6860035	107617	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	8	3.0	COc1ccc(OC)c(/C=N/n2c(S)nnc2COc2ccccc2)c1	nan
	CHEMBL3195667	107617	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	8	3.0	COc1ccc(OC)c(/C=N/n2c(S)nnc2COc2ccccc2)c1	nan
	135467322	108197	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	6	4.3	COC(=O)/C(Nc1ccccc1)=C(\C(=O)C(=O)N(C)c1ccccc1)C(=O)c1ccc(Cl)cc1	nan
	CHEMBL3208147	108197	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	6	4.3	COC(=O)/C(Nc1ccccc1)=C(\C(=O)C(=O)N(C)c1ccccc1)C(=O)c1ccc(Cl)cc1	nan
	2805193	108310	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	5	1	7	2.6	CCO/C(O)=C(C#N)/C=N/c1ccsc1C(=O)OC	nan
	CHEMBL3209558	108310	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	5	1	7	2.6	CCO/C(O)=C(C#N)/C=N/c1ccsc1C(=O)OC	nan
	5867179	108518	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.1	C/C(N)=C(/C#N)C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL3212349	108518	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.1	C/C(N)=C(/C#N)C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	3221537	112109	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	CHEMBL3209727	112109	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	CHEMBL3302425	112109	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	264006	177978	14	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	4	9	-1.0	C=CCNc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	CHEMBL46703	177978	14	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	4	9	-1.0	C=CCNc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	833435	195983	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	3	4	2.9	Cc1sc(NC(=S)NC(=O)C2CCCCC2)c(C(N)=O)c1C	nan
	CHEMBL571065	195983	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	3	4	2.9	Cc1sc(NC(=S)NC(=O)C2CCCCC2)c(C(N)=O)c1C	nan
	22334103	199215	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	9	2	8	1.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1Cl	nan
	CHEMBL601585	199215	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	9	2	8	1.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1Cl	nan
	4167655	28024	11	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.3	Brc1ccc(-c2nnc3sc(CNC4CCCC4)cn23)cc1	nan
	CHEMBL1374064	28024	11	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.3	Brc1ccc(-c2nnc3sc(CNC4CCCC4)cn23)cc1	nan
	16018920	28258	5	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	6	4.8	CCc1nnc(SCC(=O)Nc2ccc(F)cc2F)c2cc3sc(C)cc3n12	nan
	CHEMBL1375688	28258	5	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	6	4.8	CCc1nnc(SCC(=O)Nc2ccc(F)cc2F)c2cc3sc(C)cc3n12	nan
	3348974	38940	9	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	11	0.5	CCc1nnc(NC(=O)CSc2nc(C)nc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1469832	38940	9	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	11	0.5	CCc1nnc(NC(=O)CSc2nc(C)nc3c2c(=O)n(C)c(=O)n3C)s1	nan
	4351083	46888	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	8	3.0	O=C(NN1C(=O)c2ccccc2NC1c1ccc([N+](=O)[O-])o1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1543122	46888	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	8	3.0	O=C(NN1C(=O)c2ccccc2NC1c1ccc([N+](=O)[O-])o1)c1ccc([N+](=O)[O-])cc1	nan
	3241486	49639	5	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	6	4.2	COc1ccc(C(=O)Nc2ccc(N3CCN(c4ccc(OC)cc4)CC3)c(C#N)c2)cc1	nan
	CHEMBL1568468	49639	5	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	6	4.2	COc1ccc(C(=O)Nc2ccc(N3CCN(c4ccc(OC)cc4)CC3)c(C#N)c2)cc1	nan
	1261644	49795	10	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	1	4	4.7	O=C(Nc1ccncc1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	CHEMBL1569872	49795	10	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	1	4	4.7	O=C(Nc1ccncc1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	759120	52268	31	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1592299	52268	31	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	16010305	7577	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	3.2	COCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccc(Cl)cc12	nan
	CHEMBL1088575	7577	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	3.2	COCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccc(Cl)cc12	nan
	16019548	10766	9	None	-23	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	8	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(Cl)cc1)c1sccc12	nan
	CHEMBL1172597	10766	9	None	-23	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	8	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(Cl)cc1)c1sccc12	nan
	16019364	10840	5	None	-53	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	8	4.5	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1C	nan
	CHEMBL1173283	10840	5	None	-53	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	8	4.5	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1C	nan
	5721990	14642	23	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	0	2	4.5	CN(C)c1ccc(/C=C/c2ccc3ccccc3n2)cc1	nan
	CHEMBL120734	14642	23	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	0	2	4.5	CN(C)c1ccc(/C=C/c2ccc3ccccc3n2)cc1	nan
	3565	19161	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	CHEMBL129177	19161	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	CHEMBL1473205	19161	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	2803232	19304	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	2	4.3	S=C(Nc1ccccc1)Nc1ccccc1-n1cccc1	nan
	CHEMBL1299459	19304	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	2	4.3	S=C(Nc1ccccc1)Nc1ccccc1-n1cccc1	nan
	1305405	19460	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	3	4	4.4	O=C(O)c1ccccc1NC(=S)NC(=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1300720	19460	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	3	4	4.4	O=C(O)c1ccccc1NC(=S)NC(=O)c1sc2ccccc2c1Cl	nan
	24790327	19495	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	5	4.4	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cnn(C(C)C)c4)C3)ccc2c1	nan
	CHEMBL1300972	19495	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	5	4.4	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cnn(C(C)C)c4)C3)ccc2c1	nan
	5826640	19563	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	7	4.1	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1301431	19563	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	7	4.1	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	2410711	19582	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	3.5	CCOc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	CHEMBL1301615	19582	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	3.5	CCOc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	5918716	19651	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	7	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NC)CC1	nan
	CHEMBL1302267	19651	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	7	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NC)CC1	nan
	910973	19778	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	1	2	6	1.6	N#CC(C#N)=C1NC(N)=C(C#N)C(c2ccccc2)=C1C#N	nan
	CHEMBL1303255	19778	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	1	2	6	1.6	N#CC(C#N)=C1NC(N)=C(C#N)C(c2ccccc2)=C1C#N	nan
	2472728	19952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	7	2.7	Cc1sc2ncnc(SCC(=O)NC(=O)c3cccn3C)c2c1C	nan
	CHEMBL1304667	19952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	7	2.7	Cc1sc2ncnc(SCC(=O)NC(=O)c3cccn3C)c2c1C	nan
	3544771	19974	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	0	9	3.2	O=c1c2sccc2nc(SCc2cc(=O)n3ccccc3n2)n1Cc1ccccn1	nan
	CHEMBL1304859	19974	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	0	9	3.2	O=c1c2sccc2nc(SCc2cc(=O)n3ccccc3n2)n1Cc1ccccn1	nan
	7295015	20114	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.6	CSc1ccccc1-c1nnc(NC(=O)Cc2ccccc2)o1	nan
	CHEMBL1305973	20114	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.6	CSc1ccccc1-c1nnc(NC(=O)Cc2ccccc2)o1	nan
	654420	20117	4	None	-28	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	5	0	5	2.8	CCOC(=O)CSc1nc(CC)nc2ccccc12	nan
	CHEMBL1305990	20117	4	None	-28	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	5	0	5	2.8	CCOC(=O)CSc1nc(CC)nc2ccccc12	nan
	4021231	20127	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.7	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc(F)cc4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1306067	20127	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.7	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc(F)cc4)c(=N)n(CC4CCCO4)c3nc12	nan
	833786	20178	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	3	1	4	4.2	Sc1nc(SCc2ccccc2)nc2ccccc12	nan
	CHEMBL1306480	20178	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	3	1	4	4.2	Sc1nc(SCc2ccccc2)nc2ccccc12	nan
	865618	20189	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	0	4	3.6	CN(C)c1ccc(-c2nnc(-c3ccccc3F)o2)cc1	nan
	CHEMBL1306590	20189	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	0	4	3.6	CN(C)c1ccc(-c2nnc(-c3ccccc3F)o2)cc1	nan
	6078291	20296	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1307444	20296	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2820469	20375	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	3.4	CSc1sc(C(=O)NCC2CC2)c2c1S(=O)(=O)N(C)c1ccccc1-2	nan
	CHEMBL1308054	20375	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	3.4	CSc1sc(C(=O)NCC2CC2)c2c1S(=O)(=O)N(C)c1ccccc1-2	nan
	5012705	20385	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	9	2	6	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCCc1ccccc1	nan
	CHEMBL1308124	20385	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	9	2	6	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCCc1ccccc1	nan
	1201985	20535	9	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	6	3.8	O=C(CSc1nc2ccccc2nc1SCC(=O)N1CCCCC1)N1CCCCC1	nan
	CHEMBL1309335	20535	9	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	6	3.8	O=C(CSc1nc2ccccc2nc1SCC(=O)N1CCCCC1)N1CCCCC1	nan
	24891893	20543	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	9	-0.0	CCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1309394	20543	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	9	-0.0	CCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	1596915	20557	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	7	4.6	Cc1csc(NC(=O)c2sc3nc(-c4cccs4)ccc3c2N)n1	nan
	CHEMBL1309478	20557	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	7	4.6	Cc1csc(NC(=O)c2sc3nc(-c4cccs4)ccc3c2N)n1	nan
	3236246	20639	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	7	1	8	2.8	CCC(Sc1ccc2nnc(-c3ccc(OC)c(OC)c3)n2n1)C(=O)O	nan
	CHEMBL1310295	20639	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	7	1	8	2.8	CCC(Sc1ccc2nnc(-c3ccc(OC)c(OC)c3)n2n1)C(=O)O	nan
	4881170	20746	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	0	6	3.0	Cc1nc(SC2CCOC2=O)c2c(C)c(C)sc2n1	nan
	CHEMBL1311178	20746	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	0	6	3.0	Cc1nc(SC2CCOC2=O)c2c(C)c(C)sc2n1	nan
	5813760	20792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccc(Br)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1311567	20792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccc(Br)cc1)c1ccc2c(c1)OCCO2	nan
	3682235	20867	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1312109	20867	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	3588555	20946	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	580	5	1	8	3.8	Cc1cc(Br)ccc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	CHEMBL1312634	20946	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	580	5	1	8	3.8	Cc1cc(Br)ccc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	2332949	20957	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	2	5	4.7	Cc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2C)o1	nan
	CHEMBL1312698	20957	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	2	5	4.7	Cc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2C)o1	nan
	20957089	20966	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	9	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCc4ccco4)nn23)CC1	nan
	CHEMBL1312760	20966	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	9	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCc4ccco4)nn23)CC1	nan
	7064857	21258	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	5.1	CCc1cccc(C)c1Nc1c(-c2ccc(N(C)C)cc2)nc2cnccn12	nan
	CHEMBL1315626	21258	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	5.1	CCc1cccc(C)c1Nc1c(-c2ccc(N(C)C)cc2)nc2cnccn12	nan
	16299684	21269	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(NC(=O)c2nn(C)c(=O)c3ccccc23)c1	nan
	CHEMBL1315774	21269	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(NC(=O)c2nn(C)c(=O)c3ccccc23)c1	nan
	16010795	21279	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	1	8	2.8	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	CHEMBL1315899	21279	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	1	8	2.8	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	16018148	21359	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	4	4.4	CCn1cc2c(n1)-c1c(oc(C(=O)Nc3cccc(C)c3C)c1C)CC2	nan
	CHEMBL1316992	21359	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	4	4.4	CCn1cc2c(n1)-c1c(oc(C(=O)Nc3cccc(C)c3C)c1C)CC2	nan
	5921518	21417	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	8	2.1	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(c3ccccc3)CC2)nc2ccccn2c1=O	nan
	CHEMBL1317700	21417	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	8	2.1	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(c3ccccc3)CC2)nc2ccccn2c1=O	nan
	4062026	21464	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	6	4.5	Cc1ccc(Cl)cc1NC(=O)c1oc2ccc(S(=O)(=O)N3CCC4(CC3)OCCO4)cc2c1C	nan
	CHEMBL1318364	21464	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	6	4.5	Cc1ccc(Cl)cc1NC(=O)c1oc2ccc(S(=O)(=O)N3CCC4(CC3)OCCO4)cc2c1C	nan
	16027568	21465	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	CHEMBL1318374	21465	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	16028281	21479	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	7	3.4	CCc1cccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)c1	nan
	CHEMBL1318465	21479	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	7	3.4	CCc1cccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)c1	nan
	16017220	21500	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	8	1	6	4.8	Cc1nn(CCCC(=O)NCc2ccc(OC(C)C)cc2)c(=O)c2c1sc1ccccc12	nan
	CHEMBL1318645	21500	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	8	1	6	4.8	Cc1nn(CCCC(=O)NCc2ccc(OC(C)C)cc2)c(=O)c2c1sc1ccccc12	nan
	16027652	21551	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	8	4.3	CC(C)Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1319006	21551	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	8	4.3	CC(C)Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	2998240	21658	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	5	4.2	O=C(NCc1ccc(Cl)cc1)c1cc2c(nc3sccn32)s1	nan
	CHEMBL1319990	21658	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	5	4.2	O=C(NCc1ccc(Cl)cc1)c1cc2c(nc3sccn32)s1	nan
	16007411	21676	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	2	3	4.4	CC(C)c1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1	nan
	CHEMBL1320105	21676	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	2	3	4.4	CC(C)c1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1	nan
	7692481	21714	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	3	3.4	COc1cc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2cc1OC	nan
	CHEMBL1320436	21714	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	3	3.4	COc1cc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2cc1OC	nan
	16019337	21784	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)cc1C	nan
	CHEMBL1321011	21784	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)cc1C	nan
	16017632	21827	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	3	2	6	5.0	Cc1c(C(=O)Nc2ccccc2)sc2nc(-c3cc4cc(Cl)ccc4oc3=O)[nH]c(=O)c12	nan
	CHEMBL1321440	21827	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	3	2	6	5.0	Cc1c(C(=O)Nc2ccccc2)sc2nc(-c3cc4cc(Cl)ccc4oc3=O)[nH]c(=O)c12	nan
	15988428	21829	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	5	3.6	Cn1c(=O)n(-c2cccc(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1321495	21829	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	5	3.6	Cn1c(=O)n(-c2cccc(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	2988303	21831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	6	3.2	Cn1c2ccc(F)cc2c2nnc(SCCN3CCCCC3)nc21	nan
	CHEMBL1321509	21831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	6	3.2	Cn1c2ccc(F)cc2c2nnc(SCCN3CCCCC3)nc21	nan
	16017566	21862	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1321733	21862	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	2158383	22015	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1323129	22015	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	6076700	22147	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	10	2	7	2.1	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2cccnc2)cc1	nan
	CHEMBL1324242	22147	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	10	2	7	2.1	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2cccnc2)cc1	nan
	16805712	22191	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	2	9	1.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccc(S(N)(=O)=O)cc3)nnc12	nan
	CHEMBL1324587	22191	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	2	9	1.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccc(S(N)(=O)=O)cc3)nnc12	nan
	3152453	22429	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	8	1.1	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CCCO)c3nc12	nan
	CHEMBL1326883	22429	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	8	1.1	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CCCO)c3nc12	nan
	5048043	22651	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1328648	22651	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	135706200	22674	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	3.2	CN(Cc1nc(O)c2ccccc2n1)C(=O)c1cccc(S(=O)(=O)N2CCCCCC2)c1	nan
	CHEMBL1328897	22674	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	3.2	CN(Cc1nc(O)c2ccccc2n1)C(=O)c1cccc(S(=O)(=O)N2CCCCCC2)c1	nan
	5730619	22699	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C\C(=O)c3ccncc3)cc2)c1C	nan
	CHEMBL1329130	22699	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C\C(=O)c3ccncc3)cc2)c1C	nan
	2937900	22734	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	4.3	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1ccccc1F)c1cccs1	nan
	CHEMBL1329400	22734	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	4.3	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1ccccc1F)c1cccs1	nan
	2765497	22748	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	2.4	Cc1ccc(S(=O)(=O)C(C)C(=O)NCCS(=O)(=O)c2ccc(Cl)cc2)cc1	nan
	CHEMBL1329544	22748	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	2.4	Cc1ccc(S(=O)(=O)C(C)C(=O)NCCS(=O)(=O)c2ccc(Cl)cc2)cc1	nan
	44142302	22751	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	2.8	CN(C)c1ccc(C#Cc2ccc3cc(CCO)oc(=O)c3c2)cc1	nan
	CHEMBL1329575	22751	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	2.8	CN(C)c1ccc(C#Cc2ccc3cc(CCO)oc(=O)c3c2)cc1	nan
	16011595	22804	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	7	4.7	CCCCOc1ccc(CNC(=O)C2CCCN(c3nnc(-n4c(C)ccc4C)s3)C2)cc1	nan
	CHEMBL1330008	22804	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	7	4.7	CCCCOc1ccc(CNC(=O)C2CCCN(c3nnc(-n4c(C)ccc4C)s3)C2)cc1	nan
	4181210	22828	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	3.9	Cc1ccc(NC(=O)CSc2nnc3ccc4ccccc4n23)cc1	nan
	CHEMBL1330254	22828	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	3.9	Cc1ccc(NC(=O)CSc2nnc3ccc4ccccc4n23)cc1	nan
	1548033	22830	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	3	3	7	-0.6	CN(C)C(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1330266	22830	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	3	3	7	-0.6	CN(C)C(=O)CNc1nnc(S)nc1O	nan
	1960924	22922	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	4	6	2.4	COc1ccc(C(=O)NC(=S)Nc2ccc3[nH]c(O)nc3c2)c(OC)c1	nan
	CHEMBL1330933	22922	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	4	6	2.4	COc1ccc(C(=O)NC(=S)Nc2ccc3[nH]c(O)nc3c2)c(OC)c1	nan
	16022880	22991	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	2	7	4.3	COc1ccccc1NC(=O)Cn1c(=O)c(CNc2ccccc2)cc2cc(OC)c(OC)cc21	nan
	CHEMBL1331405	22991	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	2	7	4.3	COc1ccccc1NC(=O)Cn1c(=O)c(CNc2ccccc2)cc2cc(OC)c(OC)cc21	nan
	995088	23030	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	4	4.9	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3C)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1331738	23030	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	4	4.9	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3C)c3cc(Br)ccc3n2)cc1	nan
	4975488	23213	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	0	8	1.8	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(C)CC4)o3)nnc2c2ccccc12	nan
	CHEMBL1333127	23213	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	0	8	1.8	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(C)CC4)o3)nnc2c2ccccc12	nan
	5219389	23272	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	2.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc3ccccc3oc2=O)c1	nan
	CHEMBL1333624	23272	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	2.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc3ccccc3oc2=O)c1	nan
	1298840	23282	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.1	CCn1c(SCC(=O)Nc2nc3ccccc3s2)nnc1-c1ccc(Br)cc1	nan
	CHEMBL1333690	23282	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.1	CCn1c(SCC(=O)Nc2nc3ccccc3s2)nnc1-c1ccc(Br)cc1	nan
	3586634	23303	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	5.2	CCCCn1c(SCC(=O)Nc2cccc(OC)c2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1333854	23303	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	5.2	CCCCn1c(SCC(=O)Nc2cccc(OC)c2)nc2c(sc3ccccc32)c1=O	nan
	1088584	23308	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	3	3.8	CC(=O)c1cn(CC(=O)Nc2ccc(C)cc2)c2ccccc12	nan
	CHEMBL1333897	23308	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	3	3.8	CC(=O)c1cn(CC(=O)Nc2ccc(C)cc2)c2ccccc12	nan
	1912959	23417	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5728937	23417	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5925428	23417	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	CHEMBL1334749	23417	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5302178	23434	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	CHEMBL1334923	23434	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	15988344	23524	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	7	4.6	COc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2Cl)cc1	nan
	CHEMBL1335550	23524	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	7	4.6	COc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2Cl)cc1	nan
	3236871	23564	7	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	0	2	3.7	CCn1c(C)cc(=S)c2ccccc21	nan
	CHEMBL1335833	23564	7	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	0	2	3.7	CCn1c(C)cc(=S)c2ccccc21	nan
	3323389	23583	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	2	7	4.0	CC(=O)c1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	CHEMBL1336041	23583	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	2	7	4.0	CC(=O)c1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	135413771	23674	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	4.9	COc1cc(C2CC(c3c(C)cc(C)nc3O)=NN2c2ccccc2F)cc(OC)c1OC	nan
	CHEMBL1336821	23674	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	4.9	COc1cc(C2CC(c3c(C)cc(C)nc3O)=NN2c2ccccc2F)cc(OC)c1OC	nan
	2140203	23679	1	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	3	0	7	2.9	COc1ccc(-n2nnnc2-c2nc3ccccc3s2)cc1	nan
	CHEMBL1336848	23679	1	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	3	0	7	2.9	COc1ccc(-n2nnnc2-c2nc3ccccc3s2)cc1	nan
	2088251	23725	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	6	3.1	CCOc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1	nan
	CHEMBL1337298	23725	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	6	3.1	CCOc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1	nan
	1301366	23740	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	5	4.1	O=C(CCSc1nnc2ccc3ccccc3n12)Nc1ccc(F)cc1	nan
	CHEMBL1337428	23740	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	5	4.1	O=C(CCSc1nnc2ccc3ccccc3n12)Nc1ccc(F)cc1	nan
	16015123	23782	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1cccc(C)c1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	CHEMBL1337810	23782	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1cccc(C)c1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	16034823	23807	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	1	4	4.9	Cc1oc(-c2cccc(Br)c2)nc1CN1CCC(C(=O)NCc2ccccc2)CC1	nan
	CHEMBL1338052	23807	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	1	4	4.9	Cc1oc(-c2cccc(Br)c2)nc1CN1CCC(C(=O)NCc2ccccc2)CC1	nan
	2137854	23911	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1338842	23911	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	16023227	23925	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	2	6	4.7	O=C(Cn1c(=O)c(CNc2ccccc2)cc2cc3c(cc21)OCCO3)Nc1ccccc1Cl	nan
	CHEMBL1339042	23925	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	2	6	4.7	O=C(Cn1c(=O)c(CNc2ccccc2)cc2cc3c(cc21)OCCO3)Nc1ccccc1Cl	nan
	4012037	23995	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	5	4.3	c1coc(CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1339672	23995	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	5	4.3	c1coc(CSc2ncnc3c2oc2ccccc23)c1	nan
	16406923	24134	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	3	6	2.3	Cc1coc2c1c(C)cc1oc(=O)c(CC(=O)NCC(=O)N[C@H](C(=O)O)C(C)C)c(C)c12	nan
	CHEMBL1340985	24134	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	3	6	2.3	Cc1coc2c1c(C)cc1oc(=O)c(CC(=O)NCC(=O)N[C@H](C(=O)O)C(C)C)c(C)c12	nan
	1859832	24181	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	0	7	4.3	COc1ccc(CCn2c(-c3ccc(F)cc3)nc3c(c(=O)c4ccccc4n3C)c2=O)cc1OC	nan
	CHEMBL1341311	24181	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	0	7	4.3	COc1ccc(CCn2c(-c3ccc(F)cc3)nc3c(c(=O)c4ccccc4n3C)c2=O)cc1OC	nan
	6402475	24416	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	4	4.2	Nc1nc(-c2ccc(Cl)cc2)nnc1-c1ccc(Br)cc1	nan
	CHEMBL1343242	24416	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	4	4.2	Nc1nc(-c2ccc(Cl)cc2)nnc1-c1ccc(Br)cc1	nan
	1831284	24446	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	4401304	24446	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	CHEMBL1343474	24446	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	3238813	24459	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	5	3.8	COc1ccc(-c2cc(C(=O)Nc3cccc(C(C)=O)c3)no2)cc1	nan
	CHEMBL1343596	24459	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	5	3.8	COc1ccc(-c2cc(C(=O)Nc3cccc(C(C)=O)c3)no2)cc1	nan
	2821813	24528	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	3	4.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc2ncsc2c1	nan
	CHEMBL1344238	24528	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	3	4.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc2ncsc2c1	nan
	3158796	24604	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	2	2	5	2.9	Cc1cccc(N2C(S)=C(C#N)C(=O)NC2c2ccco2)c1	nan
	CHEMBL1344888	24604	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	2	2	5	2.9	Cc1cccc(N2C(S)=C(C#N)C(=O)NC2c2ccco2)c1	nan
	2558333	24672	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	9	4.8	CCc1cc2c(SCc3nc(O)c4c(C)c(C(C)=O)sc4n3)ncnc2s1	nan
	CHEMBL1345471	24672	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	9	4.8	CCc1cc2c(SCc3nc(O)c4c(C)c(C(C)=O)sc4n3)ncnc2s1	nan
	7708092	24729	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	7	2.8	COc1ccc(C(=O)Nc2nnc(S(=O)(=O)Cc3ccccc3)s2)cc1	nan
	CHEMBL1346001	24729	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	7	2.8	COc1ccc(C(=O)Nc2nnc(S(=O)(=O)Cc3ccccc3)s2)cc1	nan
	4519571	24880	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	6	2.9	O=c1c2cc(Cl)ccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	CHEMBL1347185	24880	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	6	2.9	O=c1c2cc(Cl)ccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	24790251	25044	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	4	4.2	O=C(NCC1CCOCC1)c1ccc2nc(Cc3cccc(Cl)c3)oc2c1	nan
	CHEMBL1348671	25044	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	4	4.2	O=C(NCC1CCOCC1)c1ccc2nc(Cc3cccc(Cl)c3)oc2c1	nan
	16194270	25150	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.6	COc1cccc(CNC(=O)CSc2ccc(-c3cccs3)nn2)c1	nan
	CHEMBL1349515	25150	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.6	COc1cccc(CNC(=O)CSc2ccc(-c3cccs3)nn2)c1	nan
	2308471	25225	6	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	0	5	5.7	N#Cc1c(-c2ccc(F)cc2)cc(C2CC2)nc1SCC(=O)c1cccs1	nan
	CHEMBL1350179	25225	6	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	0	5	5.7	N#Cc1c(-c2ccc(F)cc2)cc(C2CC2)nc1SCC(=O)c1cccs1	nan
	1246228	25299	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	4.5	Cc1sc(NC(=O)c2oc3ccccc3c2C)c(C#N)c1C	nan
	CHEMBL1350806	25299	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	4.5	Cc1sc(NC(=O)c2oc3ccccc3c2C)c(C#N)c1C	nan
	3810755	25477	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	5224304	25477	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	CHEMBL1352306	25477	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	3710699	25589	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	0	5	3.2	CSc1nnc(-c2ccccc2SC)o1	nan
	CHEMBL1353167	25589	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	0	5	3.2	CSc1nnc(-c2ccccc2SC)o1	nan
	2408978	25684	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	4	3.8	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(Br)cc1	nan
	CHEMBL1353794	25684	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	4	3.8	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(Br)cc1	nan
	2137114	25773	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	5	4.4	Cc1ccc(C)c(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)c1	nan
	CHEMBL1354500	25773	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	5	4.4	Cc1ccc(C)c(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)c1	nan
	7177775	25802	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	4	0	7	1.8	Cc1ccc2nc(SCC(=O)N3CCN(c4ccccc4)CC3)nc(=O)n2c1	nan
	CHEMBL1354880	25802	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	4	0	7	1.8	Cc1ccc2nc(SCC(=O)N3CCN(c4ccccc4)CC3)nc(=O)n2c1	nan
	16015313	25806	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	5.8	COc1cccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4Cl)c3C)nc2C)c1	nan
	CHEMBL1354922	25806	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	5.8	COc1cccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4Cl)c3C)nc2C)c1	nan
	16019333	25807	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.8	CCc1ccc(Nc2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)cc1	nan
	CHEMBL1354928	25807	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.8	CCc1ccc(Nc2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)cc1	nan
	15988332	25837	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	0	9	2.1	CC(=O)c1ccc(N2CCN(C(=O)CCc3nnc4n(C)c(=O)c5sccc5n34)CC2)cc1	nan
	CHEMBL1355272	25837	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	0	9	2.1	CC(=O)c1ccc(N2CCN(C(=O)CCc3nnc4n(C)c(=O)c5sccc5n34)CC2)cc1	nan
	15988502	25870	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	4	4.5	O=C(Cn1c(=O)nc(-c2ccccc2)c2ccccc21)Nc1ccc(Cl)cc1F	nan
	CHEMBL1355773	25870	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	4	4.5	O=C(Cn1c(=O)nc(-c2ccccc2)c2ccccc21)Nc1ccc(Cl)cc1F	nan
	2893260	25975	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	9	4.0	CCC(Sc1nnc2c3ccccc3n(C)c2n1)C(=O)Nc1nnc(C(C)C)s1	nan
	CHEMBL1357131	25975	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	9	4.0	CCC(Sc1nnc2c3ccccc3n(C)c2n1)C(=O)Nc1nnc(C(C)C)s1	nan
	16018894	25983	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	0	7	5.8	CCc1nnc(SCc2nc(-c3ccccc3)oc2C)c2cc3sccc3n12	nan
	CHEMBL1357169	25983	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	0	7	5.8	CCc1nnc(SCc2nc(-c3ccccc3)oc2C)c2cc3sccc3n12	nan
	16012142	26019	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	5.0	CC(CNC(=O)Cn1ncc2c3ccccc3n(Cc3cccc(Cl)c3)c2c1=O)c1ccccc1	nan
	CHEMBL1357797	26019	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	5.0	CC(CNC(=O)Cn1ncc2c3ccccc3n(Cc3cccc(Cl)c3)c2c1=O)c1ccccc1	nan
	16018042	26037	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	5	3.2	CN(C)c1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1358052	26037	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	5	3.2	CN(C)c1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	7711889	26097	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	0.2	Cn1c(CNS(=O)(=O)c2ccc(Cl)cc2)cc(=O)n(C)c1=O	nan
	CHEMBL1358800	26097	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	0.2	Cn1c(CNS(=O)(=O)c2ccc(Cl)cc2)cc(=O)n(C)c1=O	nan
	16018591	26160	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.7	COc1cc(NS(=O)(=O)c2cc3c(cc2C)N(C)CCO3)cc(OC)c1OC	nan
	CHEMBL1359260	26160	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.7	COc1cc(NS(=O)(=O)c2cc3c(cc2C)N(C)CCO3)cc(OC)c1OC	nan
	4302860	26171	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	4302861	26171	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1359331	26171	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	1270409	26181	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	11	-0.4	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC(C)(C)C)n2C)n(C)c1=O	nan
	CHEMBL1359403	26181	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	11	-0.4	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC(C)(C)C)n2C)n(C)c1=O	nan
	1472977	26248	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	3	5.3	Brc1cc(Br)c2nc(-c3ccc(N4CCOCC4)cc3)ccc2c1	nan
	CHEMBL1360031	26248	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	3	5.3	Brc1cc(Br)c2nc(-c3ccc(N4CCOCC4)cc3)ccc2c1	nan
	5910118	26283	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1360299	26283	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	2519123	26342	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	1	5	2.2	Cc1cccc(-c2nnc(SCC(=O)NC3CC3)n2C)c1	nan
	CHEMBL1360828	26342	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	1	5	2.2	Cc1cccc(-c2nnc(SCC(=O)NC3CC3)n2C)c1	nan
	1637639	26400	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	7	1	5	3.8	CC(=O)c1sc(NC(=O)CCCOc2ccccc2C)nc1C	nan
	CHEMBL1361423	26400	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	7	1	5	3.8	CC(=O)c1sc(NC(=O)CCCOc2ccccc2C)nc1C	nan
	16029936	26412	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.5	Cc1cc(C(=O)Nc2c(C)nc3ccccn3c2=O)ccc1[N+](=O)[O-]	nan
	CHEMBL1361527	26412	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.5	Cc1cc(C(=O)Nc2c(C)nc3ccccn3c2=O)ccc1[N+](=O)[O-]	nan
	16021826	26428	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cc(Cl)ccc2C)c(-c2ccccc2)n1	nan
	CHEMBL1361623	26428	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cc(Cl)ccc2C)c(-c2ccccc2)n1	nan
	135399263	26551	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	3.7	Cc1cccc(C)c1NC(=O)CSc1nc(O)c2ccccc2n1	nan
	CHEMBL1362620	26551	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	3.7	Cc1cccc(C)c1NC(=O)CSc1nc(O)c2ccccc2n1	nan
	5225696	26664	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	2	3	2.3	CC1=C(C#N)C(NC(=O)c2ccccc2Cl)(C(F)(F)F)C(=O)N1	nan
	CHEMBL1363628	26664	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	2	3	2.3	CC1=C(C#N)C(NC(=O)c2ccccc2Cl)(C(F)(F)F)C(=O)N1	nan
	1300378	26716	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	5	3.9	CC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)Nc2ccc(C)cn2)cc1	nan
	CHEMBL1364136	26716	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	5	3.9	CC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)Nc2ccc(C)cn2)cc1	nan
	1207158	26740	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	2	5	4.7	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1cccc(C(=O)O)c1	nan
	CHEMBL1364382	26740	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	2	5	4.7	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1cccc(C(=O)O)c1	nan
	658008	26742	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.7	CCN(CC)C(=O)CSC1=C(C#N)C(c2cccs2)C=C(C)N1	nan
	CHEMBL1364397	26742	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.7	CCN(CC)C(=O)CSC1=C(C#N)C(c2cccs2)C=C(C)N1	nan
	1071060	26961	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	2	6	3.1	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2OC)c1C	nan
	CHEMBL1366254	26961	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	2	6	3.1	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2OC)c1C	nan
	711643	27010	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.7	Cc1ccc(C(=O)Nc2nnc(COc3ccccc3)s2)cc1	nan
	CHEMBL1366637	27010	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.7	Cc1ccc(C(=O)Nc2nnc(COc3ccccc3)s2)cc1	nan
	16030455	27011	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	4	6.0	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1366645	27011	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	4	6.0	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)Nc1ccccc1C(F)(F)F	nan
	16010113	27019	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	3.3	CC(C)Oc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	CHEMBL1366755	27019	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	3.3	CC(C)Oc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	2115552	27044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	3.2	Cc1[nH]c2ccccc2c1C(=O)COC(=O)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	CHEMBL1366975	27044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	3.2	Cc1[nH]c2ccccc2c1C(=O)COC(=O)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	868037	27145	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	4	3.4	COc1cccc2c(S)c(CCC(C)=O)c(C)nc12	nan
	CHEMBL1367790	27145	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	4	3.4	COc1cccc2c(S)c(CCC(C)=O)c(C)nc12	nan
	1086871	27282	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	1	8	3.4	COc1ccc(Cc2nnc(NC(=O)c3ccc(OC)c(OC)c3)s2)cc1OC	nan
	CHEMBL1368875	27282	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	1	8	3.4	COc1ccc(Cc2nnc(NC(=O)c3ccc(OC)c(OC)c3)s2)cc1OC	nan
	2054025	27568	10	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	7	4.0	COC(=O)c1ccc(CSc2ncnc3c2oc2ccccc23)o1	nan
	CHEMBL1370794	27568	10	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	7	4.0	COC(=O)c1ccc(CSc2ncnc3c2oc2ccccc23)o1	nan
	2951249	27630	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	4590179	27630	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1371319	27630	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	1520515	27720	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	3	0	7	4.4	COc1ccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)cc1	nan
	CHEMBL1372041	27720	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	3	0	7	4.4	COc1ccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)cc1	nan
	15988500	27781	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	584	13	2	9	3.7	CCCCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	CHEMBL1372455	27781	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	584	13	2	9	3.7	CCCCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	16030415	27863	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.0	Cc1ccc2nc(COc3ccccc3NC(=O)c3ccccc3F)cc(=O)n2c1	nan
	CHEMBL1372965	27863	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.0	Cc1ccc2nc(COc3ccccc3NC(=O)c3ccccc3F)cc(=O)n2c1	nan
	3141921	27889	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	4	4.1	N#CCSc1nc(-c2ccccc2)nc2ccc(F)cc12	nan
	CHEMBL1373143	27889	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	4	4.1	N#CCSc1nc(-c2ccccc2)nc2ccc(F)cc12	nan
	5740603	28000	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	3.3	COc1ccc2[nH]c(/C(C#N)=C\c3ccc(C(=O)O)cc3)nc2c1	nan
	CHEMBL1373830	28000	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	3.3	COc1ccc2[nH]c(/C(C#N)=C\c3ccc(C(=O)O)cc3)nc2c1	nan
	4965542	28029	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	11	0.2	C=CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1374122	28029	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	11	0.2	C=CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	3496625	28030	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	7	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OCc3ccccc3)cc2)no1	nan
	CHEMBL1374123	28030	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	7	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OCc3ccccc3)cc2)no1	nan
	2945949	28125	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	5	2.5	O=C(CCN1C(=O)c2cccc3cccc(c23)C1=O)Nc1ccon1	nan
	CHEMBL1374764	28125	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	5	2.5	O=C(CCN1C(=O)c2cccc3cccc(c23)C1=O)Nc1ccon1	nan
	15989514	28165	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	535	8	1	7	3.7	O=C(Cn1c(=O)n(CCCS(=O)(=O)C2CCCCC2)c(=O)c2ccccc21)Nc1ccc(F)c(Cl)c1	nan
	CHEMBL1375013	28165	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	535	8	1	7	3.7	O=C(Cn1c(=O)n(CCCS(=O)(=O)C2CCCCC2)c(=O)c2ccccc21)Nc1ccc(F)c(Cl)c1	nan
	2212703	28231	10	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	4	3.0	O=C(O)Cn1cc(C(=O)c2cccs2)c2ccccc21	nan
	CHEMBL1375453	28231	10	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	4	3.0	O=C(O)Cn1cc(C(=O)c2cccs2)c2ccccc21	nan
	2471579	28255	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	9	2	7	5.5	COc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	CHEMBL1375669	28255	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	9	2	7	5.5	COc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	3167528	28271	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	7	2.9	Cc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	CHEMBL1375776	28271	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	7	2.9	Cc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	2397772	28303	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	10	1.1	COc1cc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)ccc1OCCC(C)C	nan
	CHEMBL1376204	28303	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	10	1.1	COc1cc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)ccc1OCCC(C)C	nan
	1767629	28367	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1ccccc1Cl)C3	nan
	CHEMBL1376703	28367	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1ccccc1Cl)C3	nan
	16024679	28453	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	3.3	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)c1	nan
	CHEMBL1377672	28453	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	3.3	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)c1	nan
	135520779	28469	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	6	3.3	CCCc1nc2oc3c(O)ncnc3c2c2c1COC(C)(C)C2	nan
	CHEMBL1377764	28469	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	6	3.3	CCCc1nc2oc3c(O)ncnc3c2c2c1COC(C)(C)C2	nan
	16194561	28477	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)s1	nan
	CHEMBL1377828	28477	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)s1	nan
	16025409	28483	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	2.6	NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	CHEMBL1377886	28483	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	2.6	NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	2816168	28516	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	8	1.2	CCOC(=O)c1nnn2c1nc(N1CCN(C)CC1)c1ccccc12	nan
	CHEMBL1378192	28516	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	8	1.2	CCOC(=O)c1nnn2c1nc(N1CCN(C)CC1)c1ccccc12	nan
	16021577	28543	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	2.3	CCCNC(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	CHEMBL1378416	28543	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	2.3	CCCNC(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	20886481	28684	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	4	3.9	CC(C)Oc1ccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)cc1	nan
	CHEMBL1379683	28684	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	4	3.9	CC(C)Oc1ccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)cc1	nan
	2731492	28685	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	3	2	3	3.7	COc1cccc(NC(S)=Nc2cc(C)cc(C)n2)c1	nan
	CHEMBL1379684	28685	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	3	2	3	3.7	COc1cccc(NC(S)=Nc2cc(C)cc(C)n2)c1	nan
	614385	28731	73	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	2	4	2.7	Nc1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	CHEMBL1380161	28731	73	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	2	4	2.7	Nc1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	16187343	28770	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	0	7	4.1	CC(=O)c1ccc(-c2nnc(CCC(=O)N(C)Cc3cccc4cnccc34)o2)s1	nan
	CHEMBL1380413	28770	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	0	7	4.1	CC(=O)c1ccc(-c2nnc(CCC(=O)N(C)Cc3cccc4cnccc34)o2)s1	nan
	705209	28772	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	2	6	2.7	N#Cc1c(N)n(-c2ccc(C(=O)O)cc2)c2nc3ccccc3nc12	nan
	CHEMBL1380440	28772	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	2	6	2.7	N#Cc1c(N)n(-c2ccc(C(=O)O)cc2)c2nc3ccccc3nc12	nan
	3724835	28798	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	5033543	28798	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1380602	28798	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	1445317	28802	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	1	2	3.4	CCc1cc2ccc(C)cc2nc1S	nan
	CHEMBL1380640	28802	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	1	2	3.4	CCc1cc2ccc(C)cc2nc1S	nan
	4430260	28993	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	4	0	6	2.2	O=[N+]([O-])c1cccc(OCc2cn3cccnc3n2)c1	nan
	CHEMBL1382302	28993	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	4	0	6	2.2	O=[N+]([O-])c1cccc(OCc2cn3cccnc3n2)c1	nan
	3785801	29089	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	1	6	4.6	CCCCN(CCCC)C(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	CHEMBL1383130	29089	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	1	6	4.6	CCCCN(CCCC)C(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	3151314	29096	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	2	8	1.6	N=c1c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1383245	29096	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	2	8	1.6	N=c1c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	16241852	29154	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.6	CCc1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1.CN(C)C=O	nan
	CHEMBL1383752	29154	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.6	CCc1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1.CN(C)C=O	nan
	9550688	29188	2	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	0	6	3.2	O=c1sc(N2CCN(c3ccc(F)cc3)CC2)nc2ccsc12	nan
	CHEMBL1384034	29188	2	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	0	6	3.2	O=c1sc(N2CCN(c3ccc(F)cc3)CC2)nc2ccsc12	nan
	23004552	29212	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	0	8	0.5	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3sccn3c2=O)CC1	nan
	CHEMBL1384314	29212	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	0	8	0.5	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3sccn3c2=O)CC1	nan
	1830897	29285	11	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	5	2.7	O=c1c(Cl)c(NS(=O)(=O)c2ccccc2)cnn1-c1ccccc1	nan
	CHEMBL1384824	29285	11	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	5	2.7	O=c1c(Cl)c(NS(=O)(=O)c2ccccc2)cnn1-c1ccccc1	nan
	2488909	29410	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	7	1.6	COC(=O)CNC(=O)CSc1nnc2cc(C)c3ccccc3n12	nan
	CHEMBL1386026	29410	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	7	1.6	COC(=O)CNC(=O)CSc1nnc2cc(C)c3ccccc3n12	nan
	1301168	29572	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	6	4.6	Cc1ccc(S(=O)(=O)c2nc(Nc3ccccc3C#N)sc2Cl)cc1	nan
	CHEMBL1387246	29572	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	6	4.6	Cc1ccc(S(=O)(=O)c2nc(Nc3ccccc3C#N)sc2Cl)cc1	nan
	6264256	29585	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	1	8	4.1	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)cc1OC	nan
	CHEMBL1387384	29585	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	1	8	4.1	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)cc1OC	nan
	20904611	29670	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	10	1	9	1.8	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1388050	29670	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	10	1	9	1.8	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	2819135	29748	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	3.3	COc1cccc(-c2c(C#N)c(SC)nc3cc(C)nn23)c1	nan
	CHEMBL1388609	29748	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	3.3	COc1cccc(-c2c(C#N)c(SC)nc3cc(C)nn23)c1	nan
	900107	29831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	6	-1.0	NC(=O)Cn1cnc2nc3n(c2c1=O)CCC3	nan
	CHEMBL1389257	29831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	6	-1.0	NC(=O)Cn1cnc2nc3n(c2c1=O)CCC3	nan
	1934247	29858	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	9	2	6	5.3	COCCCNC(=O)c1c(NC(=O)c2ccccc2Cl)n(Cc2ccccc2)c2nc3ccccc3nc12	nan
	CHEMBL1389486	29858	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	9	2	6	5.3	COCCCNC(=O)c1c(NC(=O)c2ccccc2Cl)n(Cc2ccccc2)c2nc3ccccc3nc12	nan
	2012798	29948	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	4.4	Cc1ccc(Cn2c(N)c(S(=O)(=O)c3cccs3)c3nc4ccccc4nc32)cc1	nan
	CHEMBL1390254	29948	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	4.4	Cc1ccc(Cn2c(N)c(S(=O)(=O)c3cccs3)c3nc4ccccc4nc32)cc1	nan
	6290194	30058	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	1	7	3.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1391210	30058	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	1	7	3.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	16193052	30118	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(Br)cc1	nan
	CHEMBL1391769	30118	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(Br)cc1	nan
	886207	30273	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.3	CCNc1nc(C)c2cc(Br)c(=O)n(CC)c2n1	nan
	CHEMBL1393118	30273	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.3	CCNc1nc(C)c2cc(Br)c(=O)n(CC)c2n1	nan
	2889346	30288	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	1	4	3.5	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cn2)C1c1ccc(F)cc1	nan
	CHEMBL1393200	30288	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	1	4	3.5	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cn2)C1c1ccc(F)cc1	nan
	6622405	30292	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	2.9	CCn1c(=O)c2cc(C(=O)N(C)CC(OC)OC)sc2c2ccccc21	nan
	CHEMBL1393223	30292	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	2.9	CCn1c(=O)c2cc(C(=O)N(C)CC(OC)OC)sc2c2ccccc21	nan
	5181542	30320	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(Cl)cc2)no1	nan
	CHEMBL1393467	30320	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(Cl)cc2)no1	nan
	20917879	30327	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	6	2.4	CN(Cc1ccco1)S(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1393505	30327	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	6	2.4	CN(Cc1ccco1)S(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	20888749	30360	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CC(C)OC(C)C2)s1	nan
	CHEMBL1393784	30360	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CC(C)OC(C)C2)s1	nan
	2135574	30430	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	9	1	8	4.4	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OCC)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1394559	30430	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	9	1	8	4.4	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OCC)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	16033270	30431	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	5.3	Cc1ccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1394566	30431	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	5.3	Cc1ccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	16025819	30436	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	4	5.4	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1394644	30436	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	4	5.4	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	16018820	30444	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	8	4.7	CCc1nnc(SCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2cc3oc(C)cc3n12	nan
	CHEMBL1394778	30444	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	8	4.7	CCc1nnc(SCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2cc3oc(C)cc3n12	nan
	5144289	30467	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	4	3.4	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1394997	30467	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	4	3.4	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)[nH]c3ccccc3c2=O)cc1	nan
	16031990	30480	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.7	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Br)cc3)nn2)s1	nan
	CHEMBL1395113	30480	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.7	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Br)cc3)nn2)s1	nan
	6200398	30499	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	7	2.8	CNc1oc(/C=C/c2cc(OC)c(OC)c(OC)c2)nc1C#N	nan
	CHEMBL1395288	30499	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	7	2.8	CNc1oc(/C=C/c2cc(OC)c(OC)c(OC)c2)nc1C#N	nan
	16033416	30508	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	5	5.8	CCOc1ccc(-c2cc(C(=O)NCc3ccc(OC)cc3)c3c(-c4ccc(F)cc4)[nH]nc3n2)cc1	nan
	CHEMBL1395414	30508	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	5	5.8	CCOc1ccc(-c2cc(C(=O)NCc3ccc(OC)cc3)c3c(-c4ccc(F)cc4)[nH]nc3n2)cc1	nan
	5323079	30534	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	4	5.2	CCOc1ccc(NC(=O)CSc2c3c(nc4ccccc24)CCCC3)cc1	nan
	CHEMBL1395837	30534	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	4	5.2	CCOc1ccc(NC(=O)CSc2c3c(nc4ccccc24)CCCC3)cc1	nan
	16024553	30537	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1395881	30537	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	5296856	30559	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	4	2.6	Cc1cccn2c3c(c(=O)nc12)C(c1cccc(F)c1)CC(=O)N3	nan
	CHEMBL1396255	30559	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	4	2.6	Cc1cccn2c3c(c(=O)nc12)C(c1cccc(F)c1)CC(=O)N3	nan
	1730979	30562	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	3	6.9	O=C(Nc1cc(C(F)(F)F)ccc1Cl)c1cc(-c2cccs2)nc2ccccc12	nan
	CHEMBL1396294	30562	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	3	6.9	O=C(Nc1cc(C(F)(F)F)ccc1Cl)c1cc(-c2cccs2)nc2ccccc12	nan
	16019329	30566	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	0	9	2.6	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1396323	30566	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	0	9	2.6	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)CC1	nan
	16018658	30577	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.9	CCc1cccc(C)c1NC(=O)C(CC)Sc1nncn2c1cc1occc12	nan
	CHEMBL1396473	30577	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.9	CCc1cccc(C)c1NC(=O)C(CC)Sc1nncn2c1cc1occc12	nan
	20885686	30643	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	6	1.4	Cc1nn(CCCC(=O)NCc2ccc(F)cc2)c(=O)c2nccn12	nan
	CHEMBL1397376	30643	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	6	1.4	Cc1nn(CCCC(=O)NCc2ccc(F)cc2)c(=O)c2nccn12	nan
	4904384	30661	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	1	3	3.5	COc1cc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2cc1OC	nan
	CHEMBL1397630	30661	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	1	3	3.5	COc1cc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2cc1OC	nan
	22517504	30712	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	2.3	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	CHEMBL1398370	30712	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	2.3	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	15989335	30727	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	13	2	7	4.4	CCOc1ccc(NC(=O)Cn2c(=O)n(CCCCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1398481	30727	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	13	2	7	4.4	CCOc1ccc(NC(=O)Cn2c(=O)n(CCCCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3ccccc32)cc1	nan
	16022088	30736	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	0	6	4.8	COc1ccc2c(c1)c1c(c(=O)n(-c3cc(Cl)ccc3C)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	CHEMBL1398563	30736	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	0	6	4.8	COc1ccc2c(c1)c1c(c(=O)n(-c3cc(Cl)ccc3C)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	3594054	30831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	5	6.2	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Br)c1	nan
	CHEMBL1399458	30831	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	5	6.2	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Br)c1	nan
	16017733	30844	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	5	2.8	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1399598	30844	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	5	2.8	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccccc1C(F)(F)F	nan
	16023027	30954	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1400601	30954	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	2992172	31095	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	5	1	7	2.8	CCOC(=O)c1sc(NC(=O)c2ccc(OC(C)=O)cc2)nc1C	nan
	CHEMBL1401867	31095	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	5	1	7	2.8	CCOC(=O)c1sc(NC(=O)c2ccc(OC(C)=O)cc2)nc1C	nan
	3124205	31149	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	4	3.3	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(F)cc2)cc1	nan
	CHEMBL1402337	31149	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	4	3.3	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(F)cc2)cc1	nan
	3833466	31190	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	8	4.3	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1402650	31190	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	8	4.3	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	1451311	31203	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	0	5	3.4	CCOC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	CHEMBL1402735	31203	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	0	5	3.4	CCOC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	698553	31229	31	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1	nan
	CHEMBL1403001	31229	31	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1	nan
	2679217	31279	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	5	3.5	COc1ccc2oc(C(=O)Nc3nccs3)c(C)c2c1	nan
	CHEMBL1403552	31279	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	5	3.5	COc1ccc2oc(C(=O)Nc3nccs3)c(C)c2c1	nan
	3705005	31367	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	0	0	1	4.2	Brc1cc(Br)c2nc3c(cc2c1)CCC3	nan
	CHEMBL1404252	31367	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	0	0	1	4.2	Brc1cc(Br)c2nc3c(cc2c1)CCC3	nan
	738260	31428	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.1	COc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cn1	nan
	CHEMBL1404986	31428	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.1	COc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cn1	nan
	16406961	31439	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	2	1	6	2.8	Cc1c(CC(=O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c(=O)oc2cc(O)c(Cl)cc12	nan
	CHEMBL1405140	31439	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	2	1	6	2.8	Cc1c(CC(=O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c(=O)oc2cc(O)c(Cl)cc12	nan
	1277429	31500	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	0	7	3.5	c1ccc(-c2cc3c(N4CCN(c5ncccn5)CC4)ncnc3s2)cc1	nan
	CHEMBL1405710	31500	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	0	7	3.5	c1ccc(-c2cc3c(N4CCN(c5ncccn5)CC4)ncnc3s2)cc1	nan
	135681062	31515	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	2	6	0.1	O=C(NCCCN1CCCC1=O)c1c(O)nc2ccccn2c1=O	nan
	CHEMBL1405883	31515	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	2	6	0.1	O=C(NCCCN1CCCC1=O)c1c(O)nc2ccccn2c1=O	nan
	2479912	31526	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	7	1.2	Cn1c(N)c(C(=O)COc2ccc(Cl)cc2Cl)c(=O)n(C)c1=O	nan
	CHEMBL1405949	31526	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	7	1.2	Cn1c(N)c(C(=O)COc2ccc(Cl)cc2Cl)c(=O)n(C)c1=O	nan
	665818	31688	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.2	CNc1ncnc2c3cc(OC)ccc3n(C)c12	nan
	CHEMBL1407387	31688	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.2	CNc1ncnc2c3cc(OC)ccc3n(C)c12	nan
	2956880	31693	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	4	2.7	O=C(Nc1ccc(N2CCOCC2)cc1)C1CC(=O)N(c2ccc(F)cc2)C1	nan
	CHEMBL1407427	31693	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	4	2.7	O=C(Nc1ccc(N2CCOCC2)cc1)C1CC(=O)N(c2ccc(F)cc2)C1	nan
	7080333	31740	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	3.9	Cc1c(-c2cccc(NC(=O)Cc3ccccc3)c2)nc2ncccn12	nan
	CHEMBL1407681	31740	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	3.9	Cc1c(-c2cccc(NC(=O)Cc3ccccc3)c2)nc2ncccn12	nan
	16016996	31845	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	6	2.4	Cc1ccc(Cl)cc1N1CCN(C(=O)C(C)n2ncn3cccc3c2=O)CC1	nan
	CHEMBL1408470	31845	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	6	2.4	Cc1ccc(Cl)cc1N1CCN(C(=O)C(C)n2ncn3cccc3c2=O)CC1	nan
	236431	31874	62	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	1	1	3.6	CC(=O)Nc1ccc(Br)c2ccccc12	nan
	CHEMBL1408731	31874	62	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	1	1	3.6	CC(=O)Nc1ccc(Br)c2ccccc12	nan
	16019396	31974	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	10	4.2	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1ccc3c(c1)OCO3)c1sccc12	nan
	CHEMBL1409519	31974	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	10	4.2	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1ccc3c(c1)OCO3)c1sccc12	nan
	6625357	31989	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	6	1.3	Cc1nn(CCCC(=O)NCCc2ccccc2)c(=O)c2nccn12	nan
	CHEMBL1409636	31989	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	6	1.3	Cc1nn(CCCC(=O)NCCc2ccccc2)c(=O)c2nccn12	nan
	302041	32342	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	7	1.9	Cn1c2ccccc2c2nnc(SCCN3CCOCC3)nc21	nan
	CHEMBL1412491	32342	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	7	1.9	Cn1c2ccccc2c2nnc(SCCN3CCOCC3)nc21	nan
	2100500	32354	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1c(Cl)cccc1NC(=O)Cn1cc(C(F)(F)F)cc(Cl)c1=O	nan
	CHEMBL1412600	32354	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1c(Cl)cccc1NC(=O)Cn1cc(C(F)(F)F)cc(Cl)c1=O	nan
	2059848	32476	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	8	3.2	Cc1cc(C)nc(SCC(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)n1	nan
	CHEMBL1413582	32476	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	8	3.2	Cc1cc(C)nc(SCC(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)n1	nan
	16017166	32535	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	4.0	COc1cccc(CNC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	CHEMBL1414014	32535	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	4.0	COc1cccc(CNC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	2919306	32565	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(C)o2)C1c1cccc(Br)c1	nan
	CHEMBL1414306	32565	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(C)o2)C1c1cccc(Br)c1	nan
	16015068	32572	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1c(Cl)cccc1NC(=O)CSc1cc(-c2ccccc2)ncn1	nan
	CHEMBL1414379	32572	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1c(Cl)cccc1NC(=O)CSc1cc(-c2ccccc2)ncn1	nan
	16010393	32583	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	2	0	3	5.9	Cc1cccc2c1-c1sc(C(=O)N(C)c3cccc(C(F)(F)F)c3)cc1CO2	nan
	CHEMBL1414451	32583	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	2	0	3	5.9	Cc1cccc2c1-c1sc(C(=O)N(C)c3cccc(C(F)(F)F)c3)cc1CO2	nan
	3245690	32903	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	7	4.2	Cc1nc2ccc3nc(NC(=O)c4ccc5c(c4)OCCO5)sc3c2s1	nan
	CHEMBL1417231	32903	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	7	4.2	Cc1nc2ccc3nc(NC(=O)c4ccc5c(c4)OCCO5)sc3c2s1	nan
	24792497	32988	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	8	2.5	COc1ccc2cc(C#N)c(SCC(=O)Nc3nonc3C)nc2c1	nan
	CHEMBL1417975	32988	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	8	2.5	COc1ccc2cc(C#N)c(SCC(=O)Nc3nonc3C)nc2c1	nan
	2473907	33147	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.1	CCOC(=O)c1cc(-c2ccc(F)cc2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	CHEMBL1419339	33147	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.1	CCOC(=O)c1cc(-c2ccc(F)cc2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	2980984	33239	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	1	6	4.3	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccccc2)CO1	nan
	CHEMBL1420144	33239	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	1	6	4.3	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccccc2)CO1	nan
	16745931	33384	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	3	2	6	3.9	Cc1ccc(-c2csc3nc4cc(C(=O)NC5CCC(O)CC5)ccc4c(=O)n23)cc1	nan
	CHEMBL1421354	33384	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	3	2	6	3.9	Cc1ccc(-c2csc3nc4cc(C(=O)NC5CCC(O)CC5)ccc4c(=O)n23)cc1	nan
	2138543	33461	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	CHEMBL1422079	33461	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	6045016	33622	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	9	1	7	4.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1423355	33622	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	9	1	7	4.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	3725185	33659	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	4	5.2	CN(C)c1ccc(P(=O)(OCc2ccccc2)C(O)c2ccc(Cl)cc2)cc1	nan
	CHEMBL1423606	33659	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	4	5.2	CN(C)c1ccc(P(=O)(OCc2ccccc2)C(O)c2ccc(Cl)cc2)cc1	nan
	135420429	33663	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	9	3.4	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1nnc(C)s1	nan
	CHEMBL1423657	33663	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	9	3.4	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1nnc(C)s1	nan
	950417	33809	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	0	7	1.2	Cc1cccn2c(=O)c(C=C(C#N)C#N)c(N3CCN(C)CC3)nc12	nan
	CHEMBL1424893	33809	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	0	7	1.2	Cc1cccn2c(=O)c(C=C(C#N)C#N)c(N3CCN(C)CC3)nc12	nan
	4008202	34129	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	9	1.9	CCOC(=O)c1sc2nc(C)nc(SCC(=O)NC3CCS(=O)(=O)C3)c2c1C	nan
	CHEMBL1427679	34129	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	9	1.9	CCOC(=O)c1sc2nc(C)nc(SCC(=O)NC3CCS(=O)(=O)C3)c2c1C	nan
	2810151	34157	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	1	4	3.7	O=C(Nc1nc2ccccc2c(=O)s1)c1ccc(F)cc1Cl	nan
	CHEMBL1427961	34157	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	1	4	3.7	O=C(Nc1nc2ccccc2c(=O)s1)c1ccc(F)cc1Cl	nan
	4603734	34352	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	2.3	O=C(COc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl	nan
	CHEMBL1429555	34352	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	2.3	O=C(COc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl	nan
	2369101	34359	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	5	3.2	CCN1C(=O)C(=C2C=C(C)N(Cc3ccco3)C(C)=C2)C(=O)N(CC)C1=S	nan
	CHEMBL1429586	34359	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	5	3.2	CCN1C(=O)C(=C2C=C(C)N(Cc3ccco3)C(C)=C2)C(=O)N(CC)C1=S	nan
	6110891	34369	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.4	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1429670	34369	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.4	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	3186593	34591	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.3	CC1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1431426	34591	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.3	CC1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	4836291	34691	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	3	4.9	CCC1CCCCN1C(=O)COc1c(Br)cc(Br)c2cccnc12	nan
	CHEMBL1432322	34691	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	3	4.9	CCC1CCCCN1C(=O)COc1c(Br)cc(Br)c2cccnc12	nan
	3236746	34708	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	7	2	4	3.9	CCOc1ccc(OCC)c(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	CHEMBL1432463	34708	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	7	2	4	3.9	CCOc1ccc(OCC)c(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	5186080	34792	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	0	5	3.1	CC1(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)CC1(Cl)Cl	nan
	CHEMBL1433143	34792	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	0	5	3.1	CC1(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)CC1(Cl)Cl	nan
	16025762	34830	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)C1	nan
	CHEMBL1433427	34830	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)C1	nan
	16031695	34900	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	2.7	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnc3)cc2)cc1	nan
	CHEMBL1434575	34900	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	2.7	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnc3)cc2)cc1	nan
	1003863	34917	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	2	5	5.6	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(Cl)cc4F)sc3n2)c1	nan
	CHEMBL1434727	34917	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	2	5	5.6	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(Cl)cc4F)sc3n2)c1	nan
	16404473	34948	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	545	8	1	8	3.7	COc1cc(OC)c(OC)cc1/C=C1\Oc2cc(OCC(=O)N3Cc4ccccc4C[C@H]3C(=O)O)ccc2C1=O	nan
	CHEMBL1435093	34948	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	545	8	1	8	3.7	COc1cc(OC)c(OC)cc1/C=C1\Oc2cc(OCC(=O)N3Cc4ccccc4C[C@H]3C(=O)O)ccc2C1=O	nan
	24891925	34967	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	7	2.3	O=C(CSc1nnc2ccc(-c3ccc(F)cc3)nn12)NCC1CCCO1	nan
	CHEMBL1435281	34967	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	7	2.3	O=C(CSc1nnc2ccc(-c3ccc(F)cc3)nn12)NCC1CCCO1	nan
	16416480	34971	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	5457481	34971	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	CHEMBL1435346	34971	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	16034509	34975	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.6	CN(C)c1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1435377	34975	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.6	CN(C)c1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	15989215	34988	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	8	2.8	COc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1435575	34988	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	8	2.8	COc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc32)cc1	nan
	4281326	35046	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	4	5.3	Cc1cccc(C)c1OCC(=O)Nc1c(C(=O)c2ccccc2)oc2ccccc12	nan
	CHEMBL1436278	35046	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	4	5.3	Cc1cccc(C)c1OCC(=O)Nc1c(C(=O)c2ccccc2)oc2ccccc12	nan
	16009492	35137	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3cccc(NC(=O)c4ccccc4F)c3)cc(=O)n12	nan
	CHEMBL1437588	35137	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3cccc(NC(=O)c4ccccc4F)c3)cc(=O)n12	nan
	16015683	35139	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	1	5	5.9	O=C(Nc1ccc2nc(SCC(=O)N3CCc4ccccc43)sc2c1)c1ccc(Cl)cc1	nan
	CHEMBL1437631	35139	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	1	5	5.9	O=C(Nc1ccc2nc(SCC(=O)N3CCc4ccccc43)sc2c1)c1ccc(Cl)cc1	nan
	16025792	35151	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	5	4.9	COc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1437725	35151	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	5	4.9	COc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	4523316	35255	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	0	5	2.6	CN(C(=O)c1cc2c(=O)n3ccccc3nc2n1C)C1CCCCC1	nan
	CHEMBL1438580	35255	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	0	5	2.6	CN(C(=O)c1cc2c(=O)n3ccccc3nc2n1C)C1CCCCC1	nan
	16012068	35314	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	2.6	Cc1cc(=O)n2nc(N3CCC(C(=O)NCc4ccc(Cl)cc4)CC3)sc2n1	nan
	CHEMBL1439177	35314	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	2.6	Cc1cc(=O)n2nc(N3CCC(C(=O)NCc4ccc(Cl)cc4)CC3)sc2n1	nan
	3846910	35335	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	2	6	4.2	Cc1ccccc1NC(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	CHEMBL1439341	35335	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	2	6	4.2	Cc1ccccc1NC(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	4246549	35498	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	4	5.2	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCCCCC4)cc3c2C)c(C)c1	nan
	CHEMBL1440777	35498	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	4	5.2	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCCCCC4)cc3c2C)c(C)c1	nan
	4230097	35517	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	9	4.1	O=C(O)CCCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1440951	35517	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	9	4.1	O=C(O)CCCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	3272255	35650	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	2	7	0.7	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCC(C(N)=O)CC3)c(=O)c2c1C	nan
	CHEMBL1442168	35650	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	2	7	0.7	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCC(C(N)=O)CC3)c(=O)c2c1C	nan
	1077468	35679	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1442429	35679	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	20876076	35693	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	0.8	COc1ccc(C)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1442544	35693	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	0.8	COc1ccc(C)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	7217841	35738	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	6	2.9	Cc1nnc2ccc(-c3ccc(NC(=O)c4ccco4)cc3)nn12	nan
	CHEMBL1442956	35738	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	6	2.9	Cc1nnc2ccc(-c3ccc(NC(=O)c4ccco4)cc3)nn12	nan
	2975734	35747	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	CHEMBL1443010	35747	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	4611621	35903	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	4.8	COc1ccc(C2=NN(c3ccc(C(=O)O)cc3)C(c3ccc(OC)c(OC)c3)C2)cc1	nan
	CHEMBL1444507	35903	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	4.8	COc1ccc(C2=NN(c3ccc(C(=O)O)cc3)C(c3ccc(OC)c(OC)c3)C2)cc1	nan
	817359	35920	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	3	3.6	CC(=O)c1ccc(NC(=S)NC(=O)Cc2ccc(Cl)cc2)cc1	nan
	CHEMBL1444699	35920	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	3	3.6	CC(=O)c1ccc(NC(=S)NC(=O)Cc2ccc(Cl)cc2)cc1	nan
	4051948	35923	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	4.6	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccc(Cl)c2)o1	nan
	CHEMBL1444743	35923	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	4.6	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccc(Cl)c2)o1	nan
	3186591	35960	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.5	CC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1445043	35960	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.5	CC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	16187836	36054	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	10	1.1	COc1ccccc1-c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1445914	36054	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	10	1.1	COc1ccccc1-c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16017757	36169	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	2.9	CCc1ccc(NC(=O)Cn2ccn(-c3cccc(Cl)c3)c(=O)c2=O)cc1	nan
	CHEMBL1446963	36169	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	2.9	CCc1ccc(NC(=O)Cn2ccn(-c3cccc(Cl)c3)c(=O)c2=O)cc1	nan
	2769301	36326	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	4	3.7	COc1ccc(-c2cc(C(=O)Nc3ccccc3F)on2)cc1	nan
	CHEMBL1448341	36326	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	4	3.7	COc1ccc(-c2cc(C(=O)Nc3ccccc3F)on2)cc1	nan
	3658309	36480	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	11	1	8	4.8	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	CHEMBL1449439	36480	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	11	1	8	4.8	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	3652194	36544	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	1	0	2	5.5	Brc1cc(Br)c2nc(-c3cccs3)ccc2c1	nan
	CHEMBL1449966	36544	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	1	0	2	5.5	Brc1cc(Br)c2nc(-c3cccs3)ccc2c1	nan
	3244704	36652	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	7	3.3	COc1ccc(C2C=C(c3cccs3)Nc3nc(CCCO)nn32)cc1	nan
	CHEMBL1450888	36652	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	7	3.3	COc1ccc(C2C=C(c3cccs3)Nc3nc(CCCO)nn32)cc1	nan
	1774540	36829	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1cccc(Cl)c1)C3	nan
	CHEMBL1452222	36829	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1cccc(Cl)c1)C3	nan
	649434	36917	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	4.2	CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	CHEMBL1452945	36917	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	4.2	CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	16187616	37066	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	10	2.8	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4cc(C)on4)nn23)cc1OC	nan
	CHEMBL1454124	37066	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	10	2.8	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4cc(C)on4)nn23)cc1OC	nan
	17580690	37103	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	1	1	2	3.5	Cc1c(C(=O)N2CC(C)OC(C)C2)[nH]c2ccc(Br)cc12	nan
	CHEMBL1454451	37103	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	1	1	2	3.5	Cc1c(C(=O)N2CC(C)OC(C)C2)[nH]c2ccc(Br)cc12	nan
	18204435	37197	6	None	-48	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	2	6	3.5	CNC(=O)c1ccc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)cc1	nan
	CHEMBL1455259	37197	6	None	-48	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	2	6	3.5	CNC(=O)c1ccc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)cc1	nan
	1265180	37304	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	8	1.0	CCCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1456231	37304	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	8	1.0	CCCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	24793479	37422	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	6	3.3	COc1ccc(C(=O)NNC(=O)CSc2nc(C(C)C)nc3ccccc23)cc1	nan
	CHEMBL1457367	37422	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	6	3.3	COc1ccc(C(=O)NNC(=O)CSc2nc(C(C)C)nc3ccccc23)cc1	nan
	24819691	37514	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	3	4	3.2	COc1ccc2cc(OCC(=O)NNC(=O)Nc3ccc(F)cc3)ccc2c1	nan
	CHEMBL1458070	37514	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	3	4	3.2	COc1ccc2cc(OCC(=O)NNC(=O)Nc3ccc(F)cc3)ccc2c1	nan
	675984	37619	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	0	2	4.0	O=C(COc1ccc2ccccc2c1Br)N1CCCCC1	nan
	CHEMBL1458979	37619	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	0	2	4.0	O=C(COc1ccc2ccccc2c1Br)N1CCCCC1	nan
	866601	37751	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	5	3.4	O=C(NC1CCCCCC1)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1460115	37751	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	5	3.4	O=C(NC1CCCCCC1)c1cc2c(=O)n3ccccc3nc2s1	nan
	20912606	37939	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	0	7	3.4	CN(C)CCN(Cc1ccccc1)C(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	CHEMBL1461808	37939	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	0	7	3.4	CN(C)CCN(Cc1ccccc1)C(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	2745719	38162	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	2.8	CC(=O)Nc1nccc(-c2cc(-c3ccccc3)no2)n1	nan
	CHEMBL1463690	38162	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	2.8	CC(=O)Nc1nccc(-c2cc(-c3ccccc3)no2)n1	nan
	741378	38318	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	3.4	COC(=O)Sc1nnc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1464821	38318	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	3.4	COC(=O)Sc1nnc(-c2ccc(Br)cc2)o1	nan
	203396	38349	77	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	3	2.8	O=c1c(Br)c(Br)cnn1-c1ccccc1	nan
	CHEMBL1465040	38349	77	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	3	2.8	O=c1c(Br)c(Br)cnn1-c1ccccc1	nan
	3518230	38369	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	4024784	38369	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	CHEMBL1465171	38369	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	24791767	38421	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	0	6	3.5	CCN(Cc1cnn(C)c1)C(=O)c1cc(COc2ccc3c(c2)CCCC3)on1	nan
	CHEMBL1465549	38421	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	0	6	3.5	CCN(Cc1cnn(C)c1)C(=O)c1cc(COc2ccc3c(c2)CCCC3)on1	nan
	16241464	38634	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	8	2.7	CN(C)C=O.O=[N+]([O-])c1cccc(COc2ncnc3cc([N+](=O)[O-])ccc23)c1	nan
	CHEMBL1467247	38634	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	8	2.7	CN(C)C=O.O=[N+]([O-])c1cccc(COc2ncnc3cc([N+](=O)[O-])ccc23)c1	nan
	1244301	38733	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	2	3.8	Cc1c(C(=O)NCc2ccccc2F)oc2ccccc12	nan
	CHEMBL1468217	38733	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	2	3.8	Cc1c(C(=O)NCc2ccccc2F)oc2ccccc12	nan
	18561646	38781	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	9	0.6	CC(C)Cc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1468525	38781	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	9	0.6	CC(C)Cc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	4257704	38839	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	1	7	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc([N+](=O)[O-])ccc2Cl)c1	nan
	CHEMBL1468952	38839	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	1	7	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc([N+](=O)[O-])ccc2Cl)c1	nan
	20957237	38974	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	9	1.7	COc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1470126	38974	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	9	1.7	COc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	1261892	38977	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	2	5	3.7	NS(=O)(=O)c1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3ccc(Br)cc23)cc1	nan
	CHEMBL1470208	38977	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	2	5	3.7	NS(=O)(=O)c1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3ccc(Br)cc23)cc1	nan
	2725142	39089	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	7	2.4	COc1nc(N)c(C#N)c(-c2ccc(N(C)CCC#N)cc2)c1C#N	nan
	CHEMBL1471123	39089	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	7	2.4	COc1nc(N)c(C#N)c(-c2ccc(N(C)CCC#N)cc2)c1C#N	nan
	15988569	39274	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	6	5.5	Cc1ccc(-c2nc(-c3cc4cccc(OCc5ccc(F)cc5)c4oc3=O)no2)cc1	nan
	CHEMBL1472849	39274	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	6	5.5	Cc1ccc(-c2nc(-c3cc4cccc(OCc5ccc(F)cc5)c4oc3=O)no2)cc1	nan
	1166244	39285	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1cccc(C)c1NC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	CHEMBL1472996	39285	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1cccc(C)c1NC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	16025417	39302	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	8	1	7	5.3	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)cc1	nan
	CHEMBL1473284	39302	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	8	1	7	5.3	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)cc1	nan
	16009695	39368	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	4	1	6	4.5	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCCC1	nan
	CHEMBL1474245	39368	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	4	1	6	4.5	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCCC1	nan
	2158398	39374	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	6	3.8	COc1ccc(Cl)cc1NC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1474329	39374	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	6	3.8	COc1ccc(Cl)cc1NC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	16009720	39379	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(CNc2nc3c(-c4ccc(C)cc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1474419	39379	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(CNc2nc3c(-c4ccc(C)cc4)nnn3c3ccccc23)cc1	nan
	16016110	39417	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	1	7	4.8	Cc1ccc(CNc2ccc(-c3nc(-c4ccco4)no3)cc2[N+](=O)[O-])cc1	nan
	CHEMBL1474896	39417	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	1	7	4.8	Cc1ccc(CNc2ccc(-c3nc(-c4ccco4)no3)cc2[N+](=O)[O-])cc1	nan
	16033296	39419	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccccc1CNC(=O)c1sc2ncnc(N(C)C3CCCCC3)c2c1C	nan
	CHEMBL1474937	39419	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccccc1CNC(=O)c1sc2ncnc(N(C)C3CCCCC3)c2c1C	nan
	3155029	39470	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	5	2.1	COc1ccc(CCNC(=O)CN2C(=O)COc3ccc(C)cc32)cc1OC	nan
	CHEMBL1475587	39470	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	5	2.1	COc1ccc(CCNC(=O)CN2C(=O)COc3ccc(C)cc32)cc1OC	nan
	16020275	39473	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	9	2	7	4.6	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)cc3)c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc32)cc1	nan
	CHEMBL1475630	39473	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	9	2	7	4.6	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)cc3)c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc32)cc1	nan
	16415433	39475	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	5513689	39475	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	CHEMBL1475648	39475	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	3646895	39493	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	7	4.9	CCOCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1475830	39493	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	7	4.9	CCOCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	16020214	39497	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	644	7	2	8	4.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2ccc(C(=O)NCc3ccc4c(c3)OCO4)cc21)Nc1ccc(Br)cc1F	nan
	CHEMBL1475923	39497	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	644	7	2	8	4.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2ccc(C(=O)NCc3ccc4c(c3)OCO4)cc21)Nc1ccc(Br)cc1F	nan
	15990518	39510	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.9	CCOC(=O)c1cccc(NC(=O)c2cc3cc4cc(OC)ccc4nc3s2)c1	nan
	CHEMBL1476197	39510	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.9	CCOC(=O)c1cccc(NC(=O)c2cc3cc4cc(OC)ccc4nc3s2)c1	nan
	16018050	39549	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1OC	nan
	CHEMBL1476725	39549	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1OC	nan
	18572231	39572	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	8	2.6	CCOc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1477019	39572	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	8	2.6	CCOc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	5294687	39604	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	8	2	4	5.3	CCCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1477360	39604	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	8	2	4	5.3	CCCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	3096467	39676	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	5751261	39676	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	CHEMBL1477993	39676	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	2027019	39743	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	7	5.3	CSc1nc(SCC(=O)O)c2sc3nc(-c4ccccc4)c4c(c3c2n1)CCC4	nan
	CHEMBL1478587	39743	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	7	5.3	CSc1nc(SCC(=O)O)c2sc3nc(-c4ccccc4)c4c(c3c2n1)CCC4	nan
	2487220	39858	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	3.8	CCn1cc(C(=O)OCC(=O)Nc2cccc(Cl)c2Cl)c(=O)c2ccc(C)nc21	nan
	CHEMBL1479594	39858	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	3.8	CCn1cc(C(=O)OCC(=O)Nc2cccc(Cl)c2Cl)c(=O)c2ccc(C)nc21	nan
	16024523	39919	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	5	3.6	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1480079	39919	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	5	3.6	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	16019201	39933	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3cc(C)cc(C)c3)c2=O)cc1	nan
	CHEMBL1480191	39933	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3cc(C)cc(C)c3)c2=O)cc1	nan
	5925055	40127	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1481881	40127	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCCO2	nan
	7258994	40135	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	8	1.9	Cc1ccc2nc(SCC(=O)Nc3ccc4c(c3)OCCO4)nc(=O)n2c1	nan
	CHEMBL1481935	40135	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	8	1.9	Cc1ccc2nc(SCC(=O)Nc3ccc4c(c3)OCCO4)nc(=O)n2c1	nan
	1470918	40217	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	3.7	Cc1ccccc1C(=O)NN(C)c1nc2ccccc2nc1C(F)(F)F	nan
	CHEMBL1482653	40217	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	3.7	Cc1ccccc1C(=O)NN(C)c1nc2ccccc2nc1C(F)(F)F	nan
	3122172	40261	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccccc1Cl	nan
	CHEMBL1483069	40261	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccccc1Cl	nan
	1093408	40311	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	2	5	4.3	COCc1cc(C)nc2sc(C(=O)Nc3ccccc3Br)c(N)c12	nan
	CHEMBL1483523	40311	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	2	5	4.3	COCc1cc(C)nc2sc(C(=O)Nc3ccccc3Br)c(N)c12	nan
	1868051	40343	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	3.4	CSc1nc(SCC(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1483727	40343	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	3.4	CSc1nc(SCC(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	4968512	40442	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	209	1	2	5	2.1	Nc1ccccc1-c1nnc(S)s1	nan
	CHEMBL1484500	40442	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	209	1	2	5	2.1	Nc1ccccc1-c1nnc(S)s1	nan
	1130974	40477	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	6	3.5	CCOc1ccc(NC(=O)c2sc(NC(C)=O)c(C(=O)OC)c2C)cc1	nan
	CHEMBL1484851	40477	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	6	3.5	CCOc1ccc(NC(=O)c2sc(NC(C)=O)c(C(=O)OC)c2C)cc1	nan
	16023029	40609	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	6	2.9	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccc(F)cc2)s1	nan
	CHEMBL1486082	40609	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	6	2.9	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccc(F)cc2)s1	nan
	2122608	40633	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	6	1	5	4.1	CC(=O)c1sc(NC(=O)COc2ccc(C(C)C)c(C)c2)nc1C	nan
	CHEMBL1486351	40633	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	6	1	5	4.1	CC(=O)c1sc(NC(=O)COc2ccc(C(C)C)c(C)c2)nc1C	nan
	15988496	40675	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	0	6	5.2	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(-c2ccc(F)c(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1486634	40675	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	0	6	5.2	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(-c2ccc(F)c(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	5058050	40781	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	0	5	4.0	CCCCN(CCCC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1487547	40781	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	0	5	4.0	CCCCN(CCCC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	1120443	40905	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	7	5.9	CCOc1cc(-c2nc3c(c(CC)nn3-c3ccccc3)c3cc(OC)c(OC)cc23)ccc1O	nan
	CHEMBL1488401	40905	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	7	5.9	CCOc1cc(-c2nc3c(c(CC)nn3-c3ccccc3)c3cc(OC)c(OC)cc23)ccc1O	nan
	1415522	40984	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	6.4	CCN(CC)C(=O)c1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	CHEMBL1488995	40984	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	6.4	CCN(CC)C(=O)c1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	2014552	41100	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	9	2.0	CCOc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)ccc1OCCN1CCOCC1	nan
	CHEMBL1489906	41100	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	9	2.0	CCOc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)ccc1OCCN1CCOCC1	nan
	2873834	41175	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	7	4.3	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CCCC2=N1	nan
	CHEMBL1490473	41175	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	7	4.3	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CCCC2=N1	nan
	1536777	41418	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	4.4	Cc1sc2ncnc(NC3CCN(Cc4ccccc4)CC3)c2c1C	nan
	CHEMBL1492096	41418	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	4.4	Cc1sc2ncnc(NC3CCN(Cc4ccccc4)CC3)c2c1C	nan
	2419865	41517	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	5	0	5	3.7	COc1ccc(C(C)=O)cc1COc1nc(C)nc2ccccc12	nan
	CHEMBL1492888	41517	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	5	0	5	3.7	COc1ccc(C(C)=O)cc1COc1nc(C)nc2ccccc12	nan
	1102906	41525	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	2	4	3.0	O=C(O)c1ccc(N2C(=O)c3cccc4c(C(=O)O)ccc(c34)C2=O)cc1	nan
	CHEMBL1492995	41525	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	2	4	3.0	O=C(O)c1ccc(N2C(=O)c3cccc4c(C(=O)O)ccc(c34)C2=O)cc1	nan
	3467703	41604	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	2	0	2	3.4	C=CCN1C(=O)c2cccc3c(Br)ccc(c23)C1=O	nan
	CHEMBL1493801	41604	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	2	0	2	3.4	C=CCN1C(=O)c2cccc3c(Br)ccc(c23)C1=O	nan
	7711621	41625	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	2	7	-0.5	CC(=O)Nc1ccc(S(=O)(=O)NCc2cc(=O)n(C)c(=O)n2C)cc1	nan
	CHEMBL1494013	41625	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	2	7	-0.5	CC(=O)Nc1ccc(S(=O)(=O)NCc2cc(=O)n(C)c(=O)n2C)cc1	nan
	681202	41694	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	3	3	3	3.6	Cc1sc(N=C(S)Nc2ccc(F)cc2)c(C(N)=O)c1C	nan
	CHEMBL1494694	41694	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	3	3	3	3.6	Cc1sc(N=C(S)Nc2ccc(F)cc2)c(C(N)=O)c1C	nan
	2451170	41773	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	6	2.8	CCOC(=O)c1sc2nc(C)nc(S)c2c1C	nan
	CHEMBL1495560	41773	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	6	2.8	CCOC(=O)c1sc2nc(C)nc(S)c2c1C	nan
	16017877	41815	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	4	2.6	Cc1ccccc1Cn1ccn(-c2ccc(F)c(F)c2)c(=O)c1=O	nan
	CHEMBL1495957	41815	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	4	2.6	Cc1ccccc1Cn1ccn(-c2ccc(F)c(F)c2)c(=O)c1=O	nan
	2917647	41938	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	6	3.5	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(Cl)cc1)c1ccco1	nan
	CHEMBL1497016	41938	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	6	3.5	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(Cl)cc1)c1ccco1	nan
	3493986	41959	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	8	1	6	5.3	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccccc3C)cc2)cc1	nan
	CHEMBL1497174	41959	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	8	1	6	5.3	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccccc3C)cc2)cc1	nan
	4260589	41996	6	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	9	2	6	4.8	CCCC1(c2ccccc2)NC(=O)N(CC(=O)Nc2sc(-c3ccccc3)cc2C(=O)OCC)C1=O	nan
	CHEMBL1497431	41996	6	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	9	2	6	4.8	CCCC1(c2ccccc2)NC(=O)N(CC(=O)Nc2sc(-c3ccccc3)cc2C(=O)OCC)C1=O	nan
	1234241	42057	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	1	1	5	2.9	Cc1nnc(S)c2nn(-c3ccccc3F)c(C)c12	nan
	CHEMBL1498110	42057	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	1	1	5	2.9	Cc1nnc(S)c2nn(-c3ccccc3F)c(C)c12	nan
	4056802	42260	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	2.8	Cc1cccn2c(=O)c3cc(C(=O)NCCCOC(C)C)sc3nc12	nan
	CHEMBL1499876	42260	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	2.8	Cc1cccn2c(=O)c3cc(C(=O)NCCCOC(C)C)sc3nc12	nan
	2908462	42265	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	1	6	3.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccccc1)c1ccco1	nan
	CHEMBL1499902	42265	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	1	6	3.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccccc1)c1ccco1	nan
	2551439	42397	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	0	8	1.7	COc1ccc(OCCOC(=O)c2nc3nccc(C)n3n2)cc1	nan
	CHEMBL1501099	42397	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	0	8	1.7	COc1ccc(OCCOC(=O)c2nc3nccc(C)n3n2)cc1	nan
	716763	42421	27	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	3.3	O=C(O)c1ccc(N2C(=O)c3cccc4cccc(c34)C2=O)cc1	nan
	CHEMBL1501298	42421	27	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	3.3	O=C(O)c1ccc(N2C(=O)c3cccc4cccc(c34)C2=O)cc1	nan
	5012247	42472	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	11	-2.0	CCN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1CCS(=O)(=O)C1	nan
	CHEMBL1501780	42472	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	11	-2.0	CCN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1CCS(=O)(=O)C1	nan
	2816746	42810	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	2	6	4.1	CCOC(=O)c1c(N=C(S)NCc2ccccc2)sc2c1CCN(C(=O)OCC)C2	nan
	CHEMBL1504775	42810	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	2	6	4.1	CCOC(=O)c1c(N=C(S)NCc2ccccc2)sc2c1CCN(C(=O)OCC)C2	nan
	2363951	42824	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	9	0.2	Cn1c(N)c(C(=O)COC(=O)CCC(=O)c2ccc(F)cc2)c(=O)n(C)c1=O	nan
	CHEMBL1504909	42824	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	9	0.2	Cn1c(N)c(C(=O)COC(=O)CCC(=O)c2ccc(F)cc2)c(=O)n(C)c1=O	nan
	3238944	42871	12	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.4	Cc1cccc(Nc2nn3c(=O)c4ccccc4nc3s2)c1	nan
	CHEMBL1505300	42871	12	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.4	Cc1cccc(Nc2nn3c(=O)c4ccccc4nc3s2)c1	nan
	7190519	42917	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	9	2.4	O=C(CSc1ccc2nnc(-c3ccccn3)n2n1)Nc1nccs1	nan
	CHEMBL1505657	42917	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	9	2.4	O=C(CSc1ccc2nnc(-c3ccccn3)n2n1)Nc1nccs1	nan
	3154081	43130	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	8	4.0	CCCOc1cccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1507529	43130	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	8	4.0	CCCOc1cccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	1803037	43316	9	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	5	6.1	Cc1cccc(NC(=O)CSc2nc(C)c(CC(=O)c3ccc(Br)cc3)c(C)c2C#N)c1C	nan
	CHEMBL1509120	43316	9	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	5	6.1	Cc1cccc(NC(=O)CSc2nc(C)c(CC(=O)c3ccc(Br)cc3)c(C)c2C#N)c1C	nan
	3772923	43328	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	1	3	2.4	Cc1nc(S)c(C#N)c2c1CCCC2	nan
	CHEMBL1509207	43328	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	1	3	2.4	Cc1nc(S)c(C#N)c2c1CCCC2	nan
	3150659	43461	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.3	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1510456	43461	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.3	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCCC3	nan
	2318166	43495	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	4.7	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCCC3)c2C#N)cc1	nan
	CHEMBL1510689	43495	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	4.7	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCCC3)c2C#N)cc1	nan
	4382156	43568	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	4	2.2	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccccc1F	nan
	CHEMBL1511309	43568	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	4	2.2	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccccc1F	nan
	5825936	43625	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	8	3.3	C=CCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1511801	43625	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	8	3.3	C=CCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	1234706	43654	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	6	3.5	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nc(C)cc(C)n2)cc1	nan
	CHEMBL1512389	43654	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	6	3.5	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nc(C)cc(C)n2)cc1	nan
	18572258	43665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	7	2.9	O=C(CSc1nnc2ccc(-c3ccc(Br)cc3)nn12)NCC1CCCO1	nan
	CHEMBL1512477	43665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	7	2.9	O=C(CSc1nnc2ccc(-c3ccc(Br)cc3)nn12)NCC1CCCO1	nan
	7205055	43694	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	6	3.3	CCN1CCN(Cc2c(O)ccc3cc(-c4ccc(OC)cc4)c(=O)oc23)CC1	nan
	CHEMBL1512819	43694	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	6	3.3	CCN1CCN(Cc2c(O)ccc3cc(-c4ccc(OC)cc4)c(=O)oc23)CC1	nan
	53229784	43696	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	5457315	43696	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	CHEMBL1512839	43696	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	16026424	43730	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	0	7	3.4	COC(=O)c1sc2ccccc2c1S(=O)(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1513424	43730	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	0	7	3.4	COC(=O)c1sc2ccccc2c1S(=O)(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	16019493	43745	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(S(=O)(=O)NCCc2nnc3ccc(SCc4ccccc4C)nn23)cc1	nan
	CHEMBL1513611	43745	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(S(=O)(=O)NCCc2nnc3ccc(SCc4ccccc4C)nn23)cc1	nan
	15989126	43749	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	11	2	7	4.7	Cc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1513634	43749	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	11	2	7	4.7	Cc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	1252356	43765	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	6	5.5	Cc1cc(C)cc(NC(=O)CSc2oc(-c3ccccc3)nc2S(=O)(=O)c2ccccc2)c1	nan
	CHEMBL1513969	43765	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	6	5.5	Cc1cc(C)cc(NC(=O)CSc2oc(-c3ccccc3)nc2S(=O)(=O)c2ccccc2)c1	nan
	16406807	43769	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	3	6	2.7	CC[C@@H](C)[C@H](NC(=O)CNC(=O)Cc1c(C)c2c(cc(C)c3c(C)coc32)oc1=O)C(=O)O	nan
	CHEMBL1514043	43769	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	3	6	2.7	CC[C@@H](C)[C@H](NC(=O)CNC(=O)Cc1c(C)c2c(cc(C)c3c(C)coc32)oc1=O)C(=O)O	nan
	2135573	43800	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	8	1	8	4.1	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1514550	43800	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	8	1	8	4.1	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	16018084	43842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1515147	43842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	4302940	43843	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	5.4	CCn1cc(CNC(=O)c2cc(-c3ccc(C)cc3)nc3ccc(Br)cc23)c(C)n1	nan
	CHEMBL1515178	43843	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	5.4	CCn1cc(CNC(=O)c2cc(-c3ccc(C)cc3)nc3ccc(Br)cc23)c(C)n1	nan
	15989010	43858	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	1	8	3.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c1	nan
	CHEMBL1515330	43858	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	1	8	3.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c1	nan
	20885696	44018	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	9	1	8	1.4	COc1ccc(CCNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1OC	nan
	CHEMBL1517314	44018	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	9	1	8	1.4	COc1ccc(CCNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1OC	nan
	1488779	44242	21	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	4	4.6	COc1ccc(Oc2nccc(-c3ccc(F)cc3)c2C#N)cc1	nan
	CHEMBL1519391	44242	21	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	4	4.6	COc1ccc(Oc2nccc(-c3ccc(F)cc3)c2C#N)cc1	nan
	3154197	44243	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	8	0.6	Cn1c(=O)c2c(ncn2CC(O)CNc2cccc(Cl)c2)n(C)c1=O	nan
	CHEMBL1519401	44243	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	8	0.6	Cn1c(=O)c2c(ncn2CC(O)CNc2cccc(Cl)c2)n(C)c1=O	nan
	5309980	44285	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	1	6	2.5	CC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	CHEMBL1519790	44285	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	1	6	2.5	CC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	20873023	44373	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccc(OC)cc2)c1=O	nan
	CHEMBL1520622	44373	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccc(OC)cc2)c1=O	nan
	135407280	44401	32	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	2	1	5	2.4	CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1520797	44401	32	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	2	1	5	2.4	CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	2868262	44465	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Br)cc1	nan
	CHEMBL1521342	44465	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Br)cc1	nan
	646901	44515	3	None	-4	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	3.6	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cc(C)on1)OCO3	nan
	CHEMBL1521729	44515	3	None	-4	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	3.6	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cc(C)on1)OCO3	nan
	16012248	44531	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.0	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)Nc3ccc(C)c(Cl)c3)c(C)nc21	nan
	CHEMBL1521906	44531	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.0	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)Nc3ccc(C)c(Cl)c3)c(C)nc21	nan
	5086217	44553	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.6	CCOC(=O)c1c(N=C(S)Nc2ccc(F)cc2)sc2c1CCC2	nan
	CHEMBL1522109	44553	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.6	CCOC(=O)c1c(N=C(S)Nc2ccc(F)cc2)sc2c1CCC2	nan
	2929681	44624	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	2	7	2.6	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CCc4ccccc4)c3nc12	nan
	CHEMBL1522811	44624	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	2	7	2.6	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CCc4ccccc4)c3nc12	nan
	352022	44666	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	0	7	0.5	CCCSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1523163	44666	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	0	7	0.5	CCCSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	861889	44676	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.0	Cc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	CHEMBL1523239	44676	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.0	Cc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	4099138	44681	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	9	2	8	3.5	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1523295	44681	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	9	2	8	3.5	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccc2c(c1)OCO2	nan
	5760985	44961	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	4	4.8	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(F)cc1)c1ccc(Br)cc1	nan
	CHEMBL1525962	44961	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	4	4.8	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(F)cc1)c1ccc(Br)cc1	nan
	3186625	45183	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	2	9	0.7	CC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	CHEMBL1527889	45183	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	2	9	0.7	CC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	1166606	45255	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	8	1	6	5.3	COc1ccc(NC(=O)CCSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)n2)cc1	nan
	CHEMBL1528550	45255	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	8	1	6	5.3	COc1ccc(NC(=O)CCSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)n2)cc1	nan
	1109837	45336	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ncccc3o2)cc1	nan
	CHEMBL1529226	45336	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ncccc3o2)cc1	nan
	4413149	45359	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1ccc(Cl)cc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1529453	45359	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1ccc(Cl)cc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	6086754	45422	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1529980	45422	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	4881121	45461	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	0	7	2.0	CCc1cc2c(SCC(=O)N(C)C3CCS(=O)(=O)C3)ncnc2s1	nan
	CHEMBL1530432	45461	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	0	7	2.0	CCc1cc2c(SCC(=O)N(C)C3CCS(=O)(=O)C3)ncnc2s1	nan
	15988929	45514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	12	2	8	3.7	COc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1530799	45514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	12	2	8	3.7	COc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	2956077	45579	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	3	3.4	COc1ccc2cc(Br)ccc2c1CC(=O)NCC1CCCO1	nan
	CHEMBL1531449	45579	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	3	3.4	COc1ccc2cc(Br)ccc2c1CC(=O)NCC1CCCO1	nan
	646794	45997	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	6	2.4	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccnc1)c1ccco1	nan
	CHEMBL1535358	45997	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	6	2.4	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccnc1)c1ccco1	nan
	9551120	46132	0	None	-14	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	3.0	CCOC(=O)Cn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	CHEMBL1536779	46132	0	None	-14	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	3.0	CCOC(=O)Cn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	5297702	46232	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	1	3	4.2	Nc1c2c(nc3cccc(Cl)c13)N(c1ccccc1)CC2	nan
	CHEMBL1537611	46232	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	1	3	4.2	Nc1c2c(nc3cccc(Cl)c13)N(c1ccccc1)CC2	nan
	5069161	46426	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	CHEMBL1539200	46426	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	1373674	46496	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	8	0.1	Cn1c(=O)c2c(nc(SCC(=O)NC3CCCC3)n2C)n(C)c1=O	nan
	CHEMBL1539818	46496	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	8	0.1	Cn1c(=O)c2c(nc(SCC(=O)NC3CCCC3)n2C)n(C)c1=O	nan
	20888840	46537	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	0	8	2.2	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	CHEMBL1540109	46537	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	0	8	2.2	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	2823604	46617	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	3	0	4	3.2	COC(=O)CSc1ccnc2cc(Cl)ccc12	nan
	CHEMBL1540846	46617	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	3	0	4	3.2	COC(=O)CSc1ccnc2cc(Cl)ccc12	nan
	2502748	46651	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	7	3.0	COc1cc(CN(C)Cc2cc(=O)n3ccsc3n2)ccc1OC(F)F	nan
	CHEMBL1541111	46651	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	7	3.0	COc1cc(CN(C)Cc2cc(=O)n3ccsc3n2)ccc1OC(F)F	nan
	3119316	46709	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	4	3.9	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(Br)cc2)cc1	nan
	CHEMBL1541516	46709	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	4	3.9	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(Br)cc2)cc1	nan
	4885704	46762	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccccc1F	nan
	CHEMBL1541978	46762	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccccc1F	nan
	20884256	46944	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	0.5	Cc1nn(CC(=O)NCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	CHEMBL1543621	46944	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	0.5	Cc1nn(CC(=O)NCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	1451421	47045	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	0	6	3.9	CCOC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1544289	47045	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	0	6	3.9	CCOC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	7120054	47121	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	CHEMBL1544911	47121	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	3192298	47141	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	2	0	5	1.3	Cc1nc2ccccn2c1C(=O)OCC#N	nan
	CHEMBL1545062	47141	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	2	0	5	1.3	Cc1nc2ccccn2c1C(=O)OCC#N	nan
	976399	47149	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	4	4.1	Cc1ccc(OC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	CHEMBL1545103	47149	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	4	4.1	Cc1ccc(OC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	3455851	47247	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	3.2	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(F)cc1	nan
	CHEMBL1545899	47247	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	3.2	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(F)cc1	nan
	2431161	47456	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	6	3.6	CC(C)[C@H](NC(=O)c1ccccc1Cl)C(=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1547817	47456	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	6	3.6	CC(C)[C@H](NC(=O)c1ccccc1Cl)C(=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	3111438	47512	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	0	4	3.2	CC(=O)OCCCN1C(=O)c2cccc3cc(Br)cc(c23)C1=O	nan
	CHEMBL1548381	47512	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	0	4	3.2	CC(=O)OCCCN1C(=O)c2cccc3cc(Br)cc(c23)C1=O	nan
	24792694	47513	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	6	1.9	Cn1c2ccccc2c2nnc(SCC(=O)NC3CC3)nc21	nan
	CHEMBL1548382	47513	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	6	1.9	Cn1c2ccccc2c2nnc(SCC(=O)NC3CC3)nc21	nan
	664646	47528	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	3.6	COc1ccc(C(=O)OCc2cc3cccc(C)c3nc2O)cc1	nan
	CHEMBL1548510	47528	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	3.6	COc1ccc(C(=O)OCc2cc3cccc(C)c3nc2O)cc1	nan
	839503	47549	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	3	3	3.0	O=C(Nc1ccccc1C(=O)O)c1ccc(NC(=O)C2CC2)cc1	nan
	CHEMBL1548673	47549	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	3	3	3.0	O=C(Nc1ccccc1C(=O)O)c1ccc(NC(=O)C2CC2)cc1	nan
	4839425	47642	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	10	0.2	CN(C)S(=O)(=O)c1cc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1Cl	nan
	CHEMBL1549482	47642	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	10	0.2	CN(C)S(=O)(=O)c1cc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1Cl	nan
	838258	47725	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	1	1	3	3.6	Sc1nc(-c2ccccc2)nc2ccccc12	nan
	CHEMBL1550135	47725	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	1	1	3	3.6	Sc1nc(-c2ccccc2)nc2ccccc12	nan
	2794423	47754	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	2	2.3	NC1=CC(=O)c2cccc3cccc1c23	nan
	CHEMBL1550366	47754	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	2	2.3	NC1=CC(=O)c2cccc3cccc1c23	nan
	16187761	47778	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	7	2.2	Cc1cc(C)n2nc(C(=O)N3CCCC(CNS(=O)(=O)c4cccs4)C3)cc2n1	nan
	CHEMBL1550610	47778	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	7	2.2	Cc1cc(C)n2nc(C(=O)N3CCCC(CNS(=O)(=O)c4cccs4)C3)cc2n1	nan
	4969856	47853	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	2	6	2.1	CC(=O)Nc1ccc(Nc2ncnc3c2cnn3C)cc1	nan
	CHEMBL1551291	47853	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	2	6	2.1	CC(=O)Nc1ccc(Nc2ncnc3c2cnn3C)cc1	nan
	16009663	47856	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	7	4.8	CSc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1551326	47856	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	7	4.8	CSc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)c1	nan
	7184893	47932	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	8	3.7	CCCCNc1nc2c(S(=O)(=O)c3ccc(C)cc3)nnn2c2ccsc12	nan
	CHEMBL1552371	47932	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	8	3.7	CCCCNc1nc2c(S(=O)(=O)c3ccc(C)cc3)nnn2c2ccsc12	nan
	1003444	47943	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	2	5	5.7	Nc1c(C(=O)Nc2ccc(Cl)cc2F)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1552586	47943	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	2	5	5.7	Nc1c(C(=O)Nc2ccc(Cl)cc2F)sc2nc(-c3cccs3)ccc12	nan
	1841026	47973	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	0	8	1.6	CCOC(=O)/C(C#N)=C/c1c(N2CCN(CC)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1553005	47973	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	0	8	1.6	CCOC(=O)/C(C#N)=C/c1c(N2CCN(CC)CC2)nc2c(C)cccn2c1=O	nan
	15988107	47975	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	0	7	3.8	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(Cc2ccccc2)c(=O)c2c1c1cc(OC)ccc1n2C	nan
	CHEMBL1553031	47975	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	0	7	3.8	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(Cc2ccccc2)c(=O)c2c1c1cc(OC)ccc1n2C	nan
	16009750	47979	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	Cc1cccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)c1	nan
	CHEMBL1553063	47979	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	Cc1cccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)c1	nan
	15988172	47997	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	2	4	2.2	CCCCNC(=O)c1ccc2c(=O)n(-c3ccccc3)c(=O)[nH]c2c1	nan
	CHEMBL1553275	47997	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	2	4	2.2	CCCCNC(=O)c1ccc2c(=O)n(-c3ccccc3)c(=O)[nH]c2c1	nan
	135697665	48007	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	9	1.8	O=C(OCc1nc(O)c2sccc2n1)c1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1553392	48007	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	9	1.8	O=C(OCc1nc(O)c2sccc2n1)c1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	5927505	48201	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	7	4.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1556043	48201	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	7	4.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCCO2	nan
	2195056	48234	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	2	4.7	O=C(Nc1ccc(F)cc1)c1ccc(COc2ccccc2)cc1	nan
	CHEMBL1556330	48234	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	2	4.7	O=C(Nc1ccc(F)cc1)c1ccc(COc2ccccc2)cc1	nan
	5301777	48251	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	2	6	5.9	COC(=O)c1ccccc1NC(=O)c1sc2nc(C)cc(C)c2c1NC(=O)c1ccccc1Cl	nan
	CHEMBL1556556	48251	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	2	6	5.9	COC(=O)c1ccccc1NC(=O)c1sc2nc(C)cc(C)c2c1NC(=O)c1ccccc1Cl	nan
	3404081	48274	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2c(C)cc(S)nc2c1	nan
	CHEMBL1556798	48274	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2c(C)cc(S)nc2c1	nan
	1348154	48281	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	4	4.9	O=C(Cc1ccc(Cl)cc1)Nc1ccc2nn(-c3ccc(Cl)cc3)nc2c1	nan
	CHEMBL1556858	48281	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	4	4.9	O=C(Cc1ccc(Cl)cc1)Nc1ccc2nn(-c3ccc(Cl)cc3)nc2c1	nan
	3708288	48293	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	1	4	7	2.3	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1ccccc1	nan
	CHEMBL1556915	48293	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	1	4	7	2.3	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1ccccc1	nan
	285470	48334	24	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CCNc1nc(Cl)nc(-c2cn(-c3ccccc3)c3ccccc23)n1	nan
	CHEMBL1557270	48334	24	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CCNc1nc(Cl)nc(-c2cn(-c3ccccc3)c3ccccc23)n1	nan
	16009846	48379	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	8	1.7	COc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)c(OC)c1	nan
	CHEMBL1557614	48379	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	8	1.7	COc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)c(OC)c1	nan
	16010737	48388	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	CCc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(C)cc3)c(=O)c3cccnc32)cc1	nan
	CHEMBL1557693	48388	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	CCc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(C)cc3)c(=O)c3cccnc32)cc1	nan
	3333649	48547	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cccs1	nan
	CHEMBL1559037	48547	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cccs1	nan
	1166246	48602	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)c(C)c1	nan
	CHEMBL1559537	48602	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)c(C)c1	nan
	16009080	48804	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	7	1	7	6.7	CCOc1ccc(-c2cc3nc(C4CCN(C(=O)OC(C)(C)C)CC4)c(C(=O)Nc4cccc(CC)c4)cn3n2)cc1	nan
	CHEMBL1561508	48804	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	7	1	7	6.7	CCOc1ccc(-c2cc3nc(C4CCN(C(=O)OC(C)(C)C)CC4)c(C(=O)Nc4cccc(CC)c4)cn3n2)cc1	nan
	3141845	48862	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	4	6.0	COc1cc(NC(=O)c2ccc(Cl)cc2Cl)ccc1-c1cc2ccccc2oc1=O	nan
	CHEMBL1562003	48862	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	4	6.0	COc1cc(NC(=O)c2ccc(Cl)cc2Cl)ccc1-c1cc2ccccc2oc1=O	nan
	2510921	48968	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	5	2.8	O=C(CNC(=O)C1CCCCC1)OCC(=O)c1ccc(Cl)s1	nan
	CHEMBL1562941	48968	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	5	2.8	O=C(CNC(=O)C1CCCCC1)OCC(=O)c1ccc(Cl)s1	nan
	4800554	49090	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	6	3.8	COc1cc(C(C)=O)ccc1OCC(=O)Nc1ccc2nc(C)sc2c1	nan
	CHEMBL1563979	49090	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	6	3.8	COc1cc(C(C)=O)ccc1OCC(=O)Nc1ccc2nc(C)sc2c1	nan
	16009343	49109	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	0	5	4.3	Cc1ccccc1OCc1cc(=O)n2c(-c3ccccc3)csc2n1	nan
	CHEMBL1564149	49109	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	0	5	4.3	Cc1ccccc1OCc1cc(=O)n2c(-c3ccccc3)csc2n1	nan
	4911790	49220	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	1	2	3.4	COc1ccc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2c1	nan
	CHEMBL1565220	49220	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	1	2	3.4	COc1ccc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2c1	nan
	974361	49275	12	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	3.9	Cc1onc(-c2ccccc2)c1C(=O)Nc1cccc2nsnc12	nan
	CHEMBL1565576	49275	12	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	3.9	Cc1onc(-c2ccccc2)c1C(=O)Nc1cccc2nsnc12	nan
	15989682	49302	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	1	8	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1565778	49302	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	1	8	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	1977639	49305	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	5	5.2	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1ccccc1Cl	nan
	CHEMBL1565785	49305	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	5	5.2	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1ccccc1Cl	nan
	789538	49440	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	0	1	4	2.0	CC1=C(C)C(C)=C(C#N)C(=C(C#N)C#N)N1	nan
	CHEMBL1566885	49440	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	0	1	4	2.0	CC1=C(C)C(C)=C(C#N)C(=C(C#N)C#N)N1	nan
	3442888	49544	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	1	0	5	3.1	Cc1cccn2c(=O)c3cc(C(=O)N4CCCC(C)C4)sc3nc12	nan
	CHEMBL1567700	49544	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	1	0	5	3.1	Cc1cccn2c(=O)c3cc(C(=O)N4CCCC(C)C4)sc3nc12	nan
	16009353	49856	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1C	nan
	CHEMBL1570398	49856	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1C	nan
	16019299	49870	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	1	5	4.2	Cc1cc(C)c(NC(=O)CSc2ccc(-c3ccccn3)nn2)c(C)c1	nan
	CHEMBL1570518	49870	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	1	5	4.2	Cc1cc(C)c(NC(=O)CSc2ccc(-c3ccccn3)nn2)c(C)c1	nan
	4917201	49942	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	6	1.4	CC(C(=O)Nc1cccnc1)n1cc([N+](=O)[O-])cn1	nan
	CHEMBL1571073	49942	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	6	1.4	CC(C(=O)Nc1cccnc1)n1cc([N+](=O)[O-])cn1	nan
	15990163	49944	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	7	3.3	COc1ccc(S(=O)(=O)Nc2cc3c(cc2NCc2ccccc2)n(C)c(=O)n3C)cc1	nan
	CHEMBL1571094	49944	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	7	3.3	COc1ccc(S(=O)(=O)Nc2cc3c(cc2NCc2ccccc2)n(C)c(=O)n3C)cc1	nan
	16194623	50029	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	0	8	1.8	CC(=O)C(Sc1ccc2nnc(-c3cccnc3)n2n1)C(C)=O	nan
	CHEMBL1572020	50029	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	0	8	1.8	CC(=O)C(Sc1ccc2nnc(-c3cccnc3)n2n1)C(C)=O	nan
	135408736	50084	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	228	1	1	5	2.1	Sc1ncnc2c1cnn2-c1ccccc1	nan
	CHEMBL1572500	50084	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	228	1	1	5	2.1	Sc1ncnc2c1cnn2-c1ccccc1	nan
	2769007	50400	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	0	7	1.4	CCOC(=O)C(C)Sc1nc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1575703	50400	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	0	7	1.4	CCOC(=O)C(C)Sc1nc(=O)n2cc(C)ccc2n1	nan
	2808306	50416	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	5	2	4	3.1	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)CCC(=O)O	nan
	CHEMBL1575844	50416	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	5	2	4	3.1	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)CCC(=O)O	nan
	4356534	50519	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	4.4	COc1ccc2nc(Cl)c(C3CC(c4ccco4)=NN3C(=O)CCCC(=O)O)cc2c1	nan
	CHEMBL1576687	50519	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	4.4	COc1ccc2nc(Cl)c(C3CC(c4ccco4)=NN3C(=O)CCCC(=O)O)cc2c1	nan
	22517522	50642	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	7	2.1	CC(Oc1ccccc1)C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	CHEMBL1577822	50642	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	7	2.1	CC(Oc1ccccc1)C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	20856926	50832	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	4	3.0	CC(=O)c1cccc(NC(=O)CNC(=O)c2cc3ccccc3o2)c1	nan
	CHEMBL1579387	50832	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	4	3.0	CC(=O)c1cccc(NC(=O)CNC(=O)c2cc3ccccc3o2)c1	nan
	4368409	50923	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	8	4.7	CCCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1580198	50923	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	8	4.7	CCCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	990451	50988	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	0	7	3.2	Cc1ccc(-n2nc3c(SCCN4CCOCC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1580766	50988	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	0	7	3.2	Cc1ccc(-n2nc3c(SCCN4CCOCC4)nnc(C)c3c2C)cc1	nan
	661914	51075	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1581469	51075	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	679340	51087	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	2	6	1.8	Cc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)o1	nan
	CHEMBL1581638	51087	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	2	6	1.8	Cc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)o1	nan
	990454	51106	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	7	3.0	Cc1nnc(SCCN2CCOCC2)c2nn(-c3ccccc3F)c(C)c12	nan
	CHEMBL1581794	51106	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	7	3.0	Cc1nnc(SCCN2CCOCC2)c2nn(-c3ccccc3F)c(C)c12	nan
	2666708	51152	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	7	3.3	COc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc(OC)c1C	nan
	CHEMBL1582108	51152	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	7	3.3	COc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc(OC)c1C	nan
	1943119	51427	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	0	10	2.9	COCCn1c(-c2cc(OC)c(OC)c(OC)c2)nc2oc3cc(OC)ccc3c(=O)c2c1=O	nan
	CHEMBL1584456	51427	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	0	10	2.9	COCCn1c(-c2cc(OC)c(OC)c(OC)c2)nc2oc3cc(OC)ccc3c(=O)c2c1=O	nan
	5923696	51606	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	1	9	-0.3	N#C/C(=C\c1c(N2CCOCC2)nc2ccccn2c1=O)C(=O)NC1CCS(=O)(=O)C1	nan
	CHEMBL1585817	51606	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	1	9	-0.3	N#C/C(=C\c1c(N2CCOCC2)nc2ccccn2c1=O)C(=O)NC1CCS(=O)(=O)C1	nan
	11957204	51653	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	5.1	O=C(Nc1nccs1)c1cc2sccc2n1Cc1ccc(Cl)cc1	nan
	CHEMBL1586282	51653	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	5.1	O=C(Nc1nccs1)c1cc2sccc2n1Cc1ccc(Cl)cc1	nan
	2534667	51665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	0	6	2.4	COc1ccc(C(C)=O)cc1COC(=O)c1cnc(C)cn1	nan
	CHEMBL1586370	51665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	0	6	2.4	COc1ccc(C(C)=O)cc1COC(=O)c1cnc(C)cn1	nan
	2048070	51669	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	4	4.0	Cc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1C	nan
	CHEMBL1586414	51669	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	4	4.0	Cc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1C	nan
	4382155	51715	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	6	1	4	2.7	CCc1ccccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1586776	51715	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	6	1	4	2.7	CCc1ccccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	3548898	51749	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	2	6	1.7	CC(=O)N1CCc2c(sc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)c2C(N)=O)C1	nan
	CHEMBL1587022	51749	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	2	6	1.7	CC(=O)N1CCc2c(sc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)c2C(N)=O)C1	nan
	3565925	51820	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.9	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCC(C)C3	nan
	CHEMBL1587609	51820	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.9	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCC(C)C3	nan
	661736	51839	14	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	6	3.5	Cc1ccccc1N1C(=O)CC(Sc2nnc(-c3ccccc3)o2)C1=O	nan
	CHEMBL1587764	51839	14	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	6	3.5	Cc1ccccc1N1C(=O)CC(Sc2nnc(-c3ccccc3)o2)C1=O	nan
	5919084	51892	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	2.9	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(F)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1588231	51892	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	2.9	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(F)cc1)c1ccc2c(c1)OCCO2	nan
	859793	51920	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	9	-0.6	Cn1c(=O)c2c(nc(SCCN3CCOCC3)n2C)n(C)c1=O	nan
	CHEMBL1588519	51920	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	9	-0.6	Cn1c(=O)c2c(nc(SCCN3CCOCC3)n2C)n(C)c1=O	nan
	4203923	51990	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	4573010	51990	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	CHEMBL1589149	51990	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	16016946	52071	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	5	4.5	Cc1c(Cl)cccc1NC(=O)Cn1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1589855	52071	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	5	4.5	Cc1c(Cl)cccc1NC(=O)Cn1nc(C)c2sc3ccccc3c2c1=O	nan
	16014998	52073	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2ccc(C)cc2)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1589876	52073	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2ccc(C)cc2)c(C#N)c(-c2ccccc2)n1	nan
	16017572	52085	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.7	CCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1589962	52085	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.7	CCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	16019870	52090	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.8	COc1ccc(OC)c(NC(=O)CSc2cn(CC(=O)N3CCCCCC3)c3ccccc23)c1	nan
	CHEMBL1590046	52090	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.8	COc1ccc(OC)c(NC(=O)CSc2cn(CC(=O)N3CCCCCC3)c3ccccc23)c1	nan
	8070199	52102	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	8	1	7	3.5	Cn1nnnc1SCCCNCc1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1590182	52102	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	8	1	7	3.5	Cn1nnnc1SCCCNCc1ccc(-c2ccc(Br)cc2)o1	nan
	1252599	52121	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	1.9	COC(=O)c1cc(CN2C(=O)c3ccccc3C2=O)c(O)c([N+](=O)[O-])c1	nan
	CHEMBL1590469	52121	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	1.9	COC(=O)c1cc(CN2C(=O)c3ccccc3C2=O)c(O)c([N+](=O)[O-])c1	nan
	3438312	52140	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	5	3.3	COc1ccccc1Cn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	CHEMBL1590737	52140	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	5	3.3	COc1ccccc1Cn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	8391566	52168	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	0	7	2.5	Cc1nnc(SCc2cc(=O)n3c(C)cccc3n2)s1	nan
	CHEMBL1590986	52168	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	0	7	2.5	Cc1nnc(SCc2cc(=O)n3c(C)cccc3n2)s1	nan
	16017932	52195	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	1	6	5.8	CCN(CC)c1ccc2cc(-c3nc4sc5c(c4c(=O)[nH]3)CCC(C(C)(C)C)C5)c(=O)oc2c1	nan
	CHEMBL1591378	52195	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	1	6	5.8	CCN(CC)c1ccc2cc(-c3nc4sc5c(c4c(=O)[nH]3)CCC(C(C)(C)C)C5)c(=O)oc2c1	nan
	7152123	52293	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	4.3	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccccc4F)ccc3n2)cc1	nan
	CHEMBL1592684	52293	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	4.3	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccccc4F)ccc3n2)cc1	nan
	20885677	52317	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	6	1	6	1.3	Cc1nn(CCCC(=O)NCc2ccccc2)c(=O)c2nccn12	nan
	CHEMBL1592977	52317	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	6	1	6	1.3	Cc1nn(CCCC(=O)NCc2ccccc2)c(=O)c2nccn12	nan
	16403621	52320	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	7	3.0	COc1ccc(OC)c(/C=C2\Oc3cc(OCC(=O)N4CCC(C(=O)O)CC4)ccc3C2=O)c1	nan
	CHEMBL1593051	52320	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	7	3.0	COc1ccc(OC)c(/C=C2\Oc3cc(OCC(=O)N4CCC(C(=O)O)CC4)ccc3C2=O)c1	nan
	20893093	52329	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	1	7	3.0	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(Cl)c3C)sc2n1	nan
	CHEMBL1593179	52329	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	1	7	3.0	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(Cl)c3C)sc2n1	nan
	16018628	52389	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	0	7	5.4	Cc1oc(-c2ccccc2Cl)nc1CSc1nncn2c1cc1occc12	nan
	CHEMBL1594061	52389	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	0	7	5.4	Cc1oc(-c2ccccc2Cl)nc1CSc1nncn2c1cc1occc12	nan
	16025303	52540	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.2	Cc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1595335	52540	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.2	Cc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	5310070	52548	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	0	8	1.8	CCOC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1595390	52548	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	0	8	1.8	CCOC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	15991139	52580	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	0	4	5.2	CCC(C)OC(=O)/C(C#N)=C\c1ccc(-c2cccc(C(F)(F)F)c2)o1	nan
	CHEMBL1595672	52580	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	0	4	5.2	CCC(C)OC(=O)/C(C#N)=C\c1ccc(-c2cccc(C(F)(F)F)c2)o1	nan
	5135766	52672	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	3	5.0	O=C(COc1ccc2oc3c(c2c1)CCCC3)Nc1ccc(Cl)cc1	nan
	CHEMBL1596555	52672	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	3	5.0	O=C(COc1ccc2oc3c(c2c1)CCCC3)Nc1ccc(Cl)cc1	nan
	3653425	52761	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	661006	52761	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	CHEMBL1597383	52761	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	2991609	52765	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	7	2	4	1.6	Cc1ccc(OCC(=O)NCCNC(=O)c2cccnc2)cc1C	nan
	CHEMBL1597415	52765	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	7	2	4	1.6	Cc1ccc(OCC(=O)NCCNC(=O)c2cccnc2)cc1C	nan
	20893092	52824	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.4	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3ccccc3C)sc2n1	nan
	CHEMBL1597947	52824	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.4	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3ccccc3C)sc2n1	nan
	44666769	52846	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	5289738	52846	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	CHEMBL1598157	52846	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	5310246	52857	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.0	COc1ccc(-c2cn3c(C)c(C(=O)Nc4ccncc4)sc3n2)cc1	nan
	CHEMBL1598249	52857	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.0	COc1ccc(-c2cn3c(C)c(C(=O)Nc4ccncc4)sc3n2)cc1	nan
	2807627	52912	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	1	0	5	1.4	CC1CCCN(c2ccc3nncn3n2)C1	nan
	CHEMBL1598761	52912	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	1	0	5	1.4	CC1CCCN(c2ccc3nncn3n2)C1	nan
	22514515	52996	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	0	7	0.9	CCOC(=O)C1CCN(C(=O)Cn2nc(CC)n3cccc3c2=O)CC1	nan
	CHEMBL1599442	52996	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	0	7	0.9	CCOC(=O)C1CCN(C(=O)Cn2nc(CC)n3cccc3c2=O)CC1	nan
	2913046	53182	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	5.1	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)c(Cl)c2)o1	nan
	CHEMBL1601179	53182	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	5.1	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)c(Cl)c2)o1	nan
	3152554	53209	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.3	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1Cl)c1ccco1	nan
	CHEMBL1601448	53209	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.3	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1Cl)c1ccco1	nan
	3733422	53255	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.2	COc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	CHEMBL1602024	53255	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.2	COc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	3185717	53258	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	8	3.2	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1C	nan
	CHEMBL1602063	53258	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	8	3.2	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1C	nan
	1541054	53585	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	5	4.3	CCOc1cccc(NC(=O)CSc2nc(C)c3c(c2C#N)CCCC3)c1	nan
	CHEMBL1604887	53585	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	5	4.3	CCOc1cccc(NC(=O)CSc2nc(C)c3c(c2C#N)CCCC3)c1	nan
	20885689	53650	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1605440	53650	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	2890303	53749	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	2.7	CC(=O)C1=C(O)C(=O)N(c2ccccn2)C1c1cccc(F)c1	nan
	CHEMBL1606210	53749	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	2.7	CC(=O)C1=C(O)C(=O)N(c2ccccn2)C1c1cccc(F)c1	nan
	16030495	53790	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	5.9	Cc1ccc(Cl)cc1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1606531	53790	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	5.9	Cc1ccc(Cl)cc1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	855274	53922	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	0	5	2.0	COc1ccc2cc(C#N)c(N3CCOCC3)nc2c1	nan
	CHEMBL1607471	53922	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	0	5	2.0	COc1ccc2cc(C#N)c(N3CCOCC3)nc2c1	nan
	3663093	53946	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.6	CCc1nnc(NC(=O)CSc2nc3c([nH]c4ccccc43)c(=O)n2-c2cc(C)cc(C)c2)s1	nan
	CHEMBL1607685	53946	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.6	CCc1nnc(NC(=O)CSc2nc3c([nH]c4ccccc43)c(=O)n2-c2cc(C)cc(C)c2)s1	nan
	889917	54047	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	5	1	3	3.7	CCc1c(SCCC(=O)O)nc2ccccc2c1C	nan
	CHEMBL1608598	54047	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	5	1	3	3.7	CCc1c(SCCC(=O)O)nc2ccccc2c1C	nan
	7120053	54198	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	CHEMBL1609827	54198	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	2371304	54237	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	6	2.8	O=C(CSc1ncnc2ccccc12)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1610145	54237	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	6	2.8	O=C(CSc1ncnc2ccccc12)NCc1ccc2c(c1)OCO2	nan
	4380426	54284	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1nnc(-c2ccccc2Cl)s1)c1ccccc1F	nan
	CHEMBL1610533	54284	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1nnc(-c2ccccc2Cl)s1)c1ccccc1F	nan
	2813334	54368	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	6	3.2	CCOC(=O)C1CCCN(C(=O)c2csc(-c3ccc4c(c3)CCO4)n2)C1	nan
	CHEMBL1611317	54368	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	6	3.2	CCOC(=O)C1CCCN(C(=O)c2csc(-c3ccc4c(c3)CCO4)n2)C1	nan
	16014906	54414	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc(CNC(=O)c2cc3cc(C)ccc3n2C)cc1	nan
	CHEMBL1611737	54414	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc(CNC(=O)c2cc3cc(C)ccc3n2C)cc1	nan
	4853715	54425	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.6	CC(=O)c1sc(NC(=O)c2cnc(Cl)c(Cl)c2)nc1C	nan
	CHEMBL1611812	54425	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.6	CC(=O)c1sc(NC(=O)c2cnc(Cl)c(Cl)c2)nc1C	nan
	16009370	54438	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	0	5	5.3	O=c1cc(COc2ccc(Cl)cc2Cl)nc2scc(-c3ccccc3)n12	nan
	CHEMBL1611935	54438	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	0	5	5.3	O=c1cc(COc2ccc(Cl)cc2Cl)nc2scc(-c3ccccc3)n12	nan
	24892471	54735	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	CHEMBL1356182	54735	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	CHEMBL1616404	54735	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	24789689	55093	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	CHEMBL1395742	55093	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	CHEMBL1619301	55093	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	6489920	55239	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1428082	55239	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1620517	55239	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	5064206	55286	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	CHEMBL1455685	55286	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	CHEMBL1621049	55286	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	820476	55539	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	CHEMBL1522563	55539	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	CHEMBL1623170	55539	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	1560419	55543	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	CHEMBL1517106	55543	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	CHEMBL1623202	55543	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	1567753	55555	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	CHEMBL1534121	55555	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	CHEMBL1623318	55555	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	818329	55719	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	CHEMBL1568356	55719	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	CHEMBL1624703	55719	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	3146476	69453	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	5767654	69453	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	6248042	69453	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	CHEMBL193627	69453	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	CHEMBL584458	69453	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	2152519	71628	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	7	0	9	3.6	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1ccccc1OCC	nan
	CHEMBL1973861	71628	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	7	0	9	3.6	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1ccccc1OCC	nan
	2003230	71882	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	0	8	1.2	CCOC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CCOC)/c1=N\C(C)=O	nan
	CHEMBL1981685	71882	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	0	8	1.2	CCOC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CCOC)/c1=N\C(C)=O	nan
	9580624	72030	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	6	1	7	2.5	COc1cccc(/C=N/Nc2ncccc2[N+](=O)[O-])c1OC	nan
	CHEMBL1986514	72030	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	6	1	7	2.5	COc1cccc(/C=N/Nc2ncccc2[N+](=O)[O-])c1OC	nan
	9564678	72174	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1991163	72174	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	135406177	72198	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	2	2	4	3.6	Cc1ccc(O)c(/N=C/C2=C(O)c3ccccc3C2=O)c1	nan
	CHEMBL1991885	72198	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	2	2	4	3.6	Cc1ccc(O)c(/N=C/C2=C(O)c3ccccc3C2=O)c1	nan
	9583975	72285	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	2	6	5.8	Nc1c(C(=O)N/N=C/c2ccccc2Cl)oc2nc(-c3ccccc3)cc(-c3ccco3)c12	nan
	CHEMBL1995041	72285	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	2	6	5.8	Nc1c(C(=O)N/N=C/c2ccccc2Cl)oc2nc(-c3ccccc3)cc(-c3ccco3)c12	nan
	5936993	72456	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	0	2	6.9	CCN(CC)c1ccc(/C=C/c2cc(-c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL2001294	72456	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	0	2	6.9	CCN(CC)c1ccc(/C=C/c2cc(-c3ccccc3)c3ccccc3n2)cc1	nan
	735993	87568	36	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.1	CN(C)c1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	CHEMBL234378	87568	36	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.1	CN(C)c1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	9638128	107254	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	7	0	5	3.4	CCN(CC)c1ccc(C(=O)c2cnc(/N=C/N(C)C)s2)cc1	nan
	CHEMBL3191439	107254	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	7	0	5	3.4	CCN(CC)c1ccc(C(=O)c2cnc(/N=C/N(C)C)s2)cc1	nan
	24892228	107358	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	0	8	2.7	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3192568	107358	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	0	8	2.7	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	46497908	107518	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	10	0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C\c2ccccc2[N+](=O)[O-])n(C)c1=O	nan
	CHEMBL3194459	107518	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	10	0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C\c2ccccc2[N+](=O)[O-])n(C)c1=O	nan
	135412189	107743	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	3	10	1.0	COc1cc(/C=N/Nc2nc(O)nnc2C)cc([N+](=O)[O-])c1O	nan
	CHEMBL3197005	107743	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	3	10	1.0	COc1cc(/C=N/Nc2nc(O)nnc2C)cc([N+](=O)[O-])c1O	nan
	4122444	108007	11	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	2.4	CCOC(=O)c1s/c(=N\C(=O)c2cccs2)n(C)c1C	nan
	CHEMBL3199794	108007	11	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	2.4	CCOC(=O)c1s/c(=N\C(=O)c2cccs2)n(C)c1C	nan
	5343366	108012	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	4	0	7	1.8	CSc1nncn1/N=C/c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3199842	108012	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	4	0	7	1.8	CSc1nncn1/N=C/c1ccc([N+](=O)[O-])cc1	nan
	135411619	108022	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	4	1	8	1.5	Cc1nn(-c2ccc([N+](=O)[O-])cc2)c(O)c1/C=N/N1CCOCC1	nan
	CHEMBL3199911	108022	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	4	1	8	1.5	Cc1nn(-c2ccc([N+](=O)[O-])cc2)c(O)c1/C=N/N1CCOCC1	nan
	9955	141793	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	CHEMBL1356616	141793	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	CHEMBL388594	141793	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	154730799	167104	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	65191	167104	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	CHEMBL1306565	167104	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	CHEMBL4302011	167104	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	21551	183658	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	2	0	6	0.6	Cn1c(=O)c2c(nc(Cc3ccccc3)n2C)n(C)c1=O	nan
	CHEMBL483661	183658	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	2	0	6	0.6	Cn1c(=O)c2c(nc(Cc3ccccc3)n2C)n(C)c1=O	nan
	4380636	199311	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	5.3	CC(C)c1ccc(Nc2c(-c3ccccn3)nc3ccccn23)cc1	nan
	CHEMBL602150	199311	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	5.3	CC(C)c1ccc(Nc2c(-c3ccccn3)nc3ccccn23)cc1	nan
	1499	2052	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	3779	2052	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	536	2052	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	CHEMBL434	2052	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	DB01064	2052	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	3762	14316	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	CHEMBL1201153	14316	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	CHEMBL1201213	14316	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	1214032	19547	13	None	-2	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	6	1	7	6.1	CC1(C)Cc2nc3sc4c(SCC(=O)NC(c5ccccc5)c5ccccc5)ncnc4c3cc2CO1	nan
	CHEMBL1301335	19547	13	None	-2	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	6	1	7	6.1	CC1(C)Cc2nc3sc4c(SCC(=O)NC(c5ccccc5)c5ccccc5)ncnc4c3cc2CO1	nan
	15990933	21558	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	3	6.2	CC(C)c1ccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)cc1	nan
	CHEMBL1319127	21558	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	3	6.2	CC(C)c1ccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)cc1	nan
	1716420	21857	14	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	5	6.5	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(C(F)(F)F)c4)c(Br)c3n2)cc1	nan
	CHEMBL1321710	21857	14	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	5	6.5	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(C(F)(F)F)c4)c(Br)c3n2)cc1	nan
	2919028	24154	15	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	10	3.9	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OC)c(OC)c2)nc1C	nan
	CHEMBL1341127	24154	15	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	10	3.9	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OC)c(OC)c2)nc1C	nan
	16019314	30669	12	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	5	1	9	4.9	COc1ccc(C)cc1Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	CHEMBL1397774	30669	12	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	5	1	9	4.9	COc1ccc(C)cc1Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	944832	31330	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	0	2	3	3.0	Sc1[nH]cnc2c3cc(Cl)ccc3nc1-2	nan
	CHEMBL1404042	31330	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	0	2	3	3.0	Sc1[nH]cnc2c3cc(Cl)ccc3nc1-2	nan
	4024853	31471	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.6	CCCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc(N(C)C)cc4)nc3c2)cc1	nan
	CHEMBL1405437	31471	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.6	CCCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc(N(C)C)cc4)nc3c2)cc1	nan
	24892224	33867	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	9	0.5	CC(C)c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1425449	33867	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	9	0.5	CC(C)c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16033262	36029	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	1	5	5.9	Cc1c(C(=O)Nc2ccc(Br)cc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1445708	36029	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	1	5	5.9	Cc1c(C(=O)Nc2ccc(Br)cc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	4179349	39342	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	8	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1473745	39342	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	8	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	2810065	42698	6	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	2	1	5	4.0	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)c1ccco1	nan
	CHEMBL1503612	42698	6	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	2	1	5	4.0	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)c1ccco1	nan
	16019583	43823	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	4	0	9	3.1	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1514816	43823	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	4	0	9	3.1	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	16023031	44355	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	3.1	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(F)cc3)s2)cc1	nan
	CHEMBL1520434	44355	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	3.1	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(F)cc3)s2)cc1	nan
	16030551	47843	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	4	5.1	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	CHEMBL1551173	47843	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	4	5.1	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	16009713	53679	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(-c2nnn3c2nc(NCc2ccc(C)cc2)c2ccccc23)cc1	nan
	CHEMBL1605623	53679	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(-c2nnn3c2nc(NCc2ccc(C)cc2)c2ccccc23)cc1	nan
	49858523	89090	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	0	5	5.0	CCCC[C@]12Cc3cc(C#N)ccc3[C@H](O1)c1c(cc(C)n(Cc3ccccc3)c1=O)O2	nan
	CHEMBL2373613	89090	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	0	5	5.0	CCCC[C@]12Cc3cc(C#N)ccc3[C@H](O1)c1c(cc(C)n(Cc3ccccc3)c1=O)O2	nan
	16010255	5880	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.1	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccc(Cl)cc23)c(C)c1	nan
	CHEMBL1079970	5880	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.1	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccc(Cl)cc23)c(C)c1	nan
	16010278	6039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	7	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1cc(Cl)ccc12	nan
	CHEMBL1080898	6039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	7	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1cc(Cl)ccc12	nan
	18560284	6254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	7	1	8	3.3	O=C1CCCN1CCCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccccc12	nan
	CHEMBL1082027	6254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	7	1	8	3.3	O=C1CCCN1CCCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccccc12	nan
	16010337	6292	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	4.1	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2cc(Cl)ccc23)cc1	nan
	CHEMBL1082207	6292	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	4.1	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2cc(Cl)ccc23)cc1	nan
	7185123	10562	7	None	-851	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	CHEMBL1170673	10562	7	None	-851	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	16019553	10591	7	None	-912	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	8	4.4	CC(C)CCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccsc12	nan
	CHEMBL1170871	10591	7	None	-912	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	8	4.4	CC(C)CCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccsc12	nan
	16019312	10782	0	None	-144	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	9	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1172727	10782	0	None	-144	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	9	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	4968664	19484	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3cc(C)ccc3C)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1300883	19484	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3cc(C)ccc3C)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	16435505	19520	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CC3CCCO3)c(=O)n2c1	nan
	CHEMBL1301161	19520	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CC3CCCO3)c(=O)n2c1	nan
	1451395	19546	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.6	Cc1cccc(NC(=O)CSc2nc(COc3ccccc3)nc3ccccc23)c1C	nan
	CHEMBL1301326	19546	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.6	Cc1cccc(NC(=O)CSc2nc(COc3ccccc3)nc3ccccc23)c1C	nan
	1019237	19707	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	6	2	5	3.6	COc1ccccc1C(=O)Nc1cccc(NC(=O)c2ccccc2OC)n1	nan
	CHEMBL1302646	19707	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	6	2	5	3.6	COc1ccccc1C(=O)Nc1cccc(NC(=O)c2ccccc2OC)n1	nan
	1176215	19890	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	7	3.7	CCc1nnc(NC(=O)CSc2nc3cc(OC)ccc3cc2C)s1	nan
	CHEMBL1304139	19890	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	7	3.7	CCc1nnc(NC(=O)CSc2nc3cc(OC)ccc3cc2C)s1	nan
	706653	19896	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	5	3.5	N#Cc1c(-c2ccccc2)c(C#N)c2nc3ccccc3n2c1N	nan
	CHEMBL1304187	19896	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	5	3.5	N#Cc1c(-c2ccccc2)c(C#N)c2nc3ccccc3n2c1N	nan
	2060107	19942	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.7	COc1ccc(NC(=O)CSc2nnc(-c3cccs3)n2-c2ccccc2)cc1	nan
	CHEMBL1304585	19942	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.7	COc1ccc(NC(=O)CSc2nnc(-c3cccs3)n2-c2ccccc2)cc1	nan
	16034541	20153	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	6	3.5	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Br)s1	nan
	CHEMBL1306241	20153	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	6	3.5	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Br)s1	nan
	12005386	20235	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	6	4.7	CCCCOc1ccc(C(=O)Nn2c(-c3cccs3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1306967	20235	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	6	4.7	CCCCOc1ccc(C(=O)Nn2c(-c3cccs3)nc3ccccc3c2=O)cc1	nan
	24818410	20487	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	6	0	6	4.2	COc1cccc(COC(=O)c2c(C)nn(-c3ccccc3)c2Cl)c1OC	nan
	CHEMBL1308959	20487	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	6	0	6	4.2	COc1cccc(COC(=O)c2c(C)nn(-c3ccccc3)c2Cl)c1OC	nan
	2081889	20760	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(Cc3ccccc3)c(=O)c2c1C	nan
	CHEMBL1311321	20760	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(Cc3ccccc3)c(=O)c2c1C	nan
	2102674	20786	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	3.6	Cc1cc(NC(=O)CSc2nc3ccccc3c(=O)n2Cc2ccc(F)cc2)no1	nan
	CHEMBL1311532	20786	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	3.6	Cc1cc(NC(=O)CSc2nc3ccccc3c(=O)n2Cc2ccc(F)cc2)no1	nan
	651309	21124	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	CHEMBL1314039	21124	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	16028453	21191	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	3	4	5.4	CCc1ccccc1NC(=O)Nc1cc(C(=O)NCc2ccc(OC)cc2)ccc1N1CCCC1	nan
	CHEMBL1314777	21191	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	3	4	5.4	CCc1ccccc1NC(=O)Nc1cc(C(=O)NCc2ccc(OC)cc2)ccc1N1CCCC1	nan
	15990013	21204	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	2	8	3.4	COc1ccccc1CNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1314976	21204	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	2	8	3.4	COc1ccccc1CNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	16025439	21225	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	7	1	6	4.6	Cc1ccccc1CN1c2ccccc2-c2nc(SCC(=O)NCc3ccccc3)ncc2S1(=O)=O	nan
	CHEMBL1315303	21225	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	7	1	6	4.6	Cc1ccccc1CN1c2ccccc2-c2nc(SCC(=O)NCc3ccccc3)ncc2S1(=O)=O	nan
	18579745	21247	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	2.9	CCOC(=O)c1nn(-c2ccc(F)cc2)c(=O)cc1OCC(=O)Nc1cccc(C)c1	nan
	CHEMBL1315496	21247	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	2.9	CCOC(=O)c1nn(-c2ccc(F)cc2)c(=O)cc1OCC(=O)Nc1cccc(C)c1	nan
	135455826	21298	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	1	5	4.9	Cc1ccc(-c2cc(C(F)F)nc3sc4c(O)ncnc4c23)cc1	nan
	CHEMBL1316104	21298	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	1	5	4.9	Cc1ccc(-c2cc(C(F)F)nc3sc4c(O)ncnc4c23)cc1	nan
	16008870	21312	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	2	1	4	3.9	Cn1c(C(=O)Nc2cccc(Cl)c2)cc2c(=O)n(C)c3ccccc3c21	nan
	CHEMBL1316241	21312	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	2	1	4	3.9	Cn1c(C(=O)Nc2cccc(Cl)c2)cc2c(=O)n(C)c3ccccc3c21	nan
	16024585	21317	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1316336	21317	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	16023032	21321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	2	5	4.7	CC(=O)c1ccc(NC(=O)c2cccc(NC(=O)N3CCSc4ncccc43)c2)cc1	nan
	CHEMBL1316423	21321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	2	5	4.7	CC(=O)c1ccc(NC(=O)c2cccc(NC(=O)N3CCSc4ncccc43)c2)cc1	nan
	937929	21334	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	4	3.6	Cc1nc(N)c(C#N)c(-c2cccnc2)c1-c1ccccc1	nan
	CHEMBL1316609	21334	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	4	3.6	Cc1nc(N)c(C#N)c(-c2cccnc2)c1-c1ccccc1	nan
	16009522	21371	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4)cc3)cc(=O)n12	nan
	CHEMBL1317126	21371	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4)cc3)cc(=O)n12	nan
	16020239	21436	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	6	1	5	5.2	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(Cc3cccc(F)c3)c2=O)cc1	nan
	CHEMBL1317963	21436	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	6	1	5	5.2	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(Cc3cccc(F)c3)c2=O)cc1	nan
	16022974	21437	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.8	Cc1nnc(N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1317977	21437	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.8	Cc1nnc(N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	3450154	21473	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.6	CC(=O)c1sc(NC(=O)C2CCCN2S(=O)(=O)c2ccccc2F)nc1C	nan
	CHEMBL1318435	21473	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.6	CC(=O)c1sc(NC(=O)C2CCCN2S(=O)(=O)c2ccccc2F)nc1C	nan
	15988872	21474	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	5.4	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)sc2c1CCCC2	nan
	CHEMBL1318439	21474	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	5.4	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)sc2c1CCCC2	nan
	16008607	21477	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	6	1.6	Cc1nc2c(c(C)c1CCC(=O)NCc1ccc(F)cc1)c(=O)n(C)c(=O)n2C	nan
	CHEMBL1318457	21477	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	6	1.6	Cc1nc2c(c(C)c1CCC(=O)NCc1ccc(F)cc1)c(=O)n(C)c(=O)n2C	nan
	15991398	21495	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	4	6.3	Cc1ccc(NC(=O)c2cc3c(-c4ccccc4)nn(-c4ccccc4)c3s2)cc1	nan
	CHEMBL1318575	21495	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	4	6.3	Cc1ccc(NC(=O)c2cc3c(-c4ccccc4)nn(-c4ccccc4)c3s2)cc1	nan
	3144686	21522	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	4	4.3	CCC(C)NC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)n1	nan
	CHEMBL1318807	21522	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	4	4.3	CCC(C)NC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)n1	nan
	1329083	21568	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	4	4.7	Cc1cccc(C)c1NC(=O)COc1ccccc1C(=O)Nc1ccc(Br)cn1	nan
	CHEMBL1319204	21568	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	4	4.7	Cc1cccc(C)c1NC(=O)COc1ccccc1C(=O)Nc1ccc(Br)cn1	nan
	1983515	21596	8	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	1	6	5.3	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)cc1)c1cccs1	nan
	CHEMBL1319447	21596	8	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	1	6	5.3	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)cc1)c1cccs1	nan
	20889080	21642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	4.1	CC(CNc1nc2ccc(Cl)cc2n2cnnc12)c1ccccc1	nan
	CHEMBL1319804	21642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	4.1	CC(CNc1nc2ccc(Cl)cc2n2cnnc12)c1ccccc1	nan
	16017559	21748	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCC(C)CC3)s2)c1	nan
	CHEMBL1320668	21748	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCC(C)CC3)s2)c1	nan
	16029569	21886	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	5	4.5	Cc1cc2c(=O)c(C(=O)c3ccncc3)cn(CC(=O)Nc3cccc(C)c3C)c2cc1C	nan
	CHEMBL1321921	21886	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	5	4.5	Cc1cc2c(=O)c(C(=O)c3ccncc3)cn(CC(=O)Nc3cccc(C)c3C)c2cc1C	nan
	15989030	21918	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	3.9	Cc1ccc(CNC(=O)CCCn2c(=O)c3sccc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	CHEMBL1322214	21918	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	3.9	Cc1ccc(CNC(=O)CCCn2c(=O)c3sccc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	4412940	21983	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	5.1	CCOc1ccc(-n2cc(C(=O)Nc3ccccc3OCC)c3cc(OC)c(OC)cc3c2=O)cc1	nan
	CHEMBL1322786	21983	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	5.1	CCOc1ccc(-n2cc(C(=O)Nc3ccccc3OCC)c3cc(OC)c(OC)cc3c2=O)cc1	nan
	3197538	22031	5	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	5.3	CCCc1nc(SCC(=O)N2c3ccccc3CC2C)c2c(C)c(C)sc2n1	nan
	CHEMBL1323376	22031	5	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	5.3	CCCc1nc(SCC(=O)N2c3ccccc3CC2C)c2c(C)c(C)sc2n1	nan
	3223224	22160	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.5	Cc1ccnc(N2CCC(C(=O)NCc3ccccc3F)CC2)n1	nan
	CHEMBL1324395	22160	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.5	Cc1ccnc(N2CCC(C(=O)NCc3ccccc3F)CC2)n1	nan
	16025301	22171	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	594	8	1	8	5.4	CCOC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1324479	22171	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	594	8	1	8	5.4	CCOC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	24818748	22214	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	3	5	3.9	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)c(OC)c1	nan
	CHEMBL1324786	22214	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	3	5	3.9	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)c(OC)c1	nan
	15991180	22289	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	4	6.4	CCOc1ccc(C(=O)Nc2ccc(Cl)c(-c3nc4cc(C)cc(C)c4o3)c2)cc1	nan
	CHEMBL1325481	22289	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	4	6.4	CCOc1ccc(C(=O)Nc2ccc(Cl)c(-c3nc4cc(C)cc(C)c4o3)c2)cc1	nan
	794333	22413	52	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	0	2	3.7	COc1ccc(C(=O)c2ccc(Br)cc2)cc1	nan
	CHEMBL1326786	22413	52	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	0	2	3.7	COc1ccc(C(=O)c2ccc(Br)cc2)cc1	nan
	16012102	22434	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	CHEMBL1326931	22434	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	2097459	22450	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1ccc(NC(=O)Cn2cc(C(F)(F)F)cc(Cl)c2=O)cc1Cl	nan
	CHEMBL1327066	22450	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1ccc(NC(=O)Cn2cc(C(F)(F)F)cc(Cl)c2=O)cc1Cl	nan
	15988236	22471	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	7	2.1	CCC(C)NC(=O)Cn1c(=O)n(-c2cc(OC)cc(OC)c2)c(=O)c2ccccc21	nan
	CHEMBL1327218	22471	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	7	2.1	CCC(C)NC(=O)Cn1c(=O)n(-c2cc(OC)cc(OC)c2)c(=O)c2ccccc21	nan
	6825246	22508	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	8	2	8	1.9	CCOc1ccc(-n2c([S-])c(C(=O)Nc3ccc(S(=O)(=O)N4CCOCC4)cc3)[n+]3cc(C(N)=O)ccc23)cc1	nan
	CHEMBL1327580	22508	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	8	2	8	1.9	CCOc1ccc(-n2c([S-])c(C(=O)Nc3ccc(S(=O)(=O)N4CCOCC4)cc3)[n+]3cc(C(N)=O)ccc23)cc1	nan
	3192843	22540	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	6	2.8	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccccc2F)n1)NC1CCCC1	nan
	CHEMBL1327798	22540	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	6	2.8	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccccc2F)n1)NC1CCCC1	nan
	2816102	22601	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	2	0	5	3.3	CCOc1ncnc2c1sc1nc(C)cc(C)c12	nan
	CHEMBL1328179	22601	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	2	0	5	3.3	CCOc1ncnc2c1sc1nc(C)cc(C)c12	nan
	16009635	22747	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	8	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1OC	nan
	CHEMBL1329536	22747	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	8	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1OC	nan
	753116	22808	49	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	3	4.3	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)o1	nan
	CHEMBL1330042	22808	49	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	3	4.3	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)o1	nan
	4246541	22917	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	4	4.9	CCN(CC)S(=O)(=O)c1ccc2oc(C(=O)Nc3ccc(Br)cc3F)c(C)c2c1	nan
	CHEMBL1330918	22917	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	4	4.9	CCN(CC)S(=O)(=O)c1ccc2oc(C(=O)Nc3ccc(Br)cc3F)c(C)c2c1	nan
	701957	22982	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	3	3.4	CCOc1cc(C)cc2oc(=O)c3c(c12)CCCC3	nan
	CHEMBL1331353	22982	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	3	3.4	CCOc1cc(C)cc2oc(=O)c3c(c12)CCCC3	nan
	16014559	22983	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.9	COc1ccc(-c2nc3nc(C)cc(Nc4cccc(C(F)(F)F)c4)n3n2)cc1	nan
	CHEMBL1331359	22983	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.9	COc1ccc(-c2nc3nc(C)cc(Nc4cccc(C(F)(F)F)c4)n3n2)cc1	nan
	16009329	23058	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	1	7	3.3	O=C(Cn1cc(S(=O)(=O)c2ccc(F)cc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	CHEMBL1331963	23058	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	1	7	3.3	O=C(Cn1cc(S(=O)(=O)c2ccc(F)cc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	2151601	23105	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1332323	23105	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	5310234	23198	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	8	2.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)NCc1ccco1	nan
	CHEMBL1333013	23198	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	8	2.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)NCc1ccco1	nan
	16018028	23317	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	4	2.6	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccccc1	nan
	CHEMBL1333957	23317	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	4	2.6	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccccc1	nan
	3174233	23375	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	10	3	7	3.1	CCCCOc1ccc(N(CC(=O)NC2CCCCC2)C(=O)c2snc(C(N)=O)c2N)cc1	nan
	CHEMBL1334365	23375	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	10	3	7	3.1	CCCCOc1ccc(N(CC(=O)NC2CCCCC2)C(=O)c2snc(C(N)=O)c2N)cc1	nan
	2237458	23383	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.3	COCc1cc(C)nc(SCC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1C#N	nan
	CHEMBL1334406	23383	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.3	COCc1cc(C)nc(SCC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1C#N	nan
	16030555	23438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	5.9	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCCc2ccccc21	nan
	CHEMBL1334948	23438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	5.9	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCCc2ccccc21	nan
	1257917	23458	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	1	4	3.0	O=C(Nc1ccc(F)cc1F)c1cc2ncc(Br)cn2n1	nan
	CHEMBL1335101	23458	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	1	4	3.0	O=C(Nc1ccc(F)cc1F)c1cc2ncc(Br)cn2n1	nan
	16010812	23490	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	0	7	3.8	Fc1ccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)cc1	nan
	CHEMBL1335280	23490	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	0	7	3.8	Fc1ccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)cc1	nan
	16015336	23519	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccc5c(c4)OCO5)c3C)nc2C)cc1	nan
	CHEMBL1335512	23519	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccc5c(c4)OCO5)c3C)nc2C)cc1	nan
	1450291	23596	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	CHEMBL1336163	23596	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	5115564	23600	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	3	7	5.7	N#Cc1ccccc1NC(=O)C1SC(Nc2ccccc2)=C(c2nc3ccccc3s2)C1=N	nan
	CHEMBL1336187	23600	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	3	7	5.7	N#Cc1ccccc1NC(=O)C1SC(Nc2ccccc2)=C(c2nc3ccccc3s2)C1=N	nan
	1366812	23939	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	4	5.3	Cc1ccc(-c2nc3ccccc3s2)cc1NC(=O)COc1ccccc1	nan
	CHEMBL1339140	23939	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	4	5.3	Cc1ccc(-c2nc3ccccc3s2)cc1NC(=O)COc1ccccc1	nan
	1860843	24066	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	2	5	5.2	Nc1c(C(=O)Nc2ccc(Br)cc2)sc2nc(-c3ccco3)ccc12	nan
	CHEMBL1340363	24066	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	2	5	5.2	Nc1c(C(=O)Nc2ccc(Br)cc2)sc2nc(-c3ccco3)ccc12	nan
	1258323	24132	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	2	6	3.6	Nc1c(C(=O)NCCc2ccccc2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1340956	24132	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	2	6	3.6	Nc1c(C(=O)NCCc2ccccc2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	1248113	24144	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	0	7	3.3	CCOC(=O)c1cc(OC(=O)c2cccs2)n(-c2ccccc2)n1	nan
	CHEMBL1341066	24144	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	0	7	3.3	CCOC(=O)c1cc(OC(=O)c2cccs2)n(-c2ccccc2)n1	nan
	2478762	24392	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	3.3	Cc1c(C(=O)OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2c1ccc1ccccc12	nan
	CHEMBL1343023	24392	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	3.3	Cc1c(C(=O)OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2c1ccc1ccccc12	nan
	3243891	24405	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	6	2.6	Cc1ccc(CNc2nc3ccccc3n3nnnc23)cc1	nan
	CHEMBL1343134	24405	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	6	2.6	Cc1ccc(CNc2nc3ccccc3n3nnnc23)cc1	nan
	2242090	24598	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	2	5	3.5	CS(=O)(=O)c1ccc2nc(NC(=O)Nc3ccccc3F)sc2c1	nan
	CHEMBL1344848	24598	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	2	5	3.5	CS(=O)(=O)c1ccc2nc(NC(=O)Nc3ccccc3F)sc2c1	nan
	665134	24634	7	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.7	O=C1CC(c2ccc(F)cc2)Cc2nc(NCc3ccco3)ncc21	nan
	CHEMBL1345142	24634	7	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.7	O=C1CC(c2ccc(F)cc2)Cc2nc(NCc3ccco3)ncc21	nan
	1096895	24683	45	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	2	5	0.6	O=C(O)c1nn2cc(CCO)cnc2c1Cl	nan
	CHEMBL1345601	24683	45	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	2	5	0.6	O=C(O)c1nn2cc(CCO)cnc2c1Cl	nan
	3640616	24754	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	6	3.4	O=C(OC1CCOC1=O)c1cc(-c2cccs2)nc2ccccc12	nan
	CHEMBL1346240	24754	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	6	3.4	O=C(OC1CCOC1=O)c1cc(-c2cccs2)nc2ccccc12	nan
	4846975	24926	21	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1-c1ccccc1	nan
	CHEMBL1347553	24926	21	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1-c1ccccc1	nan
	5219047	24972	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	5	2	4	2.1	CCC(C)NC(=O)COC(=O)c1ccc(Cl)cc1O	nan
	CHEMBL1347937	24972	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	5	2	4	2.1	CCC(C)NC(=O)COC(=O)c1ccc(Cl)cc1O	nan
	16193959	25008	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	11	2	9	2.0	NS(=O)(=O)c1ccc(CCNC(=O)CCCn2c(SCC(=O)N3CCCC3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1348274	25008	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	11	2	9	2.0	NS(=O)(=O)c1ccc(CCNC(=O)CCCn2c(SCC(=O)N3CCCC3)nc3ccsc3c2=O)cc1	nan
	3342394	25253	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	1	5	3.3	C=CCN1C(=O)c2ccccc2Sc2ccc(C(=O)NCC(OC)OC)cc21	nan
	CHEMBL1350401	25253	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	1	5	3.3	C=CCN1C(=O)c2ccccc2Sc2ccc(C(=O)NCC(OC)OC)cc21	nan
	16011056	25754	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	6	4.1	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Br)c4)ncn32)s1	nan
	CHEMBL1354311	25754	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	6	4.1	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Br)c4)ncn32)s1	nan
	16025634	25763	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	4.1	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)cc1F	nan
	CHEMBL1354359	25763	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	4.1	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)cc1F	nan
	16009946	25797	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	1.6	CCc1cccc(CC)c1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1354862	25797	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	1.6	CCc1cccc(CC)c1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	16018892	25821	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	7	5.9	CCc1nnc(SCc2nc(-c3ccccc3F)oc2C)c2cc3sccc3n12	nan
	CHEMBL1355121	25821	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	7	5.9	CCc1nnc(SCc2nc(-c3ccccc3F)oc2C)c2cc3sccc3n12	nan
	4363763	25892	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	5	0	8	4.0	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1ccc(C(C)(C)C)cc1	nan
	CHEMBL1356044	25892	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	5	0	8	4.0	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1ccc(C(C)(C)C)cc1	nan
	16024946	25908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	4	4.1	O=C(NCc1ccccc1Cl)c1ccc2c(c1)nnn2C1CCCC1	nan
	CHEMBL1356218	25908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	4	4.1	O=C(NCc1ccccc1Cl)c1ccc2c(c1)nnn2C1CCCC1	nan
	15990261	25911	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	7	4.1	Cc1nnc2c(N3CCN(c4ccccc4)CC3)nc3ccc(C(=O)c4ccccc4)cc3n12	nan
	CHEMBL1356236	25911	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	7	4.1	Cc1nnc2c(N3CCN(c4ccccc4)CC3)nc3ccc(C(=O)c4ccccc4)cc3n12	nan
	16031511	25915	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(F)cc3)s2)cc1	nan
	CHEMBL1356303	25915	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(F)cc3)s2)cc1	nan
	16030397	25931	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	5	3.4	COCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1356573	25931	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	5	3.4	COCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16009450	25948	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	3.5	O=C(COc1ccc(F)cc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1356791	25948	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	3.5	O=C(COc1ccc(F)cc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	756766	25960	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	1	4	3.8	Cn1c(SCc2cccc(F)c2)nc2c([nH]c3ccccc32)c1=O	nan
	CHEMBL1356946	25960	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	1	4	3.8	Cn1c(SCc2cccc(F)c2)nc2c([nH]c3ccccc32)c1=O	nan
	2141078	25972	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	6	4.7	COc1ccc(CNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1	nan
	CHEMBL1357087	25972	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	6	4.7	COc1ccc(CNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1	nan
	15988374	26003	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	6	0	6	5.7	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)c1ccc(Br)cc1	nan
	CHEMBL1357521	26003	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	6	0	6	5.7	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)c1ccc(Br)cc1	nan
	16020301	26017	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(F)cc3)c2=O)cc1	nan
	CHEMBL1357758	26017	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(F)cc3)c2=O)cc1	nan
	16024673	26027	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	3.9	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)c1	nan
	CHEMBL1357949	26027	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	3.9	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)c1	nan
	16016274	26045	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	0	6	4.2	Cc1cccc(-c2noc(-c3ccc(N4CCCC4)c([N+](=O)[O-])c3)n2)c1	nan
	CHEMBL1358183	26045	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	0	6	4.2	Cc1cccc(-c2noc(-c3ccc(N4CCCC4)c([N+](=O)[O-])c3)n2)c1	nan
	20880782	26057	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	7	3.0	CC1CCCCN1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	CHEMBL1358259	26057	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	7	3.0	CC1CCCCN1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	15988865	26073	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	1	5	3.6	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1	nan
	CHEMBL1358506	26073	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	1	5	3.6	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1	nan
	16009824	26090	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	2	7	4.0	NS(=O)(=O)c1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccc(Cl)cc23)cc1	nan
	CHEMBL1358725	26090	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	2	7	4.0	NS(=O)(=O)c1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccc(Cl)cc23)cc1	nan
	1231059	26093	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.7	CC(=O)Nc1cccc(-c2nnc(-c3ccc(C)cc3)o2)c1	nan
	CHEMBL1358793	26093	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.7	CC(=O)Nc1cccc(-c2nnc(-c3ccc(C)cc3)o2)c1	nan
	1317893	26137	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.2	Cc1cc(OCC(=O)Nc2cc(-c3nc4ncccc4o3)ccc2C)ccc1Cl	nan
	CHEMBL1359048	26137	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.2	Cc1cc(OCC(=O)Nc2cc(-c3nc4ncccc4o3)ccc2C)ccc1Cl	nan
	3410425	26251	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	0	7	3.7	CCOCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OCC)ccc21	nan
	CHEMBL1360046	26251	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	0	7	3.7	CCOCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OCC)ccc21	nan
	2335932	26333	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(C)c1NC(=O)COC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1360771	26333	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(C)c1NC(=O)COC(=O)c1ccc2c(c1)OCO2	nan
	16009752	26396	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	5	4.5	CCCCNc1nc2c(-c3cccc(C)c3)nnn2c2ccccc12	nan
	CHEMBL1361402	26396	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	5	4.5	CCCCNc1nc2c(-c3cccc(C)c3)nnn2c2ccccc12	nan
	16022921	26409	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	CHEMBL1361507	26409	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	2345644	26481	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.5	COc1cccc(C(=O)Nc2nnc(-c3ccc(OC)cc3OC)s2)c1	nan
	CHEMBL1362103	26481	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.5	COc1cccc(C(=O)Nc2nnc(-c3ccc(OC)cc3OC)s2)c1	nan
	16022913	26524	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	4.3	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1362452	26524	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	4.3	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	1313404	26538	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	7	4.0	CCOc1cc(C2C(C(=O)OC)=CN(C3CCCC3)C=C2C(=O)OC)cc(Br)c1O	nan
	CHEMBL1362550	26538	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	7	4.0	CCOc1cc(C2C(C(=O)OC)=CN(C3CCCC3)C=C2C(=O)OC)cc(Br)c1O	nan
	3448294	26559	23	None	-19	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	0	3	5.0	O=Cc1cc2ccccc2nc1SCc1ccc(Cl)cc1	nan
	CHEMBL1362687	26559	23	None	-19	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	0	3	5.0	O=Cc1cc2ccccc2nc1SCc1ccc(Cl)cc1	nan
	16026537	26683	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	6	4.2	CC(=O)c1cccc(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	CHEMBL1363862	26683	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	6	4.2	CC(=O)c1cccc(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	16009886	26693	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	7	4.3	COc1cccc(-n2c(=O)c3sc4ccccc4c3n(CC(=O)Nc3ccccc3C)c2=O)c1	nan
	CHEMBL1363941	26693	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	7	4.3	COc1cccc(-n2c(=O)c3sc4ccccc4c3n(CC(=O)Nc3ccccc3C)c2=O)c1	nan
	3359750	26761	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.2	O=C(CSc1nc(-c2ccccc2)c2ccccc2n1)Nc1ccc(F)cc1	nan
	CHEMBL1364552	26761	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.2	O=C(CSc1nc(-c2ccccc2)c2ccccc2n1)Nc1ccc(F)cc1	nan
	16019445	26815	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	8	5.7	Cc1ccc(C)c(Nc2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)c1	nan
	CHEMBL1365021	26815	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	8	5.7	Cc1ccc(C)c(Nc2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)c1	nan
	1152421	27014	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	6	5.4	CCOc1ccccc1NC(=O)CSc1nc(-c2cccs2)cc(C(F)(F)F)n1	nan
	CHEMBL1366693	27014	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	6	5.4	CCOc1ccccc1NC(=O)CSc1nc(-c2cccs2)cc(C(F)(F)F)n1	nan
	1080694	27042	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	5	3.2	CC1(C)CC(=O)c2sc(NS(=O)(=O)c3ccc(F)cc3)nc2C1	nan
	CHEMBL1366962	27042	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	5	3.2	CC1(C)CC(=O)c2sc(NS(=O)(=O)c3ccc(F)cc3)nc2C1	nan
	16022984	27116	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1367585	27116	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	16015654	27269	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	6	1	5	4.7	CC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	CHEMBL1368731	27269	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	6	1	5	4.7	CC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	2918354	27563	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	5	3.7	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1cccc(Br)c1	nan
	CHEMBL1370753	27563	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	5	3.7	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1cccc(Br)c1	nan
	1005238	27599	18	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	3.5	Cc1cc(NC(=O)CSc2nc3c(c(-c4cccnc4)c2C#N)CCC3)no1	nan
	CHEMBL1371055	27599	18	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	3.5	Cc1cc(NC(=O)CSc2nc3c(c(-c4cccnc4)c2C#N)CCC3)no1	nan
	1442423	27895	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	4.0	Cc1cc(NC(=O)CSc2nc(C(C)(C)C)nc3ccccc23)no1	nan
	CHEMBL1373175	27895	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	4.0	Cc1cc(NC(=O)CSc2nc(C(C)(C)C)nc3ccccc23)no1	nan
	6615570	27951	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	4	1	7	3.7	COc1ccc(C)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	CHEMBL1373530	27951	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	4	1	7	3.7	COc1ccc(C)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	2410746	27971	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	5	3.0	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	CHEMBL1373647	27971	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	5	3.0	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	16009969	28097	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	7	1.3	CN(CC(=O)Nc1ccc(Cl)cc1F)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1374581	28097	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	7	1.3	CN(CC(=O)Nc1ccc(Cl)cc1F)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	9547710	28099	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	9	0.3	Cn1c(N)c(C(=O)COC(=O)c2ccnc3ccccc23)c(=O)n(C)c1=O	nan
	CHEMBL1374591	28099	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	9	0.3	Cn1c(N)c(C(=O)COC(=O)c2ccnc3ccccc23)c(=O)n(C)c1=O	nan
	4414022	28129	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	6	4.0	CCOC(=O)c1c(NC(=O)C(C)Oc2ccccc2F)sc(C(C)=O)c1C	nan
	CHEMBL1374782	28129	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	6	4.0	CCOC(=O)c1c(NC(=O)C(C)Oc2ccccc2F)sc(C(C)=O)c1C	nan
	679950	28192	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.9	CCN(CC)c1ccc(-c2c(C#N)c(N)nc(OC)c2C#N)cc1	nan
	CHEMBL1375207	28192	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.9	CCN(CC)c1ccc(-c2c(C#N)c(N)nc(OC)c2C#N)cc1	nan
	5297522	28203	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	2	7	4.0	CCOC(=O)c1ccc(NC(=O)c2sc3nc4c(cc3c2N)N2CCC4CC2)cc1	nan
	CHEMBL1375280	28203	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	2	7	4.0	CCOC(=O)c1ccc(NC(=O)c2sc3nc4c(cc3c2N)N2CCC4CC2)cc1	nan
	16022988	28250	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	7	2.8	CCNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(OC)cc4)nc23)CC1	nan
	CHEMBL1375625	28250	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	7	2.8	CCNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(OC)cc4)nc23)CC1	nan
	1224964	28254	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	2	3	4.2	O=C(Nc1ccc(C(=O)NC2CCCCC2)cc1)c1cncc(Br)c1	nan
	CHEMBL1375663	28254	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	2	3	4.2	O=C(Nc1ccc(C(=O)NC2CCCCC2)cc1)c1cncc(Br)c1	nan
	16009514	28337	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1	nan
	CHEMBL1376473	28337	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1	nan
	16010769	28410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	3.6	Cc1ccc(Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cccnc32)cc1	nan
	CHEMBL1377217	28410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	3.6	Cc1ccc(Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cccnc32)cc1	nan
	16024487	28464	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.2	Cc1cc(C)cc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)c1	nan
	CHEMBL1377738	28464	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.2	Cc1cc(C)cc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)c1	nan
	20887350	28756	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	7	1.3	Cc1nn(CC(=O)N2CCC3(CC2)OCCO3)c(=O)c2cc3ccccc3n12	nan
	CHEMBL1380351	28756	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	7	1.3	Cc1nn(CC(=O)N2CCC3(CC2)OCCO3)c(=O)c2cc3ccccc3n12	nan
	1943710	28915	8	None	-6	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	5.1	CCCCc1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	CHEMBL1381564	28915	8	None	-6	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	5.1	CCCCc1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	2220993	28952	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	4.5	Cc1cc(NC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)no1	nan
	CHEMBL1381905	28952	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	4.5	Cc1cc(NC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)no1	nan
	2551678	28960	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.3	Cc1[nH]c2ccccc2c1C(=O)CSc1nc2ccccc2c(=O)n1-c1ccccc1F	nan
	CHEMBL1381998	28960	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.3	Cc1[nH]c2ccccc2c1C(=O)CSc1nc2ccccc2c(=O)n1-c1ccccc1F	nan
	15997541	29230	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	2	7	3.4	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cccc(Cl)c3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1384419	29230	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	2	7	3.4	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cccc(Cl)c3)c3ccccc3c2=O)cc1OC	nan
	2412434	29303	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1ccc(NC(=O)CSc2ncnc3ccccc23)cc1	nan
	CHEMBL1385049	29303	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1ccc(NC(=O)CSc2ncnc3ccccc23)cc1	nan
	1490540	29310	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	4	3.9	COc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	CHEMBL1385084	29310	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	4	3.9	COc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	1442725	29353	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	4	3.9	CC(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1385478	29353	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	4	3.9	CC(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	660521	29432	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCCCC2	nan
	CHEMBL1386214	29432	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCCCC2	nan
	658023	29757	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	2	7	2.7	CCOc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)c(OCC)c1	nan
	CHEMBL1388744	29757	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	2	7	2.7	CCOc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)c(OCC)c1	nan
	5913531	29810	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	8	1	8	3.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1389094	29810	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	8	1	8	3.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	135749817	29955	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	2	4	4.9	N#C/C(=C(\O)c1cc(Cl)sc1Cl)c1nc2ccccc2[nH]1	nan
	CHEMBL1390333	29955	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	2	4	4.9	N#C/C(=C(\O)c1cc(Cl)sc1Cl)c1nc2ccccc2[nH]1	nan
	135468428	30133	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	5	2	7	5.1	Cc1cc(-n2c(SCC(=O)Nc3ccc(Br)cc3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1391897	30133	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	5	2	7	5.1	Cc1cc(-n2c(SCC(=O)Nc3ccc(Br)cc3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	5393174	30159	38	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	4	3.2	COc1ccc(-c2cc3ccc(O)cc3oc2=O)cc1	nan
	CHEMBL1392132	30159	38	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	4	3.2	COc1ccc(-c2cc3ccc(O)cc3oc2=O)cc1	nan
	738837	30185	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	1	2	3.9	Cc1occc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL1392331	30185	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	1	2	3.9	Cc1occc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	16194581	30253	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	9	0.9	CC(Sc1nc(-c2ccco2)nc2c1c(=O)n(C)c(=O)n2C)C(=O)O	nan
	CHEMBL1392938	30253	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	9	0.9	CC(Sc1nc(-c2ccco2)nc2c1c(=O)n(C)c(=O)n2C)C(=O)O	nan
	16029022	30476	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	2.5	COC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCC(C)CC3)cn2C)cc1	nan
	CHEMBL1395073	30476	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	2.5	COC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCC(C)CC3)cn2C)cc1	nan
	16024525	30524	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1395642	30524	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	16009355	30530	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	0	5	5.1	CC(C)c1ccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)cc1	nan
	CHEMBL1395773	30530	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	0	5	5.1	CC(C)c1ccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)cc1	nan
	16012262	30583	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(NC(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1C	nan
	CHEMBL1396597	30583	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(NC(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1C	nan
	16425494	30602	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	5522461	30602	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	CHEMBL1396834	30602	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	15988387	30606	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	2	4	2.2	COc1cccc(C(=O)NC2=NC(c3ccccc3F)CC(=O)N2)c1	nan
	CHEMBL1396902	30606	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	2	4	2.2	COc1cccc(C(=O)NC2=NC(c3ccccc3F)CC(=O)N2)c1	nan
	16030463	30626	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	CC1CCN(C(=O)CSc2nc3ccccc3nc2Cc2ccccc2)CC1	nan
	CHEMBL1397149	30626	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	CC1CCN(C(=O)CSc2nc3ccccc3nc2Cc2ccccc2)CC1	nan
	16011758	30636	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.8	COc1ccc(OC)c(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1397253	30636	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.8	COc1ccc(OC)c(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	15988254	30694	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	0	7	3.1	COc1cc(OC)cc(-n2c(=O)c3ccccc3n(Cc3ccccc3C#N)c2=O)c1	nan
	CHEMBL1398033	30694	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	0	7	3.1	COc1cc(OC)cc(-n2c(=O)c3ccccc3n(Cc3ccccc3C#N)c2=O)c1	nan
	5089883	30703	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	6	5.9	O=C(CSc1oc(-c2ccc(F)cc2)nc1S(=O)(=O)c1ccccc1)c1ccc(Cl)cc1	nan
	CHEMBL1398184	30703	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	6	5.9	O=C(CSc1oc(-c2ccc(F)cc2)nc1S(=O)(=O)c1ccccc1)c1ccc(Cl)cc1	nan
	16020303	30708	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3cccc(F)c3)c2=O)cc1	nan
	CHEMBL1398259	30708	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3cccc(F)c3)c2=O)cc1	nan
	16025636	30714	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	4	1	6	3.9	CN1c2cc(Cl)ccc2-c2nc(SCC(=O)Nc3ccc(F)cc3F)ncc2S1(=O)=O	nan
	CHEMBL1398402	30714	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	4	1	6	3.9	CN1c2cc(Cl)ccc2-c2nc(SCC(=O)Nc3ccc(F)cc3F)ncc2S1(=O)=O	nan
	16030333	30723	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	6	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2OC)cc1	nan
	CHEMBL1398464	30723	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	6	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2OC)cc1	nan
	16022444	30749	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	7	4.8	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3nc2s1	nan
	CHEMBL1398653	30749	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	7	4.8	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3nc2s1	nan
	4135187	30802	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	6	4.4	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2F)cc1	nan
	CHEMBL1399236	30802	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	6	4.4	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2F)cc1	nan
	2135591	30806	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.7	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(Cl)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1399275	30806	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.7	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(Cl)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	135546815	30813	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	5	4.0	Cc1ccc(NC(=O)C(C)Sc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)c(C)c1	nan
	CHEMBL1399310	30813	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	5	4.0	Cc1ccc(NC(=O)C(C)Sc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)c(C)c1	nan
	135513990	30860	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	5	4.4	Cc1c(Br)ccc(NC(=O)CSc2nc(O)c3ccccc3n2)c1C	nan
	CHEMBL1399762	30860	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	5	4.4	Cc1c(Br)ccc(NC(=O)CSc2nc(O)c3ccccc3n2)c1C	nan
	6484563	30936	33	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	0	2	2	3.4	SC1=NC2(CCCCC2)Nc2ccccc21	nan
	CHEMBL1400466	30936	33	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	0	2	2	3.4	SC1=NC2(CCCCC2)Nc2ccccc21	nan
	16011170	30958	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.6	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(Cl)cc1F	nan
	CHEMBL1400646	30958	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.6	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(Cl)cc1F	nan
	2404851	30984	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	1	7	1.0	O=S(=O)(c1cccc(-c2nnc(S)o2)c1)N1CCOCC1	nan
	CHEMBL1400922	30984	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	1	7	1.0	O=S(=O)(c1cccc(-c2nnc(S)o2)c1)N1CCOCC1	nan
	659778	31009	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1F	nan
	CHEMBL1401137	31009	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1F	nan
	4852309	31024	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	3	4.5	COc1cc(C(=O)NC(c2ccccc2)c2ccccc2)cc(OC)c1C	nan
	CHEMBL1401266	31024	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	3	4.5	COc1cc(C(=O)NC(c2ccccc2)c2ccccc2)cc(OC)c1C	nan
	1994854	31027	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	8	3.6	CCn1c(SCC(=O)Nc2ccc(C(C)=O)cc2)nc2nc3c(cc2c1=O)COC(C)(C)C3	nan
	CHEMBL1401292	31027	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	8	3.6	CCn1c(SCC(=O)Nc2ccc(C(C)=O)cc2)nc2nc3c(cc2c1=O)COC(C)(C)C3	nan
	16011439	31327	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	6	6.3	COc1ccc(Cn2c(SCc3ccc(C(=O)NC(C)c4ccccc4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1404015	31327	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	6	6.3	COc1ccc(Cn2c(SCc3ccc(C(=O)NC(C)c4ccccc4)cc3)nc3cccnc32)cc1	nan
	2456084	31332	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	2	8	4.0	COc1cc(NC(=O)c2ccco2)c(C(=O)OCC(=O)Nc2ncc(Cl)cc2Cl)cc1OC	nan
	CHEMBL1404053	31332	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	2	8	4.0	COc1cc(NC(=O)c2ccco2)c(C(=O)OCC(=O)Nc2ncc(Cl)cc2Cl)cc1OC	nan
	2826390	31424	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	5	2.9	COC(=O)c1sccc1NC(=O)C1CC(C)=C(C)CC1C(=O)O	nan
	CHEMBL1404933	31424	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	5	2.9	COC(=O)c1sccc1NC(=O)C1CC(C)=C(C)CC1C(=O)O	nan
	16007508	31436	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	3	5.7	CCc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1405105	31436	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	3	5.7	CCc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	1930124	31527	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nc3ccccc3nc21	nan
	CHEMBL1405964	31527	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nc3ccccc3nc21	nan
	135464462	31681	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	6	3.1	CN(C)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	CHEMBL1407344	31681	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	6	3.1	CN(C)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	3221573	31712	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	8	3	5	3.0	COCCCN=C(S)NCCNc1nc2c(C)c(C)ccc2cc1C#N	nan
	CHEMBL1407546	31712	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	8	3	5	3.0	COCCCN=C(S)NCCNc1nc2c(C)c(C)ccc2cc1C#N	nan
	266900	31726	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	3	4.3	COC(=O)c1cc(C)nc2c(C)cc3[nH]c4ccccc4c3c12	nan
	CHEMBL1407610	31726	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	3	4.3	COC(=O)c1cc(C)nc2c(C)cc3[nH]c4ccccc4c3c12	nan
	16018228	31789	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	5	1.1	CN(C)CCNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	CHEMBL1408060	31789	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	5	1.1	CN(C)CCNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	800213	31821	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	4.8	CC(C)(C)c1ccc(-c2nnc(NC(=O)c3ccccc3)s2)cc1	nan
	CHEMBL1408281	31821	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	4.8	CC(C)(C)c1ccc(-c2nnc(NC(=O)c3ccccc3)s2)cc1	nan
	4837904	31885	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.1	COc1ccc(CCNC(=O)Cc2c(C)c3cc4c(C)coc4cc3oc2=O)cc1OC	nan
	CHEMBL1408806	31885	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.1	COc1ccc(CCNC(=O)Cc2c(C)c3cc4c(C)coc4cc3oc2=O)cc1OC	nan
	915456	31888	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	4	4.6	Oc1ccccc1-c1nc(NCc2ccccc2)c2ccccc2n1	nan
	CHEMBL1408828	31888	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	4	4.6	Oc1ccccc1-c1nc(NCc2ccccc2)c2ccccc2n1	nan
	15988127	32018	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	6	3	6	7.6	COc1ccccc1NC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(C)cc3C)c(-c3ccccc3Cl)c2c1N	nan
	CHEMBL1409862	32018	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	6	3	6	7.6	COc1ccccc1NC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(C)cc3C)c(-c3ccccc3Cl)c2c1N	nan
	649505	32021	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	2.3	O=C(Nc1ccc2c(c1)OCO2)C1CCN(c2ccc(S(=O)(=O)N3CCOCC3)cc2)CC1	nan
	CHEMBL1409886	32021	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	2.3	O=C(Nc1ccc2c(c1)OCO2)C1CCN(c2ccc(S(=O)(=O)N3CCOCC3)cc2)CC1	nan
	688670	32039	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	4	3.5	COc1ccc(-c2cc(=O)c3cc(OC)ccc3o2)cc1	nan
	CHEMBL1410006	32039	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	4	3.5	COc1ccc(-c2cc(=O)c3cc(OC)ccc3o2)cc1	nan
	4137223	32147	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	5	5.2	Cc1nc(N2CCC(C)CC2)c2c(C)c(C(=O)Nc3ccc(C)c(F)c3)sc2n1	nan
	CHEMBL1410912	32147	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	5	5.2	Cc1nc(N2CCC(C)CC2)c2c(C)c(C(=O)Nc3ccc(C)c(F)c3)sc2n1	nan
	1088392	32338	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	7	3.0	COC(=O)c1sc(NC(=O)c2c(OC)cccc2OC)c(C#N)c1C	nan
	CHEMBL1412474	32338	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	7	3.0	COC(=O)c1sc(NC(=O)c2c(OC)cccc2OC)c(C#N)c1C	nan
	790792	32496	36	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	3	3.4	CCc1c(C)nc2ccc(OC)cc2c1S	nan
	CHEMBL1413735	32496	36	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	3	3.4	CCc1c(C)nc2ccc(OC)cc2c1S	nan
	16015840	32529	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	4	5.0	Cc1cccc(-c2nc3cc(NC(=O)COc4ccccc4F)ccc3o2)c1	nan
	CHEMBL1413987	32529	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	4	5.0	Cc1cccc(-c2nc3cc(NC(=O)COc4ccccc4F)ccc3o2)c1	nan
	655034	32625	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	2	7	2.4	COc1cc(CC(NC(C)=O)C(=O)NC2CCN(c3nc(C)cc(C)c3C#N)CC2)cc(OC)c1	nan
	CHEMBL1414774	32625	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	2	7	2.4	COc1cc(CC(NC(C)=O)C(=O)NC2CCN(c3nc(C)cc(C)c3C#N)CC2)cc(OC)c1	nan
	16016268	32627	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	0	8	5.0	COc1ccccc1N1CCN(c2ccc(-c3nc(-c4ccccc4C)no3)cc2[N+](=O)[O-])CC1	nan
	CHEMBL1414801	32627	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	0	8	5.0	COc1ccccc1N1CCN(c2ccc(-c3nc(-c4ccccc4C)no3)cc2[N+](=O)[O-])CC1	nan
	2156145	32724	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	9	4.3	COc1ccc(-n2c(SCC(=O)Nc3cc(C)on3)nc3c4ccccc4nc-3c2O)cc1	nan
	CHEMBL1415709	32724	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	9	4.3	COc1ccc(-n2c(SCC(=O)Nc3cc(C)on3)nc3c4ccccc4nc-3c2O)cc1	nan
	7190669	32785	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1	nan
	CHEMBL1416264	32785	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1	nan
	16012962	32800	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	0	6	3.9	Fc1cccc(-n2ncc3c2ncn2nc(-c4ccccc4Cl)nc32)c1	nan
	CHEMBL1416375	32800	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	0	6	3.9	Fc1cccc(-n2ncc3c2ncn2nc(-c4ccccc4Cl)nc32)c1	nan
	4808145	32957	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	7	1.3	Cn1c(=O)c2c(ncn2CCOc2ccc(Br)cc2)n(C)c1=O	nan
	CHEMBL1417778	32957	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	7	1.3	Cn1c(=O)c2c(ncn2CCOc2ccc(Br)cc2)n(C)c1=O	nan
	16009664	33036	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1418446	33036	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	4625060	33107	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	4	2.2	O=C(CC1N=C2c3ccccc3NC(=S)N2C1=O)NC1CCCCC1	nan
	CHEMBL1419028	33107	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	4	2.2	O=C(CC1N=C2c3ccccc3NC(=S)N2C1=O)NC1CCCCC1	nan
	665236	33153	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	4.4	CCc1nc(SCC(=O)Nc2ccc3c(c2)OCCO3)c2oc3ccccc3c2n1	nan
	CHEMBL1419387	33153	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	4.4	CCc1nc(SCC(=O)Nc2ccc3c(c2)OCCO3)c2oc3ccccc3c2n1	nan
	20927027	33170	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	2.0	O=S(=O)(c1ccc(-c2ccc(O)nn2)o1)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1419593	33170	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	2.0	O=S(=O)(c1ccc(-c2ccc(O)nn2)o1)N1CCN(c2ccccc2)CC1	nan
	16024782	33329	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4F)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1420848	33329	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4F)CC3)ccc2c1)N1CCCCC1	nan
	3185701	33352	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	541	10	3	8	3.0	CCOc1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2F)cc1	nan
	CHEMBL1421091	33352	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	541	10	3	8	3.0	CCOc1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2F)cc1	nan
	1078539	33603	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	7	2.5	Cc1cccc(-n2ncc3c(N4CCC5(CC4)OCCO5)ncnc32)c1	nan
	CHEMBL1423202	33603	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	7	2.5	Cc1cccc(-n2ncc3c(N4CCC5(CC4)OCCO5)ncnc32)c1	nan
	993322	33642	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	4.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)Nc3cc(C)on3)n2)cc1	nan
	CHEMBL1423477	33642	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	4.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)Nc3cc(C)on3)n2)cc1	nan
	16194711	33852	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	9	1.5	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(CCNC(=O)c4ccccc4)n3n2)CC1	nan
	CHEMBL1425185	33852	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	9	1.5	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(CCNC(=O)c4ccccc4)n3n2)CC1	nan
	661193	34035	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	5	1	7	1.9	Cc1cccc(-n2ncc3c(NCCN4CCOCC4)ncnc32)c1	nan
	CHEMBL1426726	34035	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	5	1	7	1.9	Cc1cccc(-n2ncc3c(NCCN4CCOCC4)ncnc32)c1	nan
	2999700	34180	3	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	5	4.6	Cn1c(/C(C#N)=C(\O)COc2ccc3ccccc3c2)nc2ccccc21	nan
	CHEMBL1428087	34180	3	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	5	4.6	Cn1c(/C(C#N)=C(\O)COc2ccc3ccccc3c2)nc2ccccc21	nan
	1371384	34303	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	1	4	2.7	Cc1ccc(/C=C2/SC(=O)NC2=S)o1	nan
	CHEMBL1429158	34303	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	1	4	2.7	Cc1ccc(/C=C2/SC(=O)NC2=S)o1	nan
	2815019	34599	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	8	0.7	Cn1c(=O)c2c(nc(Sc3ccccc3N)n2C)n(C)c1=O	nan
	CHEMBL1431497	34599	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	8	0.7	Cn1c(=O)c2c(nc(Sc3ccccc3N)n2C)n(C)c1=O	nan
	2114663	34642	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	5	5.3	Cc1onc(-c2ccccc2)c1C(=O)Nc1nc(-c2cc(F)ccc2F)cs1	nan
	CHEMBL1431887	34642	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	5	5.3	Cc1onc(-c2ccccc2)c1C(=O)Nc1nc(-c2cc(F)ccc2F)cs1	nan
	650995	34745	13	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	6	4.2	Cc1nonc1NC(=O)CSc1nc2cc(Cl)ccc2c2c1CCCC2	nan
	CHEMBL1432773	34745	13	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	6	4.2	Cc1nonc1NC(=O)CSc1nc2cc(Cl)ccc2c2c1CCCC2	nan
	15989049	34833	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	529	8	1	8	3.9	O=C(CCCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1433448	34833	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	529	8	1	8	3.9	O=C(CCCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	16009658	34847	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1cccc(F)c1	nan
	CHEMBL1433649	34847	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1cccc(F)c1	nan
	16030989	34853	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	4.3	COC(=O)c1c(-c2ccc(Cl)cc2)noc1N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1433722	34853	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	4.3	COC(=O)c1c(-c2ccc(Cl)cc2)noc1N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	15990910	34866	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	4	5.8	CSc1cccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	CHEMBL1433922	34866	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	4	5.8	CSc1cccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	16008787	34907	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.3	COc1ccccc1CNC(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1	nan
	CHEMBL1434647	34907	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.3	COc1ccccc1CNC(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1	nan
	16022785	34908	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)c(C)c1	nan
	CHEMBL1434648	34908	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)c(C)c1	nan
	24819144	34913	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	6	6.0	COC(=O)c1ccc(/C=C/c2c(-c3ccsc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	CHEMBL1434681	34913	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	6	6.0	COC(=O)c1ccc(/C=C/c2c(-c3ccsc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	135546816	34919	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	2	6	3.8	CCOc1ccccc1NC(=O)C(C)Sc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1	nan
	CHEMBL1434743	34919	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	2	6	3.8	CCOc1ccccc1NC(=O)C(C)Sc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1	nan
	16024519	34937	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	7	3.7	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1435013	34937	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	7	3.7	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3nc(C)ccc3c2=O)cc1	nan
	16018510	34941	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	5.3	COc1cccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)c1	nan
	CHEMBL1435044	34941	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	5.3	COc1cccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)c1	nan
	15988487	34951	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	4	4.3	CC1(C)CC(=O)c2cc(-c3nc(-c4ccccc4)cs3)c(=O)[nH]c2C1	nan
	CHEMBL1435109	34951	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	4	4.3	CC1(C)CC(=O)c2cc(-c3nc(-c4ccccc4)cs3)c(=O)[nH]c2C1	nan
	6225711	35016	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	4	3.6	Cc1cc(O)c2c(C)c(CC(=O)NCc3ccccc3Cl)c(=O)oc2c1	nan
	CHEMBL1435970	35016	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	4	3.6	Cc1cc(O)c2c(C)c(CC(=O)NCc3ccccc3Cl)c(=O)oc2c1	nan
	15987771	35020	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	0	5	3.5	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)c21	nan
	CHEMBL1436008	35020	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	0	5	3.5	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)c21	nan
	5059361	35039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	6	4.7	Cc1cccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)c1	nan
	CHEMBL1436184	35039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	6	4.7	Cc1cccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)c1	nan
	4230972	35110	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	9	2	7	4.8	CC(C)c1ccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccco4)C(=O)N23)cc1	nan
	CHEMBL1437178	35110	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	9	2	7	4.8	CC(C)c1ccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccco4)C(=O)N23)cc1	nan
	16007712	35111	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.5	CCN(CC)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)N1CCN(c3cc(Cl)ccc3C)CC1)cn2C	nan
	CHEMBL1437207	35111	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.5	CCN(CC)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)N1CCN(c3cc(Cl)ccc3C)CC1)cn2C	nan
	15988469	35191	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	4.8	COc1ccc(NC(=O)C2CCN(c3ccc(Sc4ccc(C)cc4)nn3)CC2)cc1	nan
	CHEMBL1438027	35191	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	4.8	COc1ccc(NC(=O)C2CCN(c3ccc(Sc4ccc(C)cc4)nn3)CC2)cc1	nan
	3230795	35205	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	0	6	4.6	CN(C(=O)CSC1=NC2C(N=N1)c1cc(Br)ccc1N2C)C1CCCCC1	nan
	CHEMBL1438136	35205	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	0	6	4.6	CN(C(=O)CSC1=NC2C(N=N1)c1cc(Br)ccc1N2C)C1CCCCC1	nan
	16017737	35416	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	1.9	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccc(F)cc1	nan
	CHEMBL1440044	35416	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	1.9	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccc(F)cc1	nan
	16024943	35461	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	4.0	CC(=O)c1ccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)cc1	nan
	CHEMBL1440442	35461	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	4.0	CC(=O)c1ccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)cc1	nan
	16195917	35534	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	8	0.2	Cn1c(N)c(C(=O)COC(=O)CC2CC3CCC2C3)c(=O)n(C)c1=O	nan
	CHEMBL1441131	35534	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	8	0.2	Cn1c(N)c(C(=O)COC(=O)CC2CC3CCC2C3)c(=O)n(C)c1=O	nan
	16009208	35629	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	3.2	CCOc1ccc(CNC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c32)cc1	nan
	CHEMBL1441997	35629	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	3.2	CCOc1ccc(CNC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c32)cc1	nan
	2980137	35841	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	7	2.7	COc1ccc(-n2c(SC(C)C(=O)N3CCOCC3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1443960	35841	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	7	2.7	COc1ccc(-n2c(SC(C)C(=O)N3CCOCC3)nc3ccccc3c2=O)cc1	nan
	2421482	35908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	9	3.0	CCOC(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	CHEMBL1444560	35908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	9	3.0	CCOC(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	2136705	35953	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	7	3.8	COc1cc2c(=O)c(S(=O)(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2cc1OC	nan
	CHEMBL1444994	35953	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	7	3.8	COc1cc2c(=O)c(S(=O)(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2cc1OC	nan
	4154281	35975	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	5	5.3	O=C(CSc1ncnc2c1sc1ccccc12)Nc1ccc(Br)cc1	nan
	CHEMBL1445182	35975	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	5	5.3	O=C(CSc1ncnc2c1sc1ccccc12)Nc1ccc(Br)cc1	nan
	738863	36002	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	3.6	O=C(Nc1nc(=O)c2ccccc2s1)c1ccc(Cl)cc1	nan
	CHEMBL1445436	36002	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	3.6	O=C(Nc1nc(=O)c2ccccc2s1)c1ccc(Cl)cc1	nan
	3151463	36362	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	7	1.8	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1448581	36362	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	7	1.8	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc21	nan
	20903711	36434	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	7	1.1	COCCNC(=O)CCc1nnc2ccc(N3CCC(C)CC3)nn12	nan
	CHEMBL1449064	36434	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	7	1.1	COCCNC(=O)CCc1nnc2ccc(N3CCC(C)CC3)nn12	nan
	9550466	36446	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.5	Cc1ccc(-n2nc(C)c3c(C)c(CCC(=O)NC(C)c4ccccc4)c(C)nc32)cc1	nan
	CHEMBL1449158	36446	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.5	Cc1ccc(-n2nc(C)c3c(C)c(CCC(=O)NC(C)c4ccccc4)c(C)nc32)cc1	nan
	1440341	36452	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	3	4.8	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1ccccc1)CCC3	nan
	CHEMBL1449215	36452	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	3	4.8	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1ccccc1)CCC3	nan
	1034641	36569	10	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	5	3.8	Cc1ccc(-n2c(N)c(C#N)c(-c3ccc(Cl)cc3)c(C#N)c2=O)cc1	nan
	CHEMBL1450150	36569	10	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	5	3.8	Cc1ccc(-n2c(N)c(C#N)c(-c3ccc(Cl)cc3)c(C#N)c2=O)cc1	nan
	16009195	36589	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	3.5	CCN(Cc1ccccc1)C(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c21	nan
	CHEMBL1450283	36589	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	3.5	CCN(Cc1ccccc1)C(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c21	nan
	1341628	36651	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	4	5.8	CC(=O)c1ccc(NC(=O)c2cn(-c3ccccc3)nc2-c2ccc(Br)cc2)cc1	nan
	CHEMBL1450882	36651	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	4	5.8	CC(=O)c1ccc(NC(=O)c2cn(-c3ccccc3)nc2-c2ccc(Br)cc2)cc1	nan
	16019140	37063	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	8	3.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)c3oc4ccccc4c32)c1	nan
	CHEMBL1454100	37063	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	8	3.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)c3oc4ccccc4c32)c1	nan
	16009221	37107	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	4.6	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1454484	37107	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	4.6	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	16026522	37135	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	5	4.3	CCOC(=O)c1sc2cccc(F)c2c1S(=O)(=O)NCc1ccccc1Cl	nan
	CHEMBL1454707	37135	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	5	4.3	CCOC(=O)c1sc2cccc(F)c2c1S(=O)(=O)NCc1ccccc1Cl	nan
	6011252	37177	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	12	1	8	4.5	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCN2CCOCC2)cc1OC	nan
	CHEMBL1455062	37177	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	12	1	8	4.5	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCN2CCOCC2)cc1OC	nan
	16026066	37193	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.7	CCc1ccccc1NC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	CHEMBL1455235	37193	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.7	CCc1ccccc1NC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	24819160	37302	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	6	5.9	COC(=O)c1ccc(/C=C/c2c(-c3ccc(OC)cc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	CHEMBL1456226	37302	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	6	5.9	COC(=O)c1ccc(/C=C/c2c(-c3ccc(OC)cc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	135520065	37497	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	2.5	COC(=O)C(CC(C)C)NC(=O)CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1457936	37497	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	2.5	COC(=O)C(CC(C)C)NC(=O)CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	2125831	37544	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	2	2	3.9	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)cc2F)c1C	nan
	CHEMBL1458351	37544	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	2	2	3.9	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)cc2F)c1C	nan
	1110886	37814	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	3	5	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccc(NC(C)=O)cc3)nc(-c3ccc(NC(C)=O)cc3)n2)cc1	nan
	CHEMBL1460618	37814	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	3	5	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccc(NC(C)=O)cc3)nc(-c3ccc(NC(C)=O)cc3)n2)cc1	nan
	17255621	37869	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	6	3.7	CCOc1ccc(NC(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	CHEMBL1461095	37869	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	6	3.7	CCOc1ccc(NC(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	4437250	37872	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	2	2	4.2	CCN=C(S)N(CCc1c(C)[nH]c2ccccc12)Cc1cccnc1	nan
	CHEMBL1461107	37872	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	2	2	4.2	CCN=C(S)N(CCc1c(C)[nH]c2ccccc12)Cc1cccnc1	nan
	2784799	37998	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	1	1	4	2.5	O=C1C([N+](=O)[O-])=C(O)c2cccc3cccc1c23	nan
	CHEMBL1462267	37998	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	1	1	4	2.5	O=C1C([N+](=O)[O-])=C(O)c2cccc3cccc1c23	nan
	1442463	38163	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	5	4.0	CC(C)(C)c1nc(SCC(=O)N2CC(=O)Nc3ccccc32)c2ccccc2n1	nan
	CHEMBL1463696	38163	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	5	4.0	CC(C)(C)c1nc(SCC(=O)N2CC(=O)Nc3ccccc32)c2ccccc2n1	nan
	664194	38191	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	0	7	2.7	c1ccc(-n2ncc3c2ncn2nc(-c4ccco4)nc32)cc1	nan
	CHEMBL1463869	38191	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	0	7	2.7	c1ccc(-n2ncc3c2ncn2nc(-c4ccco4)nc32)cc1	nan
	2370579	38256	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	8	-0.4	Cn1c(N)c(C(=O)COC(=O)C2CCCC2)c(=O)n(C)c1=O	nan
	CHEMBL1464368	38256	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	8	-0.4	Cn1c(N)c(C(=O)COC(=O)C2CCCC2)c(=O)n(C)c1=O	nan
	4230513	38298	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	9	0.6	CC(C)Cn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1464655	38298	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	9	0.6	CC(C)Cn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1214727	38434	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	5	4.2	Cc1c(-c2ccc(Cl)cc2)oc(=O)c2c(N)n(-c3ccccc3)nc12	nan
	CHEMBL1465659	38434	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	5	4.2	Cc1c(-c2ccc(Cl)cc2)oc(=O)c2c(N)n(-c3ccccc3)nc12	nan
	4225516	38539	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	5	3.5	O=C(O)c1cccnc1SCc1cn2cc(Br)ccc2n1	nan
	CHEMBL1466534	38539	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	5	3.5	O=C(O)c1cccnc1SCc1cn2cc(Br)ccc2n1	nan
	16020097	38650	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	9	1	7	3.3	CCCCN(C)CCNC(=O)c1nn(-c2ccc(OC)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1467366	38650	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	9	1	7	3.3	CCCCN(C)CCNC(=O)c1nn(-c2ccc(OC)cc2)c(=O)c2c1c1ccccc1n2C	nan
	3137696	38666	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	0	7	-0.2	COCCn1c(Br)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1467508	38666	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	0	7	-0.2	COCCn1c(Br)nc2c1c(=O)n(C)c(=O)n2C	nan
	2396532	38765	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	2	9	-0.1	CC(=O)c1c(C)[nH]c(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	CHEMBL1468416	38765	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	2	9	-0.1	CC(=O)c1c(C)[nH]c(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	4994172	38890	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	2	5	4.0	Nc1cc(C(=O)Nc2ccc(Cl)cc2)ccc1N1CC2CC(C1)c1cccc(=O)n1C2	nan
	CHEMBL1469442	38890	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	2	5	4.0	Nc1cc(C(=O)Nc2ccc(Cl)cc2)ccc1N1CC2CC(C1)c1cccc(=O)n1C2	nan
	2517516	39042	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	2.7	CC(C)COc1ccc(C(=O)N2C(=O)c3ccc(N)cc3C2=O)cc1	nan
	CHEMBL1470757	39042	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	2.7	CC(C)COc1ccc(C(=O)N2C(=O)c3ccc(N)cc3C2=O)cc1	nan
	4968659	39171	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	9	2	6	6.1	CCc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	CHEMBL1471857	39171	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	9	2	6	6.1	CCc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	16032187	39281	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	8	2.7	Cc1cc(NC(=O)CSc2ncc(C(=O)Nc3ccc(Cl)cc3)c(=O)n2C)no1	nan
	CHEMBL1472946	39281	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	8	2.7	Cc1cc(NC(=O)CSc2ncc(C(=O)Nc3ccc(Cl)cc3)c(=O)n2C)no1	nan
	16416626	39323	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	7205030	39323	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	CHEMBL1473511	39323	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	16022561	39325	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	CHEMBL1473551	39325	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	16025981	39361	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	5	4.3	O=c1cc2nc(-c3ccccc3F)nc(SCc3ccc(Br)cc3)n2[nH]1	nan
	CHEMBL1474099	39361	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	5	4.3	O=c1cc2nc(-c3ccccc3F)nc(SCc3ccc(Br)cc3)n2[nH]1	nan
	5302625	39392	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	2	5	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	CHEMBL1474507	39392	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	2	5	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	20893081	39430	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	8	2.1	COc1ccc(NC(=O)C2CCCN2c2nn3c(=O)cc(C)nc3s2)cc1	nan
	CHEMBL1475089	39430	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	8	2.1	COc1ccc(NC(=O)C2CCCN2c2nn3c(=O)cc(C)nc3s2)cc1	nan
	15988958	39448	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(CNC(=O)CCCCCn2c(=O)c3sccc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	CHEMBL1475354	39448	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(CNC(=O)CCCCCn2c(=O)c3sccc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	16020297	39469	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	557	7	1	6	5.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3ccc(F)cc3Cl)c2=O)cc1	nan
	CHEMBL1475582	39469	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	557	7	1	6	5.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3ccc(F)cc3Cl)c2=O)cc1	nan
	16015655	39522	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.6	COc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)N3CCCc4ccccc43)sc2c1	nan
	CHEMBL1476387	39522	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.6	COc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)N3CCCc4ccccc43)sc2c1	nan
	15988828	39554	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	4.0	O=C(Nc1cccc(Cl)c1)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	CHEMBL1476787	39554	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	4.0	O=C(Nc1cccc(Cl)c1)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	15988909	39594	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	0	7	3.4	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)c1	nan
	CHEMBL1477251	39594	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	0	7	3.4	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)c1	nan
	16027484	39610	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1cccc(F)c1	nan
	CHEMBL1477385	39610	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1cccc(F)c1	nan
	16009837	39618	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	7	4.7	COc1cccc(NC(=O)Cn2c(=O)n(-c3ccc(Cl)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1477435	39618	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	7	4.7	COc1cccc(NC(=O)Cn2c(=O)n(-c3ccc(Cl)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	663717	39673	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	7	4.0	CCOCCCn1cnc2c(c1=O)c1nc3ccccc3nc1n2-c1ccc(C)cc1	nan
	CHEMBL1477914	39673	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	7	4.0	CCOCCCn1cnc2c(c1=O)c1nc3ccccc3nc1n2-c1ccc(C)cc1	nan
	16018985	39688	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1478117	39688	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	15988423	39768	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	4	2.8	COc1ccccc1NC(=O)c1cc2c([nH]c1=O)CC(C)(C)CC2=O	nan
	CHEMBL1478841	39768	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	4	2.8	COc1ccccc1NC(=O)c1cc2c([nH]c1=O)CC(C)(C)CC2=O	nan
	24819115	39819	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	5	6	2.9	Nc1c(Cl)cc(-c2nc3cc(C(=O)NCCO)ccc3c(O)c2O)cc1Cl	nan
	CHEMBL1479302	39819	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	5	6	2.9	Nc1c(Cl)cc(-c2nc3cc(C(=O)NCCO)ccc3c(O)c2O)cc1Cl	nan
	2511800	39843	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	2	5	4.0	CCOc1ncccc1C(=O)Nc1ccc(C(=O)Nc2ccc(OC)cc2)cc1	nan
	CHEMBL1479469	39843	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	2	5	4.0	CCOc1ncccc1C(=O)Nc1ccc(C(=O)Nc2ccc(OC)cc2)cc1	nan
	3352626	39986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	11	1	6	5.3	CCCC[S+]([O-])CC(O)CSc1nc(-c2ccc(OC)cc2)cc(-c2ccccc2)c1C#N	nan
	CHEMBL1480619	39986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	11	1	6	5.3	CCCC[S+]([O-])CC(O)CSc1nc(-c2ccc(OC)cc2)cc(-c2ccccc2)c1C#N	nan
	20957489	40131	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)n2n1	nan
	CHEMBL1481894	40131	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)n2n1	nan
	16033868	40136	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	2	9	4.0	COc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	CHEMBL1481939	40136	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	2	9	4.0	COc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	5297519	40186	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(C(F)(F)F)cc1)C1CCN2CC1	nan
	CHEMBL1482409	40186	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(C(F)(F)F)cc1)C1CCN2CC1	nan
	16030774	40248	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	1.2	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1482929	40248	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	1.2	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	16017755	40327	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	5	2.0	O=C(Cn1ccn(-c2cccc(Cl)c2)c(=O)c1=O)NCCc1ccccc1	nan
	CHEMBL1483603	40327	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	5	2.0	O=C(Cn1ccn(-c2cccc(Cl)c2)c(=O)c1=O)NCCc1ccccc1	nan
	16015423	40341	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccccc3F)cc2s1	nan
	CHEMBL1483703	40341	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccccc3F)cc2s1	nan
	1477383	40621	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	3	3	2.7	O=C(NC(=S)Nc1cccc2[nH]ncc12)c1ccccc1	nan
	CHEMBL1486203	40621	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	3	3	2.7	O=C(NC(=S)Nc1cccc2[nH]ncc12)c1ccccc1	nan
	16009820	40654	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	4.5	CC(C)Nc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1486479	40654	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	4.5	CC(C)Nc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	646986	40739	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	5	3.5	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccnc1)c1ccco1	nan
	CHEMBL1487207	40739	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	5	3.5	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccnc1)c1ccco1	nan
	15996976	40838	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	2	4	3.0	CC1CCN(S(=O)(=O)c2ccc3[nH]cc(C(=O)NCc4ccc(F)cc4)c(=O)c3c2)CC1	nan
	CHEMBL1487954	40838	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	2	4	3.0	CC1CCN(S(=O)(=O)c2ccc3[nH]cc(C(=O)NCc4ccc(F)cc4)c(=O)c3c2)CC1	nan
	24260	40997	82	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	3	3	2.4	Nc1ccc(-c2nc3cc(N)ccc3[nH]2)cc1	nan
	CHEMBL1489074	40997	82	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	3	3	2.4	Nc1ccc(-c2nc3cc(N)ccc3[nH]2)cc1	nan
	3144653	41004	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	5	3.8	CCCNC(=O)CSc1nc(-c2ccc(OC)cc2)cc(C(F)(F)F)n1	nan
	CHEMBL1489101	41004	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	5	3.8	CCCNC(=O)CSc1nc(-c2ccc(OC)cc2)cc(C(F)(F)F)n1	nan
	5079958	41005	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	3	4.6	CCc1ccc(Sc2cc(C(=O)O)c3ccccc3n2)cc1	nan
	CHEMBL1489124	41005	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	3	4.6	CCc1ccc(Sc2cc(C(=O)O)c3ccccc3n2)cc1	nan
	16001343	41047	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	1	7	3.3	COc1cc(NC(=O)CSc2cc(=O)n(C)c3ccccc23)cc(OC)c1OC	nan
	CHEMBL1489463	41047	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	1	7	3.3	COc1cc(NC(=O)CSc2cc(=O)n(C)c3ccccc23)cc(OC)c1OC	nan
	1327191	41074	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	2	6	4.8	COc1ccc(OC)c(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	CHEMBL1489694	41074	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	2	6	4.8	COc1ccc(OC)c(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	3151460	41095	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.2	COCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1489888	41095	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.2	COCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	4282213	41159	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	CHEMBL1490341	41159	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	28358990	41366	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	5451590	41366	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	CHEMBL1491733	41366	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	16025965	41445	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	10	1.4	CCOC(=O)c1cccc(NC(=O)c2cnc3sc(N4CCOCC4)nn3c2=O)c1	nan
	CHEMBL1492345	41445	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	10	1.4	CCOC(=O)c1cccc(NC(=O)c2cnc3sc(N4CCOCC4)nn3c2=O)c1	nan
	6157069	41511	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1OC	nan
	CHEMBL1492815	41511	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1OC	nan
	12005902	41547	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	10	4.1	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4nc5ccccc5s4)nn23)cc1OC	nan
	CHEMBL1493244	41547	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	10	4.1	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4nc5ccccc5s4)nn23)cc1OC	nan
	16022789	41558	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)cc1C	nan
	CHEMBL1493335	41558	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)cc1C	nan
	2096572	41623	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.0	COc1ccc2c(C)cc(SCC(=O)Nc3ncc(Cl)cc3Cl)nc2c1	nan
	CHEMBL1493965	41623	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.0	COc1ccc2c(C)cc(SCC(=O)Nc3ncc(Cl)cc3Cl)nc2c1	nan
	16026311	41770	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(F)cc4C)c32)cc1	nan
	CHEMBL1495516	41770	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(F)cc4C)c32)cc1	nan
	4258482	41894	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	0	5	5.6	Cc1cccc(Cc2c(C)nc3nc(SCc4ccccc4Cl)nn3c2C)c1	nan
	CHEMBL1496672	41894	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	0	5	5.6	Cc1cccc(Cc2c(C)nc3nc(SCc4ccccc4Cl)nn3c2C)c1	nan
	17583888	41930	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	1	5	3.5	CCCc1cc(=O)oc2c(C)c(OCC(=O)Nc3ccccn3)ccc12	nan
	CHEMBL1496919	41930	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	1	5	3.5	CCCc1cc(=O)oc2c(C)c(OCC(=O)Nc3ccccn3)ccc12	nan
	3260315	42000	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	9	0.6	Cc1ccc(Cl)cc1NC(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1497548	42000	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	9	0.6	Cc1ccc(Cl)cc1NC(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1488204	42290	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	4	0	5	5.3	O=S(=O)(c1ccccc1)c1cnc(-c2cccnc2)nc1-c1ccc(Cl)c(Cl)c1	nan
	CHEMBL1500120	42290	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	4	0	5	5.3	O=S(=O)(c1ccccc1)c1cnc(-c2cccnc2)nc1-c1ccc(Cl)c(Cl)c1	nan
	5309910	42820	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	2	7	2.2	CCOc1ccc(Cn2nnc(C(=O)NCc3ccc(OC)cc3)c2N)cc1	nan
	CHEMBL1504868	42820	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	2	7	2.2	CCOc1ccc(Cn2nnc(C(=O)NCc3ccc(OC)cc3)c2N)cc1	nan
	135422740	42868	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	5	1	7	4.8	Nc1c2cnnc-2nc(SCC(=O)c2ccc(Br)cc2)n1-c1ccc(Br)cc1	nan
	CHEMBL1505277	42868	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	5	1	7	4.8	Nc1c2cnnc-2nc(SCC(=O)c2ccc(Br)cc2)n1-c1ccc(Br)cc1	nan
	4975174	43418	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	1.2	COCCCn1c(C(=O)N2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1510079	43418	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	1.2	COCCCn1c(C(=O)N2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	6236457	43442	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	10	4.0	COc1cc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)cc(OC)c1OC	nan
	CHEMBL1510318	43442	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	10	4.0	COc1cc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)cc(OC)c1OC	nan
	135399378	43470	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	7	2.5	CCOc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	CHEMBL1510511	43470	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	7	2.5	CCOc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	16026527	43648	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.7	COc1ccc(CNC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)cc1	nan
	CHEMBL1512255	43648	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.7	COc1ccc(CNC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)cc1	nan
	16012611	43667	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	4.8	Cc1nc2c(c(C)nn2C(C)(C)C)c(C)c1CCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1512506	43667	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	4.8	Cc1nc2c(c(C)nn2C(C)(C)C)c(C)c1CCC(=O)Nc1ccc(F)cc1	nan
	4405319	43698	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccc5ccccc45)nc3c2)cc1	nan
	CHEMBL1512869	43698	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccc5ccccc45)nc3c2)cc1	nan
	16024551	43725	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	7	4.4	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1513333	43725	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	7	4.4	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	135416471	43732	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	Cc1ccc(-c2nc3c4ccccc4[nH]c(=O)n3n2)cc1	nan
	CHEMBL1513443	43732	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	Cc1ccc(-c2nc3c4ccccc4[nH]c(=O)n3n2)cc1	nan
	1306158	43754	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	5	5.2	COc1cc(OC)cc(C(=O)Nc2ccccc2-c2nc3ccccc3s2)c1	nan
	CHEMBL1513732	43754	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	5	5.2	COc1cc(OC)cc(C(=O)Nc2ccccc2-c2nc3ccccc3s2)c1	nan
	1887235	43790	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	5	4.8	COc1ccc(NC(=O)CCn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)cc1	nan
	CHEMBL1514436	43790	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	5	4.8	COc1ccc(NC(=O)CCn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)cc1	nan
	2158481	43802	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	2	1	5	4.1	Cc1cccc(NC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)c1C	nan
	CHEMBL1514582	43802	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	2	1	5	4.1	Cc1cccc(NC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)c1C	nan
	2134751	43803	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	10	1	8	4.5	O=C(CCCCCn1c(=O)c2sccc2n(Cc2ccccc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1514595	43803	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	10	1	8	4.5	O=C(CCCCCn1c(=O)c2sccc2n(Cc2ccccc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	7990486	43806	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	6	2.5	COc1cccc(CNC(=O)COC(=O)/C(C#N)=C/c2ccc(N(C)C)cc2)c1	nan
	CHEMBL1514625	43806	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	6	2.5	COc1cccc(CNC(=O)COC(=O)/C(C#N)=C/c2ccc(N(C)C)cc2)c1	nan
	16016989	43819	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.1	Cc1ccc(CNC(=O)C(C)n2nc(C)c3sc4ccccc4c3c2=O)cc1	nan
	CHEMBL1514781	43819	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.1	Cc1ccc(CNC(=O)C(C)n2nc(C)c3sc4ccccc4c3c2=O)cc1	nan
	4246910	43826	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	0	10	0.0	CCOCCn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1514858	43826	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	0	10	0.0	CCOCCn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	16030776	43830	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	10	1.9	Cc1cc(NC(=O)CSc2nc(-c3ccccc3F)nc3c2c(=O)n(C)c(=O)n3C)no1	nan
	CHEMBL1514941	43830	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	10	1.9	Cc1cc(NC(=O)CSc2nc(-c3ccccc3F)nc3c2c(=O)n(C)c(=O)n3C)no1	nan
	16022121	43853	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	4	0	7	2.9	COc1ccc2c(c1)c1c(c(=O)n(-c3cccc(Cl)c3)c(=O)n1CC(=O)N1CCCC1)n2C	nan
	CHEMBL1515298	43853	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	4	0	7	2.9	COc1ccc2c(c1)c1c(c(=O)n(-c3cccc(Cl)c3)c(=O)n1CC(=O)N1CCCC1)n2C	nan
	6418314	43859	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.4	CCC(Sc1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)n1)C(=O)NC1CCCC1	nan
	CHEMBL1515335	43859	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.4	CCC(Sc1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)n1)C(=O)NC1CCCC1	nan
	16031608	43868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)CC2)c(OC)c1	nan
	CHEMBL1515521	43868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)CC2)c(OC)c1	nan
	16014254	43875	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	2	6	3.2	NS(=O)(=O)c1ccc(CCNC(=O)c2nc(SCc3ccccc3F)ncc2Cl)cc1	nan
	CHEMBL1515689	43875	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	2	6	3.2	NS(=O)(=O)c1ccc(CCNC(=O)c2nc(SCc3ccccc3F)ncc2Cl)cc1	nan
	16009753	43886	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	1	0	5	3.8	Cn1c(=O)n(-c2ccc(Br)cc2F)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1515791	43886	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	1	0	5	3.8	Cn1c(=O)n(-c2ccc(Br)cc2F)c(=O)c2sc3ccccc3c21	nan
	16029066	43898	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.0	CC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCCCCC3)cn2C)cc1	nan
	CHEMBL1515983	43898	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.0	CC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCCCCC3)cn2C)cc1	nan
	16027656	43905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	9	4.0	CC(C)Cc1nn2c(=O)cc(COC(=O)c3cccc(NC(=O)c4cccs4)c3)nc2s1	nan
	CHEMBL1516060	43905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	9	4.0	CC(C)Cc1nn2c(=O)cc(COC(=O)c3cccc(NC(=O)c4cccs4)c3)nc2s1	nan
	16030468	43920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3ccccc3n2)cc1C	nan
	CHEMBL1516233	43920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3ccccc3n2)cc1C	nan
	15990035	43921	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	2	7	3.2	CC(C)CCNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1516237	43921	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	2	7	3.2	CC(C)CCNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	6220215	43968	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C/c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	CHEMBL1516846	43968	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C/c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	3238933	44017	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	O=C(Nc1c(C(=O)Nc2cccc(F)c2)oc2ccccc12)c1ccc2c(c1)OCO2	nan
	CHEMBL1517304	44017	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	O=C(Nc1c(C(=O)Nc2cccc(F)c2)oc2ccccc12)c1ccc2c(c1)OCO2	nan
	24687299	44079	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.9	CC(=O)c1sc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)nc1-c1ccccc1	nan
	CHEMBL1517943	44079	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.9	CC(=O)c1sc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)nc1-c1ccccc1	nan
	16009652	44095	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	2	4	5.8	O=C(Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12)c1cc2ccccc2o1	nan
	CHEMBL1518097	44095	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	2	4	5.8	O=C(Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12)c1cc2ccccc2o1	nan
	3298558	44135	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	7	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1518549	44135	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	7	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccccc2)CC1	nan
	5286935	44150	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	2	4	2.4	Cc1ccc(NC(=O)/C(C#N)=C(\N)C(Cl)(Cl)Cl)nc1	nan
	CHEMBL1518626	44150	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	2	4	2.4	Cc1ccc(NC(=O)/C(C#N)=C(\N)C(Cl)(Cl)Cl)nc1	nan
	16031509	44198	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)s2)cc1	nan
	CHEMBL1519036	44198	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)s2)cc1	nan
	938163	44238	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	5	3.2	CC(=O)Nc1cccc(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1519354	44238	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	5	3.2	CC(=O)Nc1cccc(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	2473851	44239	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	6	2.5	COc1cc(C(=O)NCCNC(=O)c2cc(OC)c(C)c(OC)c2)cc(OC)c1C	nan
	CHEMBL1519363	44239	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	6	2.5	COc1cc(C(=O)NCCNC(=O)c2cc(OC)c(C)c(OC)c2)cc(OC)c1C	nan
	24687548	44330	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	7	1	10	2.1	COc1ccc(OC)c(-c2csc(NC(=O)CSc3nnnn3C)n2)c1	nan
	CHEMBL1520201	44330	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	7	1	10	2.1	COc1ccc(OC)c(-c2csc(NC(=O)CSc3nnnn3C)n2)c1	nan
	1142116	44334	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	4	4.7	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccccc1	nan
	CHEMBL1520265	44334	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	4	4.7	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccccc1	nan
	2577415	44594	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	0	8	2.4	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)c2csc(N3CCCCC3)n2)cc1	nan
	CHEMBL1522536	44594	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	0	8	2.4	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)c2csc(N3CCCCC3)n2)cc1	nan
	16027586	44759	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	3.6	CCc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1524058	44759	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	3.6	CCc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	22581682	44784	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	6	3.9	COc1ccc(-c2cn3nc(SCC(=O)NC4CCCCC4)ccc3n2)cc1	nan
	CHEMBL1524339	44784	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	6	3.9	COc1ccc(-c2cn3nc(SCC(=O)NC4CCCCC4)ccc3n2)cc1	nan
	2814763	44796	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	1	4.2	O=C(Nc1ccc(F)cc1)c1cc2cc(Cl)ccc2[nH]1	nan
	CHEMBL1524425	44796	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	1	4.2	O=C(Nc1ccc(F)cc1)c1cc2cc(Cl)ccc2[nH]1	nan
	16012570	44863	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccccc3Cl)c(C)nc21	nan
	CHEMBL1525143	44863	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccccc3Cl)c(C)nc21	nan
	3119681	45167	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	3	6.1	O=C(Cc1ccccc1)Nc1sc2c(c1C(=O)Nc1cccc(Cl)c1)CCCCC2	nan
	CHEMBL1527765	45167	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	3	6.1	O=C(Cc1ccccc1)Nc1sc2c(c1C(=O)Nc1cccc(Cl)c1)CCCCC2	nan
	3370309	45348	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	2	7	3.5	CCN(CCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)c1cccc(C)c1	nan
	CHEMBL1529348	45348	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	2	7	3.5	CCN(CCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)c1cccc(C)c1	nan
	3178487	45403	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.8	CCn1c(SCC(=O)N2CCC(C)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1529806	45403	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.8	CCn1c(SCC(=O)N2CCC(C)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3161332	45653	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	5.4	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1ccccc1F	nan
	CHEMBL1532063	45653	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	5.4	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1ccccc1F	nan
	3787408	45756	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccc(C)cc2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	CHEMBL1532953	45756	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccc(C)cc2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	2105095	45757	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	7	3.7	Cc1cc(NC(=O)CSc2nc3cc(Cl)ccc3c(=O)n2CC(C)C)no1	nan
	CHEMBL1532957	45757	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	7	3.7	Cc1cc(NC(=O)CSc2nc3cc(Cl)ccc3c(=O)n2CC(C)C)no1	nan
	2965497	45760	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	4	0	5	4.2	O=C(c1cc(-c2ccccn2)nc2ccc(Br)cc12)N1CCN(S(=O)(=O)c2ccccc2)CC1	nan
	CHEMBL1532981	45760	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	4	0	5	4.2	O=C(c1cc(-c2ccccn2)nc2ccc(Br)cc12)N1CCN(S(=O)(=O)c2ccccc2)CC1	nan
	16019855	45813	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	3.8	Cc1ccccc1-c1noc(-c2cc3ccccc3oc2=O)n1	nan
	CHEMBL1533477	45813	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	3.8	Cc1ccccc1-c1noc(-c2cc3ccccc3oc2=O)n1	nan
	17374586	46273	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	0	4	3.5	CCC(Oc1cc(Cl)ccc1Cl)C(=O)N1CCC2(CC1)OCCO2	nan
	CHEMBL1537906	46273	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	0	4	3.5	CCC(Oc1cc(Cl)ccc1Cl)C(=O)N1CCC2(CC1)OCCO2	nan
	1078178	46579	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	2	6	3.2	COc1cc(OC)cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)c1	nan
	CHEMBL1540495	46579	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	2	6	3.2	COc1cc(OC)cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)c1	nan
	721260	46613	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	2	1	5	1.7	CCOC(=O)c1cc(C#N)c(S)nc1C	nan
	CHEMBL1540818	46613	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	2	1	5	1.7	CCOC(=O)c1cc(C#N)c(S)nc1C	nan
	657993	46625	14	None	-31	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	1	4	3.4	COc1ccc(-c2c(C#N)c(S)nc3c2CCC3)cc1	nan
	CHEMBL1540912	46625	14	None	-31	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	1	4	3.4	COc1ccc(-c2c(C#N)c(S)nc3c2CCC3)cc1	nan
	1356173	47072	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	2	4	4.8	CCOC(=O)c1c(N=C(S)Nc2ccc(C)cc2)sc2c1CCC2	nan
	CHEMBL1544543	47072	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	2	4	4.8	CCOC(=O)c1c(N=C(S)Nc2ccc(C)cc2)sc2c1CCC2	nan
	16195345	47202	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	2	8	0.4	Cn1c(=O)c2cc(S(=O)(=O)NC(Cc3ccccc3)C(=O)NCC3CCCO3)ccc2n(C)c1=O	nan
	CHEMBL1545503	47202	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	2	8	0.4	Cn1c(=O)c2cc(S(=O)(=O)NC(Cc3ccccc3)C(=O)NCC3CCCO3)ccc2n(C)c1=O	nan
	2868878	47217	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	4.1	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1cccc(F)c1	nan
	CHEMBL1545607	47217	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	4.1	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1cccc(F)c1	nan
	3186499	47237	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	8	3.5	CCc1nnc(NC(=O)CSc2nc3cc4c(cc3cc2C)OCCO4)s1	nan
	CHEMBL1545790	47237	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	8	3.5	CCc1nnc(NC(=O)CSc2nc3cc4c(cc3cc2C)OCCO4)s1	nan
	1485832	47305	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	1	4	4.6	O=C(Nc1ccccc1)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F	nan
	CHEMBL1546403	47305	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	1	4	4.6	O=C(Nc1ccccc1)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F	nan
	24892595	47484	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	7	3.8	COCCn1c(SCC(=O)Nc2cccc(F)c2)nc2c3ccccc3nc-2c1O	nan
	CHEMBL1548166	47484	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	7	3.8	COCCn1c(SCC(=O)Nc2cccc(F)c2)nc2c3ccccc3nc-2c1O	nan
	4223534	47504	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	2	4.5	CC1(C)C(CSc2nc3ccccc3[nH]2)C1(Cl)Cl	nan
	CHEMBL1548301	47504	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	2	4.5	CC1(C)C(CSc2nc3ccccc3[nH]2)C1(Cl)Cl	nan
	818439	47580	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	1	2	7	1.1	COC(=O)c1sc2nc(N)c(C#N)cc2c1N	nan
	CHEMBL1548988	47580	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	1	2	7	1.1	COC(=O)c1sc2nc(N)c(C#N)cc2c1N	nan
	1417035	47651	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	8	1.0	Cn1c(=O)c2c(nc(SCc3ccc(C(=O)O)cc3)n2C)n(C)c1=O	nan
	CHEMBL1549569	47651	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	8	1.0	Cn1c(=O)c2c(nc(SCc3ccc(C(=O)O)cc3)n2C)n(C)c1=O	nan
	1838684	47683	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	4.3	O=C(COc1ccc(Cl)cc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1549821	47683	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	4.3	O=C(COc1ccc(Cl)cc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	1777240	47836	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	5	2.3	Cc1cc(OCC(=O)N2CCC(C(=O)O)CC2)c2c3c(c(=O)oc2c1)CCC3	nan
	CHEMBL1551078	47836	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	5	2.3	Cc1cc(OCC(=O)N2CCC(C(=O)O)CC2)c2c3c(c(=O)oc2c1)CCC3	nan
	16009855	47880	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	5	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)Nc1ccc(F)cc1F	nan
	CHEMBL1551826	47880	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	5	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)Nc1ccc(F)cc1F	nan
	16030710	47886	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	5	1	9	3.3	COC(=O)c1ccc(NC(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccc(C)cc5)sc4n3)CC2)cc1	nan
	CHEMBL1551878	47886	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	5	1	9	3.3	COC(=O)c1ccc(NC(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccc(C)cc5)sc4n3)CC2)cc1	nan
	1004076	47889	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4C)sc3n2)cc1	nan
	CHEMBL1551914	47889	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4C)sc3n2)cc1	nan
	7222625	47950	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	6	4.4	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(C)c(F)c3)nn2)s1	nan
	CHEMBL1552706	47950	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	6	4.4	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(C)c(F)c3)nn2)s1	nan
	16010352	47986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	4	4.6	CCOC(=O)c1c(C)c(-c2ccccc2)n(CC(=O)NCCc2cccc(C)c2)c1C	nan
	CHEMBL1553141	47986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	4	4.6	CCOC(=O)c1c(C)c(-c2ccccc2)n(CC(=O)NCCc2cccc(C)c2)c1C	nan
	16030832	48040	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	1	4	4.2	O=C(Nc1ccccc1C(=O)N1CCCCC1)c1nsc2ccccc12	nan
	CHEMBL1553983	48040	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	1	4	4.2	O=C(Nc1ccccc1C(=O)N1CCCCC1)c1nsc2ccccc12	nan
	16012075	48046	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	4.2	CC(=O)c1ccc(NC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)cc1	nan
	CHEMBL1554061	48046	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	4.2	CC(=O)c1ccc(NC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)cc1	nan
	16008778	48048	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	9	1.9	CCOC(=O)Cn1c(=O)oc2cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)ccc21	nan
	CHEMBL1554084	48048	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	9	1.9	CCOC(=O)Cn1c(=O)oc2cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)ccc21	nan
	3147967	48052	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.6	Cc1cccc(NC(=O)CSc2nnc3c4ccccc4n(C)c3n2)c1	nan
	CHEMBL1554132	48052	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.6	Cc1cccc(NC(=O)CSc2nnc3c4ccccc4n(C)c3n2)c1	nan
	1222858	48059	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	8	3.3	COC(=O)c1sc(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c(C(=O)OC)c1C	nan
	CHEMBL1554200	48059	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	8	3.3	COC(=O)c1sc(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c(C(=O)OC)c1C	nan
	16027476	48060	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1	nan
	CHEMBL1554206	48060	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1	nan
	15989095	48061	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	7	2.2	NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1554211	48061	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	7	2.2	NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	15991109	48066	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1ccc(F)cc1F	nan
	CHEMBL1554314	48066	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1ccc(F)cc1F	nan
	3503858	48074	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	6	5.3	CCC(C)NC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1Cc1ccccc1Cl	nan
	CHEMBL1554470	48074	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	6	5.3	CCC(C)NC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1Cc1ccccc1Cl	nan
	16024920	48109	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	5	5.0	CCCOc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1555031	48109	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	5	5.0	CCCOc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16009072	48117	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	2.8	CCOc1ccc(S(=O)(=O)c2c[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1555115	48117	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	2.8	CCOc1ccc(S(=O)(=O)c2c[nH]c3ccccc3c2=O)cc1	nan
	16015125	48120	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1C	nan
	CHEMBL1555140	48120	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1C	nan
	9550626	48163	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	7	3.9	CCOC(=O)c1c(NC(=O)c2cc(CC(C)C)on2)sc(C(C)=O)c1C	nan
	CHEMBL1555685	48163	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	7	3.9	CCOC(=O)c1c(NC(=O)c2cc(CC(C)C)on2)sc(C(C)=O)c1C	nan
	2176795	48204	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	5	3.8	Cc1onc(-c2ccccc2Cl)c1C(=O)NC(=S)NCC(=O)c1ccccc1	nan
	CHEMBL1556085	48204	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	5	3.8	Cc1onc(-c2ccccc2Cl)c1C(=O)NC(=S)NCC(=O)c1ccccc1	nan
	16022893	48339	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.8	Cc1ccc(-n2nc3c(N4CCC(C(=O)NC(C)c5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1557305	48339	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.8	Cc1ccc(-n2nc3c(N4CCC(C(=O)NC(C)c5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	16011715	48407	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	6	2.9	Cc1cc(F)ccc1Nc1nc2ccccc2n2nnnc12	nan
	CHEMBL1557862	48407	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	6	2.9	Cc1cc(F)ccc1Nc1nc2ccccc2n2nnnc12	nan
	15989730	48412	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	3.6	Cc1cc(C)cc(Nc2nc3ccccc3n3cnnc23)c1	nan
	CHEMBL1557912	48412	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	3.6	Cc1cc(C)cc(Nc2nc3ccccc3n3cnnc23)c1	nan
	16011441	48497	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.9	COc1ccc(Cn2c(SCc3ccc(C(=O)NCc4ccccc4F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1558654	48497	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.9	COc1ccc(Cn2c(SCc3ccc(C(=O)NCc4ccccc4F)cc3)nc3cccnc32)cc1	nan
	16030801	48536	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.4	COc1ccc(-c2cc3ccc(O)c(CN4CCCC(C)C4)c3oc2=O)cc1	nan
	CHEMBL1558940	48536	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.4	COc1ccc(-c2cc3ccc(O)c(CN4CCCC(C)C4)c3oc2=O)cc1	nan
	1970873	48539	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(F)cc5)s4)c3nc12	nan
	CHEMBL1558965	48539	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(F)cc5)s4)c3nc12	nan
	16024619	48554	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	4.3	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1559093	48554	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	4.3	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	135448823	48656	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	2.7	Cc1cc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)no1	nan
	CHEMBL1560048	48656	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	2.7	Cc1cc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)no1	nan
	20944767	48759	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	3.3	O=C(CN1c2ccccc2S(=O)(=O)c2ccccc21)NCc1ccccc1	nan
	CHEMBL1561113	48759	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	3.3	O=C(CN1c2ccccc2S(=O)(=O)c2ccccc21)NCc1ccccc1	nan
	938228	48786	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1cccc(-c2cc(-c3cccnc3)nc(N)c2C#N)c1	nan
	CHEMBL1561334	48786	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1cccc(-c2cc(-c3cccnc3)nc(N)c2C#N)c1	nan
	2136514	49015	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1563400	49015	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	16195481	49058	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	3	8	2.2	COc1cc2nc(S)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2cc1OC	nan
	CHEMBL1563755	49058	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	3	8	2.2	COc1cc2nc(S)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2cc1OC	nan
	16010206	49203	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	CHEMBL1565063	49203	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	16017589	49422	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	7	1.5	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Cl	nan
	CHEMBL1566733	49422	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	7	1.5	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Cl	nan
	2764046	49426	46	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	3	4.8	O=C(O)Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1	nan
	CHEMBL1566761	49426	46	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	3	4.8	O=C(O)Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1	nan
	1419199	49445	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1419200	49445	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1566925	49445	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1101443	49532	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1ccc2oc(-c3cccc(F)c3)nc2c1)c1ccccc1F	nan
	CHEMBL1567607	49532	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1ccc2oc(-c3cccc(F)c3)nc2c1)c1ccccc1F	nan
	663542	49644	15	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(F)c1	nan
	CHEMBL1568508	49644	15	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(F)c1	nan
	2837061	49649	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	3	4.9	O=C(Nc1cccc(NC(=O)c2ccc(Cl)cc2)n1)c1ccc(Cl)cc1	nan
	CHEMBL1568556	49649	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	3	4.9	O=C(Nc1cccc(NC(=O)c2ccc(Cl)cc2)n1)c1ccc(Cl)cc1	nan
	6618042	49660	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	6	3.5	CCCCn1c(=O)nc2n(-c3ccc(OC)cc3)c3ccccc3cc-2c1=O	nan
	CHEMBL1568603	49660	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	6	3.5	CCCCn1c(=O)nc2n(-c3ccc(OC)cc3)c3ccccc3cc-2c1=O	nan
	648080	49723	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	3.6	COc1ccc2cc(C)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	CHEMBL1569235	49723	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	3.6	COc1ccc2cc(C)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	2726812	49768	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	0	4	3.4	COC(=O)c1cc2cc(Cl)ccc2nc1SC	nan
	CHEMBL1569571	49768	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	0	4	3.4	COC(=O)c1cc2cc(Cl)ccc2nc1SC	nan
	802608	49912	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	2	4.3	COc1ccc(Br)cc1C(=O)Nc1cccc(C)c1C	nan
	CHEMBL1570796	49912	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	2	4.3	COc1ccc(Br)cc1C(=O)Nc1cccc(C)c1C	nan
	1247683	49933	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.2	Cc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c(C)o1	nan
	CHEMBL1570956	49933	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.2	Cc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c(C)o1	nan
	2874268	49985	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	5	3.0	Cc1cc(NCCCN(C)C)n2c(nc3ccccc32)c1C#N	nan
	CHEMBL1571576	49985	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	5	3.0	Cc1cc(NCCCN(C)C)n2c(nc3ccccc32)c1C#N	nan
	15988316	49999	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	2.7	CCOC(=O)c1ccc(NC(=O)COC(=O)c2cn(CC)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1571739	49999	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	2.7	CCOC(=O)c1ccc(NC(=O)COC(=O)c2cn(CC)c3nc(C)ccc3c2=O)cc1	nan
	6037218	50069	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1572317	50069	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	995077	50154	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	4	4.3	Cn1cc(CNC(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cn1	nan
	CHEMBL1573031	50154	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	4	4.3	Cn1cc(CNC(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cn1	nan
	1927600	50254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	8	2	5	7.1	CCc1ccccc1NC(=O)CSc1nc(C)c(C(=O)Nc2ccccc2)c(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1574096	50254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	8	2	5	7.1	CCc1ccccc1NC(=O)CSc1nc(C)c(C(=O)Nc2ccccc2)c(-c2ccc(Cl)cc2)c1C#N	nan
	857532	50263	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.3	CCc1cc2cccc(C)c2nc1SCC(=O)NC1CCCC1	nan
	CHEMBL1574178	50263	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.3	CCc1cc2cccc(C)c2nc1SCC(=O)NC1CCCC1	nan
	7206308	50286	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	3.1	O=C(CSc1ccc(-c2ccc3c(c2)OCO3)nn1)Nc1nccs1	nan
	CHEMBL1574382	50286	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	3.1	O=C(CSc1ccc(-c2ccc3c(c2)OCO3)nn1)Nc1nccs1	nan
	2906920	50456	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	4.3	O=C(Nc1ccc(N2C(=O)C3CCCCC3C2=O)cc1Cl)c1cccs1	nan
	CHEMBL1576225	50456	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	4.3	O=C(Nc1ccc(N2C(=O)C3CCCCC3C2=O)cc1Cl)c1cccs1	nan
	135444827	50465	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	3.0	COc1cccc(N2CC(=O)C(c3nc4ccccc4s3)=C2N)c1	nan
	CHEMBL1576321	50465	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	3.0	COc1cccc(N2CC(=O)C(c3nc4ccccc4s3)=C2N)c1	nan
	4099135	50533	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1cccc(Cl)c1	nan
	CHEMBL1576790	50533	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1cccc(Cl)c1	nan
	652081	50737	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4cccnc4)c3nc12	nan
	CHEMBL1578543	50737	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4cccnc4)c3nc12	nan
	2040375	50761	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	0	6	4.7	COc1cc2oc(=O)c3c(c2cc1OCC(=O)c1c(C)n(C)c2ccccc12)CCCC3	nan
	CHEMBL1578721	50761	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	0	6	4.7	COc1cc2oc(=O)c3c(c2cc1OCC(=O)c1c(C)n(C)c2ccccc12)CCCC3	nan
	5100816	50915	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	10	2	6	3.0	O=C(COC(=O)c1cccnc1SCC(=O)NCc1ccccc1)NCc1ccccc1	nan
	CHEMBL1580143	50915	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	10	2	6	3.0	O=C(COC(=O)c1cccnc1SCC(=O)NCc1ccccc1)NCc1ccccc1	nan
	2823757	51451	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	2	4.4	CC(C)(C)c1ccc(C(=O)Nc2ccc(F)cc2)s1	nan
	CHEMBL1584690	51451	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	2	4.4	CC(C)(C)c1ccc(C(=O)Nc2ccc(F)cc2)s1	nan
	1447358	51664	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	6	1.7	CC(C)C(=O)NNC(=O)CN1CCN(c2nc(-c3ccccc3)cs2)CC1	nan
	CHEMBL1586366	51664	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	6	1.7	CC(C)C(=O)NNC(=O)CN1CCN(c2nc(-c3ccccc3)cs2)CC1	nan
	2123807	51837	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	7	0.9	COc1ccc(C(=O)Nc2cccc3c2C(=O)NC3=O)cc1S(=O)(=O)N1CCOCC1	nan
	CHEMBL1587750	51837	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	7	0.9	COc1ccc(C(=O)Nc2cccc3c2C(=O)NC3=O)cc1S(=O)(=O)N1CCOCC1	nan
	2639566	52046	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.1	COc1ccc(C(=O)COc2ccc3ccc(=O)oc3c2)c(OC)c1	nan
	CHEMBL1589654	52046	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.1	COc1ccc(C(=O)COc2ccc3ccc(=O)oc3c2)c(OC)c1	nan
	16027668	52075	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	8	3.4	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1589886	52075	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	8	3.4	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	16027394	52084	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	1	8	3.4	Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1589930	52084	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	1	8	3.4	Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	16007616	52100	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	5	3.6	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCc1ccc(F)cc1)cn2C	nan
	CHEMBL1590166	52100	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	5	3.6	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCc1ccc(F)cc1)cn2C	nan
	16018888	52117	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	0	5	5.2	Cc1nnc(SCc2ccccc2Cl)c2cc3sccc3n12	nan
	CHEMBL1590393	52117	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	0	5	5.2	Cc1nnc(SCc2ccccc2Cl)c2cc3sccc3n12	nan
	2058614	52120	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1cc(C)cc(C)c1	nan
	CHEMBL1590410	52120	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1cc(C)cc(C)c1	nan
	16025295	52131	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.8	CCc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1590637	52131	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.8	CCc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	16017896	52171	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	0	7	2.7	COc1ccc(N2CCN(C(=O)c3sc4nc5n(c(=O)c4c3C)CCC5)CC2)cc1	nan
	CHEMBL1591031	52171	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	0	7	2.7	COc1ccc(N2CCN(C(=O)c3sc4nc5n(c(=O)c4c3C)CCC5)CC2)cc1	nan
	16024829	52208	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	1	4	4.6	O=C(Nc1ccc(F)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1591484	52208	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	1	4	4.6	O=C(Nc1ccc(F)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	16027514	52219	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)c1	nan
	CHEMBL1591656	52219	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)c1	nan
	16012296	52226	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1cccc(NC(=O)c2ccc(-c3ccccc3)s2)c1	nan
	CHEMBL1591740	52226	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1cccc(NC(=O)c2ccc(-c3ccccc3)s2)c1	nan
	16019608	52276	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	8	3.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2sccc23)cc1	nan
	CHEMBL1592430	52276	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	8	3.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2sccc23)cc1	nan
	135546866	52332	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	4	3.7	Cc1ccc(NC(=O)C(C)Sc2nc3c(c(=O)[nH]2)CCCC3)cc1Cl	nan
	CHEMBL1593216	52332	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	4	3.7	Cc1ccc(NC(=O)C(C)Sc2nc3c(c(=O)[nH]2)CCCC3)cc1Cl	nan
	3955100	52338	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	7	4.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)ccc3OC)o2)cc1	nan
	CHEMBL1593290	52338	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	7	4.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)ccc3OC)o2)cc1	nan
	16019825	52355	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	2	4	3.2	Cc1ccc(C)c(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)c1	nan
	CHEMBL1593576	52355	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	2	4	3.2	Cc1ccc(C)c(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)c1	nan
	7598919	52549	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	5	3.5	CCOC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3F)c2=O)cc1	nan
	CHEMBL1595394	52549	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	5	3.5	CCOC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3F)c2=O)cc1	nan
	2135415	52584	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	6	2.0	Cc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)cc1	nan
	CHEMBL1595713	52584	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	6	2.0	Cc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)cc1	nan
	15988650	52631	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	5	5.6	Cc1cc(NC(=O)c2cc(-c3ccc(Br)cc3)on2)nn1Cc1ccc(Cl)cc1	nan
	CHEMBL1596161	52631	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	5	5.6	Cc1cc(NC(=O)c2cc(-c3ccc(Br)cc3)on2)nn1Cc1ccc(Cl)cc1	nan
	16009387	52650	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	1	7	3.9	O=C(Cn1cc(S(=O)(=O)c2ccc(Cl)cc2)c(=O)c2ccccc21)Nc1ccc2c(c1)OCO2	nan
	CHEMBL1596294	52650	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	1	7	3.9	O=C(Cn1cc(S(=O)(=O)c2ccc(Cl)cc2)c(=O)c2ccccc21)Nc1ccc2c(c1)OCO2	nan
	16028259	52674	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	6	3.0	CCOc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccc(F)cc4)ccn3n2)cc1	nan
	CHEMBL1596560	52674	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	6	3.0	CCOc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccc(F)cc4)ccn3n2)cc1	nan
	1450700	52688	2	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCCO3	nan
	CHEMBL1596663	52688	2	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCCO3	nan
	859504	52706	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	0	6	3.3	Cc1cc2cc3c(cc2nc1SCC(=O)OC(C)C)OCO3	nan
	CHEMBL1596835	52706	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	0	6	3.3	Cc1cc2cc3c(cc2nc1SCC(=O)OC(C)C)OCO3	nan
	20903879	52718	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)c1	nan
	CHEMBL1596921	52718	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)c1	nan
	5922522	52780	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	9	1	6	4.7	CCCCOc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccncc2)c(C)c1	nan
	CHEMBL1597564	52780	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	9	1	6	4.7	CCCCOc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccncc2)c(C)c1	nan
	16031965	52785	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	2	6	4.1	COc1ccc(-c2nc(C)c(CCNC(=O)C(=O)Nc3c(C)cccc3C)s2)cc1OC	nan
	CHEMBL1597608	52785	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	2	6	4.1	COc1ccc(-c2nc(C)c(CCNC(=O)C(=O)Nc3c(C)cccc3C)s2)cc1OC	nan
	4656755	52805	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.9	COc1ccc(C(=O)Nc2cc(C)c3c(=O)oc4ccccc4c3n2)cc1	nan
	CHEMBL1597754	52805	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.9	COc1ccc(C(=O)Nc2cc(C)c3c(=O)oc4ccccc4c3n2)cc1	nan
	16030399	52825	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	4	4.9	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCC(C)CC2)cc1	nan
	CHEMBL1597953	52825	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	4	4.9	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCC(C)CC2)cc1	nan
	23603072	52968	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	0	7	0.7	CC1CCCN(C(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)C1	nan
	CHEMBL1599245	52968	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	0	7	0.7	CC1CCCN(C(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)C1	nan
	16009708	53119	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	5	5.0	COc1ccc(CC(=O)Nc2c(C(=O)Nc3ccc(F)cc3)oc3ccccc23)cc1OC	nan
	CHEMBL1600646	53119	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	5	5.0	COc1ccc(CC(=O)Nc2c(C(=O)Nc3ccc(F)cc3)oc3ccccc23)cc1OC	nan
	1093818	53192	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1)c1cc(-c2ccc(Cl)cc2Cl)on1	nan
	CHEMBL1601278	53192	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1)c1cc(-c2ccc(Cl)cc2Cl)on1	nan
	4327872	53275	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	0	6	1.4	CC1CN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC(C)O1	nan
	CHEMBL1602225	53275	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	0	6	1.4	CC1CN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC(C)O1	nan
	7199971	53429	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	8	3.5	Cc1ccc(-n2ncc3c(SCC(=O)Nc4cc(C)on4)ncnc32)c(C)c1	nan
	CHEMBL1603605	53429	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	8	3.5	Cc1ccc(-n2ncc3c(SCC(=O)Nc4cc(C)on4)ncnc32)c(C)c1	nan
	22522531	53437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	1	4	3.5	CCc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	CHEMBL1603663	53437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	1	4	3.5	CCc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	7763635	53526	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	0	7	1.7	COc1ccc(C(=O)COC(=O)CN2C(=O)c3ccccc3C2=O)c(OC)c1	nan
	CHEMBL1604328	53526	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	0	7	1.7	COc1ccc(C(=O)COC(=O)CN2C(=O)c3ccccc3C2=O)c(OC)c1	nan
	1072346	53639	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.5	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1nccs1	nan
	CHEMBL1605363	53639	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.5	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1nccs1	nan
	1005145	53675	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.6	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCC2	nan
	CHEMBL1605614	53675	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.6	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCC2	nan
	15991041	53728	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	3	5.7	CCCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccc3)c(Br)c2)cc1	nan
	CHEMBL1606046	53728	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	3	5.7	CCCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccc3)c(Br)c2)cc1	nan
	2934348	53888	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	2	6	3.4	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccc(O)c1)c1ccco1	nan
	CHEMBL1607257	53888	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	2	6	3.4	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccc(O)c1)c1ccco1	nan
	16027345	53954	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	4.4	CCCNC(=O)Cn1nc(-c2ccc(C)c(C)c2)c2cnc3ccc(OC)cc3c21	nan
	CHEMBL1607743	53954	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	4.4	CCCNC(=O)Cn1nc(-c2ccc(C)c(C)c2)c2cnc3ccc(OC)cc3c21	nan
	753354	53964	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	0	6	2.6	O=C1c2ccccc2C(=O)N1c1nc2nccc(-c3ccccc3)n2n1	nan
	CHEMBL1607842	53964	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	0	6	2.6	O=C1c2ccccc2C(=O)N1c1nc2nccc(-c3ccccc3)n2n1	nan
	3512516	54097	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	7	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	CHEMBL1609027	54097	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	7	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	16011054	54111	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	6	4.0	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Cl)c4)ncn32)s1	nan
	CHEMBL1609118	54111	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	6	4.0	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Cl)c4)ncn32)s1	nan
	2422324	54216	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	3	8	-0.1	COCCn1c(N)c(C(=S)NC(=O)c2cccs2)c(=O)[nH]c1=O	nan
	CHEMBL1609964	54216	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	3	8	-0.1	COCCn1c(N)c(C(=S)NC(=O)c2cccs2)c(=O)[nH]c1=O	nan
	16007504	54274	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.2	COc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1610456	54274	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.2	COc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	2134793	54283	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	0	6	5.6	COCCCn1c(SCc2cccc(Cl)c2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1610529	54283	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	0	6	5.6	COCCCn1c(SCc2cccc(Cl)c2)nc2c(sc3ccccc32)c1=O	nan
	3374134	54310	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	4	2.4	O=C(Cn1c(=S)[nH]c2ccccc2c1=O)NCCc1ccccc1	nan
	CHEMBL1610861	54310	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	4	2.4	O=C(Cn1c(=S)[nH]c2ccccc2c1=O)NCCc1ccccc1	nan
	3185781	54398	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	10	3	8	2.2	COCCN(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCCC1)c1ccc(N(C)C)cc1	nan
	CHEMBL1611537	54398	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	10	3	8	2.2	COCCN(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCCC1)c1ccc(N(C)C)cc1	nan
	3353363	54411	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	6	4.1	COc1ccc(C2CC(=O)c3cnc(N4CCc5ccccc54)nc3C2)cc1OC	nan
	CHEMBL1611722	54411	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	6	4.1	COc1ccc(C2CC(=O)c3cnc(N4CCc5ccccc54)nc3C2)cc1OC	nan
	2201483	55358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	5739455	55358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	9587736	55358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	CHEMBL1442349	55358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	CHEMBL1621693	55358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	354678	55542	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL1518154	55542	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL1623188	55542	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	24792219	55673	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	CHEMBL1551405	55673	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	CHEMBL1624286	55673	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	3490356	72098	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	5	2.2	C#CCn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	CHEMBL1988684	72098	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	5	2.2	C#CCn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	1522244	85054	69	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	164	0	1	3	1.9	Cn1c(S)nc2ccccc21	nan
	CHEMBL227086	85054	69	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	164	0	1	3	1.9	Cn1c(S)nc2ccccc21	nan
	25252625	107116	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	6	1	5	1.8	COc1ccc(CC(=O)N/N=C/c2cccnc2)cc1OC	nan
	CHEMBL3189886	107116	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	6	1	5	1.8	COc1ccc(CC(=O)N/N=C/c2cccnc2)cc1OC	nan
	9701594	107272	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	6	2.1	O=C(N/N=C1\C/C(=N\NC(=O)c2ccncc2)c2ccccc21)c1ccncc1	nan
	CHEMBL3191689	107272	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	6	2.1	O=C(N/N=C1\C/C(=N\NC(=O)c2ccncc2)c2ccccc21)c1ccncc1	nan
	4141152	108366	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	5	2.6	CCOC(=O)c1s/c(=N\C(=O)c2cccc(C)c2)n(C)c1C	nan
	CHEMBL3210377	108366	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	5	2.6	CCOC(=O)c1s/c(=N\C(=O)c2cccc(C)c2)n(C)c1C	nan
	2150923	108569	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	3.1	CCn1/c(=N/C(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3212992	108569	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	3.1	CCn1/c(=N/C(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c(OC)ccc(OC)c21	nan
	1477780	197391	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	1	6	3.0	COc1cc(-c2nc3ccc(N4CCN(C)CC4)cc3[nH]2)cc(OC)c1OC	nan
	CHEMBL587856	197391	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	1	6	3.0	COc1cc(-c2nc3ccc(N4CCN(C)CC4)cc3[nH]2)cc(OC)c1OC	nan
	7190643	20841	10	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1311897	20841	10	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	1739479	21186	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	6.0	Cc1cc(Br)cc2c(C(=O)OCC(=O)c3ccccc3)cc(-c3ccccc3)nc12	nan
	CHEMBL1314681	21186	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	6.0	Cc1cc(Br)cc2c(C(=O)OCC(=O)c3ccccc3)cc(-c3ccccc3)nc12	nan
	15988299	21583	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	CHEMBL1319322	21583	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	4146227	26679	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1363837	26679	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	15988966	30629	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	10	1	4	6.5	CC(C)CN(CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12)CC(C)C	nan
	CHEMBL1397188	30629	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	10	1	4	6.5	CC(C)CN(CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12)CC(C)C	nan
	1398096	30970	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	7	2	5	2.8	CC(C)c1nnc(NC(=O)CCC(=O)NCc2ccc(F)cc2)s1	nan
	CHEMBL1400798	30970	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	7	2	5	2.8	CC(C)c1nnc(NC(=O)CCC(=O)NCc2ccc(F)cc2)s1	nan
	24792315	31306	2	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	9	1.9	CCc1nnc(NC(=O)CSc2nnc3nc(C)cc(C)n23)s1	nan
	CHEMBL1403815	31306	2	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	9	1.9	CCc1nnc(NC(=O)CSc2nnc3nc(C)cc(C)n23)s1	nan
	15991483	39326	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	0	6	6.1	CCOc1ccc(-c2nnc(SCC(=O)c3ccc(Br)cc3)n2-c2ccccc2)cc1	nan
	CHEMBL1473564	39326	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	0	6	6.1	CCOc1ccc(-c2nnc(SCC(=O)c3ccc(Br)cc3)n2-c2ccccc2)cc1	nan
	4299978	43593	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	9	1.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nnc2ccccn12	nan
	CHEMBL1511455	43593	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	9	1.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nnc2ccccn12	nan
	16019368	52382	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	10	4.5	COc1cc(Nc2nc3c(S(=O)(=O)c4ccc(C)c(C)c4)nnn3c3ccsc23)cc(OC)c1	nan
	CHEMBL1593977	52382	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	10	4.5	COc1cc(Nc2nc3c(S(=O)(=O)c4ccc(C)c(C)c4)nnn3c3ccsc23)cc(OC)c1	nan
	814542	52811	22	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	0	2	3	2.7	Cc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	CHEMBL1597829	52811	22	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	0	2	3	2.7	Cc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	9619102	72082	8	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	11	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1OC	nan
	CHEMBL1988156	72082	8	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	11	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1OC	nan
	16010435	6106	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	8	5.0	COc1ccccc1CNc1nc2c(S(=O)(=O)c3ccc(C)c(C)c3)nnn2c2ccc(Cl)cc12	nan
	CHEMBL1081265	6106	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	8	5.0	COc1ccccc1CNc1nc2c(S(=O)(=O)c3ccc(C)c(C)c3)nnn2c2ccc(Cl)cc12	nan
	1375940	7460	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	5	1.0	COc1ccccc1NC=C1C(=O)N(C)C(=O)N(C)C1=O	nan
	CHEMBL1087646	7460	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	5	1.0	COc1ccccc1NC=C1C(=O)N(C)C(=O)N(C)C1=O	nan
	16019310	10644	10	None	-47	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	8	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1	nan
	CHEMBL1171436	10644	10	None	-47	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	8	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1	nan
	16019394	10749	8	None	-37	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	8	4.6	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	CHEMBL1172405	10749	8	None	-37	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	8	4.6	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	16019397	10842	11	None	-54	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	9	4.5	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1173286	10842	11	None	-54	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	9	4.5	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	684664	15251	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	2.7	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccccc1	nan
	CHEMBL1215029	15251	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	2.7	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccccc1	nan
	34768	16209	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	CHEMBL1230732	16209	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	CHEMBL3392220	16209	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	3733180	19464	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.7	O=C(Nc1nnc(-c2ccccc2F)s1)c1ccccc1F	nan
	CHEMBL1300733	19464	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.7	O=C(Nc1nnc(-c2ccccc2F)s1)c1ccccc1F	nan
	3815083	19503	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	1	5	2.5	N#Cc1cnn2c(N)c(-c3ccc(Cl)cc3)cnc12	nan
	CHEMBL1301028	19503	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	1	5	2.5	N#Cc1cnn2c(N)c(-c3ccc(Cl)cc3)cnc12	nan
	2219338	19656	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	2	3	5.0	O=C(Nc1cccc(C(F)(F)F)c1)c1cccnc1NCCc1ccccc1	nan
	CHEMBL1302293	19656	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	2	3	5.0	O=C(Nc1cccc(C(F)(F)F)c1)c1cccnc1NCCc1ccccc1	nan
	1217579	19662	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	6	4.5	N#Cc1ccc(-c2nc3cc(C#N)c(C#N)cc3nc2-c2ccccc2)cc1C#N	nan
	CHEMBL1302356	19662	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	6	4.5	N#Cc1ccc(-c2nc3cc(C#N)c(C#N)cc3nc2-c2ccccc2)cc1C#N	nan
	1244329	19736	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	3.6	COC(=O)c1c(-c2cccnc2)csc1NC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1302889	19736	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	3.6	COC(=O)c1c(-c2cccnc2)csc1NC(=O)c1ccc2c(c1)OCO2	nan
	2740109	19873	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.5	N#Cc1c(N2CCOCC2)nsc1-c1ccc(C(F)(F)F)cc1	nan
	CHEMBL1303994	19873	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.5	N#Cc1c(N2CCOCC2)nsc1-c1ccc(C(F)(F)F)cc1	nan
	1462693	20143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	8	2	7	2.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)C3CC3)s2)cc1	nan
	CHEMBL1306151	20143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	8	2	7	2.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)C3CC3)s2)cc1	nan
	2158311	20145	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	5	5.1	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1306166	20145	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	5	5.1	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1C(F)(F)F	nan
	940263	20180	37	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	1	2	2.8	Cc1cc(S)c2ccccc2n1	nan
	CHEMBL1306515	20180	37	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	1	2	2.8	Cc1cc(S)c2ccccc2n1	nan
	3678328	20477	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	4.0	O=C(COC(=O)c1cccc(Br)c1)Nc1cccc2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1308878	20477	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	4.0	O=C(COC(=O)c1cccc(Br)c1)Nc1cccc2c1C(=O)c1ccccc1C2=O	nan
	3942275	20614	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	7	4.6	CC1CN(S(=O)(=O)c2ccc(C(=O)Nc3nc(-c4cc5ccccc5o4)cs3)cc2)CC(C)O1	nan
	CHEMBL1310132	20614	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	7	4.6	CC1CN(S(=O)(=O)c2ccc(C(=O)Nc3nc(-c4cc5ccccc5o4)cs3)cc2)CC(C)O1	nan
	2744150	21069	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	7	4.3	Cc1nc(-c2nnc(SCC(=O)Nc3cc(Cl)cc(Cl)c3)n2C)cs1	nan
	CHEMBL1313563	21069	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	7	4.3	Cc1nc(-c2nnc(SCC(=O)Nc3cc(Cl)cc(Cl)c3)n2C)cs1	nan
	2997549	21140	9	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	8	2.9	Cc1ccc(S(=O)(=O)c2c(N)n(CCN3CCOCC3)c3nc4ccccc4nc23)cc1C	nan
	CHEMBL1314156	21140	9	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	8	2.9	Cc1ccc(S(=O)(=O)c2c(N)n(CCN3CCOCC3)c3nc4ccccc4nc23)cc1C	nan
	16009918	21151	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	7	1.5	Cc1ccc(Cl)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1314250	21151	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	7	1.5	Cc1ccc(Cl)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	135458483	21165	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	1.7	Cc1ccn2c(=O)c(C(=O)NCCc3ccccc3)c(O)nc2c1	nan
	CHEMBL1314355	21165	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	1.7	Cc1ccn2c(=O)c(C(=O)NCCc3ccccc3)c(O)nc2c1	nan
	16024181	21187	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	4	3.9	Cc1cccc(N2C(=O)CS(=O)(=O)C23C(=O)N(Cc2c(F)cccc2Cl)c2ccccc23)c1	nan
	CHEMBL1314689	21187	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	4	3.9	Cc1cccc(N2C(=O)CS(=O)(=O)C23C(=O)N(Cc2c(F)cccc2Cl)c2ccccc23)c1	nan
	4913767	21198	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	0	7	3.2	COC(=O)Cc1c(C)c2ccc3c(c2oc1=O)CN(Cc1ccccc1OC)CO3	nan
	CHEMBL1314916	21198	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	0	7	3.2	COC(=O)Cc1c(C)c2ccc3c(c2oc1=O)CN(Cc1ccccc1OC)CO3	nan
	16027662	21209	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.5	O=C(Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1)c1ccc(F)cc1	nan
	CHEMBL1315065	21209	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.5	O=C(Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1)c1ccc(F)cc1	nan
	16021060	21242	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)cc1OC	nan
	CHEMBL1315440	21242	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)cc1OC	nan
	4524401	21254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	1	8	4.0	COC(=O)c1ccccc1NC(=O)CSc1nc2ccsc2c(=O)n1CCC(C)C	nan
	CHEMBL1315570	21254	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	1	8	4.0	COC(=O)c1ccccc1NC(=O)CSc1nc2ccsc2c(=O)n1CCC(C)C	nan
	16020822	21256	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1315619	21256	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	16016226	21272	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	5.0	CC(=O)c1cccc(NC(=O)c2nc(-c3ccccc3)n(-c3cccc(Cl)c3)n2)c1	nan
	CHEMBL1315816	21272	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	5.0	CC(=O)c1cccc(NC(=O)c2nc(-c3ccccc3)n(-c3cccc(Cl)c3)n2)c1	nan
	16009840	21275	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	5.2	COc1ccccc1NC(=O)c1oc2ccccc2c1NC(=O)C1CCCCC1	nan
	CHEMBL1315829	21275	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	5.2	COc1ccccc1NC(=O)c1oc2ccccc2c1NC(=O)C1CCCCC1	nan
	16025104	21293	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	5	4.4	CC(=O)c1cccc(NC(=O)c2cnn(-c3cccc(C)c3)c2-n2cccc2)c1	nan
	CHEMBL1316030	21293	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	5	4.4	CC(=O)c1cccc(NC(=O)c2cnn(-c3cccc(C)c3)c2-n2cccc2)c1	nan
	1083262	21301	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	0	5	4.4	CCOC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1316119	21301	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	0	5	4.4	CCOC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)c1C#N	nan
	20940443	21320	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.5	CCCNC(=O)c1cc(-c2ccccc2)c(N2CCCCC2)s1	nan
	CHEMBL1316420	21320	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.5	CCCNC(=O)c1cc(-c2ccccc2)c(N2CCCCC2)s1	nan
	16022216	21365	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	4	4.7	CC(=O)c1ccc(NC(=O)CC(c2cccs2)N2Cc3ccccc3C2=O)cc1	nan
	CHEMBL1317049	21365	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	4	4.7	CC(=O)c1ccc(NC(=O)CC(c2cccs2)N2Cc3ccccc3C2=O)cc1	nan
	16027421	21372	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	CHEMBL1317129	21372	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	2159322	21386	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	0	6	3.6	CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2c(C)ccc(OC)c21	nan
	CHEMBL1317343	21386	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	0	6	3.6	CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2c(C)ccc(OC)c21	nan
	16028188	21403	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	3	3.8	Cc1cccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)c1	nan
	CHEMBL1317555	21403	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	3	3.8	Cc1cccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)c1	nan
	16023037	21418	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	6	3.6	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(Cl)cc3)s2)cc1	nan
	CHEMBL1317727	21418	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	6	3.6	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(Cl)cc3)s2)cc1	nan
	2227086	21425	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	3	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cccc(Cl)c1	nan
	CHEMBL1317881	21425	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	3	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cccc(Cl)c1	nan
	16024891	21461	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	5	4.9	CSc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1318327	21461	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	5	4.9	CSc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16025877	21488	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	8	2.9	CC(C)Oc1ccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)cc1	nan
	CHEMBL1318545	21488	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	8	2.9	CC(C)Oc1ccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)cc1	nan
	16445400	21511	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	2	1	5	2.8	Cc1nonc1NC(=O)c1oc2ccc(F)cc2c1C	nan
	CHEMBL1318745	21511	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	2	1	5	2.8	Cc1nonc1NC(=O)c1oc2ccc(F)cc2c1C	nan
	16022946	21606	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1319510	21606	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	16022818	21672	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(Cl)cc1NC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)CC1	nan
	CHEMBL1320089	21672	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(Cl)cc1NC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)CC1	nan
	4183241	21677	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccc(F)cc3)n2)cc1	nan
	CHEMBL1320138	21677	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccc(F)cc3)n2)cc1	nan
	3167480	21687	6	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	5.1	Cc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	CHEMBL1320193	21687	6	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	5.1	Cc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	16023651	21690	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	3	5	3.6	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(C)c2)N3)cc1	nan
	CHEMBL1320214	21690	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	3	5	3.6	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(C)c2)N3)cc1	nan
	16009865	21719	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	1	6	3.6	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1320479	21719	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	1	6	3.6	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	3613580	21854	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	1	5	3.7	CNc1nc(-c2ccccc2)nc(-c2ccc(OC)cc2)c1C#N	nan
	CHEMBL1321693	21854	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	1	5	3.7	CNc1nc(-c2ccccc2)nc(-c2ccc(OC)cc2)c1C#N	nan
	16026062	22019	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.6	Cc1cccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1C	nan
	CHEMBL1323207	22019	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.6	Cc1cccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1C	nan
	720155	22049	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	2	2	4.8	Cc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(C)c3)c2)c1	nan
	CHEMBL1323476	22049	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	2	2	4.8	Cc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(C)c3)c2)c1	nan
	866639	22072	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	6	2.4	Cc1cccn2c(=O)c3cc(C(=O)N4COCC4(C)C)sc3nc12	nan
	CHEMBL1323660	22072	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	6	2.4	Cc1cccn2c(=O)c3cc(C(=O)N4COCC4(C)C)sc3nc12	nan
	7597258	22197	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	4	3.7	Cc1ccc(-c2nnc(NC(=O)Cc3ccc(F)cc3)o2)c(C)c1	nan
	CHEMBL1324652	22197	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	4	3.7	Cc1ccc(-c2nnc(NC(=O)Cc3ccc(F)cc3)o2)c(C)c1	nan
	20903561	22254	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	2	5	3.1	O=C(Nc1ccc(F)cc1)C1CCCN(S(=O)(=O)c2ccc3nc(O)ccc3c2)C1	nan
	CHEMBL1325113	22254	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	2	5	3.1	O=C(Nc1ccc(F)cc1)C1CCCN(S(=O)(=O)c2ccc3nc(O)ccc3c2)C1	nan
	1239703	22271	8	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.0	CCc1nnc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)s1	nan
	CHEMBL1325279	22271	8	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.0	CCc1nnc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)s1	nan
	4053254	22367	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	2	5	3.1	COc1ccc(NC(=O)CCn2c(=S)[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1326345	22367	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	2	5	3.1	COc1ccc(NC(=O)CCn2c(=S)[nH]c3ccccc3c2=O)cc1	nan
	2742890	22452	5	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	2	2	4.3	COc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	CHEMBL1327081	22452	5	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	2	2	4.3	COc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	16030465	22517	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)N1CCCCC1	nan
	CHEMBL1327646	22517	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)N1CCCCC1	nan
	2330460	22575	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	7	5.0	Cc1nn(-c2ccccc2Cl)c2sc(C(=O)Nc3nnc(C4CC4)s3)cc12	nan
	CHEMBL1328005	22575	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	7	5.0	Cc1nn(-c2ccccc2Cl)c2sc(C(=O)Nc3nnc(C4CC4)s3)cc12	nan
	1048410	23017	8	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	4	5.6	COc1cc(NC(=O)c2ccc(-c3ccc(Br)cc3)o2)ccc1NC(=O)C(C)C	nan
	CHEMBL1331632	23017	8	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	4	5.6	COc1cc(NC(=O)c2ccc(-c3ccc(Br)cc3)o2)ccc1NC(=O)C(C)C	nan
	1088560	23026	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	1	3	4.1	CC(=O)c1cn(CC(=O)Nc2ccc(C)c(C)c2)c2ccccc12	nan
	CHEMBL1331684	23026	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	1	3	4.1	CC(=O)c1cn(CC(=O)Nc2ccc(C)c(C)c2)c2ccccc12	nan
	16022830	23128	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)c(Cl)c1	nan
	CHEMBL1332482	23128	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)c(Cl)c1	nan
	4443607	23332	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	3.3	COc1cc2[nH]c(=S)n(Cc3ccc(F)cc3)c(=O)c2cc1OC	nan
	CHEMBL1334074	23332	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	3.3	COc1cc2[nH]c(=S)n(Cc3ccc(F)cc3)c(=O)c2cc1OC	nan
	3245441	23376	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	3.1	O=C(CCCN1C(=O)c2ccccc2C1=O)Nc1c2c(nc3c1CCC3)CCC2	nan
	CHEMBL1334367	23376	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	3.1	O=C(CCCN1C(=O)c2ccccc2C1=O)Nc1c2c(nc3c1CCC3)CCC2	nan
	16009378	23452	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	5	3.8	Cc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c(C)c1	nan
	CHEMBL1335076	23452	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	5	3.8	Cc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c(C)c1	nan
	135454500	23699	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.6	Cc1cc(-n2c(SCC(=O)Nc3ccc(F)c(F)c3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1337074	23699	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.6	Cc1cc(-n2c(SCC(=O)Nc3ccc(F)c(F)c3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	16023881	23785	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	2	4.2	O=C(Nc1ccc(F)cc1F)c1cc2ccc3cccnc3c2[nH]1	nan
	CHEMBL1337846	23785	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	2	4.2	O=C(Nc1ccc(F)cc1F)c1cc2ccc3cccnc3c2[nH]1	nan
	3458131	23951	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	CHEMBL1339257	23951	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	3677224	23979	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	6	3.3	O=C(NCCc1ccccc1)c1cc(-c2ccncc2)nc2ccc(S(=O)(=O)N3CCOCC3)cc12	nan
	CHEMBL1339543	23979	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	6	3.3	O=C(NCCc1ccccc1)c1cc(-c2ccncc2)nc2ccc(S(=O)(=O)N3CCOCC3)cc12	nan
	4625935	24038	14	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccc(F)cc2)nc1-c1ccccc1	nan
	CHEMBL1340080	24038	14	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccc(F)cc2)nc1-c1ccccc1	nan
	1873236	24313	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	7	2.6	COC(=O)c1ccc2c(=O)n(Cc3ccc4c(c3)OCO4)c(=S)[nH]c2c1	nan
	CHEMBL1342433	24313	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	7	2.6	COC(=O)c1ccc2c(=O)n(Cc3ccc4c(c3)OCO4)c(=S)[nH]c2c1	nan
	1302080	24373	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	2	4	2.8	O=C(CCc1ccccc1)NC(=S)Nc1ccc2c(c1)C(=O)OC2	nan
	CHEMBL1342849	24373	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	2	4	2.8	O=C(CCc1ccccc1)NC(=S)Nc1ccc2c(c1)C(=O)OC2	nan
	3185654	24418	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	3.3	COc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCC1)c1ccc(N(C)C)cc1	nan
	CHEMBL1343261	24418	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	3.3	COc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCC1)c1ccc(N(C)C)cc1	nan
	1164441	24469	6	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	7	4.8	COc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	CHEMBL1343720	24469	6	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	7	4.8	COc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	653965	24494	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	4	3.8	Cc1cc(C)c2nc(SCC(=O)N3CCCCC3)c(C#N)cc2c1	nan
	CHEMBL1343941	24494	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	4	3.8	Cc1cc(C)c2nc(SCC(=O)N3CCCCC3)c(C#N)cc2c1	nan
	5068572	24960	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	6	3.1	COc1ccc(Cn2c(=S)[nH]c3cc(OC)c(OC)cc3c2=O)cc1	nan
	CHEMBL1347842	24960	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	6	3.1	COc1ccc(Cn2c(=S)[nH]c3cc(OC)c(OC)cc3c2=O)cc1	nan
	2992621	25005	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	4	3.0	COc1cccc2cc(C(=O)NCc3ccc(C)cc3)c(=O)oc12	nan
	CHEMBL1348238	25005	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	4	3.0	COc1cccc2cc(C(=O)NCc3ccc(C)cc3)c(=O)oc12	nan
	2785932	25081	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	0	0	5	1.4	Cn1c(=O)c2cc3ccc(Cl)cc3nc2n(C)c1=O	nan
	CHEMBL1348983	25081	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	0	0	5	1.4	Cn1c(=O)c2cc3ccc(Cl)cc3nc2n(C)c1=O	nan
	20929691	25106	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	3.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccco3)c2n1	nan
	CHEMBL1349170	25106	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	3.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccco3)c2n1	nan
	1261778	25338	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	1	3	5.6	Cc1cccc2c(C(=O)Nc3ccc(Br)cc3)cc(-c3ccccn3)nc12	nan
	CHEMBL1351124	25338	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	1	3	5.6	Cc1cccc2c(C(=O)Nc3ccc(Br)cc3)cc(-c3ccccn3)nc12	nan
	2309203	25341	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	4	4.3	O=C(NCCCCNC(=O)c1ccc(Br)s1)c1ccc(Br)s1	nan
	CHEMBL1351160	25341	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	4	4.3	O=C(NCCCCNC(=O)c1ccc(Br)s1)c1ccc(Br)s1	nan
	1945599	25474	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	6	3.7	COc1cc(C(=O)NC(=S)Nc2cccc3nc(C)ccc23)cc(OC)c1OC	nan
	CHEMBL1352289	25474	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	6	3.7	COc1cc(C(=O)NC(=S)Nc2cccc3nc(C)ccc23)cc(OC)c1OC	nan
	2345662	25583	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	6	2.8	COc1ccc(-c2nnc(NC(=O)C(C)C)s2)c(OC)c1	nan
	CHEMBL1353144	25583	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	6	2.8	COc1ccc(-c2nnc(NC(=O)C(C)C)s2)c(OC)c1	nan
	2588947	25619	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.2	COc1ccc2c(-c3ccccc3)cc(SCC(=O)NC(N)=O)nc2c1	nan
	CHEMBL1353338	25619	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.2	COc1ccc2c(-c3ccccc3)cc(SCC(=O)NC(N)=O)nc2c1	nan
	16024589	25752	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3Cl)c2n1	nan
	CHEMBL1354308	25752	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3Cl)c2n1	nan
	24981187	25760	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	0	7	2.0	CCOC(=O)C1CCN(C(=O)COC(=O)C2CCN(S(=O)(=O)c3ccc(C)c(C)c3)CC2)CC1	nan
	CHEMBL1354340	25760	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	0	7	2.0	CCOC(=O)C1CCN(C(=O)COC(=O)C2CCN(S(=O)(=O)c3ccc(C)c(C)c3)CC2)CC1	nan
	16015624	25790	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	6	5.8	Cc1ccccc1OCC(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	CHEMBL1354759	25790	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	6	5.8	Cc1ccccc1OCC(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	16022729	25848	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	2.5	Cc1noc(Cn2c(=O)c3ccccc3n(CC(=O)Nc3cc(Cl)ccc3C)c2=O)n1	nan
	CHEMBL1355436	25848	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	2.5	Cc1noc(Cn2c(=O)c3ccccc3n(CC(=O)Nc3cc(Cl)ccc3C)c2=O)n1	nan
	15989639	25851	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.4	COc1ccc(CCn2c(=O)c3ccccc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	CHEMBL1355514	25851	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.4	COc1ccc(CCn2c(=O)c3ccccc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	16023098	25856	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	5	4.1	Cc1nnc2c3ccccc3nc(Nc3ccc(F)cc3Cl)n12	nan
	CHEMBL1355617	25856	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	5	4.1	Cc1nnc2c3ccccc3nc(Nc3ccc(F)cc3Cl)n12	nan
	2150160	25857	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	6	4.2	COCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1355622	25857	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	6	4.2	COCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	135546934	25862	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	3	3	7	4.3	Cc1cccc(NC(=O)c2sc3nc(-c4cc5ccc(O)cc5oc4=O)[nH]c(=O)c3c2C)c1	nan
	CHEMBL1355684	25862	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	3	3	7	4.3	Cc1cccc(NC(=O)c2sc3nc(-c4cc5ccc(O)cc5oc4=O)[nH]c(=O)c3c2C)c1	nan
	135419178	25883	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	5	4.8	CC(=O)Nc1ccc(/C=C/c2nc(-c3ccccc3O)n(-c3ccccc3)n2)cc1	nan
	CHEMBL1355898	25883	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	5	4.8	CC(=O)Nc1ccc(/C=C/c2nc(-c3ccccc3O)n(-c3ccccc3)n2)cc1	nan
	16017045	25928	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	0	6	4.8	CCC(C(=O)N1CCN(c2cccc(C)c2C)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1356499	25928	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	0	6	4.8	CCC(C(=O)N1CCN(c2cccc(C)c2C)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	15990110	25930	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	5	5.3	Cc1ccc(C)c(N2CCN(C(c3ccccc3)c3nnc(-c4ccccc4)o3)CC2)c1	nan
	CHEMBL1356570	25930	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	5	5.3	Cc1ccc(C)c(N2CCN(C(c3ccccc3)c3nnc(-c4ccccc4)o3)CC2)c1	nan
	5886984	25935	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	6.8	COc1c(Cl)cc(Cl)cc1/C=C(\C#N)c1nc(-c2ccc(Cl)cc2)cs1	nan
	CHEMBL1356614	25935	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	6.8	COc1c(Cl)cc(Cl)cc1/C=C(\C#N)c1nc(-c2ccc(Cl)cc2)cs1	nan
	16018240	25957	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	5.2	Cc1c(C(=O)NCc2ccc(N(C)C)cc2)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1356884	25957	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	5.2	Cc1c(C(=O)NCc2ccc(N(C)C)cc2)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	2219490	25967	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	4	5.1	O=C(Cn1cc(C(=O)c2ccco2)c2ccccc21)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1357026	25967	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	4	5.1	O=C(Cn1cc(C(=O)c2ccco2)c2ccccc21)Nc1ccccc1C(F)(F)F	nan
	16007510	25992	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	1	4	5.6	CCOc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1357328	25992	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	1	4	5.6	CCOc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	16010573	25993	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	8	1	7	2.6	CCOc1ccccc1NC(=O)Cn1c(=O)n(CCC(C)C)c(=O)c2cccnc21	nan
	CHEMBL1357333	25993	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	8	1	7	2.6	CCOc1ccccc1NC(=O)Cn1c(=O)n(CCC(C)C)c(=O)c2cccnc21	nan
	7533493	25999	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	6	4.1	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(F)ccc3F)o2)cc1	nan
	CHEMBL1357469	25999	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	6	4.1	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(F)ccc3F)o2)cc1	nan
	16030313	26023	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	CHEMBL1357868	26023	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	7244606	26026	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	0	7	2.9	C#CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OC)c(OC)cc21	nan
	CHEMBL1357945	26026	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	0	7	2.9	C#CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OC)c(OC)cc21	nan
	16018859	26030	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.1	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1357984	26030	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.1	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1C(F)(F)F	nan
	16009434	26034	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	7	3.4	O=C(COc1ccccc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1358022	26034	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	7	3.4	O=C(COc1ccccc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	15987969	26110	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	4	4.1	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3cccc(CC)c3)c21	nan
	CHEMBL1358851	26110	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	4	4.1	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3cccc(CC)c3)c21	nan
	3799752	26111	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	2.4	COc1ccc(OC)c(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)c1	nan
	CHEMBL1358861	26111	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	2.4	COc1ccc(OC)c(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)c1	nan
	7210861	26188	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	5	3.6	CCn1c(SCC(=O)Nc2ccccc2)nc2c([nH]c3ccccc32)c1=O	nan
	CHEMBL1359450	26188	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	5	3.6	CCn1c(SCC(=O)Nc2ccccc2)nc2c([nH]c3ccccc32)c1=O	nan
	1818953	26347	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	6	5.7	C=C(C)Cn1c(SCC(=O)c2ccc(Br)cc2)nc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1360901	26347	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	6	5.7	C=C(C)Cn1c(SCC(=O)c2ccc(Br)cc2)nc2sc3c(c2c1=O)CCCC3	nan
	16022921	26409	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	CHEMBL1361507	26409	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	4329717	26422	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	2	3	4.2	CC(NC(=O)c1cc(O)nc2ccc(Br)cc12)c1ccccc1	nan
	CHEMBL1361599	26422	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	2	3	4.2	CC(NC(=O)c1cc(O)nc2ccc(Br)cc12)c1ccccc1	nan
	3475073	26460	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	2	5.4	Cc1cc2ccccc2n1CCNC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	CHEMBL1361903	26460	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	2	5.4	Cc1cc2ccccc2n1CCNC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	16022126	26489	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	4.5	COc1cc(OC)c(NC(=O)c2c(N3CCCC3=O)c3cc(C)ccc3n2C)cc1Cl	nan
	CHEMBL1362140	26489	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	4.5	COc1cc(OC)c(NC(=O)c2c(N3CCCC3=O)c3cc(C)ccc3n2C)cc1Cl	nan
	1984900	26514	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	8	1	7	5.0	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3cccs3)cc2)cc1	nan
	CHEMBL1362375	26514	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	8	1	7	5.0	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3cccs3)cc2)cc1	nan
	6471827	26545	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	9	2.4	Cc1nnc(NC(=O)C(C)Sc2nnc(-c3ccco3)n2C)s1	nan
	CHEMBL1362583	26545	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	9	2.4	Cc1nnc(NC(=O)C(C)Sc2nnc(-c3ccco3)n2C)s1	nan
	7693885	26558	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	4	1	4	3.9	COc1ccc(C(=O)Nc2cc(-c3ccc(C)cc3)no2)cc1	nan
	CHEMBL1362677	26558	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	4	1	4	3.9	COc1ccc(C(=O)Nc2cc(-c3ccc(C)cc3)no2)cc1	nan
	16019393	26569	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	4.0	CCCCNc1nc2c(S(=O)(=O)c3ccc(Cl)cc3)nnn2c2ccsc12	nan
	CHEMBL1362800	26569	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	4.0	CCCCNc1nc2c(S(=O)(=O)c3ccc(Cl)cc3)nnn2c2ccsc12	nan
	22334175	26587	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	10	2	10	2.8	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cc(OC)c(OC)c(OC)c3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1362992	26587	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	10	2	10	2.8	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cc(OC)c(OC)c(OC)c3)c3ccccc3c2=O)cc1OC	nan
	645413	26598	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	3.4	Cc1cc(C(F)F)n2nc(C(=O)Nc3ccccc3Br)nc2n1	nan
	CHEMBL1363101	26598	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	3.4	Cc1cc(C(F)F)n2nc(C(=O)Nc3ccccc3Br)nc2n1	nan
	16024545	26608	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)c1	nan
	CHEMBL1363144	26608	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)c1	nan
	4447999	26644	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	2	6	4.6	Cc1ccc(NC(=O)CSc2nc3ccccc3c(=O)n2CCC(=O)NC2CCCCC2)cc1C	nan
	CHEMBL1363483	26644	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	2	6	4.6	Cc1ccc(NC(=O)CSc2nc3ccccc3c(=O)n2CCC(=O)NC2CCCCC2)cc1C	nan
	16030946	26694	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	4.1	COc1ccc(NC(=O)CSc2ccc3nc(-c4ccccc4)cn3n2)cc1OC	nan
	CHEMBL1363950	26694	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	4.1	COc1ccc(NC(=O)CSc2ccc3nc(-c4ccccc4)cn3n2)cc1OC	nan
	1960168	26752	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	2	0	5	4.4	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccc(F)cc2)cc1	nan
	CHEMBL1364491	26752	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	2	0	5	4.4	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccc(F)cc2)cc1	nan
	1258567	26944	17	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.5	COc1ccc(-c2cc(-c3ccccc3)nc(SCC(=O)Nc3nccs3)c2C#N)cc1	nan
	CHEMBL1366086	26944	17	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.5	COc1ccc(-c2cc(-c3ccccc3)nc(SCC(=O)Nc3nccs3)c2C#N)cc1	nan
	5726342	26978	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	3.8	CN1C(=O)C(O)=C(C(=O)c2ccc(Br)cc2)C1c1ccc(F)cc1	nan
	CHEMBL1366379	26978	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	3.8	CN1C(=O)C(O)=C(C(=O)c2ccc(Br)cc2)C1c1ccc(F)cc1	nan
	16015810	26992	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cccc(-c3nc4ccccc4s3)c2C)cc1	nan
	CHEMBL1366460	26992	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cccc(-c3nc4ccccc4s3)c2C)cc1	nan
	5204153	27013	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	1.3	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3ccc4c(c3)C(=O)NC4=O)cc2)CC1	nan
	CHEMBL1366674	27013	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	1.3	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3ccc4c(c3)C(=O)NC4=O)cc2)CC1	nan
	16015685	27051	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	5.5	Cc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCc5ccccc54)sc3c2)cc1	nan
	CHEMBL1367053	27051	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	5.5	Cc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCc5ccccc54)sc3c2)cc1	nan
	561651	27164	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	0	3	4.6	c1ccc(C2=NN(c3ccccc3)C(c3ccco3)C2)cc1	nan
	CHEMBL1367925	27164	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	0	3	4.6	c1ccc(C2=NN(c3ccccc3)C(c3ccco3)C2)cc1	nan
	16022119	27393	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.9	COc1ccc2c(c1)c1c(c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	CHEMBL1369667	27393	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.9	COc1ccc2c(c1)c1c(c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	16024643	27423	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	5	3.9	CCc1ccc(C(=O)c2cn(CC(=O)NCCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1369852	27423	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	5	3.9	CCc1ccc(C(=O)c2cn(CC(=O)NCCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	16018703	27467	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	0	6	3.4	Cc1ccc(Cl)cc1N1CCN(C(=O)CCn2c(=O)c3cccn3c3cccnc32)CC1	nan
	CHEMBL1370112	27467	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	0	6	3.4	Cc1ccc(Cl)cc1N1CCN(C(=O)CCn2c(=O)c3cccn3c3cccnc32)CC1	nan
	16017844	27544	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	6	1.6	COc1cccc(-n2ccn(CC(=O)NCc3ccc(C)cc3)c(=O)c2=O)c1	nan
	CHEMBL1370655	27544	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	6	1.6	COc1cccc(-n2ccn(CC(=O)NCc3ccc(C)cc3)c(=O)c2=O)c1	nan
	2053979	27559	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	4.0	CCN(C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)C1CCCCC1	nan
	CHEMBL1370734	27559	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	4.0	CCN(C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)C1CCCCC1	nan
	2999996	27586	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	3	0	9	2.9	O=C(OCc1cc(=O)n2c(n1)sc1ccccc12)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	CHEMBL1370976	27586	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	3	0	9	2.9	O=C(OCc1cc(=O)n2c(n1)sc1ccccc12)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	2212806	27640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	4	5.1	Cc1cccc(NC(=O)c2cc(NC(=O)c3ccco3)ccc2N2CCCCC2)c1	nan
	CHEMBL1371405	27640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	4	5.1	Cc1cccc(NC(=O)c2cc(NC(=O)c3ccco3)ccc2N2CCCCC2)c1	nan
	4069120	27658	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.7	COc1ccc(OC)c(NC(=O)c2oc(=O)c3ccccc3c2-c2ccccc2)c1	nan
	CHEMBL1371548	27658	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.7	COc1ccc(OC)c(NC(=O)c2oc(=O)c3ccccc3c2-c2ccccc2)c1	nan
	862401	27671	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	3.7	COc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	CHEMBL1371650	27671	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	3.7	COc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	941550	27675	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	6	3.4	COc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	CHEMBL1371690	27675	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	6	3.4	COc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	648869	27795	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	5	3.9	CCOc1ccc2cc(C#N)c(SCC(=O)N3CCC(C)CC3)nc2c1	nan
	CHEMBL1372547	27795	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	5	3.9	CCOc1ccc2cc(C#N)c(SCC(=O)N3CCC(C)CC3)nc2c1	nan
	664361	27842	12	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1nc(SCC(=O)Nc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1372818	27842	12	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1nc(SCC(=O)Nc2ccccc2)c2oc3ccccc3c2n1	nan
	2404728	27970	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.4	O=C(COC(=O)c1ccc(Cl)cc1O)NC(=O)C1CCCCC1	nan
	CHEMBL1373640	27970	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.4	O=C(COC(=O)c1ccc(Cl)cc1O)NC(=O)C1CCCCC1	nan
	711468	28007	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	1	1	3	3.3	Cc1cc(-c2cccc(Br)c2)c(C#N)c(N)n1	nan
	CHEMBL1373906	28007	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	1	1	3	3.3	Cc1cc(-c2cccc(Br)c2)c(C#N)c(N)n1	nan
	660358	28049	18	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	8	4.8	CCOC(=O)c1sc(NC(=O)CSc2nc3c(cc2C#N)CCCCCC3)c(C#N)c1C	nan
	CHEMBL1374224	28049	18	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	8	4.8	CCOC(=O)c1sc(NC(=O)CSc2nc3c(cc2C#N)CCCCCC3)c(C#N)c1C	nan
	848636	28093	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	6	5.1	Cc1sc2ncnc(Sc3nc4ccccc4s3)c2c1C	nan
	CHEMBL1374559	28093	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	6	5.1	Cc1sc2ncnc(Sc3nc4ccccc4s3)c2c1C	nan
	22330687	28116	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	8	4.3	COc1ccc(C)cc1NC(=O)c1sc2ncnc(N3CCN(c4ccccn4)CC3)c2c1C	nan
	CHEMBL1374703	28116	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	8	4.3	COc1ccc(C)cc1NC(=O)c1sc2ncnc(N3CCN(c4ccccn4)CC3)c2c1C	nan
	16421351	28143	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	5513687	28143	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	CHEMBL1374848	28143	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	2113664	28270	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	0	8	4.2	CCc1cc2c(SCC(=O)C(C#N)=C3N(C)c4ccccc4N3C)ncnc2s1	nan
	CHEMBL1375768	28270	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	0	8	4.2	CCc1cc2c(SCC(=O)C(C#N)=C3N(C)c4ccccc4N3C)ncnc2s1	nan
	1049792	28321	21	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	0	5	5.0	COc1ccc(-c2cc(-c3ccc(OC)cc3)c(C#N)c(SC)n2)cc1	nan
	CHEMBL1376368	28321	21	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	0	5	5.0	COc1ccc(-c2cc(-c3ccc(OC)cc3)c(C#N)c(SC)n2)cc1	nan
	3141909	28326	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	2	0	4	3.0	Cc1cccc2cc(C#N)c(SCC#N)nc12	nan
	CHEMBL1376381	28326	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	2	0	4	3.0	Cc1cccc2cc(C#N)c(SCC#N)nc12	nan
	1086373	28379	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	1	6	3.6	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCc3ccco3)n2)c1	nan
	CHEMBL1376846	28379	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	1	6	3.6	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCc3ccco3)n2)c1	nan
	16024493	28468	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	5	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1377756	28468	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	5	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	16018882	28474	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	1	5	4.2	CCOc1ccc(N(CC)S(=O)(=O)N2CCCC(C(=O)Nc3ccc(OC)c(Cl)c3)C2)cc1	nan
	CHEMBL1377806	28474	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	1	5	4.2	CCOc1ccc(N(CC)S(=O)(=O)N2CCCC(C(=O)Nc3ccc(OC)c(Cl)c3)C2)cc1	nan
	2426511	28541	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	0	0	4	2.7	Cc1cc(=O)n2c(sc3ccccc32)c1C#N	nan
	CHEMBL1378393	28541	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	0	0	4	2.7	Cc1cc(=O)n2c(sc3ccccc32)c1C#N	nan
	2060585	28556	61	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	1	2	1.4	O=C(c1ccccc1Cl)N1CCNCC1	nan
	CHEMBL1378602	28556	61	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	1	2	1.4	O=C(c1ccccc1Cl)N1CCNCC1	nan
	54680441	28630	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	3	4	2.6	O=C(NCc1ccccc1)c1c(O)nc2ccccc2c1O	nan
	CHEMBL1379243	28630	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	3	4	2.6	O=C(NCc1ccccc1)c1c(O)nc2ccccc2c1O	nan
	7502810	28688	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	3.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc(Br)cc3)nn2)no1	nan
	CHEMBL1379696	28688	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	3.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc(Br)cc3)nn2)no1	nan
	663350	28748	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	9	2.9	COc1cc(OC)c(-c2nn3c(-c4cccnc4)nnc3s2)cc1OC	nan
	CHEMBL1380292	28748	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	9	2.9	COc1cc(OC)c(-c2nn3c(-c4cccnc4)nnc3s2)cc1OC	nan
	551775	28842	13	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	0	5	4.0	CCN(CC)C(=O)CSc1nc(C)cc(-c2cccs2)c1C#N	nan
	CHEMBL1380940	28842	13	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	0	5	4.0	CCN(CC)C(=O)CSc1nc(C)cc(-c2cccs2)c1C#N	nan
	6470016	28978	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	2	2	3.4	CC1=C(C)CC(C(=O)NCc2cccc(Cl)c2)C(C(=O)O)C1	nan
	CHEMBL1382205	28978	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	2	2	3.4	CC1=C(C)CC(C(=O)NCc2cccc(Cl)c2)C(C(=O)O)C1	nan
	4908628	28987	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	4	3.4	Cc1ccc(S(=O)(=O)N(C)Cc2cc3cc(C)ccc3nc2O)cc1	nan
	CHEMBL1382276	28987	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	4	3.4	Cc1ccc(S(=O)(=O)N(C)Cc2cc3cc(C)ccc3nc2O)cc1	nan
	1450725	28990	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	0	7	1.8	N#Cc1cc2cc3c(cc2nc1SCC(=O)N1CCOCC1)OCO3	nan
	CHEMBL1382288	28990	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	0	7	1.8	N#Cc1cc2cc3c(cc2nc1SCC(=O)N1CCOCC1)OCO3	nan
	5155717	29147	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	5	2.1	NS(=O)(=O)c1ccc(CCn2c(=S)[nH]c3ccc(F)cc3c2=O)cc1	nan
	CHEMBL1383680	29147	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	5	2.1	NS(=O)(=O)c1ccc(CCn2c(=S)[nH]c3ccc(F)cc3c2=O)cc1	nan
	1271521	29341	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	O=C(Nc1ccc(-c2noc(-c3ccccc3F)n2)cc1)c1cccs1	nan
	CHEMBL1385411	29341	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	O=C(Nc1ccc(-c2noc(-c3ccccc3F)n2)cc1)c1cccs1	nan
	1604314	29479	12	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	6	3.6	CCOC(=O)C1=C(c2ccccc2)O/C(=C(/C(=O)OC)C(F)(F)F)S1	nan
	CHEMBL1386476	29479	12	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	6	3.6	CCOC(=O)C1=C(c2ccccc2)O/C(=C(/C(=O)OC)C(F)(F)F)S1	nan
	2815677	29495	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	0	6	1.5	CCOC(=O)c1cn2nc(N3CCCC3)ccc2n1	nan
	CHEMBL1386622	29495	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	0	6	1.5	CCOC(=O)c1cn2nc(N3CCCC3)ccc2n1	nan
	979520	29617	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	4	4.5	COc1cc(CNCc2ccccc2Cl)ccc1OCC(=O)NC1CCCCC1	nan
	CHEMBL1387627	29617	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	4	4.5	COc1cc(CNCc2ccccc2Cl)ccc1OCC(=O)NC1CCCCC1	nan
	855469	29653	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	3.4	Cc1cc(NC(=O)CSc2nc3c(C)cccc3cc2C#N)no1	nan
	CHEMBL1387916	29653	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	3.4	Cc1cc(NC(=O)CSc2nc3c(C)cccc3cc2C#N)no1	nan
	1026561	29664	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	2	3	4.5	CCOc1ccc(Br)cc1C(=O)Nc1ccc(C(=O)NCC(C)C)cc1	nan
	CHEMBL1388002	29664	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	2	3	4.5	CCOc1ccc(Br)cc1C(=O)Nc1ccc(C(=O)NCC(C)C)cc1	nan
	2372910	29709	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	0	5	3.3	c1ccc(-c2cc(-c3nnco3)c3ccccc3n2)nc1	nan
	CHEMBL1388328	29709	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	0	5	3.3	c1ccc(-c2cc(-c3nnco3)c3ccccc3n2)nc1	nan
	4909035	29949	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	5	4.0	Cc1cccc(-c2nc3c(c(SCC(=O)N4CCCC4)n2)COC(C)(C)C3)c1	nan
	CHEMBL1390262	29949	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	5	4.0	Cc1cccc(-c2nc3c(c(SCC(=O)N4CCCC4)n2)COC(C)(C)C3)c1	nan
	20969169	29976	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	4.1	COc1ccc(Cl)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	CHEMBL1390480	29976	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	4.1	COc1ccc(Cl)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	4688970	29983	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	1	6	4.2	Cc1nc(N2CCOCC2)c2c(C)c(C(=O)Nc3ccc(F)cc3Cl)sc2n1	nan
	CHEMBL1390558	29983	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	1	6	4.2	Cc1nc(N2CCOCC2)c2c(C)c(C(=O)Nc3ccc(F)cc3Cl)sc2n1	nan
	6621188	29987	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	2	4	2.3	CCc1ccc(NC(=O)CNC(=O)Cn2ccc3ccccc3c2=O)cc1	nan
	CHEMBL1390571	29987	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	2	4	2.3	CCc1ccc(NC(=O)CNC(=O)Cn2ccc3ccccc3c2=O)cc1	nan
	24687564	30124	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	7	4.0	CCOC(=O)c1c(NC(=O)COc2ccccc2C#N)sc2c1CC(C)(C)NC2(C)C	nan
	CHEMBL1391818	30124	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	7	4.0	CCOC(=O)c1c(NC(=O)COc2ccccc2C#N)sc2c1CC(C)(C)NC2(C)C	nan
	8030390	30221	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	3.1	Cc1c(C)c2ccc(OCC(=O)Nc3ccccn3)c(C)c2oc1=O	nan
	CHEMBL1392611	30221	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	3.1	Cc1c(C)c2ccc(OCC(=O)Nc3ccccn3)c(C)c2oc1=O	nan
	649622	30291	3	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	CHEMBL1393221	30291	3	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	16024685	30389	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	5	5.2	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)Nc3ccccc3C(F)(F)F)c2n1	nan
	CHEMBL1394039	30389	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	5	5.2	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)Nc3ccccc3C(F)(F)F)c2n1	nan
	3844740	30391	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	3	7	3.8	COc1ccc(C2C=C(c3ccc(Cl)cc3)Nc3nc(NC(=O)CCC(=O)O)nn32)cc1	nan
	CHEMBL1394052	30391	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	3	7	3.8	COc1ccc(C2C=C(c3ccc(Cl)cc3)Nc3nc(NC(=O)CCC(=O)O)nn32)cc1	nan
	16024945	30403	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	O=C(Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)nnn2C1CCCC1	nan
	CHEMBL1394171	30403	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	O=C(Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)nnn2C1CCCC1	nan
	2136700	30410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	3.8	Cc1ccccc1NC(=O)Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2ccccc21	nan
	CHEMBL1394236	30410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	3.8	Cc1ccccc1NC(=O)Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2ccccc21	nan
	16017140	30448	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	5	5.0	Cc1ccc(C)c(NC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	CHEMBL1394852	30448	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	5	5.0	Cc1ccc(C)c(NC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	16022416	30449	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	7	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	CHEMBL1394859	30449	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	7	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	16030605	30456	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCCc2ccccc21	nan
	CHEMBL1394911	30456	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCCc2ccccc21	nan
	16034772	30491	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	6	4.6	Cc1nn(CCCC(=O)Nc2cccc(C(F)(F)F)c2)c(=O)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1395185	30491	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	6	4.6	Cc1nn(CCCC(=O)Nc2cccc(C(F)(F)F)c2)c(=O)c2nn(-c3ccccc3)c(C)c12	nan
	2007143	30495	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	1.9	CCOC(=O)CNC(=O)c1ccc(-c2nn(C)c(=O)c3ccccc23)cc1	nan
	CHEMBL1395237	30495	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	1.9	CCOC(=O)CNC(=O)c1ccc(-c2nn(C)c(=O)c3ccccc23)cc1	nan
	16019606	30496	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccccc2Cl)c2sccc23)cc1	nan
	CHEMBL1395245	30496	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccccc2Cl)c2sccc23)cc1	nan
	16018799	30498	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	5	3.2	CCc1cccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1395272	30498	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	5	3.2	CCc1cccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)c1	nan
	15987986	30517	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	1	4	4.0	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3ccc(C)c(F)c3)c21	nan
	CHEMBL1395557	30517	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	1	4	4.0	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3ccc(C)c(F)c3)c21	nan
	16009626	30531	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	3	5.7	Cc1cc(C)cc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)c1	nan
	CHEMBL1395778	30531	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	3	5.7	Cc1cc(C)cc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)c1	nan
	16017553	30554	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	2.7	O=C(Nc1nnc(S(=O)(=O)N2CCCCC2)s1)c1ccccc1Br	nan
	CHEMBL1396131	30554	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	2.7	O=C(Nc1nnc(S(=O)(=O)N2CCCCC2)s1)c1ccccc1Br	nan
	16033012	30579	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	4	0	7	3.3	O=C(Cn1c(=O)n2nc(-c3cccc(F)c3)nc2c2ccccc21)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1396543	30579	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	4	0	7	3.3	O=C(Cn1c(=O)n2nc(-c3cccc(F)c3)nc2c2ccccc21)N1CCN(c2ccccc2F)CC1	nan
	15989006	30586	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	8	3.5	O=C(CCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1396634	30586	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	8	3.5	O=C(CCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	16009460	30609	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	3.6	COc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1OC	nan
	CHEMBL1396932	30609	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	3.6	COc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1OC	nan
	3408184	30620	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	5	5.8	CCOc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	CHEMBL1397049	30620	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	5	5.8	CCOc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	4345038	30625	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	3	5.2	CN(Cc1ccccc1)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(Cl)c2Cl)c1	nan
	CHEMBL1397130	30625	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	3	5.2	CN(Cc1ccccc1)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(Cl)c2Cl)c1	nan
	16017005	30627	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.9	CCOc1ccc(NC(=O)C(=O)c2cc(C)n(-c3cc(C)cc(C)c3)c2C)cc1	nan
	CHEMBL1397170	30627	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.9	CCOc1ccc(NC(=O)C(=O)c2cc(C)n(-c3cc(C)cc(C)c3)c2C)cc1	nan
	16009843	30689	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	1	6	3.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1398005	30689	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	1	6	3.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	15988021	30705	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	12	2	10	1.0	COCCNC(=O)CCn1c(=O)c2cc(OC)c(OC)cc2n(CC(=O)Nc2ccccc2OC)c1=O	nan
	CHEMBL1398191	30705	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	12	2	10	1.0	COCCNC(=O)CCn1c(=O)c2cc(OC)c(OC)cc2n(CC(=O)Nc2ccccc2OC)c1=O	nan
	2288826	30888	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	3	4	0.6	O=C1NC(=O)C(=CNc2cc(F)cc(F)c2)C(=O)N1	nan
	CHEMBL1400030	30888	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	3	4	0.6	O=C1NC(=O)C(=CNc2cc(F)cc(F)c2)C(=O)N1	nan
	16009302	30972	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.7	Cn1c2ccccc2c2cnn(CC(=O)Nc3ccccc3F)c(=O)c21	nan
	CHEMBL1400803	30972	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.7	Cn1c2ccccc2c2cnn(CC(=O)Nc3ccccc3F)c(=O)c21	nan
	16010052	30986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	5	4.9	COc1ccc(CCNC(=O)Cn2c(-c3cccs3)cc3cc(F)ccc32)cc1OC	nan
	CHEMBL1400938	30986	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	5	4.9	COc1ccc(CCNC(=O)Cn2c(-c3cccs3)cc3cc(F)ccc32)cc1OC	nan
	16022925	31127	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	0	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)N(C)Cc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1402121	31127	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	0	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)N(C)Cc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	3238641	31175	35	None	-354	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	5	1	3	3.0	COc1ccc(OCc2cccc(C(=O)O)c2)cc1	nan
	CHEMBL1402510	31175	35	None	-354	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	5	1	3	3.0	COc1ccc(OCc2cccc(C(=O)O)c2)cc1	nan
	24792811	31186	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	5	4.4	Cc1cccc(N2CCN(c3ccc4cc(S(=O)(=O)N5CCCCC5)ccc4n3)CC2C)c1	nan
	CHEMBL1402620	31186	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	5	4.4	Cc1cccc(N2CCN(c3ccc4cc(S(=O)(=O)N5CCCCC5)ccc4n3)CC2C)c1	nan
	13020032	31222	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	5	2.9	COc1ccc(C[C@H]2c3cc(O)c(OC)cc3CC[N+]2(C)[O-])cc1O	nan
	CHEMBL1402907	31222	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	5	2.9	COc1ccc(C[C@H]2c3cc(O)c(OC)cc3CC[N+]2(C)[O-])cc1O	nan
	3456065	31226	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	4	4.8	Oc1nnc(Cc2ccc(-c3ccc(Cl)cc3)o2)c2ccccc12	nan
	CHEMBL1402979	31226	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	4	4.8	Oc1nnc(Cc2ccc(-c3ccc(Cl)cc3)o2)c2ccccc12	nan
	807671	31263	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	2	4	2.7	Cc1nc(NC(=O)c2ccccc2O)sc1C	nan
	CHEMBL1403354	31263	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	2	4	2.7	Cc1nc(NC(=O)c2ccccc2O)sc1C	nan
	24979173	31303	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	3.2	COc1ccccc1NC(=O)COC(=O)c1ccccc1SCC(=O)N1CCCC1	nan
	CHEMBL1403792	31303	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	3.2	COc1ccccc1NC(=O)COC(=O)c1ccccc1SCC(=O)N1CCCC1	nan
	1300573	31313	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	4.7	Cc1cccc(NC(=O)Cn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)c1	nan
	CHEMBL1403862	31313	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	4.7	Cc1cccc(NC(=O)Cn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)c1	nan
	3176404	31363	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	5	2	3	3.9	Cc1cccc(CCNCc2cc3cccc(C)c3nc2O)c1	nan
	CHEMBL1404217	31363	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	5	2	3	3.9	Cc1cccc(CCNCc2cc3cccc(C)c3nc2O)c1	nan
	2941406	31420	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	1	2	5	4.2	Cc1c(C#N)c(N)nc2c3c(sc12)NC(=O)CC3c1ccc(Cl)cc1	nan
	CHEMBL1404915	31420	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	1	2	5	4.2	Cc1c(C#N)c(N)nc2c3c(sc12)NC(=O)CC3c1ccc(Cl)cc1	nan
	663707	31505	14	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	4	4.8	Fc1ccc(CSc2ncnc3c2oc2ccccc23)cc1	nan
	CHEMBL1405769	31505	14	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	4	4.8	Fc1ccc(CSc2ncnc3c2oc2ccccc23)cc1	nan
	3207570	31514	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.1	CCc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1405871	31514	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.1	CCc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	2102520	31668	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	1	7	5.0	COc1cc(C(=O)Nc2nc3ccc(C)cc3s2)ccc1OCc1c(C)noc1C	nan
	CHEMBL1407262	31668	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	1	7	5.0	COc1cc(C(=O)Nc2nc3ccc(C)cc3s2)ccc1OCc1c(C)noc1C	nan
	672442	31753	15	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	5	3.3	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccc(Cl)cc1	nan
	CHEMBL1407760	31753	15	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	5	3.3	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccc(Cl)cc1	nan
	15989447	31764	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	1	5	4.1	O=C(CCCn1c(=O)c2ccccc2n(Cc2cccc(F)c2)c1=O)NCc1ccccc1Cl	nan
	CHEMBL1407901	31764	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	1	5	4.1	O=C(CCCn1c(=O)c2ccccc2n(Cc2cccc(F)c2)c1=O)NCc1ccccc1Cl	nan
	5524322	31800	16	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	4.5	CSc1nsc(/C=C/Nc2cccc(Cl)c2)c1C#N	nan
	CHEMBL1408147	31800	16	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	4.5	CSc1nsc(/C=C/Nc2cccc(Cl)c2)c1C#N	nan
	135454349	31884	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	2	6	2.6	CCc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	CHEMBL1408793	31884	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	2	6	2.6	CCc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	16012616	31934	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccccc5F)s4)c3nc12	nan
	CHEMBL1409190	31934	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccccc5F)s4)c3nc12	nan
	16026074	31991	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.1	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccccc2C)CC1	nan
	CHEMBL1409660	31991	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.1	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccccc2C)CC1	nan
	5294544	32000	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	1	1	4	2.4	CCn1c(=S)[nH]c2nc3c(cc2c1=O)CCCC3	nan
	CHEMBL1409738	32000	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	1	1	4	2.4	CCn1c(=S)[nH]c2nc3c(cc2c1=O)CCCC3	nan
	3208202	32042	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	3	7	3.3	CCc1cc2c(C)ccc(C)c2nc1SCC(=O)Nc1cnc(O)nc1O	nan
	CHEMBL1410014	32042	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	3	7	3.3	CCc1cc2c(C)ccc(C)c2nc1SCC(=O)Nc1cnc(O)nc1O	nan
	2136000	32051	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1410088	32051	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	2056596	32165	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	2	5	2.6	CCn1ncc(Br)c1C(=O)Nc1sc2c(c1C(N)=O)CCC2	nan
	CHEMBL1411085	32165	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	2	5	2.6	CCn1ncc(Br)c1C(=O)Nc1sc2c(c1C(N)=O)CCC2	nan
	15988949	32179	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(NC(=O)Cn2c(=O)n(CCCCCC(=O)NCc3ccc(F)cc3)c(=O)c3sccc32)cc1C	nan
	CHEMBL1411183	32179	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(NC(=O)Cn2c(=O)n(CCCCCC(=O)NCc3ccc(F)cc3)c(=O)c3sccc32)cc1C	nan
	4390376	32208	3	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1	nan
	CHEMBL1411409	32208	3	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1	nan
	627327	32268	30	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	0	3	3.6	O=c1oc(-c2ccc(Br)cc2)nc2ccccc12	nan
	CHEMBL1411919	32268	30	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	0	3	3.6	O=c1oc(-c2ccc(Br)cc2)nc2ccccc12	nan
	16017002	32306	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.8	CCOc1ccc(CNC(=O)C(C)n2ncn3cccc3c2=O)cc1	nan
	CHEMBL1412238	32306	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.8	CCOc1ccc(CNC(=O)C(C)n2ncn3cccc3c2=O)cc1	nan
	16026072	32355	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	5	4.2	CCOc1ccccc1CNC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	CHEMBL1412601	32355	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	5	4.2	CCOc1ccccc1CNC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	646655	32366	3	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1412670	32366	3	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	1246434	32370	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	5	4.7	O=C(Nc1nnc(C2CCCCC2)s1)c1ccc(Br)s1	nan
	CHEMBL1412704	32370	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	5	4.7	O=C(Nc1nnc(C2CCCCC2)s1)c1ccc(Br)s1	nan
	1952877	32390	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	2	5	2.0	Cc1cc(C)c2oc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)cc(=O)c2c1	nan
	CHEMBL1412873	32390	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	2	5	2.0	Cc1cc(C)c2oc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)cc(=O)c2c1	nan
	16017227	32414	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	6	2.2	Cc1nn(CC(=O)N2CCN(c3cccc(C(F)(F)F)c3)CC2)c(=O)c2cccn12	nan
	CHEMBL1413003	32414	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	6	2.2	Cc1nn(CC(=O)N2CCN(c3cccc(C(F)(F)F)c3)CC2)c(=O)c2cccn12	nan
	15996885	32421	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1cccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)c1	nan
	CHEMBL1413061	32421	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1cccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)c1	nan
	2314879	32469	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	6	3.3	CCCCn1c2nc3ccccc3nc2c2c(=N)oc(C)nc21	nan
	CHEMBL1413521	32469	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	6	3.3	CCCCn1c2nc3ccccc3nc2c2c(=N)oc(C)nc21	nan
	694926	32484	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	1	5	3.3	Cc1cccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c1	nan
	CHEMBL1413648	32484	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	1	5	3.3	Cc1cccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c1	nan
	16025383	32594	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	6	4.4	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)NCCc1ccccc1	nan
	CHEMBL1414539	32594	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	6	4.4	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)NCCc1ccccc1	nan
	16010143	32659	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	3	5.6	Cc1ccc(Cn2c(C(=O)NCc3ccccc3Cl)cc3sccc32)cc1	nan
	CHEMBL1415124	32659	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	3	5.6	Cc1ccc(Cn2c(C(=O)NCc3ccccc3Cl)cc3sccc32)cc1	nan
	663372	32661	14	None	-14	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	4	4.2	Cc1ccc(C2CC(=O)c3cnc(N4CC(C)CC(C)C4)nc3C2)cc1	nan
	CHEMBL1415139	32661	14	None	-14	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	4	4.2	Cc1ccc(C2CC(=O)c3cnc(N4CC(C)CC(C)C4)nc3C2)cc1	nan
	16029519	32672	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	5	0	6	2.9	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3cccc(Cl)c3)CC1)CCS2	nan
	CHEMBL1415234	32672	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	5	0	6	2.9	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3cccc(Cl)c3)CC1)CCS2	nan
	1088534	32706	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	1	4	3.9	CCOc1ccc(NC(=O)Cn2cc(C(C)=O)c3ccccc32)cc1	nan
	CHEMBL1415529	32706	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	1	4	3.9	CCOc1ccc(NC(=O)Cn2cc(C(C)=O)c3ccccc32)cc1	nan
	2701522	32729	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	6	1	6	2.8	CCSc1nnc(NC(=O)Cc2ccccc2OC)s1	nan
	CHEMBL1415759	32729	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	6	1	6	2.8	CCSc1nnc(NC(=O)Cc2ccccc2OC)s1	nan
	20880977	32833	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	8	2.5	O=C(CCc1nnc2n(Cc3ccc(Cl)cc3)c(=O)c3ccccc3n12)NCCCN1CCOCC1	nan
	CHEMBL1416665	32833	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	8	2.5	O=C(CCc1nnc2n(Cc3ccc(Cl)cc3)c(=O)c3ccccc3n12)NCCCN1CCOCC1	nan
	16025415	32850	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	1	6	5.5	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)c1	nan
	CHEMBL1416823	32850	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	1	6	5.5	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)c1	nan
	24792644	32986	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.8	CN(C)c1ccc(-c2ccc3c(=O)c4ccccc4n(C)c3c2)cn1	nan
	CHEMBL1417964	32986	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.8	CN(C)c1ccc(-c2ccc3c(=O)c4ccccc4n(C)c3c2)cn1	nan
	16030529	33001	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	0	4	5.8	CCN(C(=O)CSc1nc2ccccc2nc1Cc1ccc(F)cc1)c1cccc(C)c1	nan
	CHEMBL1418101	33001	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	0	4	5.8	CCN(C(=O)CSc1nc2ccccc2nc1Cc1ccc(F)cc1)c1cccc(C)c1	nan
	1936615	33064	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	7	4.5	CC1(C)Cc2nc3sc4c(SCC(=O)NCc5ccccc5)ncnc4c3cc2CO1	nan
	CHEMBL1418632	33064	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	7	4.5	CC1(C)Cc2nc3sc4c(SCC(=O)NCc5ccccc5)ncnc4c3cc2CO1	nan
	3574260	33137	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	CHEMBL1419267	33137	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	5069803	33602	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	4	2.2	CC(C)C(=O)N1CCN(CCN2C(=O)c3cccc4cccc(c34)C2=O)CC1	nan
	CHEMBL1423181	33602	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	4	2.2	CC(C)C(=O)N1CCN(CCN2C(=O)c3cccc4cccc(c34)C2=O)CC1	nan
	4298772	33662	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	3	1	4	2.8	Cc1ccc(NC(=O)c2ccc(-n3cccn3)nc2)cc1	nan
	CHEMBL1423637	33662	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	3	1	4	2.8	Cc1ccc(NC(=O)c2ccc(-n3cccn3)nc2)cc1	nan
	135521903	33725	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1ccc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)cc1Cl	nan
	CHEMBL1424164	33725	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1ccc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)cc1Cl	nan
	5009230	34003	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	1	3	4.6	O=c1c2ccc(Cl)cc2[nH]c(=S)n1CCC1=CCCCC1	nan
	CHEMBL1426475	34003	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	1	3	4.6	O=c1c2ccc(Cl)cc2[nH]c(=S)n1CCC1=CCCCC1	nan
	1004501	34019	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	8	1	6	5.8	COc1ccc(-c2cc(-c3cccs3)c(C#N)c(SCC(=O)NCc3ccccc3)n2)cc1	nan
	CHEMBL1426581	34019	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	8	1	6	5.8	COc1ccc(-c2cc(-c3cccs3)c(C#N)c(SCC(=O)NCc3ccccc3)n2)cc1	nan
	1398121	34042	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	4	5.1	Cc1nc(Nc2ccccc2)c2oc3ccc(Cl)cc3c2n1	nan
	CHEMBL1426816	34042	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	4	5.1	Cc1nc(Nc2ccccc2)c2oc3ccc(Cl)cc3c2n1	nan
	2916457	34101	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	0	4	2.1	O=C1c2nc3ccccn3c2C(=O)N1Cc1ccccc1	nan
	CHEMBL1427322	34101	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	0	4	2.1	O=C1c2nc3ccccn3c2C(=O)N1Cc1ccccc1	nan
	2785858	34341	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	0	5	0.8	Cn1c(=O)c2cc3ccccc3nc2n(C)c1=O	nan
	CHEMBL1429441	34341	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	0	5	0.8	Cn1c(=O)c2cc3ccccc3nc2n(C)c1=O	nan
	1474449	34589	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	5	3.8	Nc1c(-c2cccs2)cnc2c(-c3ccc(F)cc3)cnn12	nan
	CHEMBL1431364	34589	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	5	3.8	Nc1c(-c2cccs2)cnc2c(-c3ccc(F)cc3)cnn12	nan
	22548378	34594	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	6	2.0	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3cc4c(cc3C)NC(=O)CO4)CC2)cc1	nan
	CHEMBL1431452	34594	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	6	2.0	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3cc4c(cc3C)NC(=O)CO4)CC2)cc1	nan
	3239990	34650	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	3	0	7	3.1	CCOC(=O)N1CCN(C(=O)c2nn(-c3ccc(C)cc3)c(=O)c3c2c2ccccc2n3C)CC1	nan
	CHEMBL1431956	34650	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	3	0	7	3.1	CCOC(=O)N1CCN(C(=O)c2nn(-c3ccc(C)cc3)c(=O)c3c2c2ccccc2n3C)CC1	nan
	1480466	34669	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2cccnc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1432166	34669	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2cccnc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	24792375	34690	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	2.5	COc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1432321	34690	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	2.5	COc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	1049756	34820	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	5	4.3	COc1ccccc1NC(=O)c1c(NC(=O)c2ccco2)sc2c1CCC2	nan
	CHEMBL1433354	34820	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	5	4.3	COc1ccccc1NC(=O)c1c(NC(=O)c2ccco2)sc2c1CCC2	nan
	2227785	34832	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	7	5.3	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1cc(OC)c(OC)c(OC)c1	nan
	CHEMBL1433437	34832	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	7	5.3	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1cc(OC)c(OC)c(OC)c1	nan
	16027247	34844	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	4.9	COc1ccc2ncc3c(-c4ccc(C)c(C)c4)nn(CC(=O)NC4CCCC4)c3c2c1	nan
	CHEMBL1433603	34844	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	4.9	COc1ccc2ncc3c(-c4ccc(C)c(C)c4)nn(CC(=O)NC4CCCC4)c3c2c1	nan
	16024617	34865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	7	1	6	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)c(Cl)c3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1433920	34865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	7	1	6	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)c(Cl)c3)c3nc(C)ccc3c2=O)cc1	nan
	16019055	34884	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccccc1CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1434234	34884	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccccc1CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2135389	34887	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	6	4.0	COc1cccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc(OC)ccc32)c1	nan
	CHEMBL1434264	34887	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	6	4.0	COc1cccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc(OC)ccc32)c1	nan
	16026966	34893	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1434365	34893	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	16021030	34904	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	3	5.9	CC(CNC(=O)Cn1c(-c2cccs2)cc2cc(Cl)ccc21)c1ccccc1	nan
	CHEMBL1434633	34904	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	3	5.9	CC(CNC(=O)Cn1c(-c2cccs2)cc2cc(Cl)ccc21)c1ccccc1	nan
	2134800	34938	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	9	1	7	4.1	COCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1435016	34938	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	9	1	7	4.1	COCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	16022354	34965	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	6	4.9	Cc1ccc(Cn2c(SCC(=O)NCc3ccc(Cl)cc3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1435272	34965	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	6	4.9	Cc1ccc(Cn2c(SCC(=O)NCc3ccc(Cl)cc3)nc3ccsc3c2=O)cc1	nan
	16022956	35005	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.7	Cc1nnc(N2CCC(C(=O)NCCc3ccccc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1435842	35005	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.7	Cc1nnc(N2CCC(C(=O)NCCc3ccccc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	16015098	35006	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.5	Cc1nc(SCC(=O)Nc2ccccc2C)cc(-c2ccccc2)n1	nan
	CHEMBL1435853	35006	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.5	Cc1nc(SCC(=O)Nc2ccccc2C)cc(-c2ccccc2)n1	nan
	16024515	35010	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	4.5	COc1ccc(Cl)cc1NC(=O)Cn1cc(C(=O)c2ccc(C)cc2)c(=O)c2ccc(C)nc21	nan
	CHEMBL1435881	35010	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	4.5	COc1ccc(Cl)cc1NC(=O)Cn1cc(C(=O)c2ccc(C)cc2)c(=O)c2ccc(C)nc21	nan
	16025955	35019	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccccc1Cl)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1436007	35019	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccccc1Cl)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	15988055	35041	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	2	1	8	3.4	Cc1cccc(C)c1Nc1nn2c(=O)c3cc4c(cc3nc2s1)OCO4	nan
	CHEMBL1436214	35041	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	2	1	8	3.4	Cc1cccc(C)c1Nc1nn2c(=O)c3cc4c(cc3nc2s1)OCO4	nan
	1166237	35052	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	7	5.4	CCOc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)cc1	nan
	CHEMBL1436413	35052	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	7	5.4	CCOc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)cc1	nan
	4076476	35070	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1cccc(C(=O)Nc2c(C(=O)c3ccc(F)cc3)oc3ccccc23)c1	nan
	CHEMBL1436707	35070	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1cccc(C(=O)Nc2c(C(=O)c3ccc(F)cc3)oc3ccccc23)c1	nan
	16012965	35077	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	3	5.3	CCCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	CHEMBL1436801	35077	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	3	5.3	CCCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	16031323	35082	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	8	1	8	3.7	COc1cc(-c2cc3n(C)c(C)c(CCC(=O)Nc4ccc(F)cc4)c(=O)n3n2)cc(OC)c1OC	nan
	CHEMBL1436894	35082	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	8	1	8	3.7	COc1cc(-c2cc3n(C)c(C)c(CCC(=O)Nc4ccc(F)cc4)c(=O)n3n2)cc(OC)c1OC	nan
	3533132	35159	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	3.3	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cncc(Br)c1	nan
	CHEMBL1437784	35159	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	3.3	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cncc(Br)c1	nan
	4650106	35201	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	2	5	4.2	O=C(NCc1cccnc1)c1ccc(Cn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	CHEMBL1438098	35201	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	2	5	4.2	O=C(NCc1cccnc1)c1ccc(Cn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	959085	35287	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	4	3.5	CC(=O)c1sc(NC(=O)c2ccc(C)c(C)c2)nc1C	nan
	CHEMBL1438925	35287	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	4	3.5	CC(=O)c1sc(NC(=O)c2ccc(C)c(C)c2)nc1C	nan
	16026319	35308	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(C)c(F)c4)c32)cc1	nan
	CHEMBL1439096	35308	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(C)c(F)c4)c32)cc1	nan
	16015553	35310	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	2	6	5.2	Cc1ccc(NC(=O)CSc2nc3ccc(NC(=O)c4ccco4)cc3s2)cc1	nan
	CHEMBL1439122	35310	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	2	6	5.2	Cc1ccc(NC(=O)CSc2nc3ccc(NC(=O)c4ccco4)cc3s2)cc1	nan
	15988982	35431	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	524	8	2	7	3.8	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(CCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1440158	35431	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	524	8	2	7	3.8	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(CCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	2137007	35670	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.8	COCCNc1nc2c(S(=O)(=O)c3cc(C)ccc3C)nnn2c2ccccc12	nan
	CHEMBL1442335	35670	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.8	COCCNc1nc2c(S(=O)(=O)c3cc(C)ccc3C)nnn2c2ccccc12	nan
	3156591	35688	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	3.0	CCCNS(=O)(=O)c1cc(-c2nnc3c4ccccc4c(C)nn23)ccc1OC	nan
	CHEMBL1442508	35688	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	3.0	CCCNS(=O)(=O)c1cc(-c2nnc3c4ccccc4c(C)nn23)ccc1OC	nan
	16009539	35728	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4F)cc3)cc(=O)n12	nan
	CHEMBL1442799	35728	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4F)cc3)cc(=O)n12	nan
	1119348	35746	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	0	6	4.2	COc1cccc2cc(-c3nnc(-c4ccc(Cl)cc4)o3)c(=O)oc12	nan
	CHEMBL1443005	35746	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	0	6	4.2	COc1cccc2cc(-c3nnc(-c4ccc(Cl)cc4)o3)c(=O)oc12	nan
	3456574	35926	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	2	5	1.8	COCCn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	CHEMBL1444789	35926	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	2	5	1.8	COCCn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	15987577	35942	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.3	Cc1cc(Cl)ccc1OCC(=O)Nc1c(Cl)ccc2nsnc12	nan
	CHEMBL1444928	35942	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.3	Cc1cc(Cl)ccc1OCC(=O)Nc1c(Cl)ccc2nsnc12	nan
	1529015	35944	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	5.3	CCOC(=O)c1c(-c2ccc(C)s2)csc1NC(=O)c1cccs1	nan
	CHEMBL1444931	35944	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	5.3	CCOC(=O)c1c(-c2ccc(C)s2)csc1NC(=O)c1cccs1	nan
	3238506	35977	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	7	3.0	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3nc4ccccc4s3)cc2)CC1	nan
	CHEMBL1445199	35977	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	7	3.0	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3nc4ccccc4s3)cc2)CC1	nan
	629629	35994	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	3	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccccc3)nc(-c3ccccc3)n2)cc1	nan
	CHEMBL1445350	35994	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	3	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccccc3)nc(-c3ccccc3)n2)cc1	nan
	16008367	36021	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	1	6	4.6	COc1cc(OC)c(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1Cl	nan
	CHEMBL1445604	36021	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	1	6	4.6	COc1cc(OC)c(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1Cl	nan
	16031877	36048	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	4.0	CCOC(=O)C1CCCN(Cc2cn3c(-c4ccc(Br)cc4)nnc3s2)C1	nan
	CHEMBL1445888	36048	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	4.0	CCOC(=O)C1CCCN(Cc2cn3c(-c4ccc(Br)cc4)nnc3s2)C1	nan
	3116123	36068	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	CHEMBL1446094	36068	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	3462774	36104	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	2	5	3.6	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	CHEMBL1446438	36104	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	2	5	3.6	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	1478332	36333	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.1	CCOC(=O)c1cc2c(=O)c3cc(C)ccc3oc2nc1C	nan
	CHEMBL1448380	36333	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.1	CCOC(=O)c1cc2c(=O)c3cc(C)ccc3oc2nc1C	nan
	15990626	36360	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	6.1	CCOc1ccc2ncc3c(-c4ccc(C)cc4)nn(-c4cccc(F)c4)c3c2c1	nan
	CHEMBL1448570	36360	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	6.1	CCOc1ccc2ncc3c(-c4ccc(C)cc4)nn(-c4cccc(F)c4)c3c2c1	nan
	16007612	36396	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	1	5	3.8	Cc1ccc(CCNC(=O)c2cn(C)c3ccc(S(=O)(=O)N(C)C4CCCCC4)cc3c2=O)cc1	nan
	CHEMBL1448823	36396	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	1	5	3.8	Cc1ccc(CCNC(=O)c2cn(C)c3ccc(S(=O)(=O)N(C)C4CCCCC4)cc3c2=O)cc1	nan
	2201274	36438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	6	3.5	COc1cccc(-c2nnc(NC(=O)Cc3cccs3)s2)c1	nan
	CHEMBL1449110	36438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	6	3.5	COc1cccc(-c2nnc(NC(=O)Cc3cccs3)s2)c1	nan
	16017301	36611	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	7	3.2	CC(C)CN(c1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2ccco2)s1	nan
	CHEMBL1450497	36611	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	7	3.2	CC(C)CN(c1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2ccco2)s1	nan
	3646626	36628	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	5.3	CC(C)OCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1450646	36628	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	5.3	CC(C)OCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	1389502	36678	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	1	3	4.0	O=C(Nc1cc(Cl)cc(Cl)c1)c1coc(=O)c(Br)c1	nan
	CHEMBL1451156	36678	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	1	3	4.0	O=C(Nc1cc(Cl)cc(Cl)c1)c1coc(=O)c(Br)c1	nan
	653554	36736	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(-c3ccccc3)c(=O)c2c1C	nan
	CHEMBL1451583	36736	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(-c3ccccc3)c(=O)c2c1C	nan
	135476823	36740	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	2.7	Cc1cccc(-n2c(SCC(=O)N3CCCC3)nc3nnc(C)c-3c2N)c1	nan
	CHEMBL1451599	36740	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	2.7	Cc1cccc(-n2c(SCC(=O)N3CCCC3)nc3nnc(C)c-3c2N)c1	nan
	2029273	36827	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	6	5.2	COc1cccc(-c2ccc(-c3noc(-c4ccccc4Br)n3)c(OC)n2)c1	nan
	CHEMBL1452203	36827	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	6	5.2	COc1cccc(-c2ccc(-c3noc(-c4ccccc4Br)n3)c(OC)n2)c1	nan
	5058847	36838	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	CHEMBL1452293	36838	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	16027444	36868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	CHEMBL1452550	36868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	4256434	37031	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	5.1	Cc1ccc(-c2nc(NC(=O)CSc3cc(C)c4ccccc4n3)ns2)cc1	nan
	CHEMBL1453902	37031	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	5.1	Cc1ccc(-c2nc(NC(=O)CSc3cc(C)c4ccccc4n3)ns2)cc1	nan
	16008459	37037	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	0	4	4.8	CCOc1ccc2c(c1)c(=O)c(C(=O)c1ccccc1)cn2Cc1ccccc1F	nan
	CHEMBL1453936	37037	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	0	4	4.8	CCOc1ccc2c(c1)c(=O)c(C(=O)c1ccccc1)cn2Cc1ccccc1F	nan
	991456	37062	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	4	4.1	COc1ccc(C(=O)Nc2ccc(Cl)cc2C(=O)NCc2ccco2)cc1	nan
	CHEMBL1454096	37062	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	4	4.1	COc1ccc(C(=O)Nc2ccc(Cl)cc2C(=O)NCc2ccco2)cc1	nan
	808336	37130	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	0	6	1.8	Cc1ccc(-c2nn3c(=O)c(C)nnc3s2)cc1	nan
	CHEMBL1454681	37130	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	0	6	1.8	Cc1ccc(-c2nn3c(=O)c(C)nnc3s2)cc1	nan
	16017701	37133	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	3.9	CCC(Sc1nc2nccnc2c(=O)n1Cc1ccc(C)cc1)C(=O)NC1CCCCC1	nan
	CHEMBL1454690	37133	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	3.9	CCC(Sc1nc2nccnc2c(=O)n1Cc1ccc(C)cc1)C(=O)NC1CCCCC1	nan
	15988663	37153	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	5	3.9	COc1ccc(OC)c(-c2cc(C(=O)NCc3ccc(Cl)cc3)no2)c1	nan
	CHEMBL1454826	37153	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	5	3.9	COc1ccc(OC)c(-c2cc(C(=O)NCc3ccc(Cl)cc3)no2)c1	nan
	599450	37249	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	1	3	3.6	O=C(Nc1ccc2c(c1)C(=O)OC2)c1ccc(C(F)(F)F)cc1	nan
	CHEMBL1455771	37249	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	1	3	3.6	O=C(Nc1ccc2c(c1)C(=O)OC2)c1ccc(C(F)(F)F)cc1	nan
	3981165	37281	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	5	2.5	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	CHEMBL1456046	37281	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	5	2.5	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	15989547	37296	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	8	1	5	3.6	O=C(CCn1c(=O)c2ccccc2n(Cc2cccc(Cl)c2)c1=O)NCCc1ccccc1	nan
	CHEMBL1456174	37296	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	8	1	5	3.6	O=C(CCn1c(=O)c2ccccc2n(Cc2cccc(Cl)c2)c1=O)NCCc1ccccc1	nan
	16027694	37331	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1456495	37331	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2ccsc2n1	nan
	3242698	37361	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	2	7	4.2	Cc1ccccc1NC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1456820	37361	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	2	7	4.2	Cc1ccccc1NC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	16024703	37414	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1457278	37414	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	7066852	37424	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	2	3	5.8	Cc1ccc2nc(-c3c[nH]c4ccccc34)c(Nc3ccccc3C)n2c1	nan
	CHEMBL1457410	37424	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	2	3	5.8	Cc1ccc2nc(-c3c[nH]c4ccccc34)c(Nc3ccccc3C)n2c1	nan
	16030759	37440	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	0	6	4.4	O=C(c1ccc2c(c1)OCCO2)N(Cc1cccnc1)c1nc2ccc(F)cc2s1	nan
	CHEMBL1457518	37440	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	0	6	4.4	O=C(c1ccc2c(c1)OCCO2)N(Cc1cccnc1)c1nc2ccc(F)cc2s1	nan
	3347951	37446	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.5	CNC(=O)C(Sc1nc(C)nc2c1oc1ccccc12)C(C)=O	nan
	CHEMBL1457585	37446	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.5	CNC(=O)C(Sc1nc(C)nc2c1oc1ccccc12)C(C)=O	nan
	654954	37563	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	3.4	Cc1ccc2nc(SCC(=O)NCc3ccco3)c(C#N)cc2c1	nan
	CHEMBL1458514	37563	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	3.4	Cc1ccc2nc(SCC(=O)NCc3ccco3)c(C#N)cc2c1	nan
	861942	37620	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	0	6	3.7	COc1ccc(OC)c(-c2csc(N(C)C(=O)c3ccco3)n2)c1	nan
	CHEMBL1458992	37620	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	0	6	3.7	COc1ccc(OC)c(-c2csc(N(C)C(=O)c3ccco3)n2)c1	nan
	2570053	37900	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	0	7	1.8	Cc1ccnc2nc(C(=O)OCCOc3ccc(F)cc3)nn12	nan
	CHEMBL1461384	37900	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	0	7	1.8	Cc1ccnc2nc(C(=O)OCCOc3ccc(F)cc3)nn12	nan
	2109478	37926	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	4	1	5	3.9	Cc1cc(NC(=O)COc2ccc3oc4ccccc4c3c2)no1	nan
	CHEMBL1461645	37926	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	4	1	5	3.9	Cc1cc(NC(=O)COc2ccc3oc4ccccc4c3c2)no1	nan
	3243431	37934	7	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	4	5.6	CCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccco3)c(Cl)c2)cc1Br	nan
	CHEMBL1461732	37934	7	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	4	5.6	CCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccco3)c(Cl)c2)cc1Br	nan
	24789924	38025	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1ccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)cc1	nan
	CHEMBL1462423	38025	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1ccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)cc1	nan
	651585	38052	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	7	2.1	COC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	CHEMBL1462713	38052	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	7	2.1	COC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	2134888	38057	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	9	2.4	COc1ccc(C=O)cc1Cn1c(=O)n(CCC(=O)NCc2ccco2)c(=O)c2sccc21	nan
	CHEMBL1462748	38057	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	9	2.4	COc1ccc(C=O)cc1Cn1c(=O)n(CCC(=O)NCc2ccco2)c(=O)c2sccc21	nan
	658551	38352	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	7	2.0	CCCOC(=O)CSc1nc(N)c(C#N)c(CC)c1C#N	nan
	CHEMBL1465062	38352	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	7	2.0	CCCOC(=O)CSc1nc(N)c(C#N)c(CC)c1C#N	nan
	2571531	38377	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	0	10	3.3	CCCCn1c(SCc2cc(=O)n3ccsc3n2)nc2cc(C(=O)OC)ccc2c1=O	nan
	CHEMBL1465204	38377	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	0	10	3.3	CCCCn1c(SCc2cc(=O)n3ccsc3n2)nc2cc(C(=O)OC)ccc2c1=O	nan
	2207742	38379	8	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	6	3.8	CCc1c(C)sc(N=C(S)Nc2nc(C)cc(C)n2)c1C(=O)OC	nan
	CHEMBL1465216	38379	8	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	6	3.8	CCc1c(C)sc(N=C(S)Nc2nc(C)cc(C)n2)c1C(=O)OC	nan
	1299194	38561	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	8	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nnc(-c3cccs3)n2CC)cc1	nan
	CHEMBL1466656	38561	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	8	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nnc(-c3cccs3)n2CC)cc1	nan
	7502637	38615	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	3.3	COc1ccc(-c2ccc(SCC(=O)Nc3nccs3)nn2)cc1OC	nan
	CHEMBL1467089	38615	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	3.3	COc1ccc(-c2ccc(SCC(=O)Nc3nccs3)nn2)cc1OC	nan
	1086372	38631	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	5	4.7	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3cccc(Cl)c3)n2)c1	nan
	CHEMBL1467241	38631	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	5	4.7	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3cccc(Cl)c3)n2)c1	nan
	865458	38642	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	2	0	4	2.8	COc1ccc2nc(SC)c(C#N)cc2c1	nan
	CHEMBL1467309	38642	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	2	0	4	2.8	COc1ccc2nc(SC)c(C#N)cc2c1	nan
	20886167	38936	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.6	COc1cccc(CNC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	CHEMBL1469817	38936	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.6	COc1cccc(CNC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	2045894	38946	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	0	5	4.9	Cc1ccc(-c2nc(=S)c3c(n2Cc2cccnc2)CC(C)(C)OC3)cc1	nan
	CHEMBL1469903	38946	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	0	5	4.9	Cc1ccc(-c2nc(=S)c3c(n2Cc2cccnc2)CC(C)(C)OC3)cc1	nan
	1035368	39067	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	4.2	COc1ccc2nc(NC(=O)CSc3nc4ccccc4o3)sc2c1	nan
	CHEMBL1470920	39067	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	4.2	COc1ccc2nc(NC(=O)CSc3nc4ccccc4o3)sc2c1	nan
	16009198	39245	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1472528	39245	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	15988292	39257	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	586	8	3	6	6.3	COCCCNC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(Cl)cc3)c(-c3ccc(Br)cc3)c2c1N	nan
	CHEMBL1472621	39257	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	586	8	3	6	6.3	COCCCNC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(Cl)cc3)c(-c3ccc(Br)cc3)c2c1N	nan
	16027199	39278	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	3.7	CC(C)NC(=O)C1CCC(Cn2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)CC1	nan
	CHEMBL1472919	39278	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	3.7	CC(C)NC(=O)C1CCC(Cn2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)CC1	nan
	15988974	39282	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	12	2	7	4.6	CCc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc(C)cc2)c(=O)c2sccc21	nan
	CHEMBL1472973	39282	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	12	2	7	4.6	CCc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc(C)cc2)c(=O)c2sccc21	nan
	9505887	39295	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	0	6	2.3	N#Cc1ccc(OC(=O)C2CCN(C3=NS(=O)(=O)c4ccccc43)CC2)cc1	nan
	CHEMBL1473154	39295	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	0	6	2.3	N#Cc1ccc(OC(=O)C2CCN(C3=NS(=O)(=O)c4ccccc43)CC2)cc1	nan
	16021070	39299	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(OC)c(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1473236	39299	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(OC)c(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	7786274	39307	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	5	3.0	O=C(COC(=O)c1cc(Br)ccc1O)Nc1cccnc1Cl	nan
	CHEMBL1473370	39307	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	5	3.0	O=C(COC(=O)c1cc(Br)ccc1O)Nc1cccnc1Cl	nan
	16017273	39322	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	1.7	Cc1nn(CC(=O)Nc2cc(F)ccc2F)c(=O)c2cccn12	nan
	CHEMBL1473495	39322	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	1.7	Cc1nn(CC(=O)Nc2cc(F)ccc2F)c(=O)c2cccn12	nan
	15990603	39358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	5	6.2	CCOC(=O)c1ccc2ncc3c(-c4ccccc4)nn(-c4ccc(F)c(Cl)c4)c3c2c1	nan
	CHEMBL1474033	39358	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	5	6.2	CCOC(=O)c1ccc2ncc3c(-c4ccccc4)nn(-c4ccc(F)c(Cl)c4)c3c2c1	nan
	16015614	39378	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CC(C)C(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	CHEMBL1474414	39378	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CC(C)C(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	16012115	39386	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	3.7	COc1cccc(CNC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)c1	nan
	CHEMBL1474469	39386	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	3.7	COc1cccc(CNC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)c1	nan
	15987618	39405	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	0	4	5.7	CCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1474699	39405	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	0	4	5.7	CCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(C(F)(F)F)c1	nan
	16016392	39406	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	4.9	CC(C)NC(=O)N1[C@H](c2cccs2)[C@@H](C)C(=O)[C@@H](C)[C@@H]1c1cccs1	nan
	CHEMBL1474706	39406	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	4.9	CC(C)NC(=O)N1[C@H](c2cccs2)[C@@H](C)C(=O)[C@@H](C)[C@@H]1c1cccs1	nan
	15989047	39438	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	1	9	3.0	N#Cc1ccccc1Cn1c(=O)n(CCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	CHEMBL1475184	39438	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	1	9	3.0	N#Cc1ccccc1Cn1c(=O)n(CCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	1300955	39464	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1ccc(CNc2ncnc3c2cnn3-c2ccc(Cl)cc2)cc1	nan
	CHEMBL1475511	39464	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1ccc(CNc2ncnc3c2cnn3-c2ccc(Cl)cc2)cc1	nan
	16021946	39496	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	4	0	6	4.8	Cc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1CC(=O)c1ccc(Cl)cc1)n2C	nan
	CHEMBL1475915	39496	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	4	0	6	4.8	Cc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1CC(=O)c1ccc(Cl)cc1)n2C	nan
	16009716	39532	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	6	4.1	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1476522	39532	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	6	4.1	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	2387574	39620	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.0	CCS(=O)(=O)c1ccc2oc(Nc3cc(Cl)ccc3OC)nc2c1	nan
	CHEMBL1477466	39620	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.0	CCS(=O)(=O)c1ccc2oc(Nc3cc(Cl)ccc3OC)nc2c1	nan
	651813	39621	7	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	6	4.1	CCc1nc(SCC(=O)NCc2ccco2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1477471	39621	7	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	6	4.1	CCc1nc(SCC(=O)NCc2ccco2)c2c3c(sc2n1)CCCC3	nan
	135542325	39658	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.0	Cc1nnc2nc(SCC(=O)NC3CCCCC3)n(-c3ccc(Br)cc3)c(N)c1-2	nan
	CHEMBL1477773	39658	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.0	Cc1nnc2nc(SCC(=O)NC3CCCCC3)n(-c3ccc(Br)cc3)c(N)c1-2	nan
	4154279	39675	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	5	5.5	Cc1c(Cl)cccc1NC(=O)CSc1ncnc2c1sc1ccccc12	nan
	CHEMBL1477945	39675	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	5	5.5	Cc1c(Cl)cccc1NC(=O)CSc1ncnc2c1sc1ccccc12	nan
	647217	39723	1	None	1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	8	3.5	CCS(=O)(=O)Nc1ccc(-c2nnc(SCC(=O)c3cccc(OC)c3)o2)cc1	nan
	CHEMBL1478450	39723	1	None	1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	8	3.5	CCS(=O)(=O)Nc1ccc(-c2nnc(SCC(=O)c3cccc(OC)c3)o2)cc1	nan
	356316	39832	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	4	2.9	Cc1ccc(S(=O)(=O)c2cc3ccccc3oc2=O)cc1	nan
	CHEMBL1479392	39832	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	4	2.9	Cc1ccc(S(=O)(=O)c2cc3ccccc3oc2=O)cc1	nan
	16009796	39970	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	6	4.4	COc1ccc(-n2c(=O)c3sc4ccccc4c3n(Cc3ccccc3)c2=O)cc1	nan
	CHEMBL1480505	39970	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	6	4.4	COc1ccc(-n2c(=O)c3sc4ccccc4c3n(Cc3ccccc3)c2=O)cc1	nan
	16024583	39998	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	CHEMBL1480766	39998	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	3273049	40090	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	533	7	1	7	4.4	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C(C)C)C2	nan
	CHEMBL1481475	40090	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	533	7	1	7	4.4	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C(C)C)C2	nan
	3662250	40117	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	2.9	COc1ccc(-c2cc(C(=O)Nc3cc(C)on3)no2)cc1OC	nan
	CHEMBL1481783	40117	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	2.9	COc1ccc(-c2cc(C(=O)Nc3cc(C)on3)no2)cc1OC	nan
	5763301	40194	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	0	3	3.8	Cn1c(/C=C/c2ccc(Cl)cc2)nc2ccccc2c1=O	nan
	CHEMBL1482443	40194	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	0	3	3.8	Cn1c(/C=C/c2ccc(Cl)cc2)nc2ccccc2c1=O	nan
	16030274	40262	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	2	3	4.4	Cc1cccc2c(=O)cc(CSCC(=O)Nc3ccc(Cl)cc3)[nH]c12	nan
	CHEMBL1483081	40262	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	2	3	4.4	Cc1cccc2c(=O)cc(CSCC(=O)Nc3ccc(Cl)cc3)[nH]c12	nan
	135419126	40306	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	2	1	3	6.5	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2cccc(Br)c2)C1	nan
	CHEMBL1483478	40306	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	2	1	3	6.5	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2cccc(Br)c2)C1	nan
	16010346	40321	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	0	7	5.0	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N(C)Cc2ccccc2)c2cc(Cl)ccc23)cc1C	nan
	CHEMBL1483574	40321	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	0	7	5.0	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N(C)Cc2ccccc2)c2cc(Cl)ccc23)cc1C	nan
	1482113	40514	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.7	COCc1cc(O)nc2cc(NC(=O)c3cccc(OC)c3)c(C)cc12	nan
	CHEMBL1485213	40514	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.7	COCc1cc(O)nc2cc(NC(=O)c3cccc(OC)c3)c(C)cc12	nan
	848452	40550	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	4	2.9	COC(=O)c1ccc2ccn(CC(=O)NC3CCCCC3)c2c1	nan
	CHEMBL1485568	40550	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	4	2.9	COC(=O)c1ccc2ccn(CC(=O)NC3CCCCC3)c2c1	nan
	6491858	40671	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	7	3.4	COc1cccc(NC(=O)CSc2nc(O)c3c(C)csc3n2)c1	nan
	CHEMBL1486601	40671	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	7	3.4	COc1cccc(NC(=O)CSc2nc(O)c3c(C)csc3n2)c1	nan
	12005495	40706	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	2	4	4.0	Cc1cccc(C)c1NC(=O)C(NS(=O)(=O)c1cccs1)c1ccccc1	nan
	CHEMBL1486971	40706	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	2	4	4.0	Cc1cccc(C)c1NC(=O)C(NS(=O)(=O)c1cccs1)c1ccccc1	nan
	2007999	40777	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	6	3.4	CC(C)c1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	CHEMBL1487512	40777	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	6	3.4	CC(C)c1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	1604294	40804	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	4	5.9	Cc1ccc(OCCCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1487726	40804	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	4	5.9	Cc1ccc(OCCCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	3847044	40970	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	4.1	COC(=O)CSc1nc2sc3c(c2c(=O)n1-c1ccc(C)cc1)CC(C(C)C)OC3	nan
	CHEMBL1488882	40970	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	4.1	COC(=O)CSc1nc2sc3c(c2c(=O)n1-c1ccc(C)cc1)CC(C(C)C)OC3	nan
	3531068	41039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	5	1	8	4.5	COC(=O)c1ccc(C(=O)OC)c(NC(=O)c2cc3nc(-c4ccc(C)cc4)cc(C(F)(F)F)n3n2)c1	nan
	CHEMBL1489426	41039	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	5	1	8	4.5	COC(=O)c1ccc(C(=O)OC)c(NC(=O)c2cc3nc(-c4ccc(C)cc4)cc(C(F)(F)F)n3n2)c1	nan
	3149408	41125	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	6	8	-1.2	Cc1ccc(C2=NNC(C(O)C(O)C(O)C(O)CO)S2)cc1	nan
	CHEMBL1490120	41125	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	6	8	-1.2	Cc1ccc(C2=NNC(C(O)C(O)C(O)C(O)CO)S2)cc1	nan
	15996835	41193	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	6	3.9	COc1cc2nc(S)nc(NCCc3ccc(C)cc3)c2cc1OC	nan
	CHEMBL1490579	41193	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	6	3.9	COc1cc2nc(S)nc(NCCc3ccc(C)cc3)c2cc1OC	nan
	5216415	41231	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	5.2	COc1cccc2cc(-c3nc(-c4ccc(Cl)cc4)cs3)c(=O)oc12	nan
	CHEMBL1490839	41231	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	5.2	COc1cccc2cc(-c3nc(-c4ccc(Cl)cc4)cs3)c(=O)oc12	nan
	16022523	41290	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	7	2.3	Cn1cnc2c(=O)oc3ccc(S(=O)(=O)N4CCN(c5ccccc5F)CC4)cc3c21	nan
	CHEMBL1491216	41290	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	7	2.3	Cn1cnc2c(=O)oc3ccc(S(=O)(=O)N4CCN(c5ccccc5F)CC4)cc3c21	nan
	16034710	41516	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1492881	41516	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	1319924	41544	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	0	6	4.8	CCCS(=O)(=O)c1c(S(=O)(=O)CCC)c2cc(CC)ccn2c1C(=O)c1ccc(Cl)cc1	nan
	CHEMBL1493213	41544	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	0	6	4.8	CCCS(=O)(=O)c1c(S(=O)(=O)CCC)c2cc(CC)ccn2c1C(=O)c1ccc(Cl)cc1	nan
	16423380	41560	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	7205024	41560	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	CHEMBL1493339	41560	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	6823777	41586	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	8	3	6	3.3	Cc1ccc(-n2c([S-])c(C(=O)Nc3ccc(OC(F)F)cc3)[n+]3ccc(C(=O)NCCO)cc23)cc1C	nan
	CHEMBL1493546	41586	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	8	3	6	3.3	Cc1ccc(-n2c([S-])c(C(=O)Nc3ccc(OC(F)F)cc3)[n+]3ccc(C(=O)NCCO)cc23)cc1C	nan
	1091748	41590	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.5	O=C(Nc1ccccc1C(=O)Nc1ccc2c(c1)OCO2)c1ccco1	nan
	CHEMBL1493592	41590	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.5	O=C(Nc1ccccc1C(=O)Nc1ccc2c(c1)OCO2)c1ccco1	nan
	4885142	41978	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.4	CC(=O)c1ccc(N2CCN(c3ccnc4cc(Cl)ccc34)CC2)cc1	nan
	CHEMBL1497325	41978	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.4	CC(=O)c1ccc(N2CCN(c3ccnc4cc(Cl)ccc34)CC2)cc1	nan
	665746	42033	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	0	5	3.5	O=C1c2oc3ccccc3c(=O)c2C(c2cccnc2)N1Cc1ccco1	nan
	CHEMBL1497863	42033	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	0	5	3.5	O=C1c2oc3ccccc3c(=O)c2C(c2cccnc2)N1Cc1ccco1	nan
	1478337	42062	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	2	1	4	5.2	Cc1ccc2oc3nc(C)c(C(=O)Nc4cccc(C(F)(F)F)c4)cc3c(=O)c2c1	nan
	CHEMBL1498149	42062	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	2	1	4	5.2	Cc1ccc2oc3nc(C)c(C(=O)Nc4cccc(C(F)(F)F)c4)cc3c(=O)c2c1	nan
	1877175	42151	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOc1ccc(C(=O)Nc2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1498972	42151	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOc1ccc(C(=O)Nc2nc(C)c(C(=O)OC)s2)cc1	nan
	663555	42398	9	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1cccc(C(=O)OCc2cc3ccccc3nc2O)c1	nan
	CHEMBL1501108	42398	9	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1cccc(C(=O)OCc2cc3ccccc3nc2O)c1	nan
	1482342	42578	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	2	1	7	2.2	CSc1nc2ncc(-c3ccsc3)c(N)n2n1	nan
	CHEMBL1502638	42578	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	2	1	7	2.2	CSc1nc2ncc(-c3ccsc3)c(N)n2n1	nan
	6624089	42853	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	4	3.3	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccc(Cl)cc1	nan
	CHEMBL1505154	42853	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	4	3.3	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccc(Cl)cc1	nan
	1488509	42881	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	3	1	4	1.9	O=C(Nc1ccnc(-c2ccncc2)n1)C1CC1	nan
	CHEMBL1505422	42881	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	3	1	4	1.9	O=C(Nc1ccnc(-c2ccncc2)n1)C1CC1	nan
	8484069	43061	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	8	3.3	CC(=O)c1ccc(NC(=O)CSc2nnc(NC(=O)c3ccco3)s2)cc1	nan
	CHEMBL1506911	43061	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	8	3.3	CC(=O)c1ccc(NC(=O)CSc2nnc(NC(=O)c3ccco3)s2)cc1	nan
	2880344	43106	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	6	4.7	COc1ccc(CC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)cc1OC	nan
	CHEMBL1507312	43106	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	6	4.7	COc1ccc(CC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)cc1OC	nan
	1440345	43195	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	3.2	Cc1cc2cc3c(cc2nc1SCC(=O)O)CCC3	nan
	CHEMBL1508003	43195	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	3.2	Cc1cc2cc3c(cc2nc1SCC(=O)O)CCC3	nan
	4435004	43383	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	4	1	3	3.8	CCCn1c(NC(=O)c2ccc(F)cc2)nc2ccccc21	nan
	CHEMBL1509719	43383	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	4	1	3	3.8	CCCn1c(NC(=O)c2ccc(F)cc2)nc2ccccc21	nan
	2676980	43405	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	2.6	O=C(Cn1cnc2ccccc2c1=O)Nc1nc2ccccc2s1	nan
	CHEMBL1509918	43405	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	2.6	O=C(Cn1cnc2ccccc2c1=O)Nc1nc2ccccc2s1	nan
	2402709	43455	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	2	7	3.0	NS(=O)(=O)c1ccc(NC(=O)COC(=O)c2cn(-c3ccccc3)nc2-c2ccccc2)cc1	nan
	CHEMBL1510422	43455	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	2	7	3.0	NS(=O)(=O)c1ccc(NC(=O)COC(=O)c2cn(-c3ccccc3)nc2-c2ccccc2)cc1	nan
	16024491	43661	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	7	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	CHEMBL1512438	43661	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	7	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	7184798	43669	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	7	3.5	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	CHEMBL1512523	43669	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	7	3.5	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	16025847	43687	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.4	Cc1cccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)c1	nan
	CHEMBL1512717	43687	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.4	Cc1cccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)c1	nan
	16026525	43688	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.6	CCc1ccccc1NC(=O)C(C)n1c(=O)cc(C)c2c(C)nn(-c3ccccc3)c21	nan
	CHEMBL1512723	43688	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.6	CCc1ccccc1NC(=O)C(C)n1c(=O)cc(C)c2c(C)nn(-c3ccccc3)c21	nan
	16026338	43690	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	5	4.7	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4cc(Cl)ccc4C)c32)cc1	nan
	CHEMBL1512750	43690	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	5	4.7	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4cc(Cl)ccc4C)c32)cc1	nan
	7066893	43710	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	2	6	4.8	COc1cc(-c2nc3sccn3c2Nc2cccc(C)c2)ccc1O	nan
	CHEMBL1513064	43710	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	2	6	4.8	COc1cc(-c2nc3sccn3c2Nc2cccc(C)c2)ccc1O	nan
	16025357	43720	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	6	1	6	5.8	Cc1ccc(CN2c3ccccc3-c3nc(SCC(=O)Nc4c(C)cc(C)cc4C)ncc3S2(=O)=O)cc1	nan
	CHEMBL1513190	43720	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	6	1	6	5.8	Cc1ccc(CN2c3ccccc3-c3nc(SCC(=O)Nc4c(C)cc(C)cc4C)ncc3S2(=O)=O)cc1	nan
	16010879	43748	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1cc2nc(NCCc3cccc(C)c3)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	CHEMBL1513631	43748	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1cc2nc(NCCc3cccc(C)c3)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	2947326	43775	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	6	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nc3c(C)c(Br)cnc3[nH]2)cc1	nan
	CHEMBL1514184	43775	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	6	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nc3c(C)c(Br)cnc3[nH]2)cc1	nan
	15988389	43812	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	3	5.3	O=C(NCCc1ccccc1)c1cc(-c2ccccc2)nc2n[nH]c(-c3ccccc3)c12	nan
	CHEMBL1514741	43812	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	3	5.3	O=C(NCCc1ccccc1)c1cc(-c2ccccc2)nc2n[nH]c(-c3ccccc3)c12	nan
	16027439	43846	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n12	nan
	CHEMBL1515224	43846	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n12	nan
	3324743	43850	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	4	5.2	CCc1ccc(OCC(=O)Nc2c(C(=O)c3ccccc3)oc3ccccc23)cc1	nan
	CHEMBL1515282	43850	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	4	5.2	CCc1ccc(OCC(=O)Nc2c(C(=O)c3ccccc3)oc3ccccc23)cc1	nan
	1035668	43895	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	5	5.7	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1	nan
	CHEMBL1515955	43895	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	5	5.7	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1	nan
	16009680	43913	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	4	4.6	Cc1ccc(S(=O)(=O)c2cn(Cc3ccc(F)cc3)c3cc(F)c(F)cc3c2=O)cc1	nan
	CHEMBL1516142	43913	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	4	4.6	Cc1ccc(S(=O)(=O)c2cn(Cc3ccc(F)cc3)c3cc(F)c(F)cc3c2=O)cc1	nan
	1516716	43936	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	3	5	3.7	Nc1c(C(=O)Nc2ccc(C(=O)O)cc2)sc2nc3c(cc12)CCCC3	nan
	CHEMBL1516550	43936	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	3	5	3.7	Nc1c(C(=O)Nc2ccc(C(=O)O)cc2)sc2nc3c(cc12)CCCC3	nan
	15989644	43938	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)N3CCC(C)CC3)c3ccccc3c2=O)c(Br)c1	nan
	CHEMBL1516553	43938	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)N3CCC(C)CC3)c3ccccc3c2=O)c(Br)c1	nan
	16027696	43975	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1cccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1516896	43975	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1cccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	16009847	44033	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	4	0	6	5.1	O=c1c2sc3ccccc3c2n(Cc2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccco1	nan
	CHEMBL1517455	44033	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	4	0	6	5.1	O=c1c2sc3ccccc3c2n(Cc2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccco1	nan
	16010572	44035	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	4.0	COc1ccc(OC)c(CCNc2nc3ccccc3c3nc(-c4cccnc4)nn23)c1	nan
	CHEMBL1517540	44035	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	4.0	COc1ccc(OC)c(CCNc2nc3ccccc3c3nc(-c4cccnc4)nn23)c1	nan
	1073734	44043	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1C	nan
	CHEMBL1517640	44043	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1C	nan
	15990463	44114	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	8	2	6	4.6	Cc1cccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccc(F)cc4)C(=O)N23)c1	nan
	CHEMBL1518319	44114	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	8	2	6	4.6	Cc1cccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccc(F)cc4)C(=O)N23)c1	nan
	890719	44166	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	0.9	CCN1C(=O)/C(=C\NCc2ccccc2)C(=O)NC1=S	nan
	CHEMBL1518771	44166	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	0.9	CCN1C(=O)/C(=C\NCc2ccccc2)C(=O)NC1=S	nan
	4457184	44187	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	2	7	2.2	N#Cc1c(N2CCCCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	CHEMBL1518944	44187	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	2	7	2.2	N#Cc1c(N2CCCCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	16013971	44217	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	0	7	3.7	Cc1nnc(N2CCN(c3ccc(Cl)cc3)CC2)c2c1nnn2Cc1ccc(F)cc1	nan
	CHEMBL1519203	44217	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	0	7	3.7	Cc1nnc(N2CCN(c3ccc(Cl)cc3)CC2)c2c1nnn2Cc1ccc(F)cc1	nan
	1557528	44237	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	8	0	5	5.1	Cc1ccc(OCCOCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1519353	44237	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	8	0	5	5.1	Cc1ccc(OCCOCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	2158290	44271	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	9	0	9	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CCCOC)/c1=N/C(=O)C(C)(C)Oc1ccc(Cl)cc1	nan
	CHEMBL1519687	44271	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	9	0	9	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CCCOC)/c1=N/C(=O)C(C)(C)Oc1ccc(Cl)cc1	nan
	4379652	44411	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	10	1.1	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3cccs3)nc2n(C)c1=O	nan
	CHEMBL1520875	44411	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	10	1.1	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3cccs3)nc2n(C)c1=O	nan
	5925852	44457	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	10	3.2	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1521267	44457	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	10	3.2	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	16018871	44492	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.8	COc1ccc(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1521570	44492	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.8	COc1ccc(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	17252948	44593	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	5	3.9	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1C	nan
	CHEMBL1522534	44593	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	5	3.9	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1C	nan
	16009486	44630	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	9	3.9	COc1cc(C(=O)Nc2ccccc2OCc2cc(=O)n3c(C)csc3n2)cc(OC)c1OC	nan
	CHEMBL1522858	44630	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	9	3.9	COc1cc(C(=O)Nc2ccccc2OCc2cc(=O)n3c(C)csc3n2)cc(OC)c1OC	nan
	932437	44660	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.9	Cc1ccc(-c2nnc3c4ccccc4c(-c4ccccc4)nn23)cc1	nan
	CHEMBL1523117	44660	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.9	Cc1ccc(-c2nnc3c4ccccc4c(-c4ccccc4)nn23)cc1	nan
	2084813	44708	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2cc(F)ccc2C)c1C	nan
	CHEMBL1523555	44708	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2cc(F)ccc2C)c1C	nan
	663733	44751	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	8	3.1	Cc1nc2c(sc3nc4c(cc32)COC(C)(C)C4)c(=O)n1CC(=O)NCc1ccco1	nan
	CHEMBL1523984	44751	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	8	3.1	Cc1nc2c(sc3nc4c(cc32)COC(C)(C)C4)c(=O)n1CC(=O)NCc1ccco1	nan
	16027443	44855	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3ccccc3NC(=O)c3ccccc3Cl)cc(=O)n12	nan
	CHEMBL1525043	44855	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3ccccc3NC(=O)c3ccccc3Cl)cc(=O)n12	nan
	1299413	44946	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	5	3.1	C=CCn1c(SCC(=O)NC2CCCCC2)nc2ccccc2c1=O	nan
	CHEMBL1525864	44946	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	5	3.1	C=CCn1c(SCC(=O)NC2CCCCC2)nc2ccccc2c1=O	nan
	4174172	45105	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	7	0	6	4.9	COc1cc2c(cc1OC)C(COc1ccc3c(C)cc(=O)oc3c1)N(C(=O)Cc1ccccc1)CC2	nan
	CHEMBL1527205	45105	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	7	0	6	4.9	COc1cc2c(cc1OC)C(COc1ccc3c(C)cc(=O)oc3c1)N(C(=O)Cc1ccccc1)CC2	nan
	757005	45384	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	8	2	5	2.7	CCCc1cc(C(=O)OC)c(NC(=O)CCCC(=O)O)s1	nan
	CHEMBL1529664	45384	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	8	2	5	2.7	CCCc1cc(C(=O)OC)c(NC(=O)CCCC(=O)O)s1	nan
	4067774	45487	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	1	4	6.0	CCCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(C)cc3)oc3ccccc23)cc1	nan
	CHEMBL1530590	45487	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	1	4	6.0	CCCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(C)cc3)oc3ccccc23)cc1	nan
	3420293	45624	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	7	2.9	Cc1ccc(NC(=O)c2sc3ncn(CC(=O)N4CCOCC4)c(=O)c3c2C)c(Br)c1	nan
	CHEMBL1531811	45624	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	7	2.9	Cc1ccc(NC(=O)c2sc3ncn(CC(=O)N4CCOCC4)c(=O)c3c2C)c(Br)c1	nan
	821799	45650	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.1	CSc1nc2ccc(Br)cn2c(=O)c1C#N	nan
	CHEMBL1532047	45650	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.1	CSc1nc2ccc(Br)cn2c(=O)c1C#N	nan
	1475615	45679	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	6	5.0	O=C(Nc1cc2c(=O)n(-c3ccc(Oc4ccccc4)cc3)ccc2oc1=O)c1ccccc1	nan
	CHEMBL1532311	45679	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	6	5.0	O=C(Nc1cc2c(=O)n(-c3ccc(Oc4ccccc4)cc3)ccc2oc1=O)c1ccccc1	nan
	15989915	45723	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	5	4.6	COc1ccc(C2CC(=O)c3c([nH]c(C(=O)OCc4ccccc4)c3C)C2)cc1OC	nan
	CHEMBL1532686	45723	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	5	4.6	COc1ccc(C2CC(=O)c3c([nH]c(C(=O)OCc4ccccc4)c3C)C2)cc1OC	nan
	656128	45752	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	0	6	2.8	CCOc1ccc2cc(C#N)c(SCC(=O)OC)nc2c1	nan
	CHEMBL1532931	45752	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	0	6	2.8	CCOc1ccc2cc(C#N)c(SCC(=O)OC)nc2c1	nan
	3137936	45880	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	5	3.4	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2C)c1C	nan
	CHEMBL1534032	45880	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	5	3.4	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2C)c1C	nan
	16011802	45929	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	3.4	COc1ccc(C(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1OC	nan
	CHEMBL1534572	45929	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	3.4	COc1ccc(C(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1OC	nan
	3410008	45949	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	2.8	CCOc1ccc(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)cc1	nan
	CHEMBL1534800	45949	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	2.8	CCOc1ccc(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)cc1	nan
	5949916	45991	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.0	Cc1[nH]c2nc(SCC(=O)c3ccccc3)nc-2cc1Br	nan
	CHEMBL1535293	45991	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.0	Cc1[nH]c2nc(SCC(=O)c3ccccc3)nc-2cc1Br	nan
	2820834	46002	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	5.6	CSc1sc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)n2C)c2c1C=CCC2	nan
	CHEMBL1535400	46002	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	5.6	CSc1sc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)n2C)c2c1C=CCC2	nan
	16019886	46068	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	3.2	Cc1cccc(NC(=O)CN2C(=O)CSc3ccc(S(=O)(=O)N4CCCC4)cc32)c1C	nan
	CHEMBL1536151	46068	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	3.2	Cc1cccc(NC(=O)CN2C(=O)CSc3ccc(S(=O)(=O)N4CCCC4)cc32)c1C	nan
	891752	46128	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.6	COc1cc(Cl)c(C)cc1NC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1536712	46128	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.6	COc1cc(Cl)c(C)cc1NC(=O)c1ccc2c(c1)OCO2	nan
	664078	46421	1	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	1	4	3.3	COc1cccc(OCc2nc3cc(Br)c[nH]c-3n2)c1	nan
	CHEMBL1539150	46421	1	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	1	4	3.3	COc1cccc(OCc2nc3cc(Br)c[nH]c-3n2)c1	nan
	841141	46771	10	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	5	2.2	COC(=O)c1c(NC(=O)c2ccccc2)sc(C(N)=O)c1C	nan
	CHEMBL1542119	46771	10	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	5	2.2	COC(=O)c1c(NC(=O)c2ccccc2)sc(C(N)=O)c1C	nan
	664933	46933	10	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	CHEMBL1543543	46933	10	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	3240821	47005	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	8	2.9	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(C(=O)c2ccco2)CC1	nan
	CHEMBL1544051	47005	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	8	2.9	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(C(=O)c2ccco2)CC1	nan
	1861702	47062	8	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	8	2.7	CC(C)OC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	CHEMBL1544436	47062	8	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	8	2.7	CC(C)OC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	3164596	47191	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	2.7	COc1ccc2cc(C(=O)NCc3ccccc3)c(=O)oc2c1	nan
	CHEMBL1545409	47191	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	2.7	COc1ccc2cc(C(=O)NCc3ccccc3)c(=O)oc2c1	nan
	4340721	47245	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	4.0	COc1ccc2cc(C#N)c(Nc3cccc(F)c3)nc2c1	nan
	CHEMBL1545865	47245	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	4.0	COc1ccc2cc(C#N)c(Nc3cccc(F)c3)nc2c1	nan
	2106365	47248	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	5	4.1	Oc1nc(-c2cccnc2)nc2sc(-c3ccccc3)cc12	nan
	CHEMBL1545901	47248	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	5	4.1	Oc1nc(-c2cccnc2)nc2sc(-c3ccccc3)cc12	nan
	902245	47395	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	1	3	4.9	CCc1cc2cc(C(=O)Nc3ccc(F)cc3)sc2s1	nan
	CHEMBL1547204	47395	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	1	3	4.9	CCc1cc2cc(C(=O)Nc3ccc(F)cc3)sc2s1	nan
	1088622	47425	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	9	1.2	CCOc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1OC	nan
	CHEMBL1547487	47425	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	9	1.2	CCOc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1OC	nan
	2801256	47564	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	1	5	2.4	Cc1nc(-c2cc(C#N)c(O)nc2C)cs1	nan
	CHEMBL1548830	47564	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	1	5	2.4	Cc1nc(-c2cc(C#N)c(O)nc2C)cs1	nan
	4601866	47675	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	10	3	6	3.4	NS(=O)(=O)c1ccc(CCNC(=O)CCCCCn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	CHEMBL1549770	47675	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	10	3	6	3.4	NS(=O)(=O)c1ccc(CCNC(=O)CCCCCn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	2731089	47723	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	2	7	2.6	COc1ccc(CCNC(=S)NC(=O)c2cc(OC)c(OC)c(OC)c2)cc1OC	nan
	CHEMBL1550121	47723	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	2	7	2.6	COc1ccc(CCNC(=S)NC(=O)c2cc(OC)c(OC)c(OC)c2)cc1OC	nan
	5122884	47755	4	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	2.8	COc1ccc2cc(CCN3C(=O)c4ccccc4C3=O)c(O)nc2c1	nan
	CHEMBL1550382	47755	4	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	2.8	COc1ccc2cc(CCN3C(=O)c4ccccc4C3=O)c(O)nc2c1	nan
	1490541	47761	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	3	4.2	Cc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	CHEMBL1550435	47761	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	3	4.2	Cc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	15944825	47823	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	5	4.2	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1550942	47823	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	5	4.2	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	15988480	47841	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	6	2.4	COC(=O)c1cc(Cl)ccc1NC(=O)Cn1c(C)cc(C)c(C#N)c1=O	nan
	CHEMBL1551156	47841	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	6	2.4	COC(=O)c1cc(Cl)ccc1NC(=O)Cn1c(C)cc(C)c(C#N)c1=O	nan
	16025269	47844	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	2	5	4.7	COC(=O)c1c(SCC(=O)Nc2ccccc2C(F)(F)F)[nH]c2ccc(Cl)cc2c1=O	nan
	CHEMBL1551199	47844	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	2	5	4.7	COC(=O)c1c(SCC(=O)Nc2ccccc2C(F)(F)F)[nH]c2ccc(Cl)cc2c1=O	nan
	16009432	47859	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	6	3.9	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)c1	nan
	CHEMBL1551357	47859	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	6	3.9	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)c1	nan
	3151519	47862	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	8	3	8	1.4	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccccc4)c(=N)n(CCOCCO)c3nc12	nan
	CHEMBL1551451	47862	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	8	3	8	1.4	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccccc4)c(=N)n(CCOCCO)c3nc12	nan
	16007408	47868	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	2	3	3.7	Cc1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1F	nan
	CHEMBL1551538	47868	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	2	3	3.7	Cc1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1F	nan
	16021062	47878	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	6	3.5	COC(=O)c1ccccc1NC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	CHEMBL1551793	47878	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	6	3.5	COC(=O)c1ccccc1NC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	1189625	47885	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)cc1	nan
	CHEMBL1551857	47885	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)cc1	nan
	16008906	47892	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1cccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1551951	47892	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1cccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	16011042	47902	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	2	3	4.8	O=C(Nc1ccc(F)cc1)c1ccc2c(c1)NC(=O)c1ccccc1S2	nan
	CHEMBL1552027	47902	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	2	3	4.8	O=C(Nc1ccc(F)cc1)c1ccc2c(c1)NC(=O)c1ccccc1S2	nan
	4412264	47903	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	0	8	4.5	CCOC(=O)CSc1nc2c(sc3cccc(F)c32)c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1552040	47903	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	0	8	4.5	CCOC(=O)CSc1nc2c(sc3cccc(F)c32)c(=O)n1Cc1ccc(OC)cc1	nan
	1187153	47905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	3.5	CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1NCCN1CCOCC1	nan
	CHEMBL1552062	47905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	3.5	CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1NCCN1CCOCC1	nan
	16027700	47927	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1C	nan
	CHEMBL1552279	47927	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1C	nan
	16032167	47945	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	8	3.5	Cn1c(SCC(=O)Nc2nc3ccccc3s2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	CHEMBL1552642	47945	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	8	3.5	Cn1c(SCC(=O)Nc2nc3ccccc3s2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	16024489	47963	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	5	4.5	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc(C)c(Cl)c3)c2n1	nan
	CHEMBL1552935	47963	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	5	4.5	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc(C)c(Cl)c3)c2n1	nan
	16030793	47964	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	5.2	COc1ccccc1-c1cc(NC(=O)COc2ccccc2Cl)n(-c2ccccc2)n1	nan
	CHEMBL1552946	47964	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	5.2	COc1ccccc1-c1cc(NC(=O)COc2ccccc2Cl)n(-c2ccccc2)n1	nan
	16020265	47971	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	6	2.5	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(CC(N)=O)c2=O)cc1	nan
	CHEMBL1552986	47971	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	6	2.5	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(CC(N)=O)c2=O)cc1	nan
	16024860	47992	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	4	3.9	O=S(=O)(c1ccc2nc(Nc3ccc(F)cc3)ccc2c1)N1CCCC1	nan
	CHEMBL1553226	47992	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	4	3.9	O=S(=O)(c1ccc2nc(Nc3ccc(F)cc3)ccc2c1)N1CCCC1	nan
	16014611	48001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	5	3.1	CSc1ccc(NC(=O)C2CCN(c3ncccn3)CC2)cc1	nan
	CHEMBL1553334	48001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	5	3.1	CSc1ccc(NC(=O)C2CCN(c3ncccn3)CC2)cc1	nan
	16018242	48017	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1OC	nan
	CHEMBL1553551	48017	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1OC	nan
	16020219	48020	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	4	4.2	Cn1c(=O)c2cc(C(=O)NC3CCCCCC3)sc2c2ccccc21	nan
	CHEMBL1553584	48020	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	4	4.2	Cn1c(=O)c2cc(C(=O)NC3CCCCCC3)sc2c2ccccc21	nan
	3158758	48022	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	4.2	COc1cc(OC)c(C2Nc3c(C)cccc3-c3cc(C)nn32)cc1OC	nan
	CHEMBL1553632	48022	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	4.2	COc1cc(OC)c(C2Nc3c(C)cccc3-c3cc(C)nn32)cc1OC	nan
	15989000	48025	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2ccccc2F)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1553743	48025	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2ccccc2F)c1=O)NCc1ccc2c(c1)OCO2	nan
	2580267	48032	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	2.9	Cc1cc(C)cc(NC(=O)COC(=O)c2ccc3c(c2)OCCO3)c1	nan
	CHEMBL1553826	48032	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	2.9	Cc1cc(C)cc(NC(=O)COC(=O)c2ccc3c(c2)OCCO3)c1	nan
	16033854	48036	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	8	3.1	COC(=O)c1ccc2c(=O)n3nc(Nc4ccc(F)cc4F)sc3nc2c1	nan
	CHEMBL1553893	48036	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	8	3.1	COC(=O)c1ccc2c(=O)n3nc(Nc4ccc(F)cc4F)sc3nc2c1	nan
	16030113	48051	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1cccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)c1	nan
	CHEMBL1554129	48051	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1cccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)c1	nan
	4361698	48070	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1554379	48070	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1cccc(C(F)(F)F)c1	nan
	16282512	48072	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	5	3.2	Cc1ccc(NC(=O)CN(C)C(=O)COc2ncnc3ccc(Br)cc23)cc1	nan
	CHEMBL1554437	48072	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	5	3.2	Cc1ccc(NC(=O)CN(C)C(=O)COc2ncnc3ccc(Br)cc23)cc1	nan
	16009851	48075	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.2	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1554474	48075	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.2	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	16011879	48076	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	2	4.1	Cc1ccc(CNC(=O)Cc2csc3ccccc23)cc1	nan
	CHEMBL1554476	48076	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	2	4.1	Cc1ccc(CNC(=O)Cc2csc3ccccc23)cc1	nan
	15988910	48079	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	0	10	2.6	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3cc(=O)n4c(C)cccc4n3)c2=O)c1	nan
	CHEMBL1554524	48079	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	0	10	2.6	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3cc(=O)n4c(C)cccc4n3)c2=O)c1	nan
	16009798	48080	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	4.8	Fc1cccc(-c2nnn3c2nc(NC2CCCCC2)c2ccccc23)c1	nan
	CHEMBL1554525	48080	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	4.8	Fc1cccc(-c2nnn3c2nc(NC2CCCCC2)c2ccccc23)c1	nan
	16019045	48081	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	4.0	CCOc1cc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)ccc1OC	nan
	CHEMBL1554576	48081	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	4.0	CCOc1cc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)ccc1OC	nan
	16010240	48095	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	3	5.3	CC(C)c1ccc(NC(=O)c2cc3sc(Cl)cc3n2C)cc1	nan
	CHEMBL1554758	48095	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	3	5.3	CC(C)c1ccc(NC(=O)c2cc3sc(Cl)cc3n2C)cc1	nan
	16016717	48126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	3	6.0	CCc1ccccc1NC(=O)Nc1ccc2c(c1)N(CC)C(=O)c1ccccc1S2	nan
	CHEMBL1555228	48126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	3	6.0	CCc1ccccc1NC(=O)Nc1ccc2c(c1)N(CC)C(=O)c1ccccc1S2	nan
	15999699	48128	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.7	CCCCNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1555241	48128	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.7	CCCCNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	16024527	48208	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.2	COc1ccc(C(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1556147	48208	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.2	COc1ccc(C(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3nc(C)ccc3c2=O)cc1	nan
	884827	48209	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	1	5	3.8	CCOc1ccc(Nc2nc3ccccc3c(=O)s2)cc1	nan
	CHEMBL1556149	48209	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	1	5	3.8	CCOc1ccc(Nc2nc3ccccc3c(=O)s2)cc1	nan
	1299811	48230	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	0	8	3.4	COC(=O)CSc1ncnc2c1sc1nc3c(cc12)COC(C)(C)C3	nan
	CHEMBL1556306	48230	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	0	8	3.4	COC(=O)CSc1ncnc2c1sc1nc3c(cc12)COC(C)(C)C3	nan
	1297627	48260	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	3	4.1	CC(=O)c1ccc(NC(=S)N2CCN(c3cccc(Cl)c3)CC2)cc1	nan
	CHEMBL1556657	48260	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	3	4.1	CC(=O)c1ccc(NC(=S)N2CCN(c3cccc(Cl)c3)CC2)cc1	nan
	1262055	48262	7	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	5.3	CCn1c(SCC(=O)Nc2cccc(F)c2)nnc1-c1cc2cc(Br)ccc2o1	nan
	CHEMBL1556666	48262	7	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	5.3	CCn1c(SCC(=O)Nc2cccc(F)c2)nnc1-c1cc2cc(Br)ccc2o1	nan
	2769090	48422	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	0	5	2.8	CC(=O)c1cc(C#N)c(N2CCN(c3ccccc3)CC2)nc1C	nan
	CHEMBL1558006	48422	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	0	5	2.8	CC(=O)c1cc(C#N)c(N2CCN(c3ccccc3)CC2)nc1C	nan
	16015862	48593	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	5.7	Cc1ccc(SCC(=O)Nc2ccc3oc(-c4ccc(F)cc4)nc3c2)cc1	nan
	CHEMBL1559463	48593	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	5.7	Cc1ccc(SCC(=O)Nc2ccc3oc(-c4ccc(F)cc4)nc3c2)cc1	nan
	3208119	48619	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2ccc(C)c(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1559714	48619	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2ccc(C)c(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	16286863	48792	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	2	6	2.7	CC(OC(=O)c1cc(Br)ccc1O)C(=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1561413	48792	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	2	6	2.7	CC(OC(=O)c1cc(Br)ccc1O)C(=O)NCc1ccc2c(c1)OCO2	nan
	24686491	48950	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccc(C)cn1	nan
	CHEMBL1562813	48950	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccc(C)cn1	nan
	135884418	48966	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	7	3.9	COc1cc2ccccc2cc1C(=O)OCc1nc(O)c2sccc2n1	nan
	CHEMBL1562918	48966	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	7	3.9	COc1cc2ccccc2cc1C(=O)OCc1nc(O)c2sccc2n1	nan
	664089	49016	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1563407	49016	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	16008603	49017	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	1.5	COc1ccc(CNC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1563417	49017	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	1.5	COc1ccc(CNC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	16025580	49065	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	4	1	6	4.6	Cc1cc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)c(C)c1	nan
	CHEMBL1563792	49065	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	4	1	6	4.6	Cc1cc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)c(C)c1	nan
	654285	49182	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	6	1.7	N#Cc1cc2cc3c(cc2nc1N1CCOCC1)OCO3	nan
	CHEMBL1564877	49182	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	6	1.7	N#Cc1cc2cc3c(cc2nc1N1CCOCC1)OCO3	nan
	4282255	49283	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	1	6	2.6	COc1cc([N+](=O)[O-])cc2sc(NC(=O)C3CC3)nc12	nan
	CHEMBL1565614	49283	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	1	6	2.6	COc1cc([N+](=O)[O-])cc2sc(NC(=O)C3CC3)nc12	nan
	151922	49553	57	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	12	1	1	5.2	O=C(O)CCCCCCCCCCCc1ccccc1	nan
	CHEMBL1567811	49553	57	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	12	1	1	5.2	O=C(O)CCCCCCCCCCCc1ccccc1	nan
	4289114	49676	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	6.0	Cc1ccc(C(=O)c2oc3ccccc3c2NC(=O)C(C)Oc2ccccc2Cl)cc1	nan
	CHEMBL1568822	49676	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	6.0	Cc1ccc(C(=O)c2oc3ccccc3c2NC(=O)C(C)Oc2ccccc2Cl)cc1	nan
	650090	49707	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	9	2.7	Cn1c(=O)c2c(nc(SCC(=O)c3cccs3)n2Cc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1569069	49707	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	9	2.7	Cn1c(=O)c2c(nc(SCC(=O)c3cccs3)n2Cc2ccc(F)cc2)n(C)c1=O	nan
	1336265	49845	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	2	6	2.5	COC(=O)c1sc(NC(=S)NC(=O)c2ccccc2F)nc1C	nan
	CHEMBL1570262	49845	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	2	6	2.5	COC(=O)c1sc(NC(=S)NC(=O)c2ccccc2F)nc1C	nan
	1834757	49886	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	5	6.7	CCN(CC)c1ccc2cc(-c3nc(-c4ccc(Cl)cc4Cl)cs3)c(=O)oc2c1	nan
	CHEMBL1570631	49886	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	5	6.7	CCN(CC)c1ccc2cc(-c3nc(-c4ccc(Cl)cc4Cl)cs3)c(=O)oc2c1	nan
	661116	49964	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	3.2	COc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	CHEMBL1571331	49964	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	3.2	COc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	3228933	50023	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	3.5	CCc1nc(SCC(=O)Nc2c(C)nn(C)c2C)c2cnn(-c3ccccc3)c2n1	nan
	CHEMBL1571990	50023	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	3.5	CCc1nc(SCC(=O)Nc2c(C)nn(C)c2C)c2cnn(-c3ccccc3)c2n1	nan
	998563	50033	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	3	5.8	Cc1ccc(NC(=O)c2cc(-c3cccs3)nc3ccccc23)c(C)c1	nan
	CHEMBL1572046	50033	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	3	5.8	Cc1ccc(NC(=O)c2cc(-c3cccs3)nc3ccccc23)c(C)c1	nan
	5038692	50071	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	1.9	O=C(O)C1Cc2ccccc2CN1C(=O)CSc1nnc2ccccn12	nan
	CHEMBL1572334	50071	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	1.9	O=C(O)C1Cc2ccccc2CN1C(=O)CSc1nnc2ccccn12	nan
	16020271	50345	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	7	1	6	5.1	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3cccc(Cl)c3)c2=O)cc1	nan
	CHEMBL1575057	50345	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	7	1	6	5.1	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3cccc(Cl)c3)c2=O)cc1	nan
	1637692	50356	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	4.1	CC(=O)c1sc(NC(=O)CCCOc2ccc(Cl)cc2)nc1C	nan
	CHEMBL1575283	50356	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	4.1	CC(=O)c1sc(NC(=O)CCCOc2ccc(Cl)cc2)nc1C	nan
	2446441	50625	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	2	2	4.2	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(C)cc2Br)c1C	nan
	CHEMBL1577640	50625	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	2	2	4.2	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(C)cc2Br)c1C	nan
	2868371	50650	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	6	2	7	2.5	CCOc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	CHEMBL1577894	50650	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	6	2	7	2.5	CCOc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	7207360	50654	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	7	3.4	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3ccncc3)nn2)cc1	nan
	CHEMBL1577921	50654	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	7	3.4	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3ccncc3)nn2)cc1	nan
	24891931	50734	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	2	7	0.7	NS(=O)(=O)c1ccc(CCNC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	CHEMBL1578510	50734	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	2	7	0.7	NS(=O)(=O)c1ccc(CCNC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	712274	50772	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	3	5	2.2	NC(=O)c1ccc2nc(NC(=O)c3ccc(N)cc3)sc2c1	nan
	CHEMBL1578798	50772	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	3	5	2.2	NC(=O)c1ccc2nc(NC(=O)c3ccc(N)cc3)sc2c1	nan
	7416477	50922	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	4	3.5	Cc1cccc(C(=O)OCC(=O)c2cccc(Br)c2)c1O	nan
	CHEMBL1580196	50922	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	4	3.5	Cc1cccc(C(=O)OCC(=O)c2cccc(Br)c2)c1O	nan
	16193583	50951	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	10	1	8	3.3	CCCCNC(=O)CSc1nc2ccc(N3CCOCC3)cc2c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1580449	50951	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	10	1	8	3.3	CCCCNC(=O)CSc1nc2ccc(N3CCOCC3)cc2c(=O)n1Cc1ccc(OC)cc1	nan
	135421577	50995	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	2	3	2.0	C=CCN1C(=O)/C(=C/c2cc3ccccc3[nH]2)C(=O)NC1=S	nan
	CHEMBL1580833	50995	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	2	3	2.0	C=CCN1C(=O)/C(=C/c2cc3ccccc3[nH]2)C(=O)NC1=S	nan
	652265	51050	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	4.1	O=C(Nc1ccc(Oc2ccccc2)cc1)C1CCN(c2ncccn2)CC1	nan
	CHEMBL1581276	51050	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	4.1	O=C(Nc1ccc(Oc2ccccc2)cc1)C1CCN(c2ncccn2)CC1	nan
	4455225	51139	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	9	2	5	3.5	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCCc3ccccc3)ccc2c1=O	nan
	CHEMBL1582016	51139	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	9	2	5	3.5	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCCc3ccccc3)ccc2c1=O	nan
	135693216	51389	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	5	2.9	Cc1cccc(CCNC(=O)Cn2ncc3c4ccccc4nc-3c2O)c1	nan
	CHEMBL1584056	51389	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	5	2.9	Cc1cccc(CCNC(=O)Cn2ncc3c4ccccc4nc-3c2O)c1	nan
	3662539	51412	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	1	4	7	3.1	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1c(F)cccc1Cl	nan
	CHEMBL1584309	51412	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	1	4	7	3.1	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1c(F)cccc1Cl	nan
	24819718	51544	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	2	4.0	O=C(c1cc2ccccc2cc1O)N1CCCC(C(F)(F)F)C1	nan
	CHEMBL1585344	51544	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	2	4.0	O=C(c1cc2ccccc2cc1O)N1CCCC(C(F)(F)F)C1	nan
	2112635	51697	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	6	2.9	Cc1nc(NCc2ccc(S(N)(=O)=O)cc2)c2c(C)c(C)sc2n1	nan
	CHEMBL1586644	51697	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	6	2.9	Cc1nc(NCc2ccc(S(N)(=O)=O)cc2)c2c(C)c(C)sc2n1	nan
	135441025	51711	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	2	4	3.7	CCCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	CHEMBL1586724	51711	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	2	4	3.7	CCCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	2158327	51752	10	None	-17	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccc(F)cc1	nan
	CHEMBL1587044	51752	10	None	-17	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccc(F)cc1	nan
	20876043	51923	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	0.5	COc1cccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1	nan
	CHEMBL1588535	51923	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	0.5	COc1cccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1	nan
	16016041	52074	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	4	4.5	COc1ccc(CC(=O)Nc2nc3c(s2)CC(C(C)(C)C)CC3)cc1	nan
	CHEMBL1589883	52074	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	4	4.5	COc1ccc(CC(=O)Nc2nc3c(s2)CC(C(C)(C)C)CC3)cc1	nan
	4671465	52099	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	4	3.3	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccc(F)cc3)o2)cc1	nan
	CHEMBL1590137	52099	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	4	3.3	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccc(F)cc3)o2)cc1	nan
	16009149	52129	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	3	5.5	Cc1ccc(CNC(=O)CSc2c3c(nc4cc(Cl)ccc24)CCCC3)cc1	nan
	CHEMBL1590589	52129	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	3	5.5	Cc1ccc(CNC(=O)CSc2c3c(nc4cc(Cl)ccc24)CCCC3)cc1	nan
	16026741	52137	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	0	8	2.8	O=C(COc1ccc(Cl)cc1)OCc1cc(=O)n2nc(C3CC3)sc2n1	nan
	CHEMBL1590675	52137	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	0	8	2.8	O=C(COc1ccc(Cl)cc1)OCc1cc(=O)n2nc(C3CC3)sc2n1	nan
	16025957	52143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1590760	52143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	16033877	52144	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	8	4.0	O=C(NCc1cccs1)c1ccc2c(=O)n3nc(Nc4ccccc4)sc3nc2c1	nan
	CHEMBL1590761	52144	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	8	4.0	O=C(NCc1cccs1)c1ccc2c(=O)n3nc(Nc4ccccc4)sc3nc2c1	nan
	18567961	52161	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	9	2	6	3.3	COc1ccc(C(=O)Nc2nc(CC(=O)NCCc3ccccc3OC)cs2)cc1	nan
	CHEMBL1590928	52161	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	9	2	6	3.3	COc1ccc(C(=O)Nc2nc(CC(=O)NCCc3ccccc3OC)cs2)cc1	nan
	16021437	52188	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	4	6.6	Cc1cc(Nc2cccc(Cl)c2)nc2ccc(NC(=O)COc3ccc(Cl)cc3)cc12	nan
	CHEMBL1591314	52188	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	4	6.6	Cc1cc(Nc2cccc(Cl)c2)nc2ccc(NC(=O)COc3ccc(Cl)cc3)cc12	nan
	16030267	52200	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCCC2)cc1	nan
	CHEMBL1591398	52200	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCCC2)cc1	nan
	15988978	52201	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	7	3.9	COc1ccc(NC(=O)Cn2c(=O)n(-c3cccc(C(F)(F)F)c3)c(=O)c3sccc32)cc1	nan
	CHEMBL1591409	52201	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	7	3.9	COc1ccc(NC(=O)Cn2c(=O)n(-c3cccc(C(F)(F)F)c3)c(=O)c3sccc32)cc1	nan
	4905426	52204	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.4	COc1ccc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2c1	nan
	CHEMBL1591442	52204	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.4	COc1ccc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2c1	nan
	15989516	52245	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	9	2	6	4.0	O=C(Cn1c(=O)n(CC2CCC(C(=O)NCCc3ccccc3)CC2)c(=O)c2ccccc21)Nc1ccccc1	nan
	CHEMBL1592027	52245	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	9	2	6	4.0	O=C(Cn1c(=O)n(CC2CCC(C(=O)NCCc3ccccc3)CC2)c(=O)c2ccccc21)Nc1ccccc1	nan
	15991260	52265	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	7	1.4	CCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1592271	52265	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	7	1.4	CCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	16027708	52288	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	7	4.7	CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1592618	52288	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	7	4.7	CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	16027669	52289	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	7	4.9	O=C(Nc1ccccc1C(=O)OCc1cc(=O)n2c3c(sc2n1)CCCC3)c1cccc(Cl)c1	nan
	CHEMBL1592645	52289	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	7	4.9	O=C(Nc1ccccc1C(=O)OCc1cc(=O)n2c3c(sc2n1)CCCC3)c1cccc(Cl)c1	nan
	16024581	52300	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	5	3.7	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1592799	52300	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	5	3.7	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	16020979	52331	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	4.5	COc1cc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc(OC)c1	nan
	CHEMBL1593212	52331	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	4.5	COc1cc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc(OC)c1	nan
	16012982	52345	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	3	5.7	Cc1cccc(N(Cc2cc3ccccc3nc2O)C(=O)c2cccc(Cl)c2)c1	nan
	CHEMBL1593385	52345	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	3	5.7	Cc1cccc(N(Cc2cc3ccccc3nc2O)C(=O)c2cccc(Cl)c2)c1	nan
	5143379	52346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	3	5.0	CC(=O)Nc1cc(C(=O)NCc2ccc(F)cc2)ccc1Sc1ccc(F)cc1	nan
	CHEMBL1593424	52346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	3	5.0	CC(=O)Nc1cc(C(=O)NCc2ccc(F)cc2)ccc1Sc1ccc(F)cc1	nan
	16322180	52362	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	5	3.7	Cc1nc(SC(C)C(=O)NC2(C#N)CCCCC2)c(C#N)c(C)c1C	nan
	CHEMBL1593705	52362	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	5	3.7	Cc1nc(SC(C)C(=O)NC2(C#N)CCCCC2)c(C#N)c(C)c1C	nan
	16024549	52368	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	4.6	CCOc1ccccc1NC(=O)Cn1cc(C(=O)c2ccc(Cl)cc2)c(=O)c2ccc(C)nc21	nan
	CHEMBL1593798	52368	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	4.6	CCOc1ccccc1NC(=O)Cn1cc(C(=O)c2ccc(Cl)cc2)c(=O)c2ccc(C)nc21	nan
	16019841	52372	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	7	4.1	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3Cl)nnc12	nan
	CHEMBL1593835	52372	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	7	4.1	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3Cl)nnc12	nan
	16026849	52379	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.8	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(F)cc4)cc3c2=O)cc1	nan
	CHEMBL1593965	52379	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.8	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(F)cc4)cc3c2=O)cc1	nan
	16024916	52385	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.9	CSc1ccc(CCNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1594028	52385	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.9	CSc1ccc(CCNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16024610	52395	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3cccc(C)c3C)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1594130	52395	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3cccc(C)c3C)c3nc(C)ccc3c2=O)cc1	nan
	2140504	52541	20	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	6	3.4	N#Cc1cc2c(nc1SCC(=O)Nc1nccs1)CCCCC2	nan
	CHEMBL1595336	52541	20	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	6	3.4	N#Cc1cc2c(nc1SCC(=O)Nc1nccs1)CCCCC2	nan
	16024587	52624	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1596100	52624	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	865538	52662	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	4.0	Cc1ccc2nc(NCc3ccccc3)c(C#N)cc2c1	nan
	CHEMBL1596421	52662	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	4.0	Cc1ccc2nc(NCc3ccccc3)c(C#N)cc2c1	nan
	16008803	52673	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	5.8	CCOc1ccccc1NC(=O)c1cc2c(Cl)nc3ccccc3c2s1	nan
	CHEMBL1596557	52673	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	5.8	CCOc1ccccc1NC(=O)c1cc2c(Cl)nc3ccccc3c2s1	nan
	1191858	52681	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	6	3.8	COc1ccc(-c2cc(=O)c3cc(OCC(=O)OC(C)C)ccc3o2)cc1	nan
	CHEMBL1596612	52681	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	6	3.8	COc1ccc(-c2cc(=O)c3cc(OCC(=O)OC(C)C)ccc3o2)cc1	nan
	16011437	52685	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NCCc4ccccc4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1596645	52685	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NCCc4ccccc4)cc3)nc3cccnc32)cc1	nan
	2110721	52704	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(F)c(F)c2F)c1C	nan
	CHEMBL1596828	52704	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(F)c(F)c2F)c1C	nan
	15991384	52740	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	4	6.2	COc1c(C)cccc1C(=O)Nc1ccc(-c2nc3ccccc3s2)c(Cl)c1	nan
	CHEMBL1597164	52740	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	4	6.2	COc1c(C)cccc1C(=O)Nc1ccc(-c2nc3ccccc3s2)c(Cl)c1	nan
	9397360	52917	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	8	3.6	CCc1nnc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)s1	nan
	CHEMBL1598832	52917	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	8	3.6	CCc1nnc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)s1	nan
	1873710	52939	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	5.3	CCOc1nc(-c2ccc(C)cc2)ccc1-c1noc(-c2ccccc2F)n1	nan
	CHEMBL1599008	52939	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	5.3	CCOc1nc(-c2ccc(C)cc2)ccc1-c1noc(-c2ccccc2F)n1	nan
	16016553	52959	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.1	Cc1cc(C)cc(OCC(=O)Nc2nonc2-c2ccc(Br)cc2)c1	nan
	CHEMBL1599164	52959	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.1	Cc1cc(C)cc(OCC(=O)Nc2nonc2-c2ccc(Br)cc2)c1	nan
	16027417	52979	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	8	4.1	Cc1csc2nc(COC(=O)c3cccc(NC(=O)COc4ccccc4Cl)c3)cc(=O)n12	nan
	CHEMBL1599306	52979	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	8	4.1	Cc1csc2nc(COC(=O)c3cccc(NC(=O)COc4ccccc4Cl)c3)cc(=O)n12	nan
	5059359	53047	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	2	0	6	4.4	Cn1c(=O)c2c(-c3ccccc3)n3c4ccccc4nc(-c4ccccc4)c3c2n(C)c1=O	nan
	CHEMBL1599921	53047	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	2	0	6	4.4	Cn1c(=O)c2c(-c3ccccc3)n3c4ccccc4nc(-c4ccccc4)c3c2n(C)c1=O	nan
	16019821	53128	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1600701	53128	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	16021830	53256	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.4	CSc1ncc(C(=O)Nc2ccc(F)cc2F)c(-c2ccccc2)n1	nan
	CHEMBL1602038	53256	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.4	CSc1ncc(C(=O)Nc2ccc(F)cc2F)c(-c2ccccc2)n1	nan
	4197620	53277	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	6	2.7	COc1ccc(Cl)cc1NC(=O)c1cnc2sccn2c1=O	nan
	CHEMBL1602236	53277	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	6	2.7	COc1ccc(Cl)cc1NC(=O)c1cnc2sccn2c1=O	nan
	16026568	53311	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	4.8	Cc1cc(C)c(NC(=O)C(C)n2c(=O)cc(-c3ccccc3)c3c(C)nn(C)c32)c(C)c1	nan
	CHEMBL1602546	53311	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	4.8	Cc1cc(C)c(NC(=O)C(C)n2c(=O)cc(-c3ccccc3)c3c(C)nn(C)c32)c(C)c1	nan
	1482197	53342	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	5	0	4	4.0	COc1ccc(C(=O)c2ccc(-c3ccc(OC)cc3)nc2)cc1	nan
	CHEMBL1602835	53342	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	5	0	4	4.0	COc1ccc(C(=O)c2ccc(-c3ccc(OC)cc3)nc2)cc1	nan
	16023008	53356	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	7	4.1	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5cccc(F)c5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1602958	53356	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	7	4.1	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5cccc(F)c5)CC4)nnc(C)c3c2C)cc1	nan
	4077604	53422	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.1	O=C(NCC1CCCO1)c1ccc2c(=O)n(-c3ccc(F)cc3)c(=S)[nH]c2c1	nan
	CHEMBL1603522	53422	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.1	O=C(NCC1CCCO1)c1ccc2c(=O)n(-c3ccc(F)cc3)c(=S)[nH]c2c1	nan
	16008430	53498	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	6	0	6	5.0	COc1ccc(N2CCN(C(=O)CCc3c(C)nc4cc(-c5ccc(Cl)cc5)nn4c3C)CC2)cc1	nan
	CHEMBL1604039	53498	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	6	0	6	5.0	COc1ccc(N2CCN(C(=O)CCc3c(C)nc4cc(-c5ccc(Cl)cc5)nn4c3C)CC2)cc1	nan
	2319103	53508	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	7	2	6	4.7	CC(=O)Nc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccc(F)cc3)cc2)cc1	nan
	CHEMBL1604161	53508	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	7	2	6	4.7	CC(=O)Nc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccc(F)cc3)cc2)cc1	nan
	1105833	53567	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	0	2	5.2	N#Cc1c(-c2cccc(F)c2)cc(-c2ccccc2)nc1Br	nan
	CHEMBL1604724	53567	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	0	2	5.2	N#Cc1c(-c2cccc(F)c2)cc(-c2ccccc2)nc1Br	nan
	13283806	53680	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	3	4.2	O=S1(=O)c2ccccc2N(Cc2ccccc2)c2ccccc21	nan
	CHEMBL1605626	53680	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	3	4.2	O=S1(=O)c2ccccc2N(Cc2ccccc2)c2ccccc21	nan
	606829	53761	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	1	2	5.1	Cc1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1606319	53761	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	1	2	5.1	Cc1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	2877673	53801	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	0	4	4.3	CCCC(=O)N1CCN(c2ccc(C(=O)c3ccc(OC)c(Br)c3)cc2F)CC1	nan
	CHEMBL1606636	53801	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	0	4	4.3	CCCC(=O)N1CCN(c2ccc(C(=O)c3ccc(OC)c(Br)c3)cc2F)CC1	nan
	16025505	53865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.1	CC(C)c1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1607091	53865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.1	CC(C)c1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	16019209	53879	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	CHEMBL1607174	53879	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	1166591	53978	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	5.4	COc1ccc(-c2cc(C(F)(F)F)nc(SCCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1608012	53978	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	5.4	COc1ccc(-c2cc(C(F)(F)F)nc(SCCC(=O)Nc3ccccc3F)n2)cc1	nan
	939124	54200	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	6	3.6	CC(=O)c1c(C)nc(Nc2nc3ccccc3s2)nc1C	nan
	CHEMBL1609840	54200	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	6	3.6	CC(=O)c1c(C)nc(Nc2nc3ccccc3s2)nc1C	nan
	15989162	54230	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	10	2	7	3.8	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(CC(=O)Nc2c(C)cc(C)cc2C)c1=O	nan
	CHEMBL1610075	54230	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	10	2	7	3.8	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(CC(=O)Nc2c(C)cc(C)cc2C)c1=O	nan
	2542807	54267	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	4	4.2	Cc1cc(C)c(NC(=O)CSc2nc(C)cc(C)c2C#N)c(C)c1	nan
	CHEMBL1610420	54267	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	4	4.2	Cc1cc(C)c(NC(=O)CSc2nc(C)cc(C)c2C#N)c(C)c1	nan
	1192919	54396	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2ccc(F)cc2)cc1	nan
	CHEMBL1611527	54396	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2ccc(F)cc2)cc1	nan
	16024853	54517	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	4	4.2	O=C(NCCc1ccccc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1612612	54517	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	4	4.2	O=C(NCCc1ccccc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	24789826	54765	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1307717	54765	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1616626	54765	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	135448704	54958	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	CHEMBL1319156	54958	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	CHEMBL1618027	54958	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	3773369	55413	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	CHEMBL1483432	55413	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	CHEMBL1622111	55413	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	6886091	107361	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	1	6	3.2	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3cc4cc(Br)ccc4o3)ccc21	nan
	CHEMBL3192586	107361	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	1	6	3.2	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3cc4cc(Br)ccc4o3)ccc21	nan
	3221539	107420	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	8	0	6	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\CCOC)S3	nan
	CHEMBL3193316	107420	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	8	0	6	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\CCOC)S3	nan
	9615796	107749	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.3	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3ccc(Cl)cc3)ccc21	nan
	CHEMBL3197069	107749	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.3	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3ccc(Cl)cc3)ccc21	nan
	24892226	107839	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	0	9	2.2	COC(=O)Cn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3197975	107839	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	0	9	2.2	COC(=O)Cn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	6341421	107891	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	3	3.6	CCCn1c(C)cs/c1=N\C(=S)Nc1ccccc1	nan
	CHEMBL3198424	107891	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	3	3.6	CCCn1c(C)cs/c1=N\C(=S)Nc1ccccc1	nan
	6065517	108303	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	5	2	4	1.1	CC(C)NC(=O)CC(=O)N/N=C/c1cccs1	nan
	CHEMBL3209441	108303	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	5	2	4	1.1	CC(C)NC(=O)CC(=O)N/N=C/c1cccs1	nan
	135485035	108453	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.9	COc1ccc(Cl)cc1/N=C/c1c(O)oc2ccccc2c1=O	nan
	CHEMBL3211560	108453	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.9	COc1ccc(Cl)cc1/N=C/c1c(O)oc2ccccc2c1=O	nan
	17584634	108656	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	0	5	2.7	COc1ccc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2Cc2ccc(F)cc2)cc1	nan
	CHEMBL3214247	108656	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	0	5	2.7	COc1ccc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2Cc2ccc(F)cc2)cc1	nan
	6869045	112088	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	CHEMBL3194304	112088	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	CHEMBL3301898	112088	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	658981	116550	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	1	5	2.7	CCOC(=O)c1c(N)sc(=S)c2c1CCC2	nan
	CHEMBL3392035	116550	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	1	5	2.7	CCOC(=O)c1c(N)sc(=S)c2c1CCC2	nan
	2241546	119892	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.8	Cc1ccc(C(=O)Nc2nc(-c3ccccc3)ns2)cc1	nan
	CHEMBL353651	119892	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.8	Cc1ccc(C(=O)Nc2nc(-c3ccccc3)ns2)cc1	nan
	878295	172632	29	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	1	1	1	3.8	O=c1cc(-c2ccccc2)c2cc(Cl)ccc2[nH]1	nan
	CHEMBL452292	172632	29	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	1	1	1	3.8	O=c1cc(-c2ccccc2)c2cc(Cl)ccc2[nH]1	nan
	16010872	197383	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	7	4.4	COc1cc2nc(NCCC(C)C)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	CHEMBL587492	197383	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	7	4.4	COc1cc2nc(NCCC(C)C)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	16017892	197441	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	6	3.4	CCOc1ccc(NC(=O)c2sc3nc4n(c(=O)c3c2C)CCC4)cc1	nan
	CHEMBL589232	197441	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	6	3.4	CCOc1ccc(NC(=O)c2sc3nc4n(c(=O)c3c2C)CCC4)cc1	nan
	1370186	197988	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	4	4.8	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ccccc3o2)cc1	nan
	CHEMBL593119	197988	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	4	4.8	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ccccc3o2)cc1	nan
	372	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	8974	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	CHEMBL285819	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	16019683	23860	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.6	Cc1ccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1338399	23860	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.6	Cc1ccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	3486944	24782	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	0	4	2.5	Cc1cc(C=C2C(=O)N(C)C(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	CHEMBL1346519	24782	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	0	4	2.5	Cc1cc(C=C2C(=O)N(C)C(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	665622	29924	7	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	11	2.8	CC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	CHEMBL1390005	29924	7	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	11	2.8	CC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	16019552	34950	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	8	4.1	Cc1ccc(CNc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)cc1	nan
	CHEMBL1435107	34950	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	8	4.1	Cc1ccc(CNc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)cc1	nan
	665286	35337	9	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	3.2	CCC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	CHEMBL1439367	35337	9	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	3.2	CCC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	2054021	35561	15	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	7	3.6	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nccs1	nan
	CHEMBL1441380	35561	15	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	7	3.6	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nccs1	nan
	1395606	35599	9	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	1	5	4.7	CCOc1ccc(-n2nc3ccc(NC(=O)c4ccc(C)cc4C)cc3n2)cc1	nan
	CHEMBL1441729	35599	9	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	1	5	4.7	CCOc1ccc(-n2nc3ccc(NC(=O)c4ccc(C)cc4C)cc3n2)cc1	nan
	997264	38617	5	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	CHEMBL1467097	38617	5	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	1552186	39277	17	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	5	1	4	6.8	Cc1ccc2nc(-c3ccc(NC(=O)COc4ccc(Br)cc4Br)cc3)sc2c1	nan
	CHEMBL1472916	39277	17	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	5	1	4	6.8	Cc1ccc2nc(-c3ccc(NC(=O)COc4ccc(Br)cc4Br)cc3)sc2c1	nan
	16009715	41691	11	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1494680	41691	11	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	16018178	47972	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.5	Cc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	CHEMBL1552994	47972	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.5	Cc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	15991072	52127	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	4	6.3	O=C(Nc1ccc2oc(-c3ccc(Br)cc3)nc2c1)c1cc2ccccc2o1	nan
	CHEMBL1590554	52127	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	4	6.3	O=C(Nc1ccc2oc(-c3ccc(Br)cc3)nc2c1)c1cc2ccccc2o1	nan
	2988582	52315	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	5.1	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)c1ccc(Cl)cc1	nan
	CHEMBL1592961	52315	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	5.1	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)c1ccc(Cl)cc1	nan
	15988483	52378	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	2	4	3.7	CC(=O)c1ccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)cc1	nan
	CHEMBL1593961	52378	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	2	4	3.7	CC(=O)c1ccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)cc1	nan
	1367050	53685	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	6	3.8	CCOc1ccc(-n2nc3ccc(NC(=O)COc4ccccc4)cc3n2)cc1	nan
	CHEMBL1605697	53685	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	6	3.8	CCOc1ccc(-n2nc3ccc(NC(=O)COc4ccccc4)cc3n2)cc1	nan
	4429605	71335	12	None	-1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	0	7	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(S(=O)(=O)N(C)c3ccccc3)cc2)n(C)c1C	nan
	CHEMBL1964939	71335	12	None	-1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	0	7	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(S(=O)(=O)N(C)c3ccccc3)cc2)n(C)c1C	nan
	16010338	5785	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	2	8	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCCNC(C)=O)c2cc(Cl)ccc23)cc1	nan
	CHEMBL1079456	5785	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	2	8	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCCNC(C)=O)c2cc(Cl)ccc23)cc1	nan
	135446757	7955	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.9	O=c1[nH]c(/C=C/c2ccc(Br)cc2)nc2ccccc12	nan
	CHEMBL1091028	7955	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.9	O=c1[nH]c(/C=C/c2ccc(Br)cc2)nc2ccccc12	nan
	250997	10375	3	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	10	3.5	COc1cc(SSc2cc(OC)cc([N+](=O)[O-])c2N)c(N)c([N+](=O)[O-])c1	nan
	CHEMBL116548	10375	3	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	10	3.5	COc1cc(SSc2cc(OC)cc([N+](=O)[O-])c2N)c(N)c([N+](=O)[O-])c1	nan
	16019609	10497	10	None	-223	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)c2ccccc2)c2sccc23)cc1	nan
	CHEMBL1170098	10497	10	None	-223	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)c2ccccc2)c2sccc23)cc1	nan
	16019288	10576	7	None	-234	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	8	4.2	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCC1)c1sccc12	nan
	CHEMBL1170696	10576	7	None	-234	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	8	4.2	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCC1)c1sccc12	nan
	16019546	10595	6	None	-676	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	8	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1sccc12	nan
	CHEMBL1170891	10595	6	None	-676	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	8	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1sccc12	nan
	16019576	10781	6	None	-1995	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	9	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1172726	10781	6	None	-1995	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	9	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	7246142	10806	9	None	-85	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	8	3.6	CC(C)Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	CHEMBL1172934	10806	9	None	-85	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	8	3.6	CC(C)Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	747391	15474	17	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.8	CCOC(=O)c1sc(NC(=O)c2ccco2)nc1-c1ccccc1	nan
	CHEMBL1222145	15474	17	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.8	CCOC(=O)c1sc(NC(=O)c2ccco2)nc1-c1ccccc1	nan
	5309696	19343	1	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	2.8	CCn1c(=O)cc(OCC(=O)Nc2nc(C)cs2)c2ccccc21	nan
	CHEMBL1299766	19343	1	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	2.8	CCn1c(=O)cc(OCC(=O)Nc2nc(C)cs2)c2ccccc21	nan
	1716419	19418	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	5	4.7	CCCCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	CHEMBL1300444	19418	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	5	4.7	CCCCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	135468422	19444	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	2	9	4.4	COc1ccc(NC(=O)CSc2nc3nnc(C)c-3c(N)n2-c2ccc(Cl)c(C)c2)cc1OC	nan
	CHEMBL1300619	19444	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	2	9	4.4	COc1ccc(NC(=O)CSc2nc3nnc(C)c-3c(N)n2-c2ccc(Cl)c(C)c2)cc1OC	nan
	5112617	19596	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	3	4	2.2	CC(C)CC(=O)NC(=S)Nc1sc2c(c1C(N)=O)CCC2	nan
	CHEMBL1301780	19596	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	3	4	2.2	CC(C)CC(=O)NC(=S)Nc1sc2c(c1C(N)=O)CCC2	nan
	1440349	19631	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.4	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1c(C)cccc1C)CCC3	nan
	CHEMBL1302141	19631	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.4	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1c(C)cccc1C)CCC3	nan
	648939	19633	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	CHEMBL1302172	19633	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	3221134	19675	4	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	4.0	COCCN(Cc1cc2cc(C)ccc2n2nnnc12)C(S)=Nc1ccccc1C	nan
	CHEMBL1302436	19675	4	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	4.0	COCCN(Cc1cc2cc(C)ccc2n2nnnc12)C(S)=Nc1ccccc1C	nan
	1864418	19677	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	6	3.5	CC(C)Cc1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	CHEMBL1302453	19677	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	6	3.5	CC(C)Cc1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	22334119	19694	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	8	2	7	2.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCc3ccc(F)cc3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1302552	19694	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	8	2	7	2.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCc3ccc(F)cc3)c3ccccc3c2=O)cc1OC	nan
	1173246	19858	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	2	6	4.2	Cc1ccc(C)c2c1cc(C)c1nnc(SCC(=O)Nc3cccc(C(=O)O)c3)n12	nan
	CHEMBL1303849	19858	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	2	6	4.2	Cc1ccc(C)c2c1cc(C)c1nnc(SCC(=O)Nc3cccc(C(=O)O)c3)n12	nan
	135455179	19977	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	135480855	19977	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	135554164	19977	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	CHEMBL1304888	19977	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	16188302	20058	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	5.4	CCN(C(=O)c1cc2c(O)nc3ccc(C)cc3c2s1)c1cccc(C)c1	nan
	CHEMBL1305636	20058	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	5.4	CCN(C(=O)c1cc2c(O)nc3ccc(C)cc3c2s1)c1cccc(C)c1	nan
	3612019	20116	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	4	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(Cl)s1	nan
	CHEMBL1305985	20116	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	4	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(Cl)s1	nan
	4243407	20278	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	4.8	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NC(c5ccccc5)c5ccccc5)cnc4c3cc2CO1	nan
	CHEMBL1307313	20278	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	4.8	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NC(c5ccccc5)c5ccccc5)cnc4c3cc2CO1	nan
	664182	20323	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	7	4.9	CC(C)c1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	CHEMBL1307669	20323	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	7	4.9	CC(C)c1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	2823681	20434	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	1	4.9	Cc1cc(C)c2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	CHEMBL1308537	20434	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	1	4.9	Cc1cc(C)c2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	135443911	20448	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.5	COc1ccc(N2CC(=O)C(c3nc(-c4ccccc4)cs3)=C2N)cc1	nan
	CHEMBL1308652	20448	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.5	COc1ccc(N2CC(=O)C(c3nc(-c4ccccc4)cs3)=C2N)cc1	nan
	7206305	20521	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	8	2.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc4c(c3)OCO4)nn2)no1	nan
	CHEMBL1309267	20521	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	8	2.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc4c(c3)OCO4)nn2)no1	nan
	546665	20647	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	5	3.0	CC(C)(C)S(=O)(=O)c1cnc(-c2ccc(Cl)cc2)nc1N	nan
	CHEMBL1310343	20647	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	5	3.0	CC(C)(C)S(=O)(=O)c1cnc(-c2ccc(Cl)cc2)nc1N	nan
	54693834	20732	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	5	2.9	CC1CCc2cc(F)cc3c(O)c(C(=O)NCc4ccco4)c(=O)n1c23	nan
	CHEMBL1311072	20732	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	5	2.9	CC1CCc2cc(F)cc3c(O)c(C(=O)NCc4ccco4)c(=O)n1c23	nan
	16746300	20755	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	618	8	0	8	6.1	COc1cc(OC)c2c(-c3ccccc3)cc(=O)oc2c1C(CC(=O)N1CCN(c2ccccc2)CC1)c1ccc2c(c1)OCO2	nan
	CHEMBL1311273	20755	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	618	8	0	8	6.1	COc1cc(OC)c2c(-c3ccccc3)cc(=O)oc2c1C(CC(=O)N1CCN(c2ccccc2)CC1)c1ccc2c(c1)OCO2	nan
	3413238	20757	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	7	2.8	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4ncsc4c3)sc2c1	nan
	CHEMBL1311288	20757	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	7	2.8	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4ncsc4c3)sc2c1	nan
	245201	20771	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	214	3	1	7	0.9	CNc1nc(SC)n(C)c(=O)c1N=O	nan
	CHEMBL1311401	20771	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	214	3	1	7	0.9	CNc1nc(SC)n(C)c(=O)c1N=O	nan
	16194626	20820	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	6	2.6	COc1ccc(N2CCN(C(c3cccs3)C(C)NS(C)(=O)=O)CC2)cc1	nan
	CHEMBL1311746	20820	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	6	2.6	COc1ccc(N2CCN(C(c3cccs3)C(C)NS(C)(=O)=O)CC2)cc1	nan
	3586870	20931	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	3	0	4	3.4	COc1ccc(Oc2cnc3ccccc3n2)cc1	nan
	CHEMBL1312526	20931	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	3	0	4	3.4	COc1ccc(Oc2cnc3ccccc3n2)cc1	nan
	645988	20960	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.3	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccco1	nan
	CHEMBL1312719	20960	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.3	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccco1	nan
	660699	21034	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	2	7	3.6	N#Cc1c(N)nc(SCC(=O)NCCc2ccccc2)c(C#N)c1-c1cccs1	nan
	CHEMBL1313254	21034	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	2	7	3.6	N#Cc1c(N)nc(SCC(=O)NCCc2ccccc2)c(C#N)c1-c1cccs1	nan
	6619041	21036	7	None	-6	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	9	2	8	3.2	CCOc1ccc(NC(=O)CNC(=O)c2nn(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc23)cc1	nan
	CHEMBL1313270	21036	7	None	-6	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	9	2	8	3.2	CCOc1ccc(NC(=O)CNC(=O)c2nn(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc23)cc1	nan
	2731590	21076	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1-c1ccc2c(c1)OCCO2	nan
	CHEMBL1313595	21076	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1-c1ccc2c(c1)OCCO2	nan
	11957277	21093	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	0	8	3.9	O=[N+]([O-])C(/C=C(\Cl)[N+](=O)[O-])=C1N(Cc2ccc(Cl)nc2)CCN1Cc1ccc(Cl)nc1	nan
	CHEMBL1313693	21093	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	0	8	3.9	O=[N+]([O-])C(/C=C(\Cl)[N+](=O)[O-])=C1N(Cc2ccc(Cl)nc2)CCN1Cc1ccc(Cl)nc1	nan
	16012576	21153	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	7	4.1	COc1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(OC)c1	nan
	CHEMBL1314269	21153	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	7	4.1	COc1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(OC)c1	nan
	16020367	21159	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	8	4.4	COC(=O)c1ccccc1NC(=O)c1cc2c(-c3ccc(OC)c(OC)c3)nn(C)c2s1	nan
	CHEMBL1314309	21159	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	8	4.4	COC(=O)c1ccccc1NC(=O)c1cc2c(-c3ccc(OC)c(OC)c3)nn(C)c2s1	nan
	16009631	21162	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	7	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1	nan
	CHEMBL1314331	21162	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	7	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1	nan
	16008545	21163	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	6	4.3	COc1ccc(C(=O)c2cn(Cc3cccc(C)c3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1314337	21163	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	6	4.3	COc1ccc(C(=O)c2cn(Cc3cccc(C)c3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	16018962	21168	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.6	O=C(NCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1314402	21168	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.6	O=C(NCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16026094	21179	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	3.1	CC(C)c1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	CHEMBL1314533	21179	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	3.1	CC(C)c1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	2152595	21193	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	0	7	2.9	COC(=O)c1ccc2c(c1)s/c(=N/C(=O)c1ccc(S(=O)(=O)N3CCCCC3)cc1)n2C	nan
	CHEMBL1314815	21193	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	0	7	2.9	COC(=O)c1ccc2c(c1)s/c(=N/C(=O)c1ccc(S(=O)(=O)N3CCCCC3)cc1)n2C	nan
	135437061	21194	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1Cl	nan
	CHEMBL1314816	21194	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1Cl	nan
	16019424	21199	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	0	8	4.5	CC1CCCN(c2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)C1	nan
	CHEMBL1314919	21199	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	0	8	4.5	CC1CCCN(c2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)C1	nan
	16010115	21203	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	2.8	Cc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	CHEMBL1314966	21203	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	2.8	Cc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	16020210	21208	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	8	2	8	4.0	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	CHEMBL1315042	21208	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	8	2	8	4.0	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	16021834	21220	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2c(C)cccc2C)c(-c2ccccc2)n1	nan
	CHEMBL1315205	21220	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2c(C)cccc2C)c(-c2ccccc2)n1	nan
	3516704	21223	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	7	4.4	CCOCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1315294	21223	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	7	4.4	CCOCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	16009766	21239	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	2	5	6.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c2cc3ccccc3o2)cc1	nan
	CHEMBL1315409	21239	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	2	5	6.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c2cc3ccccc3o2)cc1	nan
	16018863	21246	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	5	3.8	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1Br	nan
	CHEMBL1315473	21246	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	5	3.8	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1Br	nan
	16026940	21264	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1cccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)c1	nan
	CHEMBL1315714	21264	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1cccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)c1	nan
	2808363	21286	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	5	2.7	COC(=O)c1sccc1NC(=O)c1ccc(C#N)cc1	nan
	CHEMBL1315955	21286	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	5	2.7	COC(=O)c1sccc1NC(=O)c1ccc(C#N)cc1	nan
	16019191	21300	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	2	5.2	O=C(CCc1cn(Cc2ccc(F)cc2)c2ccccc12)NC1CCCCC1	nan
	CHEMBL1316117	21300	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	2	5.2	O=C(CCc1cn(Cc2ccc(F)cc2)c2ccccc12)NC1CCCCC1	nan
	16031991	21305	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	4.1	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3sc(C)nc3C)nn2)cc1	nan
	CHEMBL1316148	21305	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	4.1	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3sc(C)nc3C)nn2)cc1	nan
	2135282	21306	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1316149	21306	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	16008335	21311	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	2	6	4.4	O=C(Nc1ccc(C(F)(F)F)cc1)C1CCC(CNS(=O)(=O)c2cccc3nsnc23)CC1	nan
	CHEMBL1316232	21311	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	2	6	4.4	O=C(Nc1ccc(C(F)(F)F)cc1)C1CCC(CNS(=O)(=O)c2cccc3nsnc23)CC1	nan
	16034305	21323	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	5	4.5	CC(C)CCNC(=O)c1cc(-c2cccnc2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12	nan
	CHEMBL1316467	21323	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	5	4.5	CC(C)CCNC(=O)c1cc(-c2cccnc2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12	nan
	3162808	21327	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	6	4.8	COc1ccc(C2CC(=O)c3cnc4c(-c5ccc(F)cc5)c(C)nn4c3C2)cc1OC	nan
	CHEMBL1316500	21327	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	6	4.8	COc1ccc(C2CC(=O)c3cnc4c(-c5ccc(F)cc5)c(C)nn4c3C2)cc1OC	nan
	3674872	21328	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	3.0	CCn1c(SCC(=O)Nc2ccccc2C(=O)OC)nc2ccsc2c1=O	nan
	CHEMBL1316511	21328	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	3.0	CCn1c(SCC(=O)Nc2ccccc2C(=O)OC)nc2ccsc2c1=O	nan
	7223037	21375	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	2	4	4.3	CCc1ccccc1NC(=O)C(=O)NCCc1sc(-c2cccc(C)c2)nc1C	nan
	CHEMBL1317197	21375	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	2	4	4.3	CCc1ccccc1NC(=O)C(=O)NCCc1sc(-c2cccc(C)c2)nc1C	nan
	16026110	21385	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	5	4.2	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	CHEMBL1317332	21385	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	5	4.2	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	7205418	21399	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1ccc(-n2ncc3c(NCc4ccccc4)ncnc32)cc1Cl	nan
	CHEMBL1317524	21399	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1ccc(-n2ncc3c(NCc4ccccc4)ncnc32)cc1Cl	nan
	16008313	21412	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	2	6	4.4	Cc1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccc4nsnc34)CC2)c(Cl)c1	nan
	CHEMBL1317641	21412	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	2	6	4.4	Cc1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccc4nsnc34)CC2)c(Cl)c1	nan
	16026429	21416	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	1	7	1.2	Cc1cc2c(cc1NS(=O)(=O)c1cccc(C#N)c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1317692	21416	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	1	7	1.2	Cc1cc2c(cc1NS(=O)(=O)c1cccc(C#N)c1)n(C)c(=O)c(=O)n2C	nan
	15989759	21428	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	5	3.3	Cc1ccc2nc(NCc3ccc(F)cc3)c3nncn3c2c1	nan
	CHEMBL1317896	21428	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	5	3.3	Cc1ccc2nc(NCc3ccc(F)cc3)c3nncn3c2c1	nan
	16016705	21445	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	2.6	O=C(CCC(=O)N1CCOc2ccccc21)NCc1cccs1	nan
	CHEMBL1318069	21445	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	2.6	O=C(CCC(=O)N1CCOc2ccccc21)NCc1cccs1	nan
	15988587	21452	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NCc1ccccc1Cl	nan
	CHEMBL1318209	21452	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NCc1ccccc1Cl	nan
	7245933	21456	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	3.4	CCOc1ccc(S(=O)(=O)c2cc3cccc(OCC)c3oc2=O)cc1	nan
	CHEMBL1318269	21456	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	3.4	CCOc1ccc(S(=O)(=O)c2cc3cccc(OCC)c3oc2=O)cc1	nan
	1164100	21494	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	0	6	3.4	COc1cccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)c1	nan
	CHEMBL1318572	21494	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	0	6	3.4	COc1cccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)c1	nan
	4077176	21504	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	3	5.6	CCC(C)NC(=O)c1cc(Sc2cccc(Cl)c2)nc2ccccc12	nan
	CHEMBL1318673	21504	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	3	5.6	CCC(C)NC(=O)c1cc(Sc2cccc(Cl)c2)nc2ccccc12	nan
	4055959	21529	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	3.6	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCOCC4)cc3c2C)c(C)c1	nan
	CHEMBL1318877	21529	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	3.6	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCOCC4)cc3c2C)c(C)c1	nan
	16022946	21606	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1319510	21606	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	2967498	21668	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	1	5	3.6	O=C(Nc1nccs1)c1ccc(COc2ccccc2)o1	nan
	CHEMBL1320036	21668	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	1	5	3.6	O=C(Nc1nccs1)c1ccc(COc2ccccc2)o1	nan
	5139336	21682	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	4.4	Cc1cccc2sc(NC(=O)c3ccc(OCC4CCCO4)cc3)nc12	nan
	CHEMBL1320175	21682	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	4.4	Cc1cccc2sc(NC(=O)c3ccc(OCC4CCCO4)cc3)nc12	nan
	16030546	21689	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	3.5	COc1ccccc1C(=O)Nc1cccc(OCc2cc(=O)n3ccccc3n2)c1	nan
	CHEMBL1320207	21689	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	3.5	COc1ccccc1C(=O)Nc1cccc(OCc2cc(=O)n3ccccc3n2)c1	nan
	16030772	21734	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.8	Cn1c(=O)c2c(SCC(=O)NCc3ccco3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1320595	21734	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.8	Cn1c(=O)c2c(SCC(=O)NCc3ccco3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	16016685	21744	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	2	3	4.3	CCCCNC(=O)Nc1ccc2c(c1)N(C)C(=O)c1ccccc1S2	nan
	CHEMBL1320647	21744	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	2	3	4.3	CCCCNC(=O)Nc1ccc2c(c1)N(C)C(=O)c1ccccc1S2	nan
	16033946	21750	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	7	4.4	CCOC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(Cl)c2)cc1	nan
	CHEMBL1320676	21750	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	7	4.4	CCOC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(Cl)c2)cc1	nan
	944701	21756	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	6	2.9	COc1ccc2nc(O)c(COC(=O)c3ccco3)cc2c1	nan
	CHEMBL1320788	21756	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	6	2.9	COc1ccc2nc(O)c(COC(=O)c3ccco3)cc2c1	nan
	5135847	21788	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	2	4	3.8	CCOC(=O)c1cc2c(nc1N=C(S)NCc1ccccc1)CCCC2	nan
	CHEMBL1321064	21788	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	2	4	3.8	CCOC(=O)c1cc2c(nc1N=C(S)NCc1ccccc1)CCCC2	nan
	3634798	21791	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	7	4.5	CCOC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1CCc1ccccc1	nan
	CHEMBL1321100	21791	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	7	4.5	CCOC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1CCc1ccccc1	nan
	6473515	21807	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	2	5	3.1	COc1ccc(S(=O)(=O)Nc2ccccn2)cc1C(=O)Nc1ccccc1	nan
	CHEMBL1321208	21807	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	2	5	3.1	COc1ccc(S(=O)(=O)Nc2ccccn2)cc1C(=O)Nc1ccccc1	nan
	16026080	21842	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1321609	21842	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	661514	21847	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	8	2.7	COc1ccc(-c2nnc3sc(CN4C(=O)c5ccccc5C4=O)nn23)cc1	nan
	CHEMBL1321633	21847	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	8	2.7	COc1ccc(-c2nnc3sc(CN4C(=O)c5ccccc5C4=O)nn23)cc1	nan
	963196	21885	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	5	1	3	4.5	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)c(C)c1	nan
	CHEMBL1321920	21885	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	5	1	3	4.5	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)c(C)c1	nan
	1034156	21888	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	2	4	2.9	Cc1cc2oc(C(=O)NCc3ccc(S(N)(=O)=O)cc3)c(C)c2cc1C	nan
	CHEMBL1321976	21888	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	2	4	2.9	Cc1cc2oc(C(=O)NCc3ccc(S(N)(=O)=O)cc3)c(C)c2cc1C	nan
	16026098	21889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	5	3.7	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	CHEMBL1321983	21889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	5	3.7	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	1480476	21942	23	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1322430	21942	23	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	16021832	22060	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2cccc(C)c2C)c(-c2ccccc2)n1	nan
	CHEMBL1323559	22060	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2cccc(C)c2C)c(-c2ccccc2)n1	nan
	4868391	22107	30	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1Cc1ccccc1	nan
	CHEMBL1323909	22107	30	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1Cc1ccccc1	nan
	7284118	22111	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	5	3.2	CCOc1ccc(CCNC(=O)Cn2ccc3ccccc3c2=O)cc1OCC	nan
	CHEMBL1323924	22111	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	5	3.2	CCOc1ccc(CCNC(=O)Cn2ccc3ccccc3c2=O)cc1OCC	nan
	2135896	22129	4	None	-158	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	2	7	2.4	COc1ccc(OC)c(NC(=O)c2nnn(CCc3ccccc3)c2N)c1	nan
	CHEMBL1324085	22129	4	None	-158	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	2	7	2.4	COc1ccc(OC)c(NC(=O)c2nnn(CCc3ccccc3)c2N)c1	nan
	3422137	22134	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	0	9	2.0	COCCn1c(CN2CCN(C(c3ccccc3)c3ccccc3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1324117	22134	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	0	9	2.0	COCCn1c(CN2CCN(C(c3ccccc3)c3ccccc3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	16015664	22184	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	6	6.6	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(Cl)cc3)on2)cc1	nan
	CHEMBL1324545	22184	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	6	6.6	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(Cl)cc3)on2)cc1	nan
	5299986	22227	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	5	5.1	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1)C1CCN2CC1	nan
	CHEMBL1324899	22227	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	5	5.1	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1)C1CCN2CC1	nan
	2967360	22248	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	4	5.3	Cc1ccc(N(Cc2cc3ccc(C)cc3nc2O)S(=O)(=O)c2ccccc2)c(C)c1	nan
	CHEMBL1325059	22248	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	4	5.3	Cc1ccc(N(Cc2cc3ccc(C)cc3nc2O)S(=O)(=O)c2ccccc2)c(C)c1	nan
	4013085	22266	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.7	CCOC(=O)c1ccc(NC2Nc3cc(C)nn3S2)cc1	nan
	CHEMBL1325232	22266	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.7	CCOC(=O)c1ccc(NC2Nc3cc(C)nn3S2)cc1	nan
	4877095	22284	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.1	CCOC(=O)c1sc(NC(=O)c2cc3c(s2)CCC(C)C3)nc1C	nan
	CHEMBL1325413	22284	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.1	CCOC(=O)c1sc(NC(=O)c2cc3c(s2)CCC(C)C3)nc1C	nan
	16012280	22294	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(C)c1NC(=O)CCS(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1325535	22294	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(C)c1NC(=O)CCS(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	16011188	22307	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.4	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(C)cc1C	nan
	CHEMBL1325716	22307	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.4	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(C)cc1C	nan
	709602	22315	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	2	5	3.6	Cc1c(NC(=O)c2nc[nH]n2)cccc1-c1nc2ccccc2s1	nan
	CHEMBL1325780	22315	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	2	5	3.6	Cc1c(NC(=O)c2nc[nH]n2)cccc1-c1nc2ccccc2s1	nan
	3619431	22378	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	0	4	5.7	O=C(c1cccs1)c1cn(CCOc2ccc(Cl)cc2)c2ccccc12	nan
	CHEMBL1326440	22378	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	0	4	5.7	O=C(c1cccs1)c1cn(CCOc2ccc(Cl)cc2)c2ccccc12	nan
	663870	22385	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1ccc(C(=O)OCc2cc3ccccc3nc2O)cc1	nan
	CHEMBL1326511	22385	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1ccc(C(=O)OCc2cc3ccccc3nc2O)cc1	nan
	16018929	22395	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	11	1	7	3.6	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1OCC	nan
	CHEMBL1326604	22395	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	11	1	7	3.6	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1OCC	nan
	17583882	22404	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	3.5	CCCCc1cc(=O)oc2cc(OCC(=O)Nc3ccccn3)ccc12	nan
	CHEMBL1326654	22404	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	3.5	CCCCc1cc(=O)oc2cc(OCC(=O)Nc3ccccn3)ccc12	nan
	1477181	22447	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	3.7	CC(=O)c1cc(C#N)c(NCc2cc(-c3ccccc3)no2)nc1C	nan
	CHEMBL1327040	22447	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	3.7	CC(=O)c1cc(C#N)c(NCc2cc(-c3ccccc3)no2)nc1C	nan
	16034758	22455	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.6	COc1ccc(NC(=O)c2sc3nc[nH]c(=O)c3c2C)cc1OC	nan
	CHEMBL1327116	22455	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.6	COc1ccc(NC(=O)c2sc3nc[nH]c(=O)c3c2C)cc1OC	nan
	16008896	22463	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1	nan
	CHEMBL1327173	22463	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1	nan
	4227789	22494	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	0	5	5.5	CCN(CC)C(=O)C1CCCN(c2ncnc3c2c(-c2ccccc2)cn3-c2cccc(C)c2)C1	nan
	CHEMBL1327499	22494	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	0	5	5.5	CCN(CC)C(=O)C1CCCN(c2ncnc3c2c(-c2ccccc2)cn3-c2cccc(C)c2)C1	nan
	16032611	22598	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	3	2.9	O=C(NC1CC(=O)N(c2ccc(Cl)cc2)C1)C(=O)c1c[nH]c2ccccc12	nan
	CHEMBL1328167	22598	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	3	2.9	O=C(NC1CC(=O)N(c2ccc(Cl)cc2)C1)C(=O)c1c[nH]c2ccccc12	nan
	1426216	22668	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.1	Cc1cc(=O)n2c(C(=O)Nc3ccc(C(=O)OC(C)C)cc3)c(C(=O)Nc3ccccc3)sc2n1	nan
	CHEMBL1328860	22668	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.1	Cc1cc(=O)n2c(C(=O)Nc3ccc(C(=O)OC(C)C)cc3)c(C(=O)Nc3ccccc3)sc2n1	nan
	857007	22669	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	4	4.2	Cc1cc2cc(C)c(SCC(=O)NCc3ccco3)nc2cc1C	nan
	CHEMBL1328861	22669	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	4	4.2	Cc1cc2cc(C)c(SCC(=O)NCc3ccco3)nc2cc1C	nan
	16015065	22682	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	6	5.3	CC(=O)c1cccc(NC(=O)c2sc(-n3nc(C)c(CCC(C)C)c3C)nc2C)c1	nan
	CHEMBL1328989	22682	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	6	5.3	CC(=O)c1cccc(NC(=O)c2sc(-n3nc(C)c(CCC(C)C)c3C)nc2C)c1	nan
	7294635	22709	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	4	4.7	Nc1c(C(=O)Nc2ccccc2Cl)c2ccccn2c1C(=O)c1ccccc1	nan
	CHEMBL1329216	22709	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	4	4.7	Nc1c(C(=O)Nc2ccccc2Cl)c2ccccn2c1C(=O)c1ccccc1	nan
	2986428	22740	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.0	CC(C)CNc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CC(C)(C)OC3	nan
	CHEMBL1329460	22740	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.0	CC(C)CNc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CC(C)(C)OC3	nan
	7422802	22744	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1ccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)cc1	nan
	CHEMBL1329510	22744	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1ccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)cc1	nan
	7889414	22790	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	10	1.5	CCCn1c(N)c(C(=O)CSc2ncnc3sccc23)c(=O)n(C)c1=O	nan
	CHEMBL1329885	22790	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	10	1.5	CCCn1c(N)c(C(=O)CSc2ncnc3sccc23)c(=O)n(C)c1=O	nan
	1038210	22800	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	0	8	2.7	CCOC(=O)CCSc1nc(N2CCOCC2)c2c(c1C#N)CC(C)(C)OC2	nan
	CHEMBL1329993	22800	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	0	8	2.7	CCOC(=O)CCSc1nc(N2CCOCC2)c2c(c1C#N)CC(C)(C)OC2	nan
	16009180	22847	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCO4)c3ccc(OC)cc3c2=O)cc1	nan
	CHEMBL1330381	22847	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCO4)c3ccc(OC)cc3c2=O)cc1	nan
	1510063	22861	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	3.4	CCC(=O)c1cc2c(cc1NC(=O)c1ccccc1F)OCCO2	nan
	CHEMBL1330472	22861	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	3.4	CCC(=O)c1cc2c(cc1NC(=O)c1ccccc1F)OCCO2	nan
	16019798	22896	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)cc1OC	nan
	CHEMBL1330797	22896	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)cc1OC	nan
	1078194	22945	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	2	5	3.5	Cc1ccc(OCC(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)cc1C	nan
	CHEMBL1331082	22945	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	2	5	3.5	Cc1ccc(OCC(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)cc1C	nan
	1367422	22947	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	6	3.6	O=C(NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1)c1ccco1	nan
	CHEMBL1331090	22947	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	6	3.6	O=C(NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1)c1ccco1	nan
	15990786	22969	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	13	2	5	6.4	CCCCN(CCCNC(=O)c1cc(Nc2ccc(OC)cc2)nc2ccccc12)Cc1ccccc1	nan
	CHEMBL1331246	22969	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	13	2	5	6.4	CCCCN(CCCNC(=O)c1cc(Nc2ccc(OC)cc2)nc2ccccc12)Cc1ccccc1	nan
	1426224	22977	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	2	6	4.1	CCc1ccc(NC(=O)c2c(C(=O)Nc3ccccc3)sc3nc(C)cc(=O)n23)cc1	nan
	CHEMBL1331302	22977	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	2	6	4.1	CCc1ccc(NC(=O)c2c(C(=O)Nc3ccccc3)sc3nc(C)cc(=O)n23)cc1	nan
	16009858	23006	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	2	6	5.7	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3OC)oc3ccccc23)cc1OCC	nan
	CHEMBL1331538	23006	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	2	6	5.7	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3OC)oc3ccccc23)cc1OCC	nan
	965763	23039	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	3.8	Cc1cc(OCC(=O)Nc2ccc3oc(=O)ccc3c2)ccc1Cl	nan
	CHEMBL1331830	23039	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	3.8	Cc1cc(OCC(=O)Nc2ccc3oc(=O)ccc3c2)ccc1Cl	nan
	4216258	23075	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	3	6	6.0	CCOc1ccccc1Nc1sc(C(=O)c2ccccc2)c(N)c1C(=O)Nc1ccccc1	nan
	CHEMBL1332095	23075	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	3	6	6.0	CCOc1ccccc1Nc1sc(C(=O)c2ccccc2)c(N)c1C(=O)Nc1ccccc1	nan
	2670204	23086	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	0	9	1.7	COc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)c(OC)c1	nan
	CHEMBL1332216	23086	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	0	9	1.7	COc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)c(OC)c1	nan
	2151601	23105	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1332323	23105	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	16012517	23109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	5	6.3	CCOc1ccc(-c2cc(NC(=O)Nc3ccccc3C(F)(F)F)c(C(=O)OC)s2)cc1	nan
	CHEMBL1332340	23109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	5	6.3	CCOc1ccc(-c2cc(NC(=O)Nc3ccccc3C(F)(F)F)c(C(=O)OC)s2)cc1	nan
	2243529	23110	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	0	3	3.7	O=C(c1cccs1)N1C(=O)c2cccc3cccc1c23	nan
	CHEMBL1332342	23110	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	0	3	3.7	O=C(c1cccs1)N1C(=O)c2cccc3cccc1c23	nan
	867009	23227	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	3	3.7	COc1ccc(Cl)cc1NC(=O)c1[nH]c(C)c(C(C)=O)c1C	nan
	CHEMBL1333261	23227	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	3	3.7	COc1ccc(Cl)cc1NC(=O)c1[nH]c(C)c(C(C)=O)c1C	nan
	677173	23254	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	2	4	3.5	CCCc1nnc(N=C(S)Nc2ccccc2)s1	nan
	CHEMBL1333504	23254	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	2	4	3.5	CCCc1nnc(N=C(S)Nc2ccccc2)s1	nan
	3623159	23288	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	1	4	5.3	CCOc1ccc(Sc2cc(C(=O)NC(C)CC)c3ccccc3n2)cc1	nan
	CHEMBL1333744	23288	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	1	4	5.3	CCOc1ccc(Sc2cc(C(=O)NC(C)CC)c3ccccc3n2)cc1	nan
	16008956	23326	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	4.2	CCn1c(=O)c2cc(C(=O)NCCc3ccc(OC)c(OC)c3)sc2c2ccccc21	nan
	CHEMBL1334014	23326	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	4.2	CCn1c(=O)c2cc(C(=O)NCCc3ccc(OC)c(OC)c3)sc2c2ccccc21	nan
	2196864	23371	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	4.2	CCn1c(Cc2ccccc2)nnc1SCC(=O)Nc1nc2ccccc2s1	nan
	CHEMBL1334332	23371	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	4.2	CCn1c(Cc2ccccc2)nnc1SCC(=O)Nc1nc2ccccc2s1	nan
	3622707	23444	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1335007	23444	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	16008370	23470	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	4	3.7	Cn1c(=O)cc(SCC(=O)NCc2ccc(F)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1335160	23470	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	4	3.7	Cn1c(=O)cc(SCC(=O)NCc2ccc(F)cc2)c2cc(Cl)ccc21	nan
	16020489	23509	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	5	3.7	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1cccc(C)c1)cn2C	nan
	CHEMBL1335441	23509	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	5	3.7	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1cccc(C)c1)cn2C	nan
	16012518	23513	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	5	5.3	CCOc1ccccc1NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccccc2)c1C	nan
	CHEMBL1335479	23513	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	5	5.3	CCOc1ccccc1NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccccc2)c1C	nan
	16018933	23520	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	7	2.8	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1335514	23520	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	7	2.8	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	16022436	23531	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.2	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3nc2s1	nan
	CHEMBL1335596	23531	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.2	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3nc2s1	nan
	3221114	23571	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	6	1	6	3.3	COCCN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)C1CCCC1	nan
	CHEMBL1335947	23571	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	6	1	6	3.3	COCCN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)C1CCCC1	nan
	16015039	23588	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccccc1NC(=O)c1sc(-n2nc(C)c(Cc3ccc4c(c3)OCO4)c2C)nc1C	nan
	CHEMBL1336092	23588	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccccc1NC(=O)c1sc(-n2nc(C)c(Cc3ccc4c(c3)OCO4)c2C)nc1C	nan
	2138945	23612	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	3.5	O=C(Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1)c1ccc(F)cc1	nan
	CHEMBL1336262	23612	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	3.5	O=C(Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1)c1ccc(F)cc1	nan
	6220215	23669	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C\c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	CHEMBL1336784	23669	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C\c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	16026936	23706	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	9	3.0	O=C(COc1ccccc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1337126	23706	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	9	3.0	O=C(COc1ccccc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	1486592	23758	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	1	7	1.7	COc1ccc(Nc2nc(N(C)C)oc(=O)c2C#N)cc1	nan
	CHEMBL1337568	23758	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	1	7	1.7	COc1ccc(Nc2nc(N(C)C)oc(=O)c2C#N)cc1	nan
	1485789	23779	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	2	4.3	O=C(c1ccc(F)cc1)c1ccc(-c2ccc(F)cc2)nc1	nan
	CHEMBL1337770	23779	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	2	4.3	O=C(c1ccc(F)cc1)c1ccc(-c2ccc(F)cc2)nc1	nan
	16033861	23813	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	8	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	CHEMBL1338096	23813	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	8	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	1265732	23865	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	4	5.4	O=C(Cn1c(S)nc(-c2ccccc2)c1-c1ccccc1)c1ccccc1	nan
	CHEMBL1338427	23865	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	4	5.4	O=C(Cn1c(S)nc(-c2ccccc2)c1-c1ccccc1)c1ccccc1	nan
	16026086	23922	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	7	2.3	Cc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1339014	23922	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	7	2.3	Cc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	15944700	24131	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	2	5	4.4	O=C(Nc1cc(Cl)cc(Cl)c1)c1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1	nan
	CHEMBL1340950	24131	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	2	5	4.4	O=C(Nc1cc(Cl)cc(Cl)c1)c1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1	nan
	5069163	24146	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	7	2.9	COc1ccc(CNC(=O)CCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1341068	24146	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	7	2.9	COc1ccc(CNC(=O)CCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)cc1	nan
	855559	24269	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	3.5	CCN(C(=O)c1ccco1)c1nnc(-c2ccc(OC)cc2)s1	nan
	CHEMBL1342076	24269	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	3.5	CCN(C(=O)c1ccco1)c1nnc(-c2ccc(OC)cc2)s1	nan
	3149126	24283	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	10	2	7	3.5	CCOCCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2ccccc2c1=O	nan
	CHEMBL1342207	24283	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	10	2	7	3.5	CCOCCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2ccccc2c1=O	nan
	1086862	24302	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	7	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccc(OC)c(OC)c3)s2)cc1	nan
	CHEMBL1342348	24302	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	7	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccc(OC)c(OC)c3)s2)cc1	nan
	5443591	24341	7	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	8	1	6	3.8	CCOC(=O)/C(C#N)=C\c1ccc(OCC(=O)Nc2ccc(C)cc2C)c(OC)c1	nan
	CHEMBL1342661	24341	7	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	8	1	6	3.8	CCOC(=O)/C(C#N)=C\c1ccc(OCC(=O)Nc2ccc(C)cc2C)c(OC)c1	nan
	665611	24378	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	6	3.9	Cc1cc(-c2nnc3sc(-c4ccc(Cl)cc4Cl)nn23)[nH]n1	nan
	CHEMBL1342889	24378	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	6	3.9	Cc1cc(-c2nnc3sc(-c4ccc(Cl)cc4Cl)nn23)[nH]n1	nan
	5063932	24436	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	5	3.6	O=C(NCc1ccco1)c1ccc2c(=O)n(-c3ccccc3)c(=S)[nH]c2c1	nan
	CHEMBL1343363	24436	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	5	3.6	O=C(NCc1ccco1)c1ccc2c(=O)n(-c3ccccc3)c(=S)[nH]c2c1	nan
	2452051	24585	4	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	4.6	N#Cc1ccc(CSc2nnc(NC(=O)c3ccc4ncsc4c3)s2)cc1	nan
	CHEMBL1344739	24585	4	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	4.6	N#Cc1ccc(CSc2nnc(NC(=O)c3ccc4ncsc4c3)s2)cc1	nan
	2335388	24673	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	2	1	5	3.0	Cc1ccnc(NC(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)c1	nan
	CHEMBL1345474	24673	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	2	1	5	3.0	Cc1ccnc(NC(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)c1	nan
	666154	24674	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	6	4.2	Cc1ccc(-n2nc(C)c3c(-c4cccs4)c(C#N)c(N)nc32)cc1	nan
	CHEMBL1345487	24674	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	6	4.2	Cc1ccc(-n2nc(C)c3c(-c4cccs4)c(C#N)c(N)nc32)cc1	nan
	2040126	24679	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	2	6	2.6	Cc1ccc(/C=C2\SC(=S)N(CCC(=O)NNS(=O)(=O)c3ccccc3)C2=O)cc1	nan
	CHEMBL1345551	24679	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	2	6	2.6	Cc1ccc(/C=C2\SC(=S)N(CCC(=O)NNS(=O)(=O)c3ccccc3)C2=O)cc1	nan
	3185713	24752	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	10	3	8	3.1	CCc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NCC1CCCO1)c1ccc(N(C)C)cc1	nan
	CHEMBL1346198	24752	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	10	3	8	3.1	CCc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NCC1CCCO1)c1ccc(N(C)C)cc1	nan
	1409877	24814	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(NC(=O)COC(=O)c2ccc3c(c2)OCO3)c1C	nan
	CHEMBL1346710	24814	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(NC(=O)COC(=O)c2ccc3c(c2)OCO3)c1C	nan
	3846689	24832	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	6	2.4	COCc1nc2oc3ccc(F)cc3c(=O)c2cc1C(=O)OC	nan
	CHEMBL1346831	24832	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	6	2.4	COCc1nc2oc3ccc(F)cc3c(=O)c2cc1C(=O)OC	nan
	2813569	24881	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	6	3.3	O=C(COc1ncnc2cc(Cl)ccc12)c1ccc2c(c1)OCCO2	nan
	CHEMBL1347186	24881	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	6	3.3	O=C(COc1ncnc2cc(Cl)ccc12)c1ccc2c(c1)OCCO2	nan
	2426514	24942	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	1	0	5	2.6	Cc1cc(=O)n2nc(-c3ccccc3)sc2c1C#N	nan
	CHEMBL1347674	24942	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	1	0	5	2.6	Cc1cc(=O)n2nc(-c3ccccc3)sc2c1C#N	nan
	2950848	25015	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.2	COCc1cc(C)nc(SCC(=O)NC2CCCCC2C)c1C#N	nan
	CHEMBL1348333	25015	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.2	COCc1cc(C)nc(SCC(=O)NC2CCCCC2C)c1C#N	nan
	664720	25060	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	7	5.4	CC(C)c1nc2sc3c(NCc4ccco4)ncnc3c2c2c1COC(C)(C)C2	nan
	CHEMBL1348840	25060	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	7	5.4	CC(C)c1nc2sc3c(NCc4ccco4)ncnc3c2c2c1COC(C)(C)C2	nan
	780682	25165	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	3	3.8	C=CCn1c(NC(=O)c2ccc(C)cc2)nc2ccccc21	nan
	CHEMBL1349635	25165	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	3	3.8	C=CCn1c(NC(=O)c2ccc(C)cc2)nc2ccccc21	nan
	7157934	25276	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	1.6	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	CHEMBL1350603	25276	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	1.6	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	16194401	25377	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	2	6	2.8	CCOC(=O)N1CCC(NC(=O)c2cc3c(O)nc4ccccc4c3n2C)CC1	nan
	CHEMBL1351462	25377	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	2	6	2.8	CCOC(=O)N1CCC(NC(=O)c2cc3c(O)nc4ccccc4c3n2C)CC1	nan
	1433829	25509	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	5	1	5	2.5	COc1ccc2nc(SCC(=O)NC3CC3)c(C#N)cc2c1	nan
	CHEMBL1352517	25509	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	5	1	5	2.5	COc1ccc2nc(SCC(=O)NC3CC3)c(C#N)cc2c1	nan
	5112429	25542	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	2	7	1.9	N#CCC(=O)NNc1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]	nan
	CHEMBL1352781	25542	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	2	7	1.9	N#CCC(=O)NNc1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]	nan
	4850085	25573	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	2	8	2.8	CCOC(=O)c1sc2nc(C)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2c1C	nan
	CHEMBL1353043	25573	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	2	8	2.8	CCOC(=O)c1sc2nc(C)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2c1C	nan
	3350830	25715	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	2	4	4.7	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(Cl)c1	nan
	CHEMBL1354025	25715	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	2	4	4.7	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(Cl)c1	nan
	16017542	25758	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	7	3.6	CCN(c1ccc(C)cc1C)S(=O)(=O)c1nnc(NC(=O)c2ccccc2OC)s1	nan
	CHEMBL1354338	25758	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	7	3.6	CCN(c1ccc(C)cc1C)S(=O)(=O)c1nnc(NC(=O)c2ccccc2OC)s1	nan
	3415736	25772	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	2	6	2.3	COc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCC4)cc23)c(OC)c1	nan
	CHEMBL1354486	25772	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	2	6	2.3	COc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCC4)cc23)c(OC)c1	nan
	16008465	25779	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	4	4.5	Cc1nc2cc(-c3cccc(F)c3)nn2c(C)c1CCC(=O)NC1CCCCC1	nan
	CHEMBL1354574	25779	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	4	4.5	Cc1nc2cc(-c3cccc(F)c3)nn2c(C)c1CCC(=O)NC1CCCCC1	nan
	16008364	25780	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	1	4	5.0	Cc1ccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c(Br)c1	nan
	CHEMBL1354597	25780	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	1	4	5.0	Cc1ccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c(Br)c1	nan
	16034362	25782	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	9	1	9	2.1	CSCCC(NS(=O)(=O)c1ccc2c(c1)oc(=O)n2C)C(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1354617	25782	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	9	1	9	2.1	CSCCC(NS(=O)(=O)c1ccc2c(c1)oc(=O)n2C)C(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	16029590	25787	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	1	3	5.8	O=C(Nc1ccc(Br)cc1F)c1ccc2nc(CCc3ccccc3)oc2c1	nan
	CHEMBL1354702	25787	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	1	3	5.8	O=C(Nc1ccc(Br)cc1F)c1ccc2nc(CCc3ccccc3)oc2c1	nan
	16024765	25792	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	1	4	3.8	O=C(Cn1c(=O)c(C(F)(F)F)nc2ccccc21)Nc1cccc(Br)c1	nan
	CHEMBL1354803	25792	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	1	4	3.8	O=C(Cn1c(=O)c(C(F)(F)F)nc2ccccc21)Nc1cccc(Br)c1	nan
	16026345	25798	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	2.6	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)NC(C)C)c32)cc1	nan
	CHEMBL1354863	25798	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	2.6	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)NC(C)C)c32)cc1	nan
	7872437	25800	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	3	6	3.8	CC(=O)Nc1ccc(NC(=O)CCc2nc(O)c3c4c(sc3n2)CCCC4)cc1	nan
	CHEMBL1354869	25800	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	3	6	3.8	CC(=O)Nc1ccc(NC(=O)CCc2nc(O)c3c4c(sc3n2)CCCC4)cc1	nan
	2135022	25810	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.3	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(C)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1354981	25810	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.3	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(C)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	135416424	25813	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	3	2	6	4.8	Cc1ccc2oc(-c3cc(NC(=O)c4ccc5c(c4)OCCO5)cc(C)c3O)nc2c1	nan
	CHEMBL1355004	25813	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	3	2	6	4.8	Cc1ccc2oc(-c3cc(NC(=O)c4ccc5c(c4)OCCO5)cc(C)c3O)nc2c1	nan
	16019041	25832	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	6	3.2	CC(C)OCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1355237	25832	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	6	3.2	CC(C)OCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	135437043	25842	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	3	7	3.3	CCOc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1	nan
	CHEMBL1355309	25842	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	3	7	3.3	CCOc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1	nan
	16011751	25847	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	7	3.3	CCOC(=O)c1ccc(NC(=O)CC(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1	nan
	CHEMBL1355424	25847	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	7	3.3	CCOC(=O)c1ccc(NC(=O)CC(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1	nan
	16027630	25850	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1355500	25850	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	16025481	25855	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	3.4	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1355611	25855	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	3.4	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	16020103	25863	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	4.2	CCOc1ccc(CNC(=O)c2nn(-c3ccc(OC)cc3)c(=O)c3c2c2ccccc2n3C)cc1	nan
	CHEMBL1355692	25863	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	4.2	CCOc1ccc(CNC(=O)c2nn(-c3ccc(OC)cc3)c(=O)c3c2c2ccccc2n3C)cc1	nan
	16026942	25869	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1ccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)cc1	nan
	CHEMBL1355764	25869	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1ccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)cc1	nan
	16011703	25873	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	3.6	COc1ccc(CCNc2nc3ccc(Cl)cc3n3cnnc23)cc1OC	nan
	CHEMBL1355798	25873	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	3.6	COc1ccc(CCNc2nc3ccc(Cl)cc3n3cnnc23)cc1OC	nan
	16026082	25874	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	CHEMBL1355799	25874	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	16027128	25901	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	3	0	4	4.6	Cc1cc(=O)n(Cc2cccc(Br)c2)c2c1c(C)nn2-c1ccccc1	nan
	CHEMBL1356158	25901	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	3	0	4	4.6	Cc1cc(=O)n(Cc2cccc(Br)c2)c2c1c(C)nn2-c1ccccc1	nan
	16020942	25909	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	3	5.4	CC(NC(=O)Cn1c(-c2cccs2)cc2cc(F)ccc21)c1ccccc1	nan
	CHEMBL1356228	25909	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	3	5.4	CC(NC(=O)Cn1c(-c2cccs2)cc2cc(F)ccc21)c1ccccc1	nan
	2869380	25926	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	2	3	5.9	O=C(Nc1sc2c(c1C(=O)Nc1ccccc1Cl)CCCC2)c1ccccc1F	nan
	CHEMBL1356452	25926	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	2	3	5.9	O=C(Nc1sc2c(c1C(=O)Nc1ccccc1Cl)CCCC2)c1ccccc1F	nan
	4802695	25932	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	3	5	2.2	O=C(COC(=O)c1cc(Cl)ccc1O)NC(=O)NCc1ccccc1	nan
	CHEMBL1356574	25932	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	3	5	2.2	O=C(COC(=O)c1cc(Cl)ccc1O)NC(=O)NCc1ccccc1	nan
	16015066	25939	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1nc(SCC(=O)Nc2ccccc2Cl)cc(-c2ccccc2)n1	nan
	CHEMBL1356682	25939	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1nc(SCC(=O)Nc2ccccc2Cl)cc(-c2ccccc2)n1	nan
	16018801	25953	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	2	7	1.0	NS(=O)(=O)c1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1356848	25953	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	2	7	1.0	NS(=O)(=O)c1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	24687225	25958	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	8	0	8	3.1	COc1cccc(COC(=O)c2cc(S(=O)(=O)N3CCCCC3)ccc2N2CCOCC2)c1OC	nan
	CHEMBL1356898	25958	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	8	0	8	3.1	COc1cccc(COC(=O)c2cc(S(=O)(=O)N3CCCCC3)ccc2N2CCOCC2)c1OC	nan
	16015534	25963	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	4.3	CCOC(=O)CSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	CHEMBL1357001	25963	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	4.3	CCOC(=O)CSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	15989556	25964	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	1	9	2.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1357013	25964	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	1	9	2.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	16025511	25978	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.0	CCN1c2ccccc2-c2nc(SCC(=O)Nc3cccc(C)c3C)ncc2S1(=O)=O	nan
	CHEMBL1357149	25978	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.0	CCN1c2ccccc2-c2nc(SCC(=O)Nc3cccc(C)c3C)ncc2S1(=O)=O	nan
	20903553	25996	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	6	3.0	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1357354	25996	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	6	3.0	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	16031127	26007	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.2	CSc1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	CHEMBL1357550	26007	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.2	CSc1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	1146087	26011	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	4.7	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(F)cc3)n2)cc1	nan
	CHEMBL1357694	26011	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	4.7	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(F)cc3)n2)cc1	nan
	16027571	26032	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	9	2.9	CS(=O)(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1358013	26032	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	9	2.9	CS(=O)(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16027432	26042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	1	9	3.1	Cc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	CHEMBL1358125	26042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	1	9	3.1	Cc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	16012175	26046	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	4.7	Cc1ccccc1Cn1c2ccccc2c2cnn(CC(=O)NCCc3ccc(Cl)cc3)c(=O)c21	nan
	CHEMBL1358188	26046	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	4.7	Cc1ccccc1Cn1c2ccccc2c2cnn(CC(=O)NCCc3ccc(Cl)cc3)c(=O)c21	nan
	16011822	26051	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.2	CCOc1ccc(NC(=O)C2CCN(c3nnc(-n4c(C)ccc4C)s3)CC2)cc1	nan
	CHEMBL1358209	26051	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.2	CCOc1ccc(NC(=O)C2CCN(c3nnc(-n4c(C)ccc4C)s3)CC2)cc1	nan
	16015787	26052	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	6	6.0	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(C)c(F)c4)oc4ccccc34)no2)cc1	nan
	CHEMBL1358232	26052	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	6	6.0	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(C)c(F)c4)oc4ccccc34)no2)cc1	nan
	16009454	26087	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	CC(Oc1ccccc1)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1358685	26087	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	CC(Oc1ccccc1)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	16022826	26109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.7	CCOc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)cc1	nan
	CHEMBL1358850	26109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.7	CCOc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)cc1	nan
	654435	26131	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	6	4.2	O=C(CSc1nc2ccccc2o1)Nc1nc2ccccc2s1	nan
	CHEMBL1359027	26131	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	6	4.2	O=C(CSc1nc2ccccc2o1)Nc1nc2ccccc2s1	nan
	16009817	26138	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	1	7	5.0	Brc1cccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)c1	nan
	CHEMBL1359062	26138	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	1	7	5.0	Brc1cccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)c1	nan
	16009648	26210	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	5	4.3	COc1ccc(Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1359678	26210	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	5	4.3	COc1ccc(Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16020569	26246	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	5	4.3	CCCn1cc(S(=O)(=O)c2ccc(C)cc2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	CHEMBL1360010	26246	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	5	4.3	CCCn1cc(S(=O)(=O)c2ccc(C)cc2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	135546909	26258	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	6	3.7	COc1ccc(CN2CCc3nc(SCC(=O)Nc4cc(C)cc(C)c4)[nH]c(=O)c3C2)cc1	nan
	CHEMBL1360113	26258	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	6	3.7	COc1ccc(CN2CCc3nc(SCC(=O)Nc4cc(C)cc(C)c4)[nH]c(=O)c3C2)cc1	nan
	3185716	26282	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	10	3	8	3.7	CC(C)c1ccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)cc1	nan
	CHEMBL1360292	26282	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	10	3	8	3.7	CC(C)c1ccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)cc1	nan
	2819025	26301	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	1	1	5	1.9	N#Cc1cnc2cc(-c3ccccc3)nn2c1N	nan
	CHEMBL1360465	26301	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	1	1	5	1.9	N#Cc1cnc2cc(-c3ccccc3)nn2c1N	nan
	2141195	26322	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.7	CCc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccccc1)cn2CC(=O)Nc1cc(C)ccc1C	nan
	CHEMBL1360707	26322	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.7	CCc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccccc1)cn2CC(=O)Nc1cc(C)ccc1C	nan
	135436940	26324	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	7	5.0	Oc1cc(-c2ccc(F)cc2)nc(SCc2nc(-c3cccc(Cl)c3)no2)n1	nan
	CHEMBL1360713	26324	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	7	5.0	Oc1cc(-c2ccc(F)cc2)nc(SCc2nc(-c3cccc(Cl)c3)no2)n1	nan
	16009483	26343	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	9	1	7	1.4	CCCCN(C)CCNC(=O)C1CCCN(S(=O)(=O)c2ccc3c(c2)oc(=O)n3C)C1	nan
	CHEMBL1360843	26343	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	9	1	7	1.4	CCCCN(C)CCNC(=O)C1CCCN(S(=O)(=O)c2ccc3c(c2)oc(=O)n3C)C1	nan
	2135565	26394	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3ccc(F)cc3c2=O)cc1	nan
	CHEMBL1361368	26394	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3ccc(F)cc3c2=O)cc1	nan
	7598414	26456	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1cccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)c1	nan
	CHEMBL1361891	26456	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1cccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)c1	nan
	1071174	26458	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	8	1	7	3.8	CCOc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1361894	26458	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	8	1	7	3.8	CCOc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3ccccc3c2=O)cc1	nan
	857565	26523	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	4.2	Cc1cc(NC(=O)CSc2nc3c(C)c(C)ccc3cc2C)no1	nan
	CHEMBL1362451	26523	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	4.2	Cc1cc(NC(=O)CSc2nc3c(C)c(C)ccc3cc2C)no1	nan
	790083	26621	50	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	0	4	4.2	COc1ccccc1-c1nc(-c2ccc(Br)cc2)no1	nan
	CHEMBL1363291	26621	50	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	0	4	4.2	COc1ccccc1-c1nc(-c2ccc(Br)cc2)no1	nan
	2137970	26680	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3ccccc3)c3ccc(Cl)cc3c2=O)cc1	nan
	CHEMBL1363852	26680	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3ccccc3)c3ccc(Cl)cc3c2=O)cc1	nan
	22522543	26729	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	1	4	3.2	Cc1ccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)cc1	nan
	CHEMBL1364334	26729	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	1	4	3.2	Cc1ccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)cc1	nan
	1581690	26770	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	10	2	6	4.6	CCCCCOc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3cc(C)on3)cc2)cc1	nan
	CHEMBL1364631	26770	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	10	2	6	4.6	CCCCCOc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3cc(C)on3)cc2)cc1	nan
	1759638	26798	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	5	1	5	5.3	Cc1c(CCC(=O)N2CCC(C(=O)O)(c3ccccc3)CC2)c(=O)oc2cc3oc4c(c3cc12)CCCC4	nan
	CHEMBL1364853	26798	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	5	1	5	5.3	Cc1c(CCC(=O)N2CCC(C(=O)O)(c3ccccc3)CC2)c(=O)oc2cc3oc4c(c3cc12)CCCC4	nan
	2137118	26899	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	1	6	4.2	COc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccc(F)cc1)cn2CC(=O)Nc1ccc(C)cc1C	nan
	CHEMBL1365673	26899	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	1	6	4.2	COc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccc(F)cc1)cn2CC(=O)Nc1ccc(C)cc1C	nan
	16008395	26925	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	6	3.7	CCn1c(=O)cc(OCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2ccccc21	nan
	CHEMBL1365942	26925	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	6	3.7	CCn1c(=O)cc(OCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2ccccc21	nan
	2155747	26934	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	7	1	8	3.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)on3)o2)cc1	nan
	CHEMBL1366006	26934	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	7	1	8	3.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)on3)o2)cc1	nan
	16012964	26936	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	3	5.0	CCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	CHEMBL1366015	26936	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	3	5.0	CCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	2474394	26988	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	3.5	CCCn1c(=O)[nH]c(=O)c2c(C(F)(F)F)cc(-c3ccc(C)cc3)nc21	nan
	CHEMBL1366444	26988	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	3.5	CCCn1c(=O)[nH]c(=O)c2c(C(F)(F)F)cc(-c3ccc(C)cc3)nc21	nan
	17757029	27020	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	0	8	4.6	CCOC(=O)COc1ccc([N+](=O)[O-])cc1-c1ccnc2cc(-c3ccc(Cl)cc3)nn12	nan
	CHEMBL1366773	27020	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	0	8	4.6	CCOC(=O)COc1ccc([N+](=O)[O-])cc1-c1ccnc2cc(-c3ccc(Cl)cc3)nn12	nan
	5087310	27172	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	7	2.8	COc1cc2c(cc1OC)n(CC(=O)NC1CCCCCC1)n1c(C)cc(=O)nc21	nan
	CHEMBL1367963	27172	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	7	2.8	COc1cc2c(cc1OC)n(CC(=O)NC1CCCCCC1)n1c(C)cc(=O)nc21	nan
	4825943	27181	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	2.8	CC(Sc1nc2ccccc2c(=O)n1C)C(=O)Nc1ccc2c(c1)OCCO2	nan
	CHEMBL1368013	27181	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	2.8	CC(Sc1nc2ccccc2c(=O)n1C)C(=O)Nc1ccc2c(c1)OCCO2	nan
	16022825	27201	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	10	1.9	Cc1ccc(C)c(NC(=O)Cn2c(=O)n(Cc3nc(C)no3)c(=O)c3cc4c(cc32)OCO4)c1	nan
	CHEMBL1368194	27201	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	10	1.9	Cc1ccc(C)c(NC(=O)Cn2c(=O)n(Cc3nc(C)no3)c(=O)c3cc4c(cc32)OCO4)c1	nan
	709853	27244	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.7	COc1ccc(CNC(=O)c2cc3cccc(OC)c3oc2=O)cc1	nan
	CHEMBL1368522	27244	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.7	COc1ccc(CNC(=O)c2cc3cccc(OC)c3oc2=O)cc1	nan
	16019023	27264	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	8	1	6	2.9	CCOCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1368698	27264	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	8	1	6	2.9	CCOCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	1898787	27279	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	1.9	COC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	CHEMBL1368847	27279	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	1.9	COC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	16746213	27293	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	11	3	5	4.4	NC(=O)CC(NC(=O)Cc1ccc(Br)cc1)c1ccc(NCCc2ccccc2F)c([N+](=O)[O-])c1	nan
	CHEMBL1368944	27293	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	11	3	5	4.4	NC(=O)CC(NC(=O)Cc1ccc(Br)cc1)c1ccc(NCCc2ccccc2F)c([N+](=O)[O-])c1	nan
	15989069	27295	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	12	1	9	2.7	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	CHEMBL1368950	27295	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	12	1	9	2.7	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	3417357	27335	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	0	6	4.9	Cc1cc(C)c(Cn2c(=O)n(-c3ccccc3Cl)c(=O)c3c(C)c(C(=O)N(C)C)sc32)c(C)c1	nan
	CHEMBL1369202	27335	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	0	6	4.9	Cc1cc(C)c(Cn2c(=O)n(-c3ccccc3Cl)c(=O)c3c(C)c(C(=O)N(C)C)sc32)c(C)c1	nan
	4454678	27363	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	4.4	Cc1cc(OCC(=O)Nc2cc(-c3nn4c(C)nnc4s3)ccc2C)ccc1Cl	nan
	CHEMBL1369422	27363	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	4.4	Cc1cc(OCC(=O)Nc2cc(-c3nn4c(C)nnc4s3)ccc2C)ccc1Cl	nan
	16034378	27441	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	7	1	4	3.5	COc1ccc(C(=O)CCC(=O)Nc2cccc(C(C)=O)c2)cc1	nan
	CHEMBL1369934	27441	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	7	1	4	3.5	COc1ccc(C(=O)CCC(=O)Nc2cccc(C(C)=O)c2)cc1	nan
	16746462	27462	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	8	1	6	3.3	COc1cc(O)c(C(CCN2CCOCC2)c2ccc(N(C)C)cc2)c(OC)c1	nan
	CHEMBL1370067	27462	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	8	1	6	3.3	COc1cc(O)c(C(CCN2CCOCC2)c2ccc(N(C)C)cc2)c(OC)c1	nan
	3236293	27464	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	8	3.3	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccsc2c1=O	nan
	CHEMBL1370078	27464	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	8	3.3	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccsc2c1=O	nan
	5310561	27516	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.8	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccc(F)cc3)c2n1	nan
	CHEMBL1370473	27516	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.8	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccc(F)cc3)c2n1	nan
	667326	27529	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	5	3.5	CCOCCCNc1ncc2c(n1)CC(c1ccc(C)cc1)CC2=O	nan
	CHEMBL1370544	27529	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	5	3.5	CCOCCCNc1ncc2c(n1)CC(c1ccc(C)cc1)CC2=O	nan
	135546918	27542	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	3.6	CCCN1CCc2nc(SCC(=O)Nc3ccc(C)c(Cl)c3)nc(O)c2C1	nan
	CHEMBL1370635	27542	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	3.6	CCCN1CCc2nc(SCC(=O)Nc3ccc(C)c(Cl)c3)nc(O)c2C1	nan
	3628612	27573	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.4	CCc1nc(SCC(=O)NCCc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1370855	27573	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.4	CCc1nc(SCC(=O)NCCc2ccccc2)c2oc3ccccc3c2n1	nan
	1348188	27719	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1cccc(-c2nc3cc(NC(=O)Cc4ccc(Cl)cc4)ccc3o2)c1	nan
	CHEMBL1372034	27719	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1cccc(-c2nc3cc(NC(=O)Cc4ccc(Cl)cc4)ccc3o2)c1	nan
	1854798	27744	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	1	0	5	3.6	Cn1c(=O)nc2n(-c3ccc(Br)cc3)c3cccc(Cl)c3cc-2c1=O	nan
	CHEMBL1372184	27744	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	1	0	5	3.6	Cn1c(=O)nc2n(-c3ccc(Br)cc3)c3cccc(Cl)c3cc-2c1=O	nan
	16019423	27814	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	9	5.0	CC(C)c1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1372659	27814	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	9	5.0	CC(C)c1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	16031591	27874	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	6	3.4	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc(-c4coc(C)n4)cc3)CC2)cc1	nan
	CHEMBL1373010	27874	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	6	3.4	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc(-c4coc(C)n4)cc3)CC2)cc1	nan
	2684697	27948	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	5	3.7	COc1ccc(C)cc1NC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3	nan
	CHEMBL1373515	27948	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	5	3.7	COc1ccc(C)cc1NC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3	nan
	652717	27964	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	5	5.1	CCN1CCCC1CN(Cc1cc2cc(C)cc(C)c2nc1O)C(=O)Nc1ccccc1OC	nan
	CHEMBL1373605	27964	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	5	5.1	CCN1CCCC1CN(Cc1cc2cc(C)cc(C)c2nc1O)C(=O)Nc1ccccc1OC	nan
	16015413	27975	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	CHEMBL1373657	27975	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	16033161	28011	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	2	5	4.6	O=C(Nc1ccc(N2CCN(CCOc3ccc(Cl)cc3)CC2)c(C(=O)O)c1)c1ccc(F)cc1	nan
	CHEMBL1373926	28011	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	2	5	4.6	O=C(Nc1ccc(N2CCN(CCOc3ccc(Cl)cc3)CC2)c(C(=O)O)c1)c1ccc(F)cc1	nan
	16030696	28017	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	2.9	CC(=O)c1ccc(NC(=O)CSc2nc(-c3ccccc3C)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1374004	28017	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	2.9	CC(=O)c1ccc(NC(=O)CSc2nc(-c3ccccc3C)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	15997814	28062	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	6	4.2	COc1cc2nc(S)nc(NCc3cccc(Cl)c3)c2cc1OC	nan
	CHEMBL1374312	28062	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	6	4.2	COc1cc2nc(S)nc(NCc3cccc(Cl)c3)c2cc1OC	nan
	4521283	28069	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	4	1	5	4.7	O=C(CN1C(=O)c2ccccc2Sc2ccc(C(=O)N3CCOCC3)cc21)Nc1ccc(Cl)cc1F	nan
	CHEMBL1374381	28069	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	4	1	5	4.7	O=C(CN1C(=O)c2ccccc2Sc2ccc(C(=O)N3CCOCC3)cc21)Nc1ccc(Cl)cc1F	nan
	3734127	28107	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	4	4.0	CCc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1	nan
	CHEMBL1374637	28107	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	4	4.0	CCc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1	nan
	669593	28122	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	1	5	2.1	O=C(Nc1nccs1)c1ccc2c(c1)OCO2	nan
	CHEMBL1374723	28122	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	1	5	2.1	O=C(Nc1nccs1)c1ccc2c(c1)OCO2	nan
	656234	28163	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	3.3	O=c1c2ccccc2nc(CSc2[nH]cnc3ncnc2-3)n1-c1ccccc1	nan
	CHEMBL1375001	28163	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	3.3	O=c1c2ccccc2nc(CSc2[nH]cnc3ncnc2-3)n1-c1ccccc1	nan
	4074625	28177	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	3	6	0.3	COC(=O)c1ccccc1NC=C1C(=O)NC(=S)NC1=O	nan
	CHEMBL1375120	28177	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	3	6	0.3	COC(=O)c1ccccc1NC=C1C(=O)NC(=S)NC1=O	nan
	828451	28277	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	1	4	4.6	CCOc1ccc(Nc2nc3c(C)cccc3cc2C#N)cc1	nan
	CHEMBL1375831	28277	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	1	4	4.6	CCOc1ccc(Nc2nc3c(C)cccc3cc2C#N)cc1	nan
	7246250	28282	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	3	0	5	3.4	COc1cc(Br)cc2cc(S(=O)(=O)c3ccccc3)c(=O)oc12	nan
	CHEMBL1375897	28282	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	3	0	5	3.4	COc1cc(Br)cc2cc(S(=O)(=O)c3ccccc3)c(=O)oc12	nan
	16029523	28304	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	0	6	2.3	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3ccc(F)cc3)CC1)CCS2	nan
	CHEMBL1376205	28304	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	0	6	2.3	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3ccc(F)cc3)CC1)CCS2	nan
	4048244	28332	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	13	1	8	4.1	CCOC(=O)c1sc(-c2ccccc2)cc1NC(=O)c1ccc(S(=O)(=O)N(CCOC)CCOC)cc1	nan
	CHEMBL1376427	28332	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	13	1	8	4.1	CCOC(=O)c1sc(-c2ccccc2)cc1NC(=O)c1ccc(S(=O)(=O)N(CCOC)CCOC)cc1	nan
	1629947	28371	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	4	1.6	O=C1NC(=S)NC(=O)C1=Cc1ccc2c(c1)CCN2CCCCl	nan
	CHEMBL1376754	28371	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	4	1.6	O=C1NC(=S)NC(=O)C1=Cc1ccc2c(c1)CCN2CCCCl	nan
	1281315	28387	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	2	6	6.1	COc1ccc(-c2c3c(nc4sc(C(=O)Nc5ccccc5F)c(N)c24)CC(C)(C)CC3=O)cc1	nan
	CHEMBL1376941	28387	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	2	6	6.1	COc1ccc(-c2c3c(nc4sc(C(=O)Nc5ccccc5F)c(N)c24)CC(C)(C)CC3=O)cc1	nan
	3640458	28411	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	1	7	3.6	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C)C2	nan
	CHEMBL1377235	28411	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	1	7	3.6	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C)C2	nan
	4307577	28447	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	10	2	4	6.4	CC(C)c1ccc(Nc2cc(C(=O)NCCCN(C)Cc3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1377592	28447	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	10	2	4	6.4	CC(C)c1ccc(Nc2cc(C(=O)NCCCN(C)Cc3ccccc3)c3ccccc3n2)cc1	nan
	16193746	28527	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	1	6	2.3	Cc1ccc(N2C(=O)C3C4C=CC(CN=C(S)N5CCN(c6ccccn6)CC5)(O4)C3C2=O)cc1	nan
	CHEMBL1378295	28527	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	1	6	2.3	Cc1ccc(N2C(=O)C3C4C=CC(CN=C(S)N5CCN(c6ccccn6)CC5)(O4)C3C2=O)cc1	nan
	2220966	28569	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	3	3.4	Cc1c(Cl)ccc2c(C(N)=O)cc(-c3ccccn3)nc12	nan
	CHEMBL1378741	28569	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	3	3.4	Cc1c(Cl)ccc2c(C(N)=O)cc(-c3ccccn3)nc12	nan
	7422753	28584	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	4	2.2	NC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1	nan
	CHEMBL1378862	28584	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	4	2.2	NC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1	nan
	2815317	28592	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.8	Cc1cc(C)c2c(n1)sc1c(=O)n(Cc3ccc(F)cc3)cnc12	nan
	CHEMBL1378935	28592	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.8	Cc1cc(C)c2c(n1)sc1c(=O)n(Cc3ccc(F)cc3)cnc12	nan
	16193948	28608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	3.5	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1379050	28608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	3.5	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(c2ccccn2)CC1	nan
	24746968	28729	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.1	Cc1nc(Nc2ccccc2F)c2nnn(Cc3ccccc3Cl)c2n1	nan
	CHEMBL1380147	28729	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.1	Cc1nc(Nc2ccccc2F)c2nnn(Cc3ccccc3Cl)c2n1	nan
	725312	28752	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	3.0	CCn1cnc2sc(C(=O)Nc3ccccc3OC)c(C)c2c1=O	nan
	CHEMBL1380313	28752	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	3.0	CCn1cnc2sc(C(=O)Nc3ccccc3OC)c(C)c2c1=O	nan
	24792708	28785	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	7	3.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)c3ccccc3F)s2)cc1	nan
	CHEMBL1380537	28785	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	7	3.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)c3ccccc3F)s2)cc1	nan
	3604840	28815	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	CHEMBL1380782	28815	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	1980822	28968	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	4	3.9	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C)n2)cc1	nan
	CHEMBL1382084	28968	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	4	3.9	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C)n2)cc1	nan
	555289	29028	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	4	3.6	Cc1cc(C)c(C#N)c(SCC(=O)Nc2ccccc2C)n1	nan
	CHEMBL1382619	29028	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	4	3.6	Cc1cc(C)c(C#N)c(SCC(=O)Nc2ccccc2C)n1	nan
	9550495	29224	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccc(-c2nc3ncccc3o2)cc1NC(=O)COc1ccccc1	nan
	CHEMBL1384380	29224	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccc(-c2nc3ncccc3o2)cc1NC(=O)COc1ccccc1	nan
	7161160	29241	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	7	0.3	CCOc1ccccc1NS(=O)(=O)c1cn(C)c(=O)n(C)c1=O	nan
	CHEMBL1384530	29241	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	7	0.3	CCOc1ccccc1NS(=O)(=O)c1cn(C)c(=O)n(C)c1=O	nan
	4271811	29296	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	0	5	3.2	CCCc1nc2ccccc2c(=O)n1CC(=O)c1ccc(OC)cc1	nan
	CHEMBL1384958	29296	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	0	5	3.2	CCCc1nc2ccccc2c(=O)n1CC(=O)c1ccc(OC)cc1	nan
	2123263	29305	7	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	9	3.5	CCCn1c(N)c(-c2nc(C3CCCC3)c(C(=O)c3ccc(NC(C)=O)cc3)s2)c(=O)n(C)c1=O	nan
	CHEMBL1385062	29305	7	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	9	3.5	CCCn1c(N)c(-c2nc(C3CCCC3)c(C(=O)c3ccc(NC(C)=O)cc3)s2)c(=O)n(C)c1=O	nan
	3243476	29351	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	3.4	CC(=O)Nc1nc2c(c3c1c(=O)oc1ccccc13)CC(C)CC2	nan
	CHEMBL1385469	29351	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	3.4	CC(=O)Nc1nc2c(c3c1c(=O)oc1ccccc13)CC(C)CC2	nan
	645034	29403	4	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.9	N#Cc1cc2cc3c(cc2nc1N1CCCCC1)OCCO3	nan
	CHEMBL1385946	29403	4	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.9	N#Cc1cc2cc3c(cc2nc1N1CCCCC1)OCCO3	nan
	1233014	29424	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.4	Cc1ccc(C#N)c(SCC(=O)Nc2nccs2)n1	nan
	CHEMBL1386142	29424	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.4	Cc1ccc(C#N)c(SCC(=O)Nc2nccs2)n1	nan
	818106	29452	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	4	4.0	COc1ccc(-c2nc3c4ccccc4ccn3c2C=O)cc1	nan
	CHEMBL1386316	29452	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	4	4.0	COc1ccc(-c2nc3c4ccccc4ccn3c2C=O)cc1	nan
	2803005	29455	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.8	NC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1386328	29455	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.8	NC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	743778	29489	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	3	3.2	Cc1cc(-c2ccc(Cl)cc2)c(C#N)c(N)n1	nan
	CHEMBL1386595	29489	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	3	3.2	Cc1cc(-c2ccc(Cl)cc2)c(C#N)c(N)n1	nan
	1078300	29493	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3cccc(C)c3)c(=O)c2c1C	nan
	CHEMBL1386617	29493	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3cccc(C)c3)c(=O)c2c1C	nan
	2197659	29545	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.6	COc1ccc2c(c1)c(=O)oc1cc(OCC(=O)NC3CC3)ccc12	nan
	CHEMBL1387003	29545	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.6	COc1ccc2c(c1)c(=O)oc1cc(OCC(=O)NC3CC3)ccc12	nan
	2368754	29567	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	0	4	2.1	CCN1C(=O)C(=C2C=C(C)OC(C)=C2)C(=O)N(CC)C1=S	nan
	CHEMBL1387204	29567	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	0	4	2.1	CCN1C(=O)C(=C2C=C(C)OC(C)=C2)C(=O)N(CC)C1=S	nan
	1590813	29612	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	1	5.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc(-c2ccccc2)cc1	nan
	CHEMBL1387594	29612	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	1	5.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc(-c2ccccc2)cc1	nan
	16194196	29625	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	8	2.6	CCOC(=O)N1CCN(C(=O)CCCCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)CC1	nan
	CHEMBL1387679	29625	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	8	2.6	CCOC(=O)N1CCN(C(=O)CCCCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)CC1	nan
	3961803	29647	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	8	-0.6	Cn1nc(C(=O)OCC(=O)NC2CCS(=O)(=O)C2)c2ccccc2c1=O	nan
	CHEMBL1387823	29647	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	8	-0.6	Cn1nc(C(=O)OCC(=O)NC2CCS(=O)(=O)C2)c2ccccc2c1=O	nan
	649021	29696	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.8	Cc1cccc2cc(C(c3nnnn3Cc3ccc4c(c3)OCO4)N3CCC(C)CC3)c(O)nc12	nan
	CHEMBL1388237	29696	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.8	Cc1cccc2cc(C(c3nnnn3Cc3ccc4c(c3)OCO4)N3CCC(C)CC3)c(O)nc12	nan
	2565451	29713	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	2.1	CCOC(=O)c1sc(NC(=O)c2ccc(S(=O)(=O)N(C)C)cc2)nc1C	nan
	CHEMBL1388388	29713	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	2.1	CCOC(=O)c1sc(NC(=O)c2ccc(S(=O)(=O)N(C)C)cc2)nc1C	nan
	20874214	29740	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	3.7	CC(C)c1nn2c(=O)cc(COc3cccc(NC(=O)c4ccco4)c3)nc2s1	nan
	CHEMBL1388517	29740	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	3.7	CC(C)c1nn2c(=O)cc(COc3cccc(NC(=O)c4ccco4)c3)nc2s1	nan
	736044	29799	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	2	5	1.3	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)OCO3)cc1	nan
	CHEMBL1389015	29799	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	2	5	1.3	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)OCO3)cc1	nan
	3581200	29868	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	5	4.9	O=C(Nc1nc(-c2ccc(F)c(F)c2)cs1)c1ccc(OCC2CCCO2)cc1	nan
	CHEMBL1389543	29868	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	5	4.9	O=C(Nc1nc(-c2ccc(F)c(F)c2)cs1)c1ccc(OCC2CCCO2)cc1	nan
	2815149	29984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	1	0	4	3.3	Cn1c2ccccc2n2c(=O)cc(-c3ccccc3)c(C#N)c12	nan
	CHEMBL1390567	29984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	1	0	4	3.3	Cn1c2ccccc2n2c(=O)cc(-c3ccccc3)c(C#N)c12	nan
	1480454	30130	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	5	3.1	CN(C)c1nc(-c2cccnc2)nc(-c2ccccc2)c1C#N	nan
	CHEMBL1391874	30130	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	5	3.1	CN(C)c1nc(-c2cccnc2)nc(-c2ccccc2)c1C#N	nan
	3151961	30140	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	6	2.6	CC(C)c1nnc(NC(=O)c2ccc3c(c2)OCO3)s1	nan
	CHEMBL1391972	30140	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	6	2.6	CC(C)c1nnc(NC(=O)c2ccc3c(c2)OCO3)s1	nan
	2818919	30280	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	5	5.2	FC(F)(F)c1cc(-c2cccs2)nc2cc(-c3cccs3)nn12	nan
	CHEMBL1393159	30280	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	5	5.2	FC(F)(F)c1cc(-c2cccs2)nc2cc(-c3cccs3)nn12	nan
	3597887	30287	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	4.2	Cc1ccc(-c2nc(S(=O)(=O)c3ccc(C)cc3)c(SCC(=O)NCC3CCCO3)o2)cc1	nan
	CHEMBL1393192	30287	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	4.2	Cc1ccc(-c2nc(S(=O)(=O)c3ccc(C)cc3)c(SCC(=O)NCC3CCCO3)o2)cc1	nan
	6498520	30337	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	6	2.9	CN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)CC(C)(C)CN(C)C	nan
	CHEMBL1393589	30337	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	6	2.9	CN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)CC(C)(C)CN(C)C	nan
	938851	30370	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	1	5	3.7	Cc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	CHEMBL1393863	30370	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	1	5	3.7	Cc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	2810066	30380	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	2.9	COc1cc2nc(NC(=O)c3ccccc3)sc(=O)c2cc1OC	nan
	CHEMBL1393944	30380	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	2.9	COc1cc2nc(NC(=O)c3ccccc3)sc(=O)c2cc1OC	nan
	16010814	30392	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	3	0	7	4.3	Clc1cccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)c1	nan
	CHEMBL1394069	30392	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	3	0	7	4.3	Clc1cccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)c1	nan
	16018745	30406	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	3	5.9	Cc1ccc(Cn2c(C(=O)O)c(CNCc3ccccc3Cl)c3ccc(C)cc32)cc1	nan
	CHEMBL1394183	30406	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	3	5.9	Cc1ccc(Cn2c(C(=O)O)c(CNCc3ccccc3Cl)c3ccc(C)cc32)cc1	nan
	16030321	30407	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	3.8	COc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	CHEMBL1394221	30407	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	3.8	COc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	16019476	30409	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	4.4	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1394231	30409	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	4.4	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	16012300	30414	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1ccc(NC(=O)c2ccc(-c3ccccc3)s2)cc1	nan
	CHEMBL1394287	30414	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1ccc(NC(=O)c2ccc(-c3ccccc3)s2)cc1	nan
	16015419	30445	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	8	1	6	6.3	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(C)cc3)cc2s1	nan
	CHEMBL1394800	30445	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	8	1	6	6.3	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(C)cc3)cc2s1	nan
	5297365	30454	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1cccc(C(F)(F)F)c1)C1CCN2CC1	nan
	CHEMBL1394905	30454	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1cccc(C(F)(F)F)c1)C1CCN2CC1	nan
	1308289	30455	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	0	6	4.2	CCS(=O)(=O)c1c(S(=O)(=O)CC)c2cc(C(C)(C)C)ccn2c1C(=O)c1ccc(F)cc1	nan
	CHEMBL1394907	30455	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	0	6	4.2	CCS(=O)(=O)c1c(S(=O)(=O)CC)c2cc(C(C)(C)C)ccn2c1C(=O)c1ccc(F)cc1	nan
	7338094	30469	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1ccn2c(Nc3ccccc3C)c(-c3ccc(N4CCOCC4)cc3)nc2c1	nan
	CHEMBL1395018	30469	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1ccn2c(Nc3ccccc3C)c(-c3ccc(N4CCOCC4)cc3)nc2c1	nan
	1598875	30471	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	7	3.4	COC(=O)c1ccccc1NC(=O)CSc1nc2sc3c(c2c(=O)[nH]1)CCCC3	nan
	CHEMBL1395042	30471	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	7	3.4	COC(=O)c1ccccc1NC(=O)CSc1nc2sc3c(c2c(=O)[nH]1)CCCC3	nan
	705204	30481	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	1	1	5	3.7	N#Cc1c(N)n(-c2cccc(Cl)c2)c2nc3ccccc3nc12	nan
	CHEMBL1395126	30481	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	1	1	5	3.7	N#Cc1c(N)n(-c2cccc(Cl)c2)c2nc3ccccc3nc12	nan
	16011870	30487	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	6	6.9	Cc1oc(-c2ccccc2F)nc1Cn1c(SCc2cccc(C(F)(F)F)c2)nc2ccncc21	nan
	CHEMBL1395173	30487	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	6	6.9	Cc1oc(-c2ccccc2F)nc1Cn1c(SCc2cccc(C(F)(F)F)c2)nc2ccncc21	nan
	16011750	30488	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	4.2	CCC(C(=O)NCc1cc(OC)ccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1395174	30488	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	4.2	CCC(C(=O)NCc1cc(OC)ccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	7150993	30490	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	Cc1ccc2nc(NC(=O)CSc3nccn3Cc3ccccc3)sc2c1	nan
	CHEMBL1395184	30490	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	Cc1ccc2nc(NC(=O)CSc3nccn3Cc3ccccc3)sc2c1	nan
	16022376	30516	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	4.7	O=C(CSc1nc2ccsc2c(=O)n1Cc1ccc(F)cc1)NCc1ccc(Cl)cc1	nan
	CHEMBL1395536	30516	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	4.7	O=C(CSc1nc2ccsc2c(=O)n1Cc1ccc(F)cc1)NCc1ccc(Cl)cc1	nan
	16008365	30543	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.9	COc1cccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c1	nan
	CHEMBL1395994	30543	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.9	COc1cccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c1	nan
	16016520	30551	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	2	2	3.4	Cc1cccc(NC(=O)c2ccc3[nH]c(C)cc(=O)c3c2)c1	nan
	CHEMBL1396103	30551	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	2	2	3.4	Cc1cccc(NC(=O)c2ccc3[nH]c(C)cc(=O)c3c2)c1	nan
	16012961	30573	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	3.2	COc1ccc(Cc2nc3c4cnn(-c5cccc(F)c5)c4ncn3n2)cc1	nan
	CHEMBL1396439	30573	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	3.2	COc1ccc(Cc2nc3c4cnn(-c5cccc(F)c5)c4ncn3n2)cc1	nan
	16011203	30593	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	3.8	CCc1nn(CC(=O)Nc2c(C)cc(C)cc2C)c(=O)c2cc3sccc3n12	nan
	CHEMBL1396725	30593	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	3.8	CCc1nn(CC(=O)Nc2c(C)cc(C)cc2C)c(=O)c2cc3sccc3n12	nan
	5300039	30617	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	2	5	4.7	Nc1c(C(=O)Nc2ccc(Br)cc2F)sc2nc3c(cc12)N1CCC3CC1	nan
	CHEMBL1397016	30617	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	2	5	4.7	Nc1c(C(=O)Nc2ccc(Br)cc2F)sc2nc3c(cc12)N1CCC3CC1	nan
	16029565	30631	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	4.0	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(F)ccc32)c1	nan
	CHEMBL1397193	30631	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	4.0	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(F)ccc32)c1	nan
	9114471	30644	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	7	1.5	N#Cc1cc(C#N)c(SCC(=O)N2CC(=O)Nc3ccccc32)nc1N	nan
	CHEMBL1397378	30644	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	7	1.5	N#Cc1cc(C#N)c(SCC(=O)N2CC(=O)Nc3ccccc32)nc1N	nan
	16029539	30648	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	5	4.7	Cc1ccc2c(c1)c(=O)c(C(=O)c1ccncc1)cn2CC(=O)Nc1ccc(C(C)C)cc1	nan
	CHEMBL1397433	30648	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	5	4.7	Cc1ccc2c(c1)c(=O)c(C(=O)c1ccncc1)cn2CC(=O)Nc1ccc(C(C)C)cc1	nan
	16021836	30651	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.1	CSc1ncc(C(=O)NCc2ccc(C)cc2)c(-c2ccccc2)n1	nan
	CHEMBL1397498	30651	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.1	CSc1ncc(C(=O)NCc2ccc(C)cc2)c(-c2ccccc2)n1	nan
	16024513	30653	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C)cc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1397525	30653	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C)cc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	4069971	30679	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	4	5.3	CCCCNC(=O)c1cc(Sc2ccc(OCC)cc2)nc2ccccc12	nan
	CHEMBL1397896	30679	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	4	5.3	CCCCNC(=O)c1cc(Sc2ccc(OCC)cc2)nc2ccccc12	nan
	402652	30697	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	6	3.7	O=c1c2ccccc2nc2sc(Nc3cccc(Cl)c3)nn12	nan
	CHEMBL1398128	30697	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	6	3.7	O=c1c2ccccc2nc2sc(Nc3cccc(Cl)c3)nn12	nan
	15988651	30698	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	4	3.8	O=C(Nc1cccc(C(F)(F)F)c1)C1CCN(S(=O)(=O)c2cccs2)CC1	nan
	CHEMBL1398130	30698	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	4	3.8	O=C(Nc1cccc(C(F)(F)F)c1)C1CCN(S(=O)(=O)c2cccs2)CC1	nan
	135455820	30709	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	5	4.6	Oc1ncnc2c1sc1nc(C(F)F)cc(-c3ccccc3)c12	nan
	CHEMBL1398293	30709	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	5	4.6	Oc1ncnc2c1sc1nc(C(F)F)cc(-c3ccccc3)c12	nan
	16019015	30720	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	6	1	5	3.5	CC(C)CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1398441	30720	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	6	1	5	3.5	CC(C)CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16032326	30737	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	6	5.9	CN1CCc2c(sc(NC(=O)CSc3ccc(F)cc3)c2-c2nc3ccccc3s2)C1	nan
	CHEMBL1398567	30737	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	6	5.9	CN1CCc2c(sc(NC(=O)CSc3ccc(F)cc3)c2-c2nc3ccccc3s2)C1	nan
	2105201	30765	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	8	1	9	4.9	CCOC(=O)c1c(NC(=O)CSc2nc3ccccc3c(=O)n2-c2ccccc2)sc(C(C)=O)c1C	nan
	CHEMBL1398840	30765	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	8	1	9	4.9	CCOC(=O)c1c(NC(=O)CSc2nc3ccccc3c(=O)n2-c2ccccc2)sc(C(C)=O)c1C	nan
	16021149	30810	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	5	5.8	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccccc3)nc3cccnc32)cc1	nan
	CHEMBL1399300	30810	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	5	5.8	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccccc3)nc3cccnc32)cc1	nan
	8351751	30838	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	0	8	2.1	CCOc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	CHEMBL1399515	30838	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	0	8	2.1	CCOc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	1386490	30852	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	0	5	4.8	COc1cccc(OCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)c1	nan
	CHEMBL1399670	30852	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	0	5	4.8	COc1cccc(OCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)c1	nan
	16007871	30863	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	1	4	5.2	O=C(NCc1ccco1)c1ccc2c(c1)N(Cc1ccc(Cl)cc1)C(=O)c1ccccc1[S+]2[O-]	nan
	CHEMBL1399777	30863	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	1	4	5.2	O=C(NCc1ccco1)c1ccc2c(c1)N(Cc1ccc(Cl)cc1)C(=O)c1ccccc1[S+]2[O-]	nan
	16011403	30865	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	5	6.0	O=C(NCc1ccc(F)cc1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1399789	30865	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	5	6.0	O=C(NCc1ccc(F)cc1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	7293305	30868	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	5	3.6	COCCn1ccc2c(OCC(=O)Nc3c(C)cc(C)cc3C)cccc2c1=O	nan
	CHEMBL1399845	30868	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	5	3.6	COCCn1ccc2c(OCC(=O)Nc3c(C)cc(C)cc3C)cccc2c1=O	nan
	16030115	31005	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.4	CCc1cccc(C)c1NC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	CHEMBL1401110	31005	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.4	CCc1cccc(C)c1NC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	1163266	31019	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	1	1	5	2.2	Cc1ccc(-c2cc3ncc(C#N)c(N)n3n2)cc1	nan
	CHEMBL1401234	31019	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	1	1	5	2.2	Cc1ccc(-c2cc3ncc(C#N)c(N)n3n2)cc1	nan
	16024855	31041	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	3	1	4	5.1	Cc1cc(C)cc(NC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	CHEMBL1401368	31041	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	3	1	4	5.1	Cc1cc(C)cc(NC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	16011339	31147	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	2	5	5.2	CCOC(=O)c1ccccc1NC(=O)NC(C)c1c(-n2cccc2)sc(C)c1C	nan
	CHEMBL1402306	31147	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	2	5	5.2	CCOC(=O)c1ccccc1NC(=O)NC(C)c1c(-n2cccc2)sc(C)c1C	nan
	16019019	31157	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	3.7	O=C(NCCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1402402	31157	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	3.7	O=C(NCCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16011789	31231	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	5	3.6	Cc1ccc(-n2ncc3c(=O)n(Cc4ccccc4C)cnc32)cc1C	nan
	CHEMBL1403021	31231	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	5	3.6	Cc1ccc(-n2ncc3c(=O)n(Cc4ccccc4C)cnc32)cc1C	nan
	7096324	31248	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	2	3	2.5	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)CCCC3)cc1	nan
	CHEMBL1403204	31248	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	2	3	2.5	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)CCCC3)cc1	nan
	135437062	31273	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	6	3.5	CCC(C)NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1ccc(C)c(Cl)c1	nan
	CHEMBL1403479	31273	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	6	3.5	CCC(C)NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1ccc(C)c(Cl)c1	nan
	16026084	31334	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	1	7	2.1	O=C(Nc1cccc(F)c1)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1404065	31334	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	1	7	2.1	O=C(Nc1cccc(F)c1)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	15999042	31370	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	2.8	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sccc21)NC1CCCCC1	nan
	CHEMBL1404291	31370	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	2.8	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sccc21)NC1CCCCC1	nan
	1617675	31412	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	3	0	5	6.2	Cc1cccc(-c2nc3c4c(-c5ccccc5)c(-c5ccccc5)oc4ncn3n2)c1	nan
	CHEMBL1404812	31412	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	3	0	5	6.2	Cc1cccc(-c2nc3c4c(-c5ccccc5)c(-c5ccccc5)oc4ncn3n2)c1	nan
	2390567	31446	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	6	2.9	N#Cc1ccsc1NC(=O)COC(=O)c1cc(Br)ccc1O	nan
	CHEMBL1405202	31446	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	6	2.9	N#Cc1ccsc1NC(=O)COC(=O)c1cc(Br)ccc1O	nan
	15988048	31506	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	10	2	9	2.1	COc1cc2c(=O)n(CCC(=O)NCC3CCCO3)c(=O)n(CC(=O)Nc3c(C)cccc3C)c2cc1OC	nan
	CHEMBL1405772	31506	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	10	2	9	2.1	COc1cc2c(=O)n(CCC(=O)NCC3CCCO3)c(=O)n(CC(=O)Nc3c(C)cccc3C)c2cc1OC	nan
	16024912	31510	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.5	Cc1ccccc1CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1405829	31510	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.5	Cc1ccccc1CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	2991576	31711	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	6	2.6	CCCCc1nc2sc3c(=O)n(N)cnc3c2c2c1CCC2	nan
	CHEMBL1407541	31711	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	6	2.6	CCCCc1nc2sc3c(=O)n(N)cnc3c2c2c1CCC2	nan
	3583749	31748	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	7	3.0	COC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)sc2c1CCN(C)C2	nan
	CHEMBL1407736	31748	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	7	3.0	COC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)sc2c1CCN(C)C2	nan
	3245299	31758	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	2	7	2.7	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccccc3)c2n1	nan
	CHEMBL1407835	31758	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	2	7	2.7	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccccc3)c2n1	nan
	6485917	31807	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	9	1	8	2.6	COc1ccc(CNCCSc2nnnn2-c2ccccc2)c(OC)c1	nan
	CHEMBL1408179	31807	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	9	1	8	2.6	COc1ccc(CNCCSc2nnnn2-c2ccccc2)c(OC)c1	nan
	2265197	31816	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	2	2	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1)c1ccccc1F	nan
	CHEMBL1408256	31816	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	2	2	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1)c1ccccc1F	nan
	15989388	31901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	7	1	6	3.3	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(=O)N3CCc4ccccc4C3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1408914	31901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	7	1	6	3.3	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(=O)N3CCc4ccccc4C3)c(=O)c3ccccc32)cc1	nan
	1082765	31990	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	8	1	6	2.9	COc1ccc(CCNC(=O)COc2ccc3c(C)cc(=O)oc3c2)cc1OC	nan
	CHEMBL1409638	31990	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	8	1	6	2.9	COc1ccc(CCNC(=O)COc2ccc3c(C)cc(=O)oc3c2)cc1OC	nan
	1913870	32017	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	2	6	3.1	O=C(/C=C\Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1)c1ccccc1	nan
	CHEMBL1409860	32017	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	2	6	3.1	O=C(/C=C\Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1)c1ccccc1	nan
	2527257	32070	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	7	2	7	1.7	COc1ccc(C(=O)OCC(=O)Nc2sccc2C(N)=O)cc1OC	nan
	CHEMBL1410234	32070	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	7	2	7	1.7	COc1ccc(C(=O)OCC(=O)Nc2sccc2C(N)=O)cc1OC	nan
	2201015	32080	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	3.3	Cc1ccc(-n2c3c(cc(C(=O)NCC(=O)c4ccccc4)c2=O)C(=O)CCC3)cc1	nan
	CHEMBL1410319	32080	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	3.3	Cc1ccc(-n2c3c(cc(C(=O)NCC(=O)c4ccccc4)c2=O)C(=O)CCC3)cc1	nan
	2135385	32112	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	7	4.1	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1410565	32112	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	7	4.1	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	1160042	32132	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	0	5	3.9	Cc1cc(C)c(C#N)c(SCCS(=O)(=O)Cc2ccc(Cl)cc2)n1	nan
	CHEMBL1410783	32132	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	0	5	3.9	Cc1cc(C)c(C#N)c(SCCS(=O)(=O)Cc2ccc(Cl)cc2)n1	nan
	16232595	32144	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.1	Cc1cc(C)c(C#N)c(SCC(=O)Nc2cccc(S(=O)(=O)N3CCCC3)c2)n1	nan
	CHEMBL1410891	32144	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.1	Cc1cc(C)c(C#N)c(SCC(=O)Nc2cccc(S(=O)(=O)N3CCCC3)c2)n1	nan
	1963060	32158	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	0	6	2.6	COCCn1c(-c2ccccc2)nc2c(c(=O)c3ccccc3n2C)c1=O	nan
	CHEMBL1411041	32158	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	0	6	2.6	COCCn1c(-c2ccccc2)nc2c(c(=O)c3ccccc3n2C)c1=O	nan
	1301263	32200	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	6	4.6	COc1ccc(CC(=O)Nc2ccc(-c3nnc(-c4ccccc4)o3)cc2)cc1OC	nan
	CHEMBL1411349	32200	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	6	4.6	COc1ccc(CC(=O)Nc2ccc(-c3nnc(-c4ccccc4)o3)cc2)cc1OC	nan
	2353143	32377	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	4.4	COc1cc(SC)ccc1C(=O)Nc1ncc(Cl)cc1Cl	nan
	CHEMBL1412778	32377	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	4.4	COc1cc(SC)ccc1C(=O)Nc1ncc(Cl)cc1Cl	nan
	135402203	32454	13	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	1	6	3.5	COc1ccc(OCCSc2nc(O)c3ccccc3n2)cc1	nan
	CHEMBL1413382	32454	13	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	1	6	3.5	COc1ccc(OCCSc2nc(O)c3ccccc3n2)cc1	nan
	8722509	32472	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	7	3.6	CC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2C2CC2)cc1	nan
	CHEMBL1413558	32472	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	7	3.6	CC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2C2CC2)cc1	nan
	3240816	32475	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	0	6	2.0	COC(=O)c1cn(C)c2ccc(S(=O)(=O)N3CC(C)CC(C)C3)cc2c1=O	nan
	CHEMBL1413578	32475	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	0	6	2.0	COC(=O)c1cn(C)c2ccc(S(=O)(=O)N3CC(C)CC(C)C3)cc2c1=O	nan
	3546772	32509	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	8	1	4	5.1	CC(C)OCCCNC(=O)c1cc(Sc2ccc(F)cc2)nc2ccccc12	nan
	CHEMBL1413820	32509	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	8	1	4	5.1	CC(C)OCCCNC(=O)c1cc(Sc2ccc(F)cc2)nc2ccccc12	nan
	2216801	32532	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.2	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCCC3)no1	nan
	CHEMBL1414005	32532	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.2	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCCC3)no1	nan
	16011480	32579	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1cccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3ccncc32)c1	nan
	CHEMBL1414437	32579	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1cccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3ccncc32)c1	nan
	3185714	32612	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	2.9	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1	nan
	CHEMBL1414702	32612	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	2.9	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1	nan
	16024849	32685	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	4.7	CC(NC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1)c1ccccc1	nan
	CHEMBL1415340	32685	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	4.7	CC(NC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1)c1ccccc1	nan
	1997619	32712	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	1	0	6	3.4	O=c1nc2sc3ccccc3n2c(=O)n1-c1ccc(Cl)c(Cl)c1	nan
	CHEMBL1415577	32712	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	1	0	6	3.4	O=c1nc2sc3ccccc3n2c(=O)n1-c1ccc(Cl)c(Cl)c1	nan
	601275	32739	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	7	2.7	CCc1nnc(NC(=O)CSc2nc(C)cc(C)c2C#N)s1	nan
	CHEMBL1415875	32739	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	7	2.7	CCc1nnc(NC(=O)CSc2nc(C)cc(C)c2C#N)s1	nan
	15988188	32764	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	2	4	2.9	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	CHEMBL1416073	32764	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	2	4	2.9	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	2135587	32818	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(F)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1416515	32818	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(F)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	1829959	32824	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	6	4.6	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1cccs1	nan
	CHEMBL1416570	32824	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	6	4.6	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1cccs1	nan
	4044817	32841	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	4	1	6	4.1	CC(OC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3)C(=O)Nc1ccc(F)cc1Cl	nan
	CHEMBL1416742	32841	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	4	1	6	4.1	CC(OC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3)C(=O)Nc1ccc(F)cc1Cl	nan
	16012432	32842	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	5	3.0	O=C(NCc1cccc(Cl)c1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	CHEMBL1416749	32842	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	5	3.0	O=C(NCc1cccc(Cl)c1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	16033988	32858	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	2	0	5	2.8	Cc1ccc(-n2ncc3c(N(C)C)ncnc32)cc1Cl	nan
	CHEMBL1416927	32858	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	2	0	5	2.8	Cc1ccc(-n2ncc3c(N(C)C)ncnc32)cc1Cl	nan
	16031129	32923	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	6	4.5	COc1ccc(OC)c(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)c1	nan
	CHEMBL1417406	32923	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	6	4.5	COc1ccc(OC)c(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)c1	nan
	16018805	32938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	6	3.3	COc1ccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1Cl	nan
	CHEMBL1417571	32938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	6	3.3	COc1ccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1Cl	nan
	1490637	32981	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	2	5	4.5	COc1ccc(NC(=O)c2ccccc2Sc2ccc(NC(C)=O)nc2)cc1	nan
	CHEMBL1417935	32981	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	2	5	4.5	COc1ccc(NC(=O)c2ccccc2Sc2ccc(NC(C)=O)nc2)cc1	nan
	5768421	33004	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	9	1	6	3.8	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)c(C)c2)C1c1ccncc1	nan
	CHEMBL1418118	33004	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	9	1	6	3.8	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)c(C)c2)C1c1ccncc1	nan
	16025701	33053	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	9	3.7	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4cccc(C)c4)n3)c2C)cc1OC	nan
	CHEMBL1418579	33053	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	9	3.7	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4cccc(C)c4)n3)c2C)cc1OC	nan
	1248279	33076	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	7	3.9	COc1ccccc1Nc1nc(N)nc(-c2oc3ccccc3c2C)n1	nan
	CHEMBL1418732	33076	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	7	3.9	COc1ccccc1Nc1nc(N)nc(-c2oc3ccccc3c2C)n1	nan
	2082778	33111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	2	3	3.6	COc1ccc(Br)c(C(=O)Nc2nc3ccccc3[nH]2)c1	nan
	CHEMBL1419051	33111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	2	3	3.6	COc1ccc(Br)c(C(=O)Nc2nc3ccccc3[nH]2)c1	nan
	7708945	33129	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	1	4	4.3	Nc1c(-c2ccc(Cl)cc2)cnc2c(-c3ccccc3)cnn12	nan
	CHEMBL1419219	33129	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	1	4	4.3	Nc1c(-c2ccc(Cl)cc2)cnc2c(-c3ccccc3)cnn12	nan
	656027	33222	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	7	4.2	COc1ccc(CCN2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccs2)cc1OC	nan
	CHEMBL1420005	33222	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	7	4.2	COc1ccc(CCN2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccs2)cc1OC	nan
	16457257	33238	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	1	1	5	3.5	Cc1ccccc1-c1nc2c3ccccc3nc(S)n2n1	nan
	CHEMBL1420123	33238	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	1	1	5	3.5	Cc1ccccc1-c1nc2c3ccccc3nc(S)n2n1	nan
	5049250	33252	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	2.6	O=C(COc1cccc2cccnc12)NNC(=S)Nc1ccccc1	nan
	CHEMBL1420194	33252	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	2.6	O=C(COc1cccc2cccnc12)NNC(=S)Nc1ccccc1	nan
	2518728	33306	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.3	Cc1nn(Cc2ccc(F)cc2)c2sc(C(=O)Nc3nccs3)cc12	nan
	CHEMBL1420654	33306	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.3	Cc1nn(Cc2ccc(F)cc2)c2sc(C(=O)Nc3nccs3)cc12	nan
	1975568	33491	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	6	4.4	COc1ccc2c(c1)c1nc3ccccc3nc1n2CCCN1C(=O)c2ccccc2C1=O	nan
	CHEMBL1422285	33491	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	6	4.4	COc1ccc2c(c1)c1nc3ccccc3nc1n2CCCN1C(=O)c2ccccc2C1=O	nan
	2952481	33611	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	2	5	3.6	CCCC(=O)Nc1ccc(C(=O)Nc2ccc([N+](=O)[O-])cc2OC)cc1	nan
	CHEMBL1423274	33611	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	2	5	3.6	CCCC(=O)Nc1ccc(C(=O)Nc2ccc([N+](=O)[O-])cc2OC)cc1	nan
	4204373	33693	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	2	6	3.5	COc1cc2nc(S)nc(NCc3ccccc3)c2cc1OC	nan
	CHEMBL1423864	33693	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	2	6	3.5	COc1cc2nc(S)nc(NCc3ccccc3)c2cc1OC	nan
	3208003	33719	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cc(C)ccc2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1424112	33719	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cc(C)ccc2nc1SCC(=O)Nc1cc(C)on1	nan
	4329755	33842	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	3	6.3	O=C(Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1)Nc1ccccc1	nan
	CHEMBL1425135	33842	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	3	6.3	O=C(Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1)Nc1ccccc1	nan
	2293921	33892	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	3	5	1.5	NS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(NC(=O)C3CC3)cc2)cc1	nan
	CHEMBL1425666	33892	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	3	5	1.5	NS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(NC(=O)C3CC3)cc2)cc1	nan
	2009311	33911	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	4.6	O=C(O)CSc1ncnc2c1sc1nc(-c3ccccc3)c3c(c12)CCC3	nan
	CHEMBL1425879	33911	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	4.6	O=C(O)CSc1ncnc2c1sc1nc(-c3ccccc3)c3c(c12)CCC3	nan
	3434681	34024	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	3	5	3.9	COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	CHEMBL1426649	34024	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	3	5	3.9	COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	3430748	34027	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	3	5	2.1	COc1ccc2c3c([nH]c2c1)C1CC2C(CC(O)C(OC)C2CO)CN1CC3	nan
	CHEMBL1426665	34027	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	3	5	2.1	COc1ccc2c3c([nH]c2c1)C1CC2C(CC(O)C(OC)C2CO)CN1CC3	nan
	16195448	34088	0	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	3	4.7	Cc1cccc(NC(=O)c2ccc3c(Cl)c4c(nc3c2)CCCC4)n1	nan
	CHEMBL1427245	34088	0	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	3	4.7	Cc1cccc(NC(=O)c2ccc3c(Cl)c4c(nc3c2)CCCC4)n1	nan
	1206713	34218	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1cccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc12	nan
	CHEMBL1428460	34218	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1cccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc12	nan
	2085163	34249	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	3.7	CCOc1ncccc1C(=O)Nc1ccc2nc(C)sc2c1	nan
	CHEMBL1428703	34249	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	3.7	CCOc1ncccc1C(=O)Nc1ccc2nc(C)sc2c1	nan
	3138587	34281	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	5	10	-2.3	CN(C)c1ccc2nc3c(=O)[nH]c(=O)nc-3n(CC(O)C(O)C(O)CO)c2c1	nan
	CHEMBL1428985	34281	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	5	10	-2.3	CN(C)c1ccc2nc3c(=O)[nH]c(=O)nc-3n(CC(O)C(O)C(O)CO)c2c1	nan
	1454920	34372	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1ccccc1C)C1CC1)c1nnnn12	nan
	CHEMBL1429692	34372	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1ccccc1C)C1CC1)c1nnnn12	nan
	748627	34399	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	4.7	Cc1ccc(Nc2nc(-c3ccncc3)nc3ccccc23)cc1	nan
	CHEMBL1429854	34399	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	4.7	Cc1ccc(Nc2nc(-c3ccncc3)nc3ccccc23)cc1	nan
	1478328	34464	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.0	CCc1nc2oc3ccc(C)cc3c(=O)c2cc1C(=O)OC	nan
	CHEMBL1430305	34464	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.0	CCc1nc2oc3ccc(C)cc3c(=O)c2cc1C(=O)OC	nan
	2950980	34518	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	4	6	3.8	O=C(O)c1cc(S(=O)(=O)O)cc(Nc2c3ccccc3nc3ccccc23)c1O	nan
	CHEMBL1430778	34518	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	4	6	3.8	O=C(O)c1cc(S(=O)(=O)O)cc(Nc2c3ccccc3nc3ccccc23)c1O	nan
	3452486	34605	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1431571	34605	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	2031268	34638	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1cccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)c1	nan
	CHEMBL1431855	34638	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1cccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)c1	nan
	16030582	34835	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	2	7	4.1	Cc1ccc2[nH]c(CSc3nnc(NC(=O)COc4ccccc4F)s3)cc(=O)c2c1	nan
	CHEMBL1433463	34835	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	2	7	4.1	Cc1ccc2[nH]c(CSc3nnc(NC(=O)COc4ccccc4F)s3)cc(=O)c2c1	nan
	16014372	34849	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccc(CSc2ncc(Cl)c(C(=O)NCc3ccccc3)n2)cc1	nan
	CHEMBL1433681	34849	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccc(CSc2ncc(Cl)c(C(=O)NCc3ccccc3)n2)cc1	nan
	24980276	34879	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	8	2.9	CCOC(=O)c1c(NC(=O)COC(=O)CCOc2ccccc2C)sc(C(=O)NC)c1C	nan
	CHEMBL1434167	34879	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	8	2.9	CCOC(=O)c1c(NC(=O)COC(=O)CCOc2ccccc2C)sc(C(=O)NC)c1C	nan
	17757032	34882	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	0	4	4.6	Clc1ccc2c(c1)-c1c(cnc3cc(-c4ccccc4)nn13)CO2	nan
	CHEMBL1434219	34882	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	0	4	4.6	Clc1ccc2c(c1)-c1c(cnc3cc(-c4ccccc4)nn13)CO2	nan
	16018775	34883	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	5	3.7	Cc1cc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)ccc1Br	nan
	CHEMBL1434221	34883	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	5	3.7	Cc1cc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)ccc1Br	nan
	16018825	34894	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	8	2.4	COc1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)c(OC)c1OC	nan
	CHEMBL1434453	34894	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	8	2.4	COc1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)c(OC)c1OC	nan
	15989503	34901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	3.2	Cc1cccc(NC(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c3ccccc32)c1	nan
	CHEMBL1434580	34901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	3.2	Cc1cccc(NC(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c3ccccc32)c1	nan
	16034196	34902	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	5.2	CCOC(=O)c1ccc(N2CCN(c3cccc(OC)c3)CC2)c(NC(=O)Nc2ccc(OCC)cc2)c1	nan
	CHEMBL1434618	34902	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	5.2	CCOC(=O)c1ccc(N2CCN(c3cccc(OC)c3)CC2)c(NC(=O)Nc2ccc(OCC)cc2)c1	nan
	16030773	34911	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	5.0	Cc1cccc(OCC(=O)Nc2cc(-c3ccccc3F)nn2-c2ccccc2)c1	nan
	CHEMBL1434674	34911	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	5.0	Cc1cccc(OCC(=O)Nc2cc(-c3ccccc3F)nn2-c2ccccc2)c1	nan
	4153411	34939	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.6	Cc1cc(C)cc(OCC(=O)Nc2ccc(-c3nc4ccccc4s3)cc2)c1	nan
	CHEMBL1435020	34939	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.6	Cc1cc(C)cc(OCC(=O)Nc2ccc(-c3nc4ccccc4s3)cc2)c1	nan
	9516939	34940	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	3	1	6	3.2	COc1ccc2oc(C(=O)Nc3nnc(C)s3)c(C)c2c1	nan
	CHEMBL1435035	34940	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	3	1	6	3.2	COc1ccc2oc(C(=O)Nc3nnc(C)s3)c(C)c2c1	nan
	16016693	34955	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	5.5	CC(C)Oc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1	nan
	CHEMBL1435186	34955	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	5.5	CC(C)Oc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1	nan
	16026116	34972	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	9	1.7	COc1cccc(CNC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1OC	nan
	CHEMBL1435357	34972	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	9	1.7	COc1cccc(CNC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1OC	nan
	1821611	34982	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	5	5.9	COc1ccc(NC(=O)c2c(NC(=O)COc3ccc(Cl)cc3)sc3c2CCCCC3)cc1	nan
	CHEMBL1435471	34982	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	5	5.9	COc1ccc(NC(=O)c2c(NC(=O)COc3ccc(Cl)cc3)sc3c2CCCCC3)cc1	nan
	1251337	34990	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.2	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)cc1	nan
	CHEMBL1435587	34990	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.2	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)cc1	nan
	16010614	35015	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(CNc2nc3ccccc3c3nc(-c4cccc(C)c4)nn23)cc1	nan
	CHEMBL1435932	35015	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(CNc2nc3ccccc3c3nc(-c4cccc(C)c4)nn23)cc1	nan
	16025971	35018	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	4.1	Cc1ccc(NC(=O)CSc2nc(-c3ccccc3Cl)nc3cc(=O)[nH]n23)c(C)c1	nan
	CHEMBL1436000	35018	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	4.1	Cc1ccc(NC(=O)CSc2nc(-c3ccccc3Cl)nc3cc(=O)[nH]n23)c(C)c1	nan
	16023620	35027	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	3	5	3.4	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(F)c2)N3)cc1	nan
	CHEMBL1436076	35027	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	3	5	3.4	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(F)c2)N3)cc1	nan
	16001329	35048	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	0	7	4.9	COc1ccc(-c2nn(C)c3sc(C(=O)N4CCN(c5cccc(C)c5C)CC4)cc23)cc1OC	nan
	CHEMBL1436335	35048	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	0	7	4.9	COc1ccc(-c2nn(C)c3sc(C(=O)N4CCN(c5cccc(C)c5C)CC4)cc23)cc1OC	nan
	16015802	35054	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	4	6.5	Cc1ccc(SCC(=O)Nc2cccc(-c3nc4cc(Cl)ccc4o3)c2C)cc1	nan
	CHEMBL1436447	35054	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	4	6.5	Cc1ccc(SCC(=O)Nc2cccc(-c3nc4cc(Cl)ccc4o3)c2C)cc1	nan
	16008886	35059	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.3	COc1ccc(CNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)c(OC)c1	nan
	CHEMBL1436510	35059	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.3	COc1ccc(CNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)c(OC)c1	nan
	16024495	35098	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	3.3	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	CHEMBL1437062	35098	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	3.3	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	16019037	35107	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	0	6	4.6	CCOC(=O)c1cnc2cc(-c3ccc(OCC)cc3)nn2c1-c1ccccc1	nan
	CHEMBL1437136	35107	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	0	6	4.6	CCOC(=O)c1cnc2cc(-c3ccc(OCC)cc3)nn2c1-c1ccccc1	nan
	16030417	35131	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1cccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3cc(C)ccc3n2)c1	nan
	CHEMBL1437458	35131	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1cccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3cc(C)ccc3n2)c1	nan
	15987619	35134	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	5.7	CCCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(Cl)c1	nan
	CHEMBL1437513	35134	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	5.7	CCCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(Cl)c1	nan
	16027516	35142	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	CHEMBL1437665	35142	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	2986974	35146	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.5	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)COc1ccccc1C	nan
	CHEMBL1437693	35146	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.5	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)COc1ccccc1C	nan
	16025598	35203	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	1	7	4.1	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1438111	35203	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	1	7	4.1	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)cc1	nan
	16012435	35216	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	0	4	3.7	CCc1nn(Cc2cccc(F)c2)c(=O)c2cc3cc(C)ccc3n12	nan
	CHEMBL1438209	35216	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	0	4	3.7	CCc1nn(Cc2cccc(F)c2)c(=O)c2cc3cc(C)ccc3n12	nan
	16014909	35306	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc2c(c1)cc(C(=O)NCc1ccccc1C)n2C	nan
	CHEMBL1439084	35306	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc2c(c1)cc(C(=O)NCc1ccccc1C)n2C	nan
	992393	35328	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	5.0	CCOC(=O)c1cnc2c(C)cc(Cl)cc2c1NCCc1ccc(OC)c(OC)c1	nan
	CHEMBL1439287	35328	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	5.0	CCOC(=O)c1cnc2c(C)cc(Cl)cc2c1NCCc1ccc(OC)c(OC)c1	nan
	2767956	35355	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	3	4.9	CSc1cc(-c2ccc(Cl)cc2)c(C(=O)NC(C)C)s1	nan
	CHEMBL1439494	35355	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	3	4.9	CSc1cc(-c2ccc(Cl)cc2)c(C(=O)NC(C)C)s1	nan
	3116122	35384	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccc(NC(=O)CSc2nc(N)c(C#N)cc2C#N)cc1	nan
	CHEMBL1439707	35384	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccc(NC(=O)CSc2nc(N)c(C#N)cc2C#N)cc1	nan
	16016094	35429	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	7	5.1	COc1ccc(-c2noc(-c3ccc(NC4CCCCC4)c([N+](=O)[O-])c3)n2)cc1	nan
	CHEMBL1440140	35429	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	7	5.1	COc1ccc(-c2noc(-c3ccc(NC4CCCCC4)c([N+](=O)[O-])c3)n2)cc1	nan
	1630787	35475	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	3.3	CC(C)(C)NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	CHEMBL1440595	35475	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	3.3	CC(C)(C)NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	16014413	35485	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccccc1CSc1ncc(Cl)c(C(=O)NCc2ccccc2)n1	nan
	CHEMBL1440676	35485	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccccc1CSc1ncc(Cl)c(C(=O)NCc2ccccc2)n1	nan
	15989176	35580	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	9	1	5	3.2	CCCCNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccccc2C)c1=O	nan
	CHEMBL1441599	35580	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	9	1	5	3.2	CCCCNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccccc2C)c1=O	nan
	16008898	35602	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	6	3.5	CCOC(=O)c1cccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1441757	35602	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	6	3.5	CCOC(=O)c1cccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	1374312	35612	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	2.6	COc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	CHEMBL1441823	35612	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	2.6	COc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	979004	35616	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	0	10	2.6	CC(C)(C)c1nnc2sc(SCC(=O)c3ccc4c(c3)OCCO4)nn2c1=O	nan
	CHEMBL1441873	35616	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	0	10	2.6	CC(C)(C)c1nnc2sc(SCC(=O)c3ccc4c(c3)OCCO4)nn2c1=O	nan
	1860569	35639	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)cc1	nan
	CHEMBL1442098	35639	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)cc1	nan
	5302651	35829	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	5	3.7	CCc1ccc(NC(=O)CSc2nc(C)cc(COC)c2C#N)cc1	nan
	CHEMBL1443840	35829	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	5	3.7	CCc1ccc(NC(=O)CSc2nc(C)cc(COC)c2C#N)cc1	nan
	12006099	35867	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	13	1	7	4.1	CCCN(CCC)C(=O)Cn1c(=O)n(CCCCCC(=O)Nc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1444172	35867	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	13	1	7	4.1	CCCN(CCC)C(=O)Cn1c(=O)n(CCCCCC(=O)Nc2ccccc2)c(=O)c2sccc21	nan
	16019024	35901	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.5	COCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1444500	35901	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.5	COCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16034708	35904	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	3.6	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3)c2n1	nan
	CHEMBL1444524	35904	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	3.6	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3)c2n1	nan
	16016687	35924	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	2	5	4.8	COc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1OC	nan
	CHEMBL1444758	35924	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	2	5	4.8	COc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1OC	nan
	3238164	35949	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	3	3.1	O=C(CCN1CCN(c2ccc(F)cc2)CC1)Nc1ccc(F)cc1	nan
	CHEMBL1444967	35949	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	3	3.1	O=C(CCN1CCN(c2ccc(F)cc2)CC1)Nc1ccc(F)cc1	nan
	2296239	35950	13	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	8	1	6	2.7	CCn1c(SCC(=O)NCCOc2ccccc2)nc2ccccc2c1=O	nan
	CHEMBL1444971	35950	13	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	8	1	6	2.7	CCn1c(SCC(=O)NCCOc2ccccc2)nc2ccccc2c1=O	nan
	657584	35961	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	5	3.9	CC(C)Cc1nc(N2CCN(C(=O)Cc3ccccc3)CC2)c(C#N)c2c1COC(C)(C)C2	nan
	CHEMBL1445051	35961	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	5	3.9	CC(C)Cc1nc(N2CCN(C(=O)Cc3ccccc3)CC2)c(C#N)c2c1COC(C)(C)C2	nan
	15988979	36014	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	7	3.2	O=C(CCn1c(=O)c2sccc2n(CC(=O)Nc2ccccc2)c1=O)NCc1ccccc1Cl	nan
	CHEMBL1445545	36014	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	7	3.2	O=C(CCn1c(=O)c2sccc2n(CC(=O)Nc2ccccc2)c1=O)NCc1ccccc1Cl	nan
	16023569	36039	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.1	CC(=O)c1ccc(N2CCN(C(=O)CCn3cnc4onc(-c5ccc(F)cc5)c4c3=O)CC2)cc1	nan
	CHEMBL1445781	36039	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.1	CC(=O)c1ccc(N2CCN(C(=O)CCn3cnc4onc(-c5ccc(F)cc5)c4c3=O)CC2)cc1	nan
	7157939	36064	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	2	3	3.1	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cc(Cl)ccc1Cl	nan
	CHEMBL1446030	36064	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	2	3	3.1	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cc(Cl)ccc1Cl	nan
	1480468	36126	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	5	3.9	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccccc2)c1C#N	nan
	CHEMBL1446611	36126	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	5	3.9	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccccc2)c1C#N	nan
	2195706	36152	5	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	8	2.8	CCOC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1446861	36152	5	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	8	2.8	CCOC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	16010637	36190	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	4.7	CCN(Cc1ccccc1)C(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1	nan
	CHEMBL1447092	36190	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	4.7	CCN(Cc1ccccc1)C(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1	nan
	2130696	36288	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.9	N#C/C(C(=O)NCc1ccco1)=C1/SC=C(c2ccccc2)N1c1ccccc1	nan
	CHEMBL1447960	36288	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.9	N#C/C(C(=O)NCc1ccco1)=C1/SC=C(c2ccccc2)N1c1ccccc1	nan
	4583349	36335	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	5	2.2	Cc1ccc(NC(=O)CCn2c(=O)[nH]c3ccsc3c2=O)cc1F	nan
	CHEMBL1448388	36335	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	5	2.2	Cc1ccc(NC(=O)CCn2c(=O)[nH]c3ccsc3c2=O)cc1F	nan
	5396132	36417	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	0	5	3.7	COc1cc(/C=C2/C(=O)ON=C2C)ccc1OCc1ccccc1F	nan
	CHEMBL1448972	36417	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	0	5	3.7	COc1cc(/C=C2/C(=O)ON=C2C)ccc1OCc1ccccc1F	nan
	1201887	36443	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	0	3	4.0	Cc1cccc(CSc2nc3c(cc2C#N)CCC3)c1	nan
	CHEMBL1449126	36443	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	0	3	4.0	Cc1cccc(CSc2nc3c(cc2C#N)CCC3)c1	nan
	649163	36447	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	5	3.0	CCN(CC)S(=O)(=O)c1ccc(Cl)c(C(=O)Oc2cccnc2)c1	nan
	CHEMBL1449162	36447	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	5	3.0	CCN(CC)S(=O)(=O)c1ccc(Cl)c(C(=O)Oc2cccnc2)c1	nan
	16019152	36504	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	7	4.0	Cc1ccccc1Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	CHEMBL1449607	36504	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	7	4.0	Cc1ccccc1Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	16017274	36522	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.6	CCN(CC)c1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	CHEMBL1449789	36522	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.6	CCN(CC)c1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	15996185	36530	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	2	4	4.7	CCC(C)NC(=O)CCC(=O)Nc1ccc2nc(N3CC(C)CC(C)C3)cc(C)c2c1	nan
	CHEMBL1449862	36530	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	2	4	4.7	CCC(C)NC(=O)CCC(=O)Nc1ccc2nc(N3CC(C)CC(C)C3)cc(C)c2c1	nan
	15989912	36534	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	7	5.4	Cc1cc(C)n(-c2nc3ccccc3nc2Nc2ccc(Cl)c(C(=O)OC(C)C)c2)n1	nan
	CHEMBL1449881	36534	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	7	5.4	Cc1cc(C)n(-c2nc3ccccc3nc2Nc2ccc(Cl)c(C(=O)OC(C)C)c2)n1	nan
	16020571	36695	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	4.2	CCn1cc(S(=O)(=O)c2cc(C)cc(C)c2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	CHEMBL1451264	36695	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	4.2	CCn1cc(S(=O)(=O)c2cc(C)cc(C)c2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	5058847	36838	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	CHEMBL1452293	36838	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	15988482	36968	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.4	Cc1ccc(C(=O)c2cn(Cc3ccc(F)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1453340	36968	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.4	Cc1ccc(C(=O)c2cn(Cc3ccc(F)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16019909	36976	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	0	8	3.8	COc1cc(-c2noc(-c3cc4cccc(C)c4oc3=O)n2)cc(OC)c1OC	nan
	CHEMBL1453424	36976	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	0	8	3.8	COc1cc(-c2noc(-c3cc4cccc(C)c4oc3=O)n2)cc(OC)c1OC	nan
	16024781	37017	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	4	1.9	O=C1C(=O)N(C2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)CCN1Cc1ccccc1	nan
	CHEMBL1453815	37017	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	4	1.9	O=C1C(=O)N(C2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)CCN1Cc1ccccc1	nan
	16024608	37027	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	1	7	3.5	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	CHEMBL1453881	37027	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	1	7	3.5	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	3940076	37040	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	1	5	3.3	Cc1ccc(CNc2nc3nc(C)c(Cl)c(C)n3n2)cc1	nan
	CHEMBL1453947	37040	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	1	5	3.3	Cc1ccc(CNc2nc3nc(C)c(Cl)c(C)n3n2)cc1	nan
	1604929	37045	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	5	4.6	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)c1	nan
	CHEMBL1453974	37045	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	5	4.6	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)c1	nan
	707946	37070	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	3.0	O=C(Nc1nc2nccc(-c3ccccc3)n2n1)c1ccccc1	nan
	CHEMBL1454141	37070	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	3.0	O=C(Nc1nc2nccc(-c3ccccc3)n2n1)c1ccccc1	nan
	16010581	37086	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c1	nan
	CHEMBL1454246	37086	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c1	nan
	15988208	37154	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	9	1.7	COC(=O)c1cccnc1-n1c(=O)c2cccnc2n(CC(=O)Nc2cccc(C)c2)c1=O	nan
	CHEMBL1454833	37154	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	9	1.7	COC(=O)c1cccnc1-n1c(=O)c2cccnc2n(CC(=O)Nc2cccc(C)c2)c1=O	nan
	5123668	37210	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	10	1	7	5.2	CCc1ccc(NC(=O)CSc2nc3c(sc4ccccc43)c(=O)n2CCN(CC)CC)cc1	nan
	CHEMBL1455415	37210	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	10	1	7	5.2	CCc1ccc(NC(=O)CSc2nc3c(sc4ccccc43)c(=O)n2CCN(CC)CC)cc1	nan
	135421575	37265	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	2	4	3.3	CCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	CHEMBL1455904	37265	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	2	4	3.3	CCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	914701	37292	8	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	4	4.3	CCc1nc2sc3c(Cl)ncnc3c2c2c1CCCC2	nan
	CHEMBL1456130	37292	8	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	4	4.3	CCc1nc2sc3c(Cl)ncnc3c2c2c1CCCC2	nan
	2023595	37416	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1457309	37416	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	16024557	37452	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(Cl)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1457615	37452	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(Cl)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	20920344	37475	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	4.4	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5cccs5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1457782	37475	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	4.4	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5cccs5)CC4)nnc(C)c3c2C)cc1	nan
	3245484	37605	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	2	7	1.9	COc1cc2[nH]c(=O)n(CCC(=O)NC3CCN(Cc4ccccc4)CC3)c(=O)c2cc1OC	nan
	CHEMBL1458892	37605	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	2	7	1.9	COc1cc2[nH]c(=O)n(CCC(=O)NC3CCN(Cc4ccccc4)CC3)c(=O)c2cc1OC	nan
	2467173	37627	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	9	1	11	1.4	C=CCn1c(SCC(=O)c2c(N)n(CCC)c(=O)n(C)c2=O)nnc1-c1ccncc1	nan
	CHEMBL1459057	37627	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	9	1	11	1.4	C=CCn1c(SCC(=O)c2c(N)n(CCC)c(=O)n(C)c2=O)nnc1-c1ccncc1	nan
	3185309	37654	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	10	3	9	3.7	COc1ccc(OC)c(C(C(=O)NC2CCCCC2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2OC)c1	nan
	CHEMBL1459257	37654	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	10	3	9	3.7	COc1ccc(OC)c(C(C(=O)NC2CCCCC2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2OC)c1	nan
	2910207	37671	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	7	1	6	3.9	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccco1	nan
	CHEMBL1459409	37671	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	7	1	6	3.9	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccco1	nan
	2138506	37804	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	2	6	3.0	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(C(=O)OCC)CC1	nan
	CHEMBL1460540	37804	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	2	6	3.0	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(C(=O)OCC)CC1	nan
	1995746	37817	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	3	8	0.9	NC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccccn3)n2N)cc1	nan
	CHEMBL1460633	37817	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	3	8	0.9	NC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccccn3)n2N)cc1	nan
	1511731	37845	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	2.9	COc1ccc(C(=O)Nc2nc(C)c3cc4c(cc3n2)OCO4)cc1	nan
	CHEMBL1460863	37845	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	2.9	COc1ccc(C(=O)Nc2nc(C)c3cc4c(cc3n2)OCO4)cc1	nan
	4340474	37895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	6	2	6	2.1	CCCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3	nan
	CHEMBL1461327	37895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	6	2	6	2.1	CCCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3	nan
	2331607	37925	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	1	5	2.7	O=C(Nc1ccccn1)c1ccc2c(c1)S(=O)(=O)c1ccccc1C2=O	nan
	CHEMBL1461642	37925	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	1	5	2.7	O=C(Nc1ccccn1)c1ccc2c(c1)S(=O)(=O)c1ccccc1C2=O	nan
	4594455	37985	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	7	3.9	CSc1nc(N2CCN(c3ccccc3)CC2)cc(N2CCN(c3ccccc3)CC2)n1	nan
	CHEMBL1462148	37985	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	7	3.9	CSc1nc(N2CCN(c3ccccc3)CC2)cc(N2CCN(c3ccccc3)CC2)n1	nan
	661296	38016	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	2	1	3.2	CCc1c(C(=O)O)[nH]c2ccc(Br)cc12	nan
	CHEMBL1462380	38016	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	2	1	3.2	CCc1c(C(=O)O)[nH]c2ccc(Br)cc12	nan
	3183779	38046	5	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.7	Oc1nc2cc3c(cc2cc1C(c1nnnn1Cc1ccccc1)N1CCCCCC1)OCCO3	nan
	CHEMBL1462671	38046	5	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.7	Oc1nc2cc3c(cc2cc1C(c1nnnn1Cc1ccccc1)N1CCCCCC1)OCCO3	nan
	5418960	38065	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	4	3.3	O=c1c2cc3c(nc2[nH]c(=S)n1-c1ccccc1)CCCC3	nan
	CHEMBL1462820	38065	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	4	3.3	O=c1c2cc3c(nc2[nH]c(=S)n1-c1ccccc1)CCCC3	nan
	2766000	38097	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	1	8	3.9	COCCCn1c(SCc2ccc(OC)cc2)nc2cc(OC)c(OC)cc2c1=N	nan
	CHEMBL1463048	38097	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	1	8	3.9	COCCCn1c(SCc2ccc(OC)cc2)nc2cc(OC)c(OC)cc2c1=N	nan
	16188024	38120	2	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1ccc2nc(O)c3cc(C(=O)N(C)c4ccccc4C)sc3c2c1	nan
	CHEMBL1463271	38120	2	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1ccc2nc(O)c3cc(C(=O)N(C)c4ccccc4C)sc3c2c1	nan
	4429285	38133	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	7	3.7	COC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(C)c2)cc1	nan
	CHEMBL1463413	38133	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	7	3.7	COC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(C)c2)cc1	nan
	1738267	38138	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	8	1	4	5.2	O=C(CCC(=O)OCC(=O)c1ccc(-c2ccccc2)cc1)Nc1cccc(Cl)c1	nan
	CHEMBL1463488	38138	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	8	1	4	5.2	O=C(CCC(=O)OCC(=O)c1ccc(-c2ccccc2)cc1)Nc1cccc(Cl)c1	nan
	3761375	38262	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	0	4	4.3	CSc1nc(C)c2c(n1)N(c1ccc(C(C)C)cc1)CC2	nan
	CHEMBL1464437	38262	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	0	4	4.3	CSc1nc(C)c2c(n1)N(c1ccc(C(C)C)cc1)CC2	nan
	2044631	38317	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	2	4	4.3	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(C)c1	nan
	CHEMBL1464810	38317	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	2	4	4.3	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(C)c1	nan
	2372173	38363	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccccc2F)nc1-c1ccccc1	nan
	CHEMBL1465138	38363	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccccc2F)nc1-c1ccccc1	nan
	2988623	38585	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	0	6	3.2	CCOc1ccc(C(=O)N2CCN(c3cnn(-c4ccccc4)c(=O)c3Cl)CC2)cc1	nan
	CHEMBL1466802	38585	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	0	6	3.2	CCOc1ccc(C(=O)N2CCN(c3cnn(-c4ccccc4)c(=O)c3Cl)CC2)cc1	nan
	2428874	38605	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	1.9	O=C(Nc1cccc2c1C(=O)NC2=O)c1cccnc1Cl	nan
	CHEMBL1466996	38605	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	1.9	O=C(Nc1cccc2c1C(=O)NC2=O)c1cccnc1Cl	nan
	3574259	38625	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	CHEMBL1467198	38625	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	16007702	38657	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	5	2.6	CCn1cc(C(=O)NCCc2ccc(C)cc2)c(=O)c2cc(S(=O)(=O)N(C)C)ccc21	nan
	CHEMBL1467433	38657	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	5	2.6	CCn1cc(C(=O)NCCc2ccc(C)cc2)c(=O)c2cc(S(=O)(=O)N(C)C)ccc21	nan
	663318	38670	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	0	6	4.3	CC1CCN(c2nc3ccccc3nc2C(C#N)C(=O)OC2CCCCC2)CC1	nan
	CHEMBL1467520	38670	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	0	6	4.3	CC1CCN(c2nc3ccccc3nc2C(C#N)C(=O)OC2CCCCC2)CC1	nan
	2820576	38769	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.4	Cc1csc2sc(-c3ccnc(SCC(=O)NCc4ccccc4)n3)c(C)c12	nan
	CHEMBL1468435	38769	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.4	Cc1csc2sc(-c3ccnc(SCC(=O)NCc4ccccc4)n3)c(C)c12	nan
	970728	38787	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	2	2	5.0	Cc1cc(C)nc(NC(S)=Nc2cccc(Cl)c2Cl)c1	nan
	CHEMBL1468575	38787	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	2	2	5.0	Cc1cc(C)nc(NC(S)=Nc2cccc(Cl)c2Cl)c1	nan
	4294342	38790	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	2	2	3.6	Cc1cc2cc(CNC(=O)NC3CCCCC3)ccc2n1C	nan
	CHEMBL1468608	38790	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	2	2	3.6	Cc1cc2cc(CNC(=O)NC3CCCCC3)ccc2n1C	nan
	648454	38797	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	4	3.4	Cc1cc(C)nc(N2CCC(C(=O)Nc3ccc4c(c3)CCC4)CC2)n1	nan
	CHEMBL1468653	38797	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	4	3.4	Cc1cc(C)nc(N2CCC(C(=O)Nc3ccc4c(c3)CCC4)CC2)n1	nan
	7202588	38880	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	7	2.9	COC(=O)c1ccc2nc(NC(=O)CCS(=O)(=O)c3ccccc3)sc2c1	nan
	CHEMBL1469363	38880	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	7	2.9	COC(=O)c1ccc2nc(NC(=O)CCS(=O)(=O)c3ccccc3)sc2c1	nan
	1073207	39020	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	0	9	2.4	COc1ccc(-n2nnnc2SCC(=O)c2ccc3c(c2)OCCO3)cc1	nan
	CHEMBL1470594	39020	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	0	9	2.4	COc1ccc(-n2nnnc2SCC(=O)c2ccc3c(c2)OCCO3)cc1	nan
	3615142	39021	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.0	Cc1c(C(=O)Nc2cccnc2Cl)oc2ccccc12	nan
	CHEMBL1470599	39021	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.0	Cc1c(C(=O)Nc2cccnc2Cl)oc2ccccc12	nan
	16009952	39258	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	7	0.9	Cc1ccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1F	nan
	CHEMBL1472658	39258	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	7	0.9	Cc1ccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1F	nan
	1892783	39266	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	3	1	5	4.8	Cc1ccc(-c2nnc3c4ccccc4c(C)nn23)cc1NC(=O)c1ccccc1	nan
	CHEMBL1472759	39266	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	3	1	5	4.8	Cc1ccc(-c2nnc3c4ccccc4c(C)nn23)cc1NC(=O)c1ccccc1	nan
	16008277	39270	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	1	5	5.8	Cc1cc(N2CCC(C(=O)Nc3ccc(F)cc3F)CC2)n2nc(C)c(-c3ccc(Cl)cc3)c2n1	nan
	CHEMBL1472790	39270	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	1	5	5.8	Cc1cc(N2CCC(C(=O)Nc3ccc(F)cc3F)CC2)n2nc(C)c(-c3ccc(Cl)cc3)c2n1	nan
	16015830	39273	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	4	5.1	O=C(COc1ccccc1F)Nc1ccc(-c2nc3ccccc3s2)cc1	nan
	CHEMBL1472798	39273	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	4	5.1	O=C(COc1ccccc1F)Nc1ccc(-c2nc3ccccc3s2)cc1	nan
	16030736	39283	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	3	5.3	CC(C)(C)C(=O)Nc1cc(-c2cccc(Br)c2)nn1-c1ccccc1	nan
	CHEMBL1472994	39283	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	3	5.3	CC(C)(C)C(=O)Nc1cc(-c2cccc(Br)c2)nn1-c1ccccc1	nan
	16015144	39286	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	1	5	4.6	O=C(/C=C/c1ccc(Cl)cc1)Nc1nc(-c2cccs2)ns1	nan
	CHEMBL1472998	39286	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	1	5	4.6	O=C(/C=C/c1ccc(Cl)cc1)Nc1nc(-c2cccs2)ns1	nan
	16010790	39313	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	7	2.7	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	CHEMBL1473410	39313	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	7	2.7	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	16009809	39315	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	2	5	5.9	COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)C23CC4CC(CC(C4)C2)C3)c(OC)c1	nan
	CHEMBL1473436	39315	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	2	5	5.9	COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)C23CC4CC(CC(C4)C2)C3)c(OC)c1	nan
	16009067	39320	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	1	3	5.5	Cc1ccc2nc(Cl)c3cc(C(=O)NC4CCCCC4)sc3c2c1	nan
	CHEMBL1473455	39320	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	1	3	5.5	Cc1ccc2nc(Cl)c3cc(C(=O)NC4CCCCC4)sc3c2c1	nan
	864758	39327	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	6	2.1	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	CHEMBL1473580	39327	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	6	2.1	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	16010866	39328	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	7	2.9	COc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1Cl	nan
	CHEMBL1473610	39328	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	7	2.9	COc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1Cl	nan
	16008902	39330	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	4	3.3	Cc1cccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1473624	39330	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	4	3.3	Cc1cccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	4425770	39336	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	4.4	Cc1cccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)o2)c1	nan
	CHEMBL1473697	39336	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	4.4	Cc1cccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)o2)c1	nan
	16025407	39341	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	6	1	6	5.2	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2cccc(F)c2)S3(=O)=O)cc1F	nan
	CHEMBL1473728	39341	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	6	1	6	5.2	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2cccc(F)c2)S3(=O)=O)cc1F	nan
	15989780	39387	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.9	Clc1ccc(CCNc2nc3cc(Cl)c(Cl)cc3n3cnnc23)cc1	nan
	CHEMBL1474477	39387	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.9	Clc1ccc(CCNc2nc3cc(Cl)c(Cl)cc3n3cnnc23)cc1	nan
	16034729	39399	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	7	5.0	COc1ccc(-c2cn3nc(N4CCC(C(=O)Nc5cccc(Cl)c5)CC4)sc3n2)cc1	nan
	CHEMBL1474594	39399	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	7	5.0	COc1ccc(-c2cn3nc(N4CCC(C(=O)Nc5cccc(Cl)c5)CC4)sc3n2)cc1	nan
	16012452	39411	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	5	2.4	O=C(NCc1ccccc1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	CHEMBL1474806	39411	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	5	2.4	O=C(NCc1ccccc1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	16020997	39413	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.9	Cc1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1F	nan
	CHEMBL1474813	39413	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.9	Cc1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1F	nan
	16012520	39441	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	5	4.9	CC(=O)Nc1ccc(NC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccccc3)c2C)cc1	nan
	CHEMBL1475217	39441	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	5	4.9	CC(=O)Nc1ccc(NC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccccc3)c2C)cc1	nan
	16008390	39446	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	4	4.2	CCc1ccc(CNC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1	nan
	CHEMBL1475336	39446	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	4	4.2	CCc1ccc(CNC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1	nan
	3225367	39450	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	3	5.8	Cc1cccc(C)c1NC(=O)c1cc2sccc2n1Cc1ccc(F)cc1	nan
	CHEMBL1475367	39450	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	3	5.8	Cc1cccc(C)c1NC(=O)c1cc2sccc2n1Cc1ccc(F)cc1	nan
	1983981	39458	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	5.2	Cc1ccc(-c2nn3c(-c4ccc(C)cc4)nnc3c3ccccc23)cc1	nan
	CHEMBL1475431	39458	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	5.2	Cc1ccc(-c2nn3c(-c4ccc(C)cc4)nnc3c3ccccc23)cc1	nan
	16030137	39472	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	7	1	7	3.6	CCOc1ccccc1CNC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	CHEMBL1475622	39472	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	7	1	7	3.6	CCOc1ccccc1CNC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	16016540	39474	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	2	3.7	Cc1cc(=O)c2cc(C(=O)Nc3cccc(C)c3C)ccc2[nH]1	nan
	CHEMBL1475643	39474	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	2	3.7	Cc1cc(=O)c2cc(C(=O)Nc3cccc(C)c3C)ccc2[nH]1	nan
	16026533	39482	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	7	4.0	COc1ccc(OC)c(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	CHEMBL1475722	39482	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	7	4.0	COc1ccc(OC)c(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	16030897	39486	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	1	6	4.8	COc1ccc(-c2cn3nc(SCC(=O)Nc4cccc(C)c4C)ccc3n2)cc1	nan
	CHEMBL1475786	39486	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	1	6	4.8	COc1ccc(-c2cn3nc(SCC(=O)Nc4cccc(C)c4C)ccc3n2)cc1	nan
	16012637	39507	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	0	10	3.3	Cc1ccc2nc3c(cc(C#N)c(=O)n3-c3nnc(SCc4ccccc4)s3)c(=O)n2c1	nan
	CHEMBL1476168	39507	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	0	10	3.3	Cc1ccc2nc3c(cc(C#N)c(=O)n3-c3nnc(SCc4ccccc4)s3)c(=O)n2c1	nan
	16009819	39517	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	8	4.3	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1Cl	nan
	CHEMBL1476323	39517	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	8	4.3	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1Cl	nan
	16009801	39523	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)c(OC)c1	nan
	CHEMBL1476410	39523	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)c(OC)c1	nan
	15987507	39528	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	6.1	Cc1cc(C)c2oc(-c3ccc(Cl)c(NC(=O)c4cccs4)c3)nc2c1	nan
	CHEMBL1476493	39528	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	6.1	Cc1cc(C)c2oc(-c3ccc(Cl)c(NC(=O)c4cccs4)c3)nc2c1	nan
	16030393	39536	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	4	5.2	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCc3ccccc32)cc1	nan
	CHEMBL1476572	39536	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	4	5.2	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCc3ccccc32)cc1	nan
	16010862	39543	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1C	nan
	CHEMBL1476637	39543	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1C	nan
	4154280	39556	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	5.9	CCc1ccccc1NC(=O)C(CC)Sc1ncnc2c1sc1ccccc12	nan
	CHEMBL1476806	39556	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	5.9	CCc1ccccc1NC(=O)C(CC)Sc1ncnc2c1sc1ccccc12	nan
	7184887	39570	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	8	3.4	CC1CCN(c2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1476979	39570	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	8	3.4	CC1CCN(c2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)CC1	nan
	666072	39671	8	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	6	4.6	CSc1ccc(-c2c(C#N)c(N)nc3c2c(C)nn3-c2ccccc2)cc1	nan
	CHEMBL1477886	39671	8	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	6	4.6	CSc1ccc(-c2c(C#N)c(N)nc3c2c(C)nn3-c2ccccc2)cc1	nan
	2810062	39686	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	1	6	2.9	Cc1csc2c(=O)sc(NC(=O)c3ccco3)nc12	nan
	CHEMBL1478110	39686	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	1	6	2.9	Cc1csc2c(=O)sc(NC(=O)c3ccco3)nc12	nan
	16014364	39718	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	4.8	Cc1ccc(CNC(=O)c2nc(SCc3ccc(F)cc3)ncc2Cl)cc1	nan
	CHEMBL1478416	39718	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	4.8	Cc1ccc(CNC(=O)c2nc(SCc3ccc(F)cc3)ncc2Cl)cc1	nan
	947086	39741	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	0	4	4.1	COc1ccc(-c2c(C#N)c(C)nc3c2C(=O)c2ccccc2-3)cc1	nan
	CHEMBL1478573	39741	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	0	4	4.1	COc1ccc(-c2c(C#N)c(C)nc3c2C(=O)c2ccccc2-3)cc1	nan
	15990421	39752	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	1	4	5.9	Cc1cc(Br)ccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1478684	39752	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	1	4	5.9	Cc1cc(Br)ccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	2150494	39764	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	7	3.8	COCCn1c(SCC(=O)Nc2ccc(C)cc2)nc2c(oc3ccccc32)c1=O	nan
	CHEMBL1478802	39764	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	7	3.8	COCCn1c(SCC(=O)Nc2ccc(C)cc2)nc2c(oc3ccccc32)c1=O	nan
	9267240	39772	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	O=C(Nc1ccc(Cl)cc1F)c1ccc(-n2cncn2)cc1	nan
	CHEMBL1478883	39772	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	O=C(Nc1ccc(Cl)cc1F)c1ccc(-n2cncn2)cc1	nan
	16015604	39812	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	6.3	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(C)cc3)on2)cc1	nan
	CHEMBL1479260	39812	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	6.3	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(C)cc3)on2)cc1	nan
	4050786	39884	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	2.8	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(NC(C)=O)ccc21	nan
	CHEMBL1479784	39884	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	2.8	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(NC(C)=O)ccc21	nan
	16009694	39886	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	8	4.6	COc1ccc(-c2nnn3c2nc(NCCc2ccc(OC)c(OC)c2)c2ccccc23)cc1	nan
	CHEMBL1479788	39886	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	8	4.6	COc1ccc(-c2nnn3c2nc(NCCc2ccc(OC)c(OC)c2)c2ccccc23)cc1	nan
	2140519	40046	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	3	6	1.2	COC(=O)CCC(=O)NC(=S)Nc1sc(C)c(C)c1C(N)=O	nan
	CHEMBL1481122	40046	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	3	6	1.2	COC(=O)CCC(=O)NC(=S)Nc1sc(C)c(C)c1C(N)=O	nan
	16189596	40059	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	4	4.5	CCN1CCCc2cc(CN(CCN3CCOCC3)C(S)=Nc3ccccc3C)ccc21	nan
	CHEMBL1481195	40059	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	4	4.5	CCN1CCCc2cc(CN(CCN3CCOCC3)C(S)=Nc3ccccc3C)ccc21	nan
	6324455	40143	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	4	3.1	CCN(CC)S(=O)(=O)c1ccc2nc(O)c3ccccc3c2c1	nan
	CHEMBL1482015	40143	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	4	3.1	CCN(CC)S(=O)(=O)c1ccc2nc(O)c3ccccc3c2c1	nan
	4898982	40168	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	5	2.9	COc1ccc2cc(C(=O)N3CCN(Cc4ccc5c(c4)OCO5)CC3)[nH]c2c1	nan
	CHEMBL1482223	40168	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	5	2.9	COc1ccc2cc(C(=O)N3CCN(Cc4ccc5c(c4)OCO5)CC3)[nH]c2c1	nan
	16194617	40178	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	6	4.4	CCOc1ncccc1C(=O)Nc1cccc(-c2nc3cccnc3s2)c1	nan
	CHEMBL1482332	40178	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	6	4.4	CCOc1ncccc1C(=O)Nc1cccc(-c2nc3cccnc3s2)c1	nan
	7598416	40282	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	2.6	Cc1cccc(Cn2cccc(C(=O)Nc3nnc(C)s3)c2=O)c1	nan
	CHEMBL1483270	40282	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	2.6	Cc1cccc(Cn2cccc(C(=O)Nc3nnc(C)s3)c2=O)c1	nan
	16033878	40294	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	6	4.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccccc3nc2s1	nan
	CHEMBL1483384	40294	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	6	4.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccccc3nc2s1	nan
	5033969	40338	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	4	3.0	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)c(S(=O)(=O)N(C)C)c2)c1C	nan
	CHEMBL1483695	40338	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	4	3.0	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)c(S(=O)(=O)N(C)C)c2)c1C	nan
	2346667	40348	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	6	0	5	2.8	COc1ccc(C(=O)COC(=O)c2ccc(N(C)C)cc2)cc1	nan
	CHEMBL1483762	40348	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	6	0	5	2.8	COc1ccc(C(=O)COC(=O)c2ccc(N(C)C)cc2)cc1	nan
	4199549	40369	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	9	0	6	4.9	CCOc1ccccc1C(=O)N1CCc2cc(OC)c(OC)cc2C1COc1ccc(OC)cc1	nan
	CHEMBL1483991	40369	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	9	0	6	4.9	CCOc1ccccc1C(=O)N1CCc2cc(OC)c(OC)cc2C1COc1ccc(OC)cc1	nan
	135399202	40434	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	5	3.1	NC1=C(c2nc3ccccc3s2)C(=O)CN1C1CCCCC1	nan
	CHEMBL1484439	40434	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	5	3.1	NC1=C(c2nc3ccccc3s2)C(=O)CN1C1CCCCC1	nan
	2377756	40470	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	6	3.4	O=C(O)c1cccnc1Sc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1484807	40470	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	6	3.4	O=C(O)c1cccnc1Sc1ncnc2sc3c(c12)CCC3	nan
	135410529	40509	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	4.7	CCS(=O)(=O)c1cccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c1	nan
	CHEMBL1485170	40509	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	4.7	CCS(=O)(=O)c1cccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c1	nan
	135521955	40548	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1cc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1485562	40548	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1cc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	15989053	40560	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	1	8	4.0	Cc1cc(C)c(Cn2c(=O)n(CCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1485622	40560	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	1	8	4.0	Cc1cc(C)c(Cn2c(=O)n(CCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	4277738	40572	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	3	4.8	Sc1nc(-c2ccc(Br)cc2)cn1CCc1ccccc1	nan
	CHEMBL1485734	40572	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	3	4.8	Sc1nc(-c2ccc(Br)cc2)cn1CCc1ccccc1	nan
	16012072	40608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	11	1	6	3.8	CCCCN(C)CCCNC(=O)Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O	nan
	CHEMBL1486036	40608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	11	1	6	3.8	CCCCN(C)CCCNC(=O)Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O	nan
	1273744	40638	11	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	7	3.8	Cc1cc(C)c(C#N)c(SCC(=O)Nc2nnc(-c3ccccc3)s2)n1	nan
	CHEMBL1486391	40638	11	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	7	3.8	Cc1cc(C)c(C#N)c(SCC(=O)Nc2nnc(-c3ccccc3)s2)n1	nan
	16021806	40661	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	4	5.1	CSc1ncc(C(=O)Nc2ccccc2C(F)(F)F)c(-c2ccccc2)n1	nan
	CHEMBL1486543	40661	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	4	5.1	CSc1ncc(C(=O)Nc2ccccc2C(F)(F)F)c(-c2ccccc2)n1	nan
	5339079	40690	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	4	4.4	Cc1nc(-c2ccccc2)nc2nc(-c3ccccc3)cc(O)c12	nan
	CHEMBL1486764	40690	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	4	4.4	Cc1nc(-c2ccccc2)nc2nc(-c3ccccc3)cc(O)c12	nan
	702036	40767	13	None	-19	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	1	0	5	4.2	N#Cc1c2c(c(-n3cnc4ccccc43)n3c1nc1ccccc13)CCC2	nan
	CHEMBL1487421	40767	13	None	-19	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	1	0	5	4.2	N#Cc1c2c(c(-n3cnc4ccccc43)n3c1nc1ccccc13)CCC2	nan
	15989752	40787	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.9	Cc1ccc2nc(NCCc3ccc(Cl)cc3)c3nncn3c2c1	nan
	CHEMBL1487625	40787	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.9	Cc1ccc2nc(NCCc3ccc(Cl)cc3)c3nncn3c2c1	nan
	16008663	40800	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	8	1.6	COC(=O)c1ccc(NC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1487699	40800	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	8	1.6	COC(=O)c1ccc(NC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	16025367	40896	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	7	1	7	5.4	COc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)cc1	nan
	CHEMBL1488348	40896	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	7	1	7	5.4	COc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)cc1	nan
	4611609	40902	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	3	6.2	CCc1ccc(OCC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)c(Br)c1	nan
	CHEMBL1488388	40902	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	3	6.2	CCc1ccc(OCC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)c(Br)c1	nan
	1726407	40923	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	4	6.4	CCOc1cccc(C(=O)Nc2ccc3oc(-c4ccc(C(C)(C)C)cc4)nc3c2)c1	nan
	CHEMBL1488581	40923	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	4	6.4	CCOc1cccc(C(=O)Nc2ccc3oc(-c4ccc(C(C)(C)C)cc4)nc3c2)c1	nan
	16030737	40959	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	10	2.0	Cc1ccc(-c2nc(SCC(=O)Nc3cc(C)on3)c3c(=O)n(C)c(=O)n(C)c3n2)cc1	nan
	CHEMBL1488787	40959	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	10	2.0	Cc1ccc(-c2nc(SCC(=O)Nc3cc(C)on3)c3c(=O)n(C)c(=O)n(C)c3n2)cc1	nan
	824820	41008	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	5	3.1	Cc1ccc(-n2c(N)c(C#N)c(-c3ccccc3)c(C#N)c2=O)cc1	nan
	CHEMBL1489157	41008	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	5	3.1	Cc1ccc(-n2c(N)c(C#N)c(-c3ccccc3)c(C#N)c2=O)cc1	nan
	2036296	41049	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	6	4.0	CCCCn1c(-c2cccs2)nc2oc3ccccc3c(=O)c2c1=O	nan
	CHEMBL1489469	41049	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	6	4.0	CCCCn1c(-c2cccs2)nc2oc3ccccc3c(=O)c2c1=O	nan
	3448820	41105	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	0	4	4.8	COc1cc2c(cc1OC)C(COc1ccc(F)cc1)N(C(=O)c1ccccc1F)CC2	nan
	CHEMBL1489934	41105	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	0	4	4.8	COc1cc2c(cc1OC)C(COc1ccc(F)cc1)N(C(=O)c1ccccc1F)CC2	nan
	655760	41180	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	4	3.0	Cc1ccc(C)c(NC(=O)Cn2nc(C)c3ccccc3c2=O)c1	nan
	CHEMBL1490512	41180	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	4	3.0	Cc1ccc(C)c(NC(=O)Cn2nc(C)c3ccccc3c2=O)c1	nan
	16007588	41212	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	5	4.1	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCCc1ccc(Cl)cc1)cn2C	nan
	CHEMBL1490705	41212	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	5	4.1	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCCc1ccc(Cl)cc1)cn2C	nan
	1483825	41219	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.3	FC(F)(F)c1cnc(-c2cnc(-c3cccnc3)nc2)c(Cl)c1	nan
	CHEMBL1490743	41219	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.3	FC(F)(F)c1cnc(-c2cnc(-c3cccnc3)nc2)c(Cl)c1	nan
	16194118	41245	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	2.0	CCOC(=O)c1ccc(NC(=S)N2CCN(c3ccc(N4CCOCC4)nn3)CC2)cc1	nan
	CHEMBL1490926	41245	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	2.0	CCOC(=O)c1ccc(NC(=S)N2CCN(c3ccc(N4CCOCC4)nn3)CC2)cc1	nan
	4578555	41266	17	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCCC1	nan
	CHEMBL1491054	41266	17	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCCC1	nan
	1147591	41327	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	CHEMBL1491533	41327	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	761949	41459	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.7	CC(=O)c1cnc2cc(-c3cccc(Br)c3)nn2c1C	nan
	CHEMBL1492474	41459	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.7	CC(=O)c1cnc2cc(-c3cccc(Br)c3)nn2c1C	nan
	16031672	41507	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	2	4	2.8	O=C(Nc1ccc(F)cc1F)C1CCN(S(=O)(=O)c2ccc3[nH]c(=O)ccc3c2)CC1	nan
	CHEMBL1492791	41507	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	2	4	2.8	O=C(Nc1ccc(F)cc1F)C1CCN(S(=O)(=O)c2ccc3[nH]c(=O)ccc3c2)CC1	nan
	3496289	41539	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	11	2	7	3.7	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCCOC)cc3)c(=O)c2cc1OCC	nan
	CHEMBL1493174	41539	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	11	2	7	3.7	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCCOC)cc3)c(=O)c2cc1OCC	nan
	16033055	41552	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	10	0	11	3.4	CCOc1ccc(C(=O)Cn2c(=O)n3nc(CCn4nc(C)cc4C)nc3c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1493282	41552	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	10	0	11	3.4	CCOc1ccc(C(=O)Cn2c(=O)n3nc(CCn4nc(C)cc4C)nc3c3cc(OC)c(OC)cc32)cc1	nan
	6324582	41606	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	3.7	Cc1ccc2cc(CCNC(=O)CC(C)(C)C)c(O)nc2c1C	nan
	CHEMBL1493825	41606	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	3.7	Cc1ccc2cc(CCNC(=O)CC(C)(C)C)c(O)nc2c1C	nan
	2337492	41676	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	5	5.2	CCOC(=O)c1c(C)oc2c1cc(NS(=O)(=O)c1ccc(C)cc1)c1ccccc12	nan
	CHEMBL1494522	41676	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	5	5.2	CCOC(=O)c1c(C)oc2c1cc(NS(=O)(=O)c1ccc(C)cc1)c1ccccc12	nan
	16030367	41744	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	5.5	CCc1ccccc1NC(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1	nan
	CHEMBL1495193	41744	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	5.5	CCc1ccccc1NC(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1	nan
	659270	41750	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	1	8	2.7	CCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OC)cc2)c1C#N	nan
	CHEMBL1495223	41750	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	1	8	2.7	CCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OC)cc2)c1C#N	nan
	1473491	41751	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	0	4	4.3	O=C1c2ccccc2C(=O)N1CCc1csc(-c2cccc(Cl)c2)n1	nan
	CHEMBL1495238	41751	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	0	4	4.3	O=C1c2ccccc2C(=O)N1CCc1csc(-c2cccc(Cl)c2)n1	nan
	803577	41774	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.6	CC(=O)c1sc(NC(=O)c2ccc3c(c2)OCO3)nc1C	nan
	CHEMBL1495561	41774	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.6	CC(=O)c1sc(NC(=O)c2ccc3c(c2)OCO3)nc1C	nan
	16015766	41781	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	2	4.9	CC(C)CC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3[nH]2)c1	nan
	CHEMBL1495596	41781	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	2	4.9	CC(C)CC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3[nH]2)c1	nan
	1394903	41791	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	6	0	5	4.9	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Br)cc1	nan
	CHEMBL1495702	41791	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	6	0	5	4.9	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Br)cc1	nan
	9550975	41874	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	6	4.1	COc1ccccc1CNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1496499	41874	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	6	4.1	COc1ccccc1CNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	7190533	41911	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	6	3.8	Cc1ccccc1CSc1ccc2nnc(-c3ccccn3)n2n1	nan
	CHEMBL1496795	41911	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	6	3.8	Cc1ccccc1CSc1ccc2nnc(-c3ccccn3)n2n1	nan
	22548523	41924	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.8	CN(Cc1ccccc1)S(=O)(=O)c1ccc2nc(O)ccc2c1	nan
	CHEMBL1496881	41924	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.8	CN(Cc1ccccc1)S(=O)(=O)c1ccc2nc(O)ccc2c1	nan
	16030464	41939	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	4	5.1	COc1ccccc1C(=O)Nc1ccccc1SCc1cc(=O)c2ccccc2[nH]1	nan
	CHEMBL1497018	41939	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	4	5.1	COc1ccccc1C(=O)Nc1ccccc1SCc1cc(=O)c2ccccc2[nH]1	nan
	3282397	41969	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	3.8	CCOc1ccc(-n2nc(C(=O)NC3CCCCC3)c3ccccc3c2=O)cc1	nan
	CHEMBL1497244	41969	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	3.8	CCOc1ccc(-n2nc(C(=O)NC3CCCCC3)c3ccccc3c2=O)cc1	nan
	2190255	41975	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	3	6	-0.1	CCN1C(=O)/C(=C/Nc2ccc(S(N)(=O)=O)cc2)C(=O)NC1=S	nan
	CHEMBL1497307	41975	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	3	6	-0.1	CCN1C(=O)/C(=C/Nc2ccc(S(N)(=O)=O)cc2)C(=O)NC1=S	nan
	860457	42046	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	6	2.6	CSc1nnc(-c2ccc(S(=O)(=O)N3CCCCC3)cc2)o1	nan
	CHEMBL1497958	42046	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	6	2.6	CSc1nnc(-c2ccc(S(=O)(=O)N3CCCCC3)cc2)o1	nan
	2815318	42125	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	7	2.2	CCOC(=O)Cn1cnc2c(sc3nc(C)cc(C)c32)c1=O	nan
	CHEMBL1498797	42125	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	7	2.2	CCOC(=O)Cn1cnc2c(sc3nc(C)cc(C)c32)c1=O	nan
	2126242	42129	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.3	COc1ccc2c(C)cc(SCC(=O)Nc3cccnc3Cl)nc2c1	nan
	CHEMBL1498813	42129	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.3	COc1ccc2c(C)cc(SCC(=O)Nc3cccnc3Cl)nc2c1	nan
	1105537	42218	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	6	3.2	CCOC(=O)/C(C#N)=C/c1ccc(OCC(=O)Nc2ccccc2)c(OC)c1	nan
	CHEMBL1499500	42218	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	6	3.2	CCOC(=O)/C(C#N)=C/c1ccc(OCC(=O)Nc2ccccc2)c(OC)c1	nan
	649649	42231	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	6	2.0	Cc1ccnc(N2CCC(C(=O)NCc3ccc4c(c3)OCO4)CC2)n1	nan
	CHEMBL1499616	42231	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	6	2.0	Cc1ccnc(N2CCC(C(=O)NCc3ccc4c(c3)OCO4)CC2)n1	nan
	866361	42232	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1499629	42232	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1Cc1ccc2c(c1)OCO2	nan
	2764824	42258	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	2	2.8	CNC(=O)c1cc(C(=O)c2ccc(C(F)(F)F)cc2F)c[nH]1	nan
	CHEMBL1499851	42258	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	2	2.8	CNC(=O)c1cc(C(=O)c2ccc(C(F)(F)F)cc2F)c[nH]1	nan
	852955	42293	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	4	5.0	Cc1sc2nc(Cc3ccccc3)nc(O)c2c1-c1ccccc1	nan
	CHEMBL1500159	42293	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	4	5.0	Cc1sc2nc(Cc3ccccc3)nc(O)c2c1-c1ccccc1	nan
	135415434	42449	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	7	2.3	Cc1ccc(S(=O)(=O)N2CCN(C(=O)CSc3nc(O)c4ccccc4n3)CC2)cc1	nan
	CHEMBL1501602	42449	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	7	2.3	Cc1ccc(S(=O)(=O)N2CCN(C(=O)CSc3nc(O)c4ccccc4n3)CC2)cc1	nan
	54676936	42470	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	2	4	3.0	O=C(Nc1cccc(F)c1)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	CHEMBL1501763	42470	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	2	4	3.0	O=C(Nc1cccc(F)c1)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	1176241	42526	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	6	4.5	CCOc1ccc2nc(SCC(=O)Nc3ccc(S(=O)(=O)N4CCCC4)cc3)c(C)cc2c1	nan
	CHEMBL1502202	42526	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	6	4.5	CCOc1ccc2nc(SCC(=O)Nc3ccc(S(=O)(=O)N4CCCC4)cc3)c(C)cc2c1	nan
	734457	42625	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	257	3	1	5	2.6	COC(=O)c1ccc(Nc2nc(C)cc(C)n2)cc1	nan
	CHEMBL1503104	42625	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	257	3	1	5	2.6	COC(=O)c1ccc(Nc2nc(C)cc(C)n2)cc1	nan
	2515869	42649	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	2.9	CCC(=O)c1ccc(OCC(=O)c2ccc3c(c2)NC(=O)CO3)cc1	nan
	CHEMBL1503299	42649	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	2.9	CCC(=O)c1ccc(OCC(=O)c2ccc3c(c2)NC(=O)CO3)cc1	nan
	5310469	42679	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	0	8	3.3	COc1ccc(-c2nnc3ccc(SCC(=O)N4CCCCCC4)nn23)cc1OC	nan
	CHEMBL1503498	42679	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	0	8	3.3	COc1ccc(-c2nnc3ccc(SCC(=O)N4CCCCCC4)nn23)cc1OC	nan
	3574258	42687	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccc(Cl)cc1	nan
	CHEMBL1503560	42687	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccc(Cl)cc1	nan
	1859366	42692	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	4	5.0	Cc1ccc(S(=O)(=O)N(Cc2cc3ccc(C)cc3nc2O)c2ccccc2)cc1	nan
	CHEMBL1503583	42692	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	4	5.0	Cc1ccc(S(=O)(=O)N(Cc2cc3ccc(C)cc3nc2O)c2ccccc2)cc1	nan
	664334	42797	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	0	4	4.2	O=C1CC(c2ccc(F)cc2)Cc2nc(N3CCc4ccccc43)ncc21	nan
	CHEMBL1504653	42797	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	0	4	4.2	O=C1CC(c2ccc(F)cc2)Cc2nc(N3CCc4ccccc43)ncc21	nan
	2980439	42856	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	7	2	4	3.2	CCc1ccc(N2CCN(CCNC(=O)Nc3ccc(OC)cc3)CC2)cc1	nan
	CHEMBL1505203	42856	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	7	2	4	3.2	CCc1ccc(N2CCN(CCNC(=O)Nc3ccc(OC)cc3)CC2)cc1	nan
	661657	42866	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	0	7	3.3	O=C1c2ccccc2C(=O)N1Cc1nn2c(-c3ccc(Cl)cc3)nnc2s1	nan
	CHEMBL1505268	42866	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	0	7	3.3	O=C1c2ccccc2C(=O)N1Cc1nn2c(-c3ccc(Cl)cc3)nnc2s1	nan
	12006071	42884	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	0	6	4.5	O=C(CSc1ccc2nnc(-c3ccc(Cl)cc3)n2n1)N1CCCc2ccccc21	nan
	CHEMBL1505466	42884	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	0	6	4.5	O=C(CSc1ccc2nnc(-c3ccc(Cl)cc3)n2n1)N1CCCc2ccccc21	nan
	834457	42948	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	2.7	NS(=O)(=O)c1ccc(NCc2c(F)cccc2Cl)cc1	nan
	CHEMBL1505860	42948	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	2.7	NS(=O)(=O)c1ccc(NCc2c(F)cccc2Cl)cc1	nan
	1804684	42954	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.8	COCc1cc(C)nc(SCC(=O)Nc2cccc(C)c2C)c1C#N	nan
	CHEMBL1505914	42954	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.8	COCc1cc(C)nc(SCC(=O)Nc2cccc(C)c2C)c1C#N	nan
	3882765	42983	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	2	1	3.9	Cc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3)cc2c1	nan
	CHEMBL1506222	42983	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	2	1	3.9	Cc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3)cc2c1	nan
	3795359	43022	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.8	CCC(C)c1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1	nan
	CHEMBL1506487	43022	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.8	CCC(C)c1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1	nan
	4118928	43027	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	7	2	5	2.1	CCCCOCCCN1C(C)=CC(=C2C(=O)NC(=S)NC2=O)C=C1C	nan
	CHEMBL1506535	43027	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	7	2	5	2.1	CCCCOCCCN1C(C)=CC(=C2C(=O)NC(=S)NC2=O)C=C1C	nan
	1078308	43083	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3ccccc3C)c(=O)c2c1C	nan
	CHEMBL1507058	43083	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3ccccc3C)c(=O)c2c1C	nan
	1390207	43091	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	0	5	4.8	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Cl)cc1	nan
	CHEMBL1507117	43091	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	0	5	4.8	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Cl)cc1	nan
	9550860	43109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	3	2.0	Cc1ccc(OC(=O)c2ccccc2P(=O)(O)O)cc1	nan
	CHEMBL1507343	43109	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	3	2.0	Cc1ccc(OC(=O)c2ccccc2P(=O)(O)O)cc1	nan
	2810073	43121	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.3	Cc1csc2c(=O)sc(NC(=O)c3cccs3)nc12	nan
	CHEMBL1507430	43121	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.3	Cc1csc2c(=O)sc(NC(=O)c3cccs3)nc12	nan
	20874463	43186	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	4.1	Cc1ccc(-c2nnn3c2nc(NC(C)C)c2ccccc23)cc1	nan
	CHEMBL1507945	43186	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	4.1	Cc1ccc(-c2nnn3c2nc(NC(C)C)c2ccccc23)cc1	nan
	5875901	43205	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	3.8	CCOC(=O)CN1C(=O)/C(=C/c2cccc(Br)c2)Oc2ccccc21	nan
	CHEMBL1508095	43205	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	3.8	CCOC(=O)CN1C(=O)/C(=C/c2cccc(Br)c2)Oc2ccccc21	nan
	649082	43236	2	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	2	7	2.6	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccco2)n1)NC1CCCCC1	nan
	CHEMBL1508376	43236	2	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	2	7	2.6	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccco2)n1)NC1CCCCC1	nan
	1735895	43537	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	7	3.2	CCc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	CHEMBL1511120	43537	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	7	3.2	CCc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	1186303	43562	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	2	6	3.3	CN(C)c1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1	nan
	CHEMBL1511271	43562	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	2	6	3.3	CN(C)c1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1	nan
	2815635	43598	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	2	4	5.7	O=C(Nc1ccccc1)Nc1sccc1-c1nc2ccccc2s1	nan
	CHEMBL1511507	43598	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	2	4	5.7	O=C(Nc1ccccc1)Nc1sccc1-c1nc2ccccc2s1	nan
	661880	43600	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	0	6	2.3	N#CCc1nc2c3c4c(sc3ncn2n1)CCCC4	nan
	CHEMBL1511519	43600	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	0	6	2.3	N#CCc1nc2c3c4c(sc3ncn2n1)CCCC4	nan
	4604131	43641	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	7	3.9	COc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1512120	43641	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	7	3.9	COc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3ccsc3c2=O)cc1	nan
	16027453	43673	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1ccccc1C(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1512551	43673	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1ccccc1C(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2c(C)csc2n1	nan
	16018474	43675	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	5.8	CCc1ccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)cc1	nan
	CHEMBL1512597	43675	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	5.8	CCc1ccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)cc1	nan
	16030606	43677	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4cccc(C)c4n3)c2)c1	nan
	CHEMBL1512611	43677	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4cccc(C)c4n3)c2)c1	nan
	16030447	43678	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4ccccc4Cl)c3)cc(=O)n2c1	nan
	CHEMBL1512613	43678	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4ccccc4Cl)c3)cc(=O)n2c1	nan
	7245878	43685	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	6	2.6	COc1ccc(S(=O)(=O)c2cc3cc(OC)ccc3oc2=O)cc1	nan
	CHEMBL1512705	43685	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	6	2.6	COc1ccc(S(=O)(=O)c2cc3cc(OC)ccc3oc2=O)cc1	nan
	16020157	43705	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	9	3.6	CCOC(=O)CSc1nc2cc(OC)c(OC)cc2c2nc(-c3ccccc3)nn12	nan
	CHEMBL1512982	43705	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	9	3.6	CCOC(=O)CSc1nc2cc(OC)c(OC)cc2c2nc(-c3ccccc3)nn12	nan
	16023839	43706	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	3	0	6	4.0	CN1CCN(C(=O)c2cnn(-c3cccc(Cl)c3)c2C2CCN(C(=O)OC(C)(C)C)CC2)CC1	nan
	CHEMBL1513006	43706	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	3	0	6	4.0	CN1CCN(C(=O)c2cnn(-c3cccc(Cl)c3)c2C2CCN(C(=O)OC(C)(C)C)CC2)CC1	nan
	3402023	43708	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	8	2	5	5.4	COc1ccc(CNC(=O)c2ccc(Sc3ccc(Cl)cc3)c(NC(C)=O)c2)c(OC)c1	nan
	CHEMBL1513023	43708	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	8	2	5	5.4	COc1ccc(CNC(=O)c2ccc(Sc3ccc(Cl)cc3)c(NC(C)=O)c2)c(OC)c1	nan
	16014785	43709	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	2	6	4.5	COC(=O)c1ccc(NC(=O)CSc2nc(C)cc(C)c2C(=O)Nc2ccccc2)cc1	nan
	CHEMBL1513057	43709	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	2	6	4.5	COC(=O)c1ccc(NC(=O)CSc2nc(C)cc(C)c2C(=O)Nc2ccccc2)cc1	nan
	16021019	43711	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(CSc2nc3cccnc3n2Cc2ccc(F)cc2)cc1	nan
	CHEMBL1513070	43711	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(CSc2nc3cccnc3n2Cc2ccc(F)cc2)cc1	nan
	16008530	43717	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	5	6.0	CSc1ccc(CCNC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccc(C)c(C)c3)c2C)cc1	nan
	CHEMBL1513168	43717	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	5	6.0	CSc1ccc(CCNC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccc(C)c(C)c3)c2C)cc1	nan
	16018739	43728	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.0	O=C(CCn1c(=O)c2cccn2c2cccnc21)NCc1ccc(Cl)cc1	nan
	CHEMBL1513371	43728	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.0	O=C(CCn1c(=O)c2cccn2c2cccnc21)NCc1ccc(Cl)cc1	nan
	16030719	43731	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	9	2.0	Cc1cccc(-c2nc(SCC(=O)NCc3ccco3)c3c(=O)n(C)c(=O)n(C)c3n2)c1	nan
	CHEMBL1513435	43731	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	9	2.0	Cc1cccc(-c2nc(SCC(=O)NCc3ccco3)c3c(=O)n(C)c(=O)n(C)c3n2)c1	nan
	16025371	43733	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	568	6	1	6	6.0	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)c1	nan
	CHEMBL1513466	43733	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	568	6	1	6	6.0	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)c1	nan
	16026779	43737	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	8	2.8	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1513507	43737	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	8	2.8	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16024940	43739	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	4.9	O=C(NCCc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1513535	43739	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	4.9	O=C(NCCc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	1316309	43751	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1ccc2oc(-c3ccc(Cl)c(NC(=O)Cc4ccccc4)c3)nc2c1	nan
	CHEMBL1513652	43751	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1ccc2oc(-c3ccc(Cl)c(NC(=O)Cc4ccccc4)c3)nc2c1	nan
	16025593	43766	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	3	0	8	3.9	Cc1c(-c2nc(-c3ccc4c(c3)OCO4)no2)nnn1-c1ccc(Br)cc1F	nan
	CHEMBL1514000	43766	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	3	0	8	3.9	Cc1c(-c2nc(-c3ccc4c(c3)OCO4)no2)nnn1-c1ccc(Br)cc1F	nan
	15989077	43781	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	10	1	8	4.8	Cc1cc(C)c(Cn2c(=O)n(CCCCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1514246	43781	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	10	1	8	4.8	Cc1cc(C)c(Cn2c(=O)n(CCCCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	2689697	43786	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	3.2	COc1ccc(C(=O)OCC(=O)c2c[nH]c3ccccc23)cc1OC	nan
	CHEMBL1514340	43786	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	3.2	COc1ccc(C(=O)OCC(=O)c2c[nH]c3ccccc23)cc1OC	nan
	24982480	43799	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	5	2.3	CCN(Cc1ccccc1)C(=O)Cc1ccc(OC)c(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1514540	43799	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	5	2.3	CCN(Cc1ccccc1)C(=O)Cc1ccc(OC)c(S(=O)(=O)N2CCOCC2)c1	nan
	16015735	43824	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	3	3	9	2.5	COC(=O)c1c(C)sc(-c2c(-c3ccc4c(c3)OCCO4)[nH]c3c2c(=O)[nH]c(=O)n3C)c1O	nan
	CHEMBL1514818	43824	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	3	3	9	2.5	COC(=O)c1c(C)sc(-c2c(-c3ccc4c(c3)OCCO4)[nH]c3c2c(=O)[nH]c(=O)n3C)c1O	nan
	16022151	43828	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	6	2.5	COc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1C)n2C	nan
	CHEMBL1514879	43828	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	6	2.5	COc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1C)n2C	nan
	16009667	43836	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	5	4.5	O=c1c2sc3ccccc3c2n(Cc2ccccc2)c(=O)n1Cc1ccccc1	nan
	CHEMBL1515036	43836	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	5	4.5	O=c1c2sc3ccccc3c2n(Cc2ccccc2)c(=O)n1Cc1ccccc1	nan
	5167801	43839	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	O=C(NC1CCCCC1)c1cc(Nc2ccccc2)nc2ccccc12	nan
	CHEMBL1515050	43839	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	O=C(NC1CCCCC1)c1cc(Nc2ccccc2)nc2ccccc12	nan
	16030854	43841	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	2	4	5.0	CC(NC(=O)c1ccc(NC(=O)c2nsc3ccccc23)cc1)c1ccccc1	nan
	CHEMBL1515130	43841	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	2	4	5.0	CC(NC(=O)c1ccc(NC(=O)c2nsc3ccccc23)cc1)c1ccccc1	nan
	135416423	43862	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	4	4.7	CCc1ccc2oc(-c3cc(NC(=O)C(C)C)cc(C)c3O)nc2c1	nan
	CHEMBL1515394	43862	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	4	4.7	CCc1ccc2oc(-c3cc(NC(=O)C(C)C)cc(C)c3O)nc2c1	nan
	8057488	43883	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	5.4	Cc1cc2nc(-c3ccc(OCc4ccccc4F)cc3)cc(C(F)(F)F)n2n1	nan
	CHEMBL1515771	43883	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	5.4	Cc1cc2nc(-c3ccc(OCc4ccccc4F)cc3)cc(C(F)(F)F)n2n1	nan
	4154278	43885	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1C	nan
	CHEMBL1515779	43885	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1C	nan
	16017003	43911	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	4	4.5	CCOc1ccccc1NC(=O)C(=O)c1cc(C)n(-c2ccc(F)cc2)c1C	nan
	CHEMBL1516117	43911	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	4	4.5	CCOc1ccccc1NC(=O)C(=O)c1cc(C)n(-c2ccc(F)cc2)c1C	nan
	7343169	43922	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	5	4.9	CCOC(=O)c1cnc2cc(-c3ccc(Cl)cc3)nn2c1-c1ccccc1	nan
	CHEMBL1516275	43922	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	5	4.9	CCOC(=O)c1cnc2cc(-c3ccc(Cl)cc3)nn2c1-c1ccccc1	nan
	3586950	43930	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	6	4.6	O=C(CSc1nc2ccsc2c(=O)n1-c1ccc(Br)cc1)NCc1ccccc1	nan
	CHEMBL1516478	43930	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	6	4.6	O=C(CSc1nc2ccsc2c(=O)n1-c1ccc(Br)cc1)NCc1ccccc1	nan
	3206747	44071	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	COc1cccc(CC(=O)Nc2nc3c(s2)C(=O)CC(C)(C)C3)c1	nan
	CHEMBL1517888	44071	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	COc1cccc(CC(=O)Nc2nc3c(s2)C(=O)CC(C)(C)C3)c1	nan
	985821	44075	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1cc(F)cc(F)c1)c1sc(Cl)nc1-c1ccccc1	nan
	CHEMBL1517907	44075	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1cc(F)cc(F)c1)c1sc(Cl)nc1-c1ccccc1	nan
	1093907	44076	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	7	1.5	CNS(=O)(=O)c1ccc(NC(=O)c2nc3nc(C)cc(C(F)F)n3n2)cc1	nan
	CHEMBL1517917	44076	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	7	1.5	CNS(=O)(=O)c1ccc(NC(=O)c2nc3nc(C)cc(C(F)F)n3n2)cc1	nan
	15991337	44099	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	0	7	4.8	CCc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1518140	44099	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	0	7	4.8	CCc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	16011836	44141	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	5.0	COc1ccc(CSc2nc3ccncc3n2CC(=O)Nc2cc(C)cc(C)c2)cc1	nan
	CHEMBL1518592	44141	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	5.0	COc1ccc(CSc2nc3ccncc3n2CC(=O)Nc2cc(C)cc(C)c2)cc1	nan
	1086869	44190	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	6	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)c(OC)c1	nan
	CHEMBL1518977	44190	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	6	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)c(OC)c1	nan
	730225	44203	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	2	6	2.2	N#CCc1c(C#N)c(N)nc(Nc2ccccc2)c1C#N	nan
	CHEMBL1519080	44203	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	2	6	2.2	N#CCc1c(C#N)c(N)nc(Nc2ccccc2)c1C#N	nan
	1008965	44215	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	4	6.1	CC(=O)c1cccc(NC(=O)c2cc(-c3ccc(Cl)s3)nc3ccccc23)c1	nan
	CHEMBL1519196	44215	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	4	6.1	CC(=O)c1cccc(NC(=O)c2cc(-c3ccc(Cl)s3)nc3ccccc23)c1	nan
	16025959	44298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	8	1.6	O=C(NCCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1519916	44298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	8	1.6	O=C(NCCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	2740242	44305	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	2	2	4	3.1	Cc1noc(C(F)(F)F)c1C(=O)NNC(=O)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1519973	44305	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	2	2	4	3.1	Cc1noc(C(F)(F)F)c1C(=O)NNC(=O)c1cccc(C(F)(F)F)c1	nan
	16020184	44397	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	8	0	9	5.3	COc1cc2nc(SCc3cccc(Cl)c3)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	CHEMBL1520786	44397	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	8	0	9	5.3	COc1cc2nc(SCc3cccc(Cl)c3)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	15989989	44400	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	8	2	9	3.4	COc1ccc(CCNC(=O)c2ccc(Nc3nc4ccccc4n4nnnc34)cc2)cc1OC	nan
	CHEMBL1520796	44400	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	8	2	9	3.4	COc1ccc(CCNC(=O)c2ccc(Nc3nc4ccccc4n4nnnc34)cc2)cc1OC	nan
	742057	44441	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	6	3.1	O=C(Nc1nc2ccc([N+](=O)[O-])cc2s1)c1ccco1	nan
	CHEMBL1521136	44441	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	6	3.1	O=C(Nc1nc2ccc([N+](=O)[O-])cc2s1)c1ccco1	nan
	16026879	44469	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	6	4.4	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(SC)cc4)cc3c2=O)cc1	nan
	CHEMBL1521365	44469	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	6	4.4	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(SC)cc4)cc3c2=O)cc1	nan
	1164118	44482	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	0	7	3.4	COc1ccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)cc1OC	nan
	CHEMBL1521488	44482	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	0	7	3.4	COc1ccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)cc1OC	nan
	3146504	44536	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	CHEMBL1521972	44536	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	16021952	44568	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	7	1	7	3.9	CCc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3c2c2cc(OC)ccc2n3C)c1	nan
	CHEMBL1522220	44568	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	7	1	7	3.9	CCc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3c2c2cc(OC)ccc2n3C)c1	nan
	4090626	44619	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	4	5.8	CCOc1ccc(NC(=O)c2c(NC(=O)Cc3ccccc3)sc3c2CCCCC3)cc1	nan
	CHEMBL1522769	44619	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	4	5.8	CCOc1ccc(NC(=O)c2c(NC(=O)Cc3ccccc3)sc3c2CCCCC3)cc1	nan
	3148294	44625	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	6	4.1	CC(C)CNC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	CHEMBL1522819	44625	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	6	4.1	CC(C)CNC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	16030650	44649	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	5	0	8	3.0	O=c1cc(CN2CCN(S(=O)(=O)c3ccccc3)CC2)nc2sc(-c3ccccc3Cl)nn12	nan
	CHEMBL1522977	44649	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	5	0	8	3.0	O=c1cc(CN2CCN(S(=O)(=O)c3ccccc3)CC2)nc2sc(-c3ccccc3Cl)nn12	nan
	16026964	44691	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccccc1F)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1523393	44691	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccccc1F)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	16027395	44715	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	10	3.4	CCOCCc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	CHEMBL1523585	44715	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	10	3.4	CCOCCc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	2465708	44724	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	6	1	9	4.8	COc1ccccc1-n1c(=O)c(C#N)c(-c2ccc([N+](=O)[O-])cc2)c2cc(C(=O)c3ccccc3O)cnc21	nan
	CHEMBL1523696	44724	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	6	1	9	4.8	COc1ccccc1-n1c(=O)c(C#N)c(-c2ccc([N+](=O)[O-])cc2)c2cc(C(=O)c3ccccc3O)cnc21	nan
	1465904	44741	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	1	7	4.8	CCc1nnc(NC(=O)CSc2nc(C3CCCCC3)nc3ccccc23)s1	nan
	CHEMBL1523892	44741	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	1	7	4.8	CCc1nnc(NC(=O)CSc2nc(C3CCCCC3)nc3ccccc23)s1	nan
	7422674	44742	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	3	4.2	O=C(Nc1ccccc1C(F)(F)F)c1cccn(Cc2ccccc2)c1=O	nan
	CHEMBL1523907	44742	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	3	4.2	O=C(Nc1ccccc1C(F)(F)F)c1cccn(Cc2ccccc2)c1=O	nan
	15989150	44786	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	6	3.6	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccc(C)cc2)c1=O	nan
	CHEMBL1524350	44786	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	6	3.6	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccc(C)cc2)c1=O	nan
	2548636	44869	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	3	7	2.5	Cc1nc(SCC(=O)Nc2cc(C(N)=O)cc(C(N)=O)c2)c2c(C)c(C)sc2n1	nan
	CHEMBL1525189	44869	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	3	7	2.5	Cc1nc(SCC(=O)Nc2cc(C(N)=O)cc(C(N)=O)c2)c2c(C)c(C)sc2n1	nan
	15989883	44873	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	3	5.4	Cc1c(C(=O)OC2CCCCC2)[nH]c2c1C(=O)CC(c1ccccc1Cl)C2	nan
	CHEMBL1525262	44873	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	3	5.4	Cc1c(C(=O)OC2CCCCC2)[nH]c2c1C(=O)CC(c1ccccc1Cl)C2	nan
	1186420	44916	10	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	7	3.8	Clc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	CHEMBL1525610	44916	10	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	7	3.8	Clc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	4154665	44920	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	2	7	3.3	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCOC)cc3)c(=O)c2cc1OCC	nan
	CHEMBL1525634	44920	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	2	7	3.3	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCOC)cc3)c(=O)c2cc1OCC	nan
	135460528	44975	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	2	5	3.5	Cc1ccc(N2C(=O)NC(=O)/C(=C/Nc3ncc(Br)cc3Br)C2=O)cc1	nan
	CHEMBL1526117	44975	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	2	5	3.5	Cc1ccc(N2C(=O)NC(=O)/C(=C/Nc3ncc(Br)cc3Br)C2=O)cc1	nan
	579848	45033	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	1	3	4.7	O=C(Nc1ccc(-c2ccc([N+](=O)[O-])cc2)cc1)c1ccccc1F	nan
	CHEMBL1526496	45033	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	1	3	4.7	O=C(Nc1ccc(-c2ccc([N+](=O)[O-])cc2)cc1)c1ccccc1F	nan
	16018883	45093	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	4	4.6	Cc1ccc(C)c(NC(=O)CCCN2C(=O)C(c3ccccc3)Oc3cccnc32)c1	nan
	CHEMBL1527105	45093	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	4	4.6	Cc1ccc(C)c(NC(=O)CCCN2C(=O)C(c3ccccc3)Oc3cccnc32)c1	nan
	2765322	45139	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	7	1.1	N#Cc1cc(C#N)c(N2CCN(c3ccccn3)CC2)nc1N	nan
	CHEMBL1527484	45139	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	7	1.1	N#Cc1cc(C#N)c(N2CCN(c3ccccn3)CC2)nc1N	nan
	16009430	45172	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.7	CCC(CC)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1527797	45172	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.7	CCC(CC)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	16015678	45173	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CCC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	CHEMBL1527810	45173	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CCC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	16009490	45221	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	CHEMBL1528261	45221	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	16016701	45224	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	2.6	COC(=O)c1ccccc1NC(=O)CCC(=O)N1CCOc2ccccc21	nan
	CHEMBL1528274	45224	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	2.6	COC(=O)c1ccccc1NC(=O)CCC(=O)N1CCOc2ccccc21	nan
	16391033	45240	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	3	3.8	COc1cc2ccccc2cc1C(=O)Nc1ccc(C)cn1	nan
	CHEMBL1528436	45240	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	3	3.8	COc1cc2ccccc2cc1C(=O)Nc1ccc(C)cn1	nan
	7185472	45262	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	2	6	2.6	CCOC(=O)c1ccccc1NC(=O)CSc1nc(=O)[nH]c2c1CCCC2	nan
	CHEMBL1528587	45262	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	2	6	2.6	CCOC(=O)c1ccccc1NC(=O)CSc1nc(=O)[nH]c2c1CCCC2	nan
	5310045	45316	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	5	4.2	Cc1c(C(=O)Nc2ccncc2)sc2nc(-c3ccc(F)cc3)cn12	nan
	CHEMBL1529086	45316	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	5	4.2	Cc1c(C(=O)Nc2ccncc2)sc2nc(-c3ccc(F)cc3)cn12	nan
	5146627	45354	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	0	6	5.1	COCCN(CCOC)c1ncnc2c1c(-c1ccccc1)cn2-c1ccc(C)c(Cl)c1	nan
	CHEMBL1529403	45354	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	0	6	5.1	COCCN(CCOC)c1ncnc2c1c(-c1ccccc1)cn2-c1ccc(C)c(Cl)c1	nan
	5181996	45368	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	4	0	6	1.0	CCOC(=O)Cc1nc2ccccc2n(CC#N)c1=O	nan
	CHEMBL1529516	45368	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	4	0	6	1.0	CCOC(=O)Cc1nc2ccccc2n(CC#N)c1=O	nan
	2099952	45395	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	4.9	Oc1nc(Cc2ccc(F)cc2)nc2scc(-c3ccc(F)cc3)c12	nan
	CHEMBL1529751	45395	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	4.9	Oc1nc(Cc2ccc(F)cc2)nc2scc(-c3ccc(F)cc3)c12	nan
	4373285	45423	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1Br	nan
	CHEMBL1529998	45423	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1Br	nan
	16024591	45467	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCCc3ccccc3)c2n1	nan
	CHEMBL1530480	45467	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCCc3ccccc3)c2n1	nan
	4994836	45616	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	Cc1ccccc1Nc1cc(C(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1531717	45616	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	Cc1ccccc1Nc1cc(C(=O)NC2CCCC2)c2ccccc2n1	nan
	982830	45661	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.7	Cc1cc2nnc(SCC(=O)Nc3ccc(F)c(Cl)c3)n2c2ccccc12	nan
	CHEMBL1532117	45661	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.7	Cc1cc2nnc(SCC(=O)Nc3ccc(F)c(Cl)c3)n2c2ccccc12	nan
	895668	45677	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	4	3.2	CC(=O)c1cccc(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	CHEMBL1532290	45677	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	4	3.2	CC(=O)c1cccc(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	2078424	45743	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	2	4	2.9	COc1cccc(CC(=O)Nc2sc3c(c2C(N)=O)CCCC3)c1	nan
	CHEMBL1532835	45743	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	2	4	2.9	COc1cccc(CC(=O)Nc2sc3c(c2C(N)=O)CCCC3)c1	nan
	718477	45746	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	1	0	6	2.1	COc1nc(C)nc2c1sc(=S)n2C	nan
	CHEMBL1532843	45746	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	1	0	6	2.1	COc1nc(C)nc2c1sc(=S)n2C	nan
	3239288	45785	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	2.9	CCC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	CHEMBL1533246	45785	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	2.9	CCC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	16025355	45824	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	7	1	6	5.5	CCc1ccccc1NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(C)cc1)S2(=O)=O	nan
	CHEMBL1533601	45824	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	7	1	6	5.5	CCc1ccccc1NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(C)cc1)S2(=O)=O	nan
	3214708	45844	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	2	8	2.5	CC(=O)Nc1ccc(S(=O)(=O)N2CCN(Cc3nc(O)c4c(C)c(C)sc4n3)CC2)cc1	nan
	CHEMBL1533736	45844	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	2	8	2.5	CC(=O)Nc1ccc(S(=O)(=O)N2CCN(Cc3nc(O)c4c(C)c(C)sc4n3)CC2)cc1	nan
	16028279	45860	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	3.2	CCOc1ccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)cc1	nan
	CHEMBL1533861	45860	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	3.2	CCOc1ccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)cc1	nan
	4046943	45877	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.5	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCC3)no1	nan
	CHEMBL1534012	45877	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.5	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCC3)no1	nan
	3932775	45893	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	3.8	CCc1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	CHEMBL1534252	45893	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	3.8	CCc1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	4658600	45928	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	7	1	6	6.0	CCN(CC)C(=O)c1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	CHEMBL1534562	45928	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	7	1	6	6.0	CCN(CC)C(=O)c1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	16025630	45974	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	1	7	3.7	COc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	CHEMBL1535077	45974	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	1	7	3.7	COc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	3185711	45987	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	9	3	8	2.6	CN(C)c1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2)cc1	nan
	CHEMBL1535224	45987	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	9	3	8	2.6	CN(C)c1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2)cc1	nan
	54677757	46024	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	4	3.4	Cn1c(=O)c(Sc2ccccc2)c(O)c2ccccc21	nan
	CHEMBL1535623	46024	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	4	3.4	Cn1c(=O)c(Sc2ccccc2)c(O)c2ccccc21	nan
	4792884	46057	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	6	2.9	COc1ccc(Br)cc1-c1nc2c(c(=O)[nH]c(=O)n2Cc2ccccc2)n1C	nan
	CHEMBL1535940	46057	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	6	2.9	COc1ccc(Br)cc1-c1nc2c(c(=O)[nH]c(=O)n2Cc2ccccc2)n1C	nan
	135516269	46088	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	3.1	CCOc1ccc(-n2c(SCC(=O)NC(C)CC)nc3nnc(C)c-3c2N)cc1	nan
	CHEMBL1536353	46088	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	3.1	CCOc1ccc(-n2c(SCC(=O)NC(C)CC)nc3nnc(C)c-3c2N)cc1	nan
	3208311	46108	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	3	9	2.5	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cnc(O)nc1O)OCO3	nan
	CHEMBL1536575	46108	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	3	9	2.5	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cnc(O)nc1O)OCO3	nan
	1965061	46163	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	0	6	4.0	CCCCCc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1536987	46163	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	0	6	4.0	CCCCCc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1Cc1ccc(OC)cc1	nan
	2296181	46205	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	3	2.4	O=C(CNC(=S)NC(=O)C1CCCCC1)c1ccccc1	nan
	CHEMBL1537419	46205	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	3	2.4	O=C(CNC(=S)NC(=O)C1CCCCC1)c1ccccc1	nan
	4358102	46237	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.8	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1537648	46237	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.8	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccc(F)cc2)CC1	nan
	16194098	46256	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	6	3.6	CSc1ccc(CNc2nc3ccccc3n3cnnc23)cc1	nan
	CHEMBL1537791	46256	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	6	3.6	CSc1ccc(CNc2nc3ccccc3n3cnnc23)cc1	nan
	1272394	46357	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	7	3.5	COc1ccc(C(=O)Nc2nnc(Cc3cccs3)s2)cc1OC	nan
	CHEMBL1538560	46357	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	7	3.5	COc1ccc(C(=O)Nc2nnc(Cc3cccs3)s2)cc1OC	nan
	921484	46453	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	4	4.1	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1	nan
	CHEMBL1539494	46453	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	4	4.1	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1	nan
	664170	46524	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	0	8	3.5	CCOC(=O)N1CCN(c2nc(SC)nc3sc4c(c23)CC(C)(C)OC4)CC1	nan
	CHEMBL1540011	46524	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	0	8	3.5	CCOC(=O)N1CCN(c2nc(SC)nc3sc4c(c23)CC(C)(C)OC4)CC1	nan
	6621296	46607	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	6	3.3	O=C(NCc1ccccc1)C1CCCN(c2nc3ccsc3c(=O)s2)C1	nan
	CHEMBL1540762	46607	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	6	3.3	O=C(NCc1ccccc1)C1CCCN(c2nc3ccsc3c(=O)s2)C1	nan
	2855521	46672	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	2	4	3.2	COc1ccc(COC(=O)C2=C(C)NC(=O)NC2c2ccc(F)cc2)cc1	nan
	CHEMBL1541261	46672	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	2	4	3.2	COc1ccc(COC(=O)C2=C(C)NC(=O)NC2c2ccc(F)cc2)cc1	nan
	687554	46700	23	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.1	CC(=O)Oc1ccc2oc(-c3ccccc3)c(C(N)=O)c2c1	nan
	CHEMBL1541470	46700	23	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.1	CC(=O)Oc1ccc2oc(-c3ccccc3)c(C(N)=O)c2c1	nan
	16746196	46880	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	10	3	5	3.2	CCCCNc1ccc(C(CC(N)=O)NC(=O)c2ccccc2)cc1[N+](=O)[O-]	nan
	CHEMBL1543039	46880	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	10	3	5	3.2	CCCCNc1ccc(C(CC(N)=O)NC(=O)c2ccccc2)cc1[N+](=O)[O-]	nan
	654907	46894	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	6	4.5	COc1ccc(C(=O)Nc2cccc(-c3nc4ncccc4o3)c2C)cc1OC	nan
	CHEMBL1543164	46894	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	6	4.5	COc1ccc(C(=O)Nc2cccc(-c3nc4ncccc4o3)c2C)cc1OC	nan
	899145	46922	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	0	5	4.1	Cc1cnn(C(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)c1	nan
	CHEMBL1543380	46922	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	0	5	4.1	Cc1cnn(C(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)c1	nan
	1337412	46926	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	146674638	46926	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	CHEMBL1543421	46926	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	1773311	46971	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.1	CCN(CC)C(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1543838	46971	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.1	CCN(CC)C(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	22553577	47042	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	5	3.5	O=C(CCCn1c(=O)c2cccn2c2cccnc21)NCc1cccc(Br)c1	nan
	CHEMBL1544274	47042	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	5	3.5	O=C(CCCn1c(=O)c2cccn2c2cccnc21)NCc1cccc(Br)c1	nan
	2150501	47222	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	8	3.5	COCCn1c(SCC(=O)Nc2ccc(OC)cc2)nc2c(oc3ccccc32)c1=O	nan
	CHEMBL1545636	47222	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	8	3.5	COCCn1c(SCC(=O)Nc2ccc(OC)cc2)nc2c(oc3ccccc32)c1=O	nan
	1131000	47230	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.2	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2F)c1C	nan
	CHEMBL1545709	47230	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.2	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2F)c1C	nan
	4975679	47326	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	1	1	1	4.0	O=C(c1cc2cc(Cl)ccc2[nH]1)N1CCc2ccccc2C1	nan
	CHEMBL1546589	47326	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	1	1	1	4.0	O=C(c1cc2cc(Cl)ccc2[nH]1)N1CCc2ccccc2C1	nan
	4099286	47373	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	8	1	4	3.8	CCOc1ccc(CNC(=O)CCc2cn(C)c3ccccc23)cc1OC	nan
	CHEMBL1547036	47373	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	8	1	4	3.8	CCOc1ccc(CNC(=O)CCc2cn(C)c3ccccc23)cc1OC	nan
	246421	47382	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	3	6	3.0	CSc1nc(O)c(Nc2cccc(Cl)c2)c(O)n1	nan
	CHEMBL1547116	47382	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	3	6	3.0	CSc1nc(O)c(Nc2cccc(Cl)c2)c(O)n1	nan
	3179963	47492	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	3	7	2.3	CCC(C(=O)NC1CCCC1)N(C(=O)c1snc(C(N)=O)c1N)c1ccc(OC)cc1	nan
	CHEMBL1548213	47492	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	3	7	2.3	CCC(C(=O)NC1CCCC1)N(C(=O)c1snc(C(N)=O)c1N)c1ccc(OC)cc1	nan
	16608827	47511	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	5	3.8	COc1ccc(S(=O)(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1NC(C)=O	nan
	CHEMBL1548379	47511	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	5	3.8	COc1ccc(S(=O)(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1NC(C)=O	nan
	1711150	47619	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	8	1	6	3.6	COc1cc(/C=C/C(=O)OCC(=O)Nc2ccccc2Cl)cc(OC)c1OC	nan
	CHEMBL1549297	47619	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	8	1	6	3.6	COc1cc(/C=C/C(=O)OCC(=O)Nc2ccccc2Cl)cc(OC)c1OC	nan
	4371420	47624	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	0	4	2.9	O=C(COC(=O)c1ccc(N2CCCC2=O)cc1)c1ccccc1	nan
	CHEMBL1549350	47624	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	0	4	2.9	O=C(COC(=O)c1ccc(N2CCCC2=O)cc1)c1ccccc1	nan
	650104	47752	2	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	3.8	CCc1cc2ccc(OC)cc2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1550363	47752	2	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	3.8	CCc1cc2ccc(OC)cc2nc1SCC(=O)Nc1cc(C)on1	nan
	891743	47797	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.5	Cc1nc(-c2ccc(C(=O)Nc3ccc(F)cc3)cc2)cs1	nan
	CHEMBL1550704	47797	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.5	Cc1nc(-c2ccc(C(=O)Nc3ccc(F)cc3)cc2)cs1	nan
	135437051	47842	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	3	6	4.1	CCc1ccccc1NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1cccc(C)c1	nan
	CHEMBL1551159	47842	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	3	6	4.1	CCc1ccccc1NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1cccc(C)c1	nan
	16030615	47846	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	0	9	3.1	COc1ccc(C(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccccc5C)sc4n3)CC2)cc1OC	nan
	CHEMBL1551229	47846	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	0	9	3.1	COc1ccc(C(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccccc5C)sc4n3)CC2)cc1OC	nan
	16018080	47849	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	6	3.5	COc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1OC	nan
	CHEMBL1551250	47849	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	6	3.5	COc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1OC	nan
	16012980	47858	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	3	5.3	Cc1ccc2nc(O)c(CN(C(=O)c3cccc(Cl)c3)C(C)(C)C)cc2c1	nan
	CHEMBL1551350	47858	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	3	5.3	Cc1ccc2nc(O)c(CN(C(=O)c3cccc(Cl)c3)C(C)(C)C)cc2c1	nan
	3534311	47865	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	6	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)COc3ccccc3)sc2c1	nan
	CHEMBL1551511	47865	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	6	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)COc3ccccc3)sc2c1	nan
	16030318	47867	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.5	CCOc1ccc(C(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)cc1	nan
	CHEMBL1551529	47867	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.5	CCOc1ccc(C(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)cc1	nan
	16031341	47873	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	2	1	5	1.9	Cc1ccccc1C(=O)Nc1nnc2n1CCS2	nan
	CHEMBL1551637	47873	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	2	1	5	1.9	Cc1ccccc1C(=O)Nc1nnc2n1CCS2	nan
	16012572	47877	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccc(Cl)cc3)c(C)nc21	nan
	CHEMBL1551773	47877	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccc(Cl)cc3)c(C)nc21	nan
	4112916	47891	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	0	5	5.2	CCOc1nc(-c2ccccc2)ccc1-c1noc(-c2ccc(C)cc2)n1	nan
	CHEMBL1551932	47891	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	0	5	5.2	CCOc1nc(-c2ccccc2)ccc1-c1noc(-c2ccc(C)cc2)n1	nan
	16030647	47893	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	6	0	8	3.6	CC(Oc1ccccc1)C(=O)N1CCN(Cc2cc(=O)n3nc(-c4ccccc4Cl)sc3n2)CC1	nan
	CHEMBL1551961	47893	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	6	0	8	3.6	CC(Oc1ccccc1)C(=O)N1CCN(Cc2cc(=O)n3nc(-c4ccccc4Cl)sc3n2)CC1	nan
	4069977	47901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.3	CCOc1ccc(Sc2cc(C(=O)NC(C)c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1552026	47901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.3	CCOc1ccc(Sc2cc(C(=O)NC(C)c3ccccc3)c3ccccc3n2)cc1	nan
	16027075	47909	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	0	8	4.8	COc1ccc(-c2nc(Cn3c(=O)cc(C)c4c(C)nn(-c5ccccc5)c43)c(C)o2)cc1OC	nan
	CHEMBL1552119	47909	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	0	8	4.8	COc1ccc(-c2nc(Cn3c(=O)cc(C)c4c(C)nn(-c5ccccc5)c43)c(C)o2)cc1OC	nan
	24792649	47913	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	0	0	3	3.5	Cn1c2ccccc2c(=O)c2ccc(C#Cc3ccccn3)cc21	nan
	CHEMBL1552163	47913	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	0	0	3	3.5	Cn1c2ccccc2c(=O)c2ccc(C#Cc3ccccn3)cc21	nan
	16020555	47935	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	0	5	4.8	O=c1c(S(=O)(=O)c2ccccc2)cn(Cc2cccc(F)c2)c2cc(N3CCCC3)c(F)cc12	nan
	CHEMBL1552450	47935	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	0	5	4.8	O=c1c(S(=O)(=O)c2ccccc2)cn(Cc2cccc(F)c2)c2cc(N3CCCC3)c(F)cc12	nan
	7217107	47938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	2.4	Cc1ccc(NC(=O)c2cnc(SCC(=O)Nc3cc(C)on3)n(C)c2=O)cc1	nan
	CHEMBL1552487	47938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	2.4	Cc1ccc(NC(=O)c2cnc(SCC(=O)Nc3cc(C)on3)n(C)c2=O)cc1	nan
	3666941	47939	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	6	1	6	4.9	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2-c2ccc(Br)cc2)cc1	nan
	CHEMBL1552556	47939	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	6	1	6	4.9	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2-c2ccc(Br)cc2)cc1	nan
	16010970	47952	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	0	7	3.6	CCc1cc2c(cc3c(=O)n(CC(=O)N4CCN(c5cc(Cl)ccc5C)CC4)ncn32)s1	nan
	CHEMBL1552740	47952	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	0	7	3.6	CCc1cc2c(cc3c(=O)n(CC(=O)N4CCN(c5cc(Cl)ccc5C)CC4)ncn32)s1	nan
	16021520	47955	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	4	4.6	CSc1ncc(C(=O)NCc2cccc(Br)c2)c(-c2ccccc2)n1	nan
	CHEMBL1552765	47955	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	4	4.6	CSc1ncc(C(=O)NCc2cccc(Br)c2)c(-c2ccccc2)n1	nan
	16024485	47974	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2n1	nan
	CHEMBL1553018	47974	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2n1	nan
	3160964	47978	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.6	Cc1cccc(OCC(=O)Nc2c(C)ccc3nsnc23)c1C	nan
	CHEMBL1553050	47978	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.6	Cc1cccc(OCC(=O)Nc2c(C)ccc3nsnc23)c1C	nan
	16012361	48026	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	5	4.2	CCc1ccccc1NC(=O)Cn1ncc2c(C)n(Cc3ccccc3F)c(C)c2c1=O	nan
	CHEMBL1553757	48026	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	5	4.2	CCc1ccccc1NC(=O)Cn1ncc2c(C)n(Cc3ccccc3F)c(C)c2c1=O	nan
	16027446	48042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(OCc1cc(=O)n2nc(C3CC3)sc2n1)c1ccc(NC(=O)c2ccccc2F)cc1	nan
	CHEMBL1553997	48042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(OCc1cc(=O)n2nc(C3CC3)sc2n1)c1ccc(NC(=O)c2ccccc2F)cc1	nan
	16030862	48069	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	3	3.1	CC(=O)N1CCc2cc(CNS(=O)(=O)c3ccccc3C(F)(F)F)ccc21	nan
	CHEMBL1554375	48069	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	3	3.1	CC(=O)N1CCc2cc(CNS(=O)(=O)c3ccccc3C(F)(F)F)ccc21	nan
	16030106	48078	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1ccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)cc1	nan
	CHEMBL1554505	48078	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1ccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)cc1	nan
	4074992	48084	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	4	5.9	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(F)cc3)c3ccccc3n2)cc1	nan
	CHEMBL1554644	48084	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	4	5.9	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(F)cc3)c3ccccc3n2)cc1	nan
	5058559	48096	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	2.9	CC(=O)c1cccc(NC(=O)c2ccc(S(=O)(=O)N3CC(C)OC(C)C3)cc2)c1	nan
	CHEMBL1554762	48096	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	2.9	CC(=O)c1cccc(NC(=O)c2ccc(S(=O)(=O)N3CC(C)OC(C)C3)cc2)c1	nan
	16026882	48097	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	8	3.5	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1554822	48097	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	8	3.5	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	4289361	48111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1cccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)c1	nan
	CHEMBL1555049	48111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1cccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)c1	nan
	3282564	48118	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	4	4.6	Cc1ccc(-c2nnc(NC(=O)c3c(F)cccc3Cl)s2)cc1	nan
	CHEMBL1555127	48118	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	4	4.6	Cc1ccc(-c2nnc(NC(=O)c3c(F)cccc3Cl)s2)cc1	nan
	16009325	48129	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	7	3.2	O=C(Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	CHEMBL1555288	48129	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	7	3.2	O=C(Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	135416425	48132	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	2	4	5.1	Cc1ccccc1C(=O)Nc1cc(C)c(O)c(-c2nc3ccccc3o2)c1	nan
	CHEMBL1555312	48132	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	2	4	5.1	Cc1ccccc1C(=O)Nc1cc(C)c(O)c(-c2nc3ccccc3o2)c1	nan
	16023840	48182	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	6	4.3	CCOC(=O)c1c(C)oc2nc(C)nc(NCc3ccccc3Cl)c12	nan
	CHEMBL1555863	48182	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	6	4.3	CCOC(=O)c1c(C)oc2nc(C)nc(NCc3ccccc3Cl)c12	nan
	4432211	48191	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	6	2.5	CC(=O)N1CCc2c(sc(NC(=O)c3ccc4c(c3)OCCO4)c2C#N)C1	nan
	CHEMBL1555967	48191	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	6	2.5	CC(=O)N1CCc2c(sc(NC(=O)c3ccc4c(c3)OCCO4)c2C#N)C1	nan
	929959	48226	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	8	0.8	COc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1556274	48226	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	8	0.8	COc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	1718133	48254	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	5	4.3	CCCCCC(=O)NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1	nan
	CHEMBL1556586	48254	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	5	4.3	CCCCCC(=O)NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1	nan
	1475314	48265	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	251	2	1	4	3.2	Cc1nc(N)ncc1Sc1ccc(Cl)cc1	nan
	CHEMBL1556672	48265	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	251	2	1	4	3.2	Cc1nc(N)ncc1Sc1ccc(Cl)cc1	nan
	1829088	48317	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	5	2.5	COCCNC(=O)Cn1nc(-c2ccc(Cl)cc2)c2ccccc2c1=O	nan
	CHEMBL1557090	48317	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	5	2.5	COCCNC(=O)Cn1nc(-c2ccc(Cl)cc2)c2ccccc2c1=O	nan
	16008924	48327	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	3	1	4	3.6	Cn1c(C(=O)NCc2ccc(Cl)cc2)cc2c(=O)n(C)c3ccccc3c21	nan
	CHEMBL1557189	48327	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	3	1	4	3.6	Cn1c(C(=O)NCc2ccc(Cl)cc2)cc2c(=O)n(C)c3ccccc3c21	nan
	20868637	48370	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	3.8	CCOc1ccc2ncc(S(=O)(=O)c3ccc(C)c(C)c3)c(O)c2c1	nan
	CHEMBL1557551	48370	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	3.8	CCOc1ccc2ncc(S(=O)(=O)c3ccc(C)c(C)c3)c(O)c2c1	nan
	16030924	48386	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	6	5.1	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccc(C)c(Cl)c4)ccc3n2)cc1	nan
	CHEMBL1557656	48386	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	6	5.1	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccc(C)c(Cl)c4)ccc3n2)cc1	nan
	899391	48391	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	2.8	O=C(Cc1ccccc1)Nc1nc(=O)c2ccccc2s1	nan
	CHEMBL1557721	48391	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	2.8	O=C(Cc1ccccc1)Nc1nc(=O)c2ccccc2s1	nan
	3846782	48393	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	4	1	7	4.1	Cc1ccc(Cn2c(=N)c(S(=O)(=O)c3ccc(Br)cc3)cc3c(=O)n4ccccc4nc32)cc1	nan
	CHEMBL1557740	48393	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	4	1	7	4.1	Cc1ccc(Cn2c(=N)c(S(=O)(=O)c3ccc(Br)cc3)cc3c(=O)n4ccccc4nc32)cc1	nan
	1485561	48415	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	3	0	5	4.4	O=S(=O)(c1ccccc1)c1cnn2c(C(F)(F)F)cc(-c3ccc(F)cc3)nc12	nan
	CHEMBL1557929	48415	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	3	0	5	4.4	O=S(=O)(c1ccccc1)c1cnn2c(C(F)(F)F)cc(-c3ccc(F)cc3)nc12	nan
	54706216	48471	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	3	4	3.5	O=C(NC1CCCCCCC1)c1c(O)nc2ccccc2c1O	nan
	CHEMBL1558469	48471	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	3	4	3.5	O=C(NC1CCCCCCC1)c1c(O)nc2ccccc2c1O	nan
	5185520	48482	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	2	4	2.5	Nc1cc(Cl)ccc1C(=O)OCC(=O)NC1CCCCC1	nan
	CHEMBL1558534	48482	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	2	4	2.5	Nc1cc(Cl)ccc1C(=O)OCC(=O)NC1CCCCC1	nan
	666603	48516	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	6	4.1	Cc1nn(-c2ccc(F)cc2)c2nc(N)c(C#N)c(-c3cccs3)c12	nan
	CHEMBL1558784	48516	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	6	4.1	Cc1nn(-c2ccc(F)cc2)c2nc(N)c(C#N)c(-c3cccs3)c12	nan
	15991438	48524	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	6	3.8	Cc1cccc(NC(=O)CSc2nc3ccccc3nc2N2CCOCC2)c1C	nan
	CHEMBL1558859	48524	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	6	3.8	Cc1cccc(NC(=O)CSc2nc3ccccc3nc2N2CCOCC2)c1C	nan
	950988	48540	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	2	5	4.8	COc1cccc(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	CHEMBL1558977	48540	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	2	5	4.8	COc1cccc(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	4345257	48551	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	2	6	3.2	Cc1cc(C)cc(NC(=O)CSc2nnc(NC(=O)C3CC3)s2)c1	nan
	CHEMBL1559060	48551	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	2	6	3.2	Cc1cc(C)cc(NC(=O)CSc2nnc(NC(=O)C3CC3)s2)c1	nan
	900716	48563	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	5	3.6	COC(=O)c1ccc(NC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	CHEMBL1559158	48563	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	5	3.6	COC(=O)c1ccc(NC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	2156049	48633	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	4	5.5	Cc1ccc(-n2c(SCc3ccccc3)nc3c([nH]c4ccccc43)c2=O)cc1	nan
	CHEMBL1559857	48633	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	4	5.5	Cc1ccc(-n2c(SCc3ccccc3)nc3c([nH]c4ccccc43)c2=O)cc1	nan
	3138574	48636	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	3	4	3.6	O=C(NNc1c2ccccc2nc2ccccc12)C(O)c1ccccc1	nan
	CHEMBL1559872	48636	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	3	4	3.6	O=C(NNc1c2ccccc2nc2ccccc12)C(O)c1ccccc1	nan
	16017814	48654	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	6	2.9	COc1ccc(Cl)cc1NC(=O)Cn1ccn(-c2cc(C)cc(C)c2)c(=O)c1=O	nan
	CHEMBL1560031	48654	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	6	2.9	COc1ccc(Cl)cc1NC(=O)Cn1ccn(-c2cc(C)cc(C)c2)c(=O)c1=O	nan
	2028031	48728	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	1	0	5	3.5	Cc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1C1CCCCCC1	nan
	CHEMBL1560823	48728	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	1	0	5	3.5	Cc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1C1CCCCCC1	nan
	4690835	48731	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	COc1ccc2oc(-c3cccc(NC(=O)c4ccc(C#N)cc4F)c3)nc2c1	nan
	CHEMBL1560860	48731	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	COc1ccc2oc(-c3cccc(NC(=O)c4ccc(C#N)cc4F)c3)nc2c1	nan
	15990056	48903	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	5	4.4	CCc1nnc2c3ccccc3nc(Nc3ccc(F)c(Cl)c3)n12	nan
	CHEMBL1562390	48903	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	5	4.4	CCc1nnc2c3ccccc3nc(Nc3ccc(F)c(Cl)c3)n12	nan
	5299641	48907	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	4.6	Cc1ccc(Cl)cc1NC(=O)CSc1nc(C)c(C)c(C)c1C#N	nan
	CHEMBL1562426	48907	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	4.6	Cc1ccc(Cl)cc1NC(=O)CSc1nc(C)c(C)c(C)c1C#N	nan
	135496880	48910	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	9	3.5	Oc1nc(SCc2nc(O)c3cnn(-c4ccccc4)c3n2)nc2ccccc12	nan
	CHEMBL1562459	48910	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	9	3.5	Oc1nc(SCc2nc(O)c3cnn(-c4ccccc4)c3n2)nc2ccccc12	nan
	1176245	48956	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	4.0	CCOc1ccc2nc(SCC(=O)Nc3cc(C)on3)c(C)cc2c1	nan
	CHEMBL1562840	48956	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	4.0	CCOc1ccc2nc(SCC(=O)Nc3cc(C)on3)c(C)cc2c1	nan
	16030293	48959	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	5	6.0	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1562857	48959	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	5	6.0	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)Nc1ccccc1C(F)(F)F	nan
	16008836	49038	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.2	O=C(NCCCN1CCN(c2ccc(F)cc2)CC1)c1cc2c(Cl)nc3ccccc3c2s1	nan
	CHEMBL1563658	49038	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.2	O=C(NCCCN1CCN(c2ccc(F)cc2)CC1)c1cc2c(Cl)nc3ccccc3c2s1	nan
	258436	49108	41	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	1	0	2	2.5	CN1C=CC(=CC=C2C=CC(=O)C=C2)C=C1	nan
	CHEMBL1564141	49108	41	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	1	0	2	2.5	CN1C=CC(=CC=C2C=CC(=O)C=C2)C=C1	nan
	16030542	49127	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2cccc(OCc3cc(=O)n4ccccc4n3)c2)cc1C	nan
	CHEMBL1564400	49127	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2cccc(OCc3cc(=O)n4ccccc4n3)c2)cc1C	nan
	2819137	49187	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	1	6	2.3	COc1cccc(-c2nc(N)nc(SC)c2C#N)c1	nan
	CHEMBL1564918	49187	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	1	6	2.3	COc1cccc(-c2nc(N)nc(SC)c2C#N)c1	nan
	3244591	49191	1	None	-100	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	6	4.3	CC(C)CCn1c(SCC#N)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1564940	49191	1	None	-100	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	6	4.3	CC(C)CCn1c(SCC#N)nc2c(sc3ccccc32)c1=O	nan
	16010206	49203	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	CHEMBL1565063	49203	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	1147655	49206	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	7	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1OC	nan
	CHEMBL1565079	49206	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	7	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1OC	nan
	694360	49255	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	5	3.1	N#Cc1c(-c2cccs2)cc(C2CC2)nc1SCC(N)=O	nan
	CHEMBL1565417	49255	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	5	3.1	N#Cc1c(-c2cccs2)cc(C2CC2)nc1SCC(N)=O	nan
	16021091	49298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1565772	49298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3cccnc32)cc1	nan
	16019049	49382	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	7	3.6	COc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c(OC)c1	nan
	CHEMBL1566421	49382	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	7	3.6	COc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c(OC)c1	nan
	2810064	49390	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	7	2.5	COc1cc2nc(NC(=O)c3ccco3)sc(=O)c2cc1OC	nan
	CHEMBL1566488	49390	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	7	2.5	COc1cc2nc(NC(=O)c3ccco3)sc(=O)c2cc1OC	nan
	15988926	49543	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	12	1	7	3.0	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1567696	49543	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	12	1	7	3.0	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	16017081	49632	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	4.5	CCC(C(=O)Nc1ccccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1568421	49632	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	4.5	CCC(C(=O)Nc1ccccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	16030322	49683	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	8	2.9	CCCC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1	nan
	CHEMBL1568901	49683	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	8	2.9	CCCC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1	nan
	713644	49699	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	5	1.4	Cc1cn(C(=O)CN2C(=O)c3ccccc3C2=O)c(C)n1	nan
	CHEMBL1569010	49699	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	5	1.4	Cc1cn(C(=O)CN2C(=O)c3ccccc3C2=O)c(C)n1	nan
	16024577	49738	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	3.7	COc1cc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc(OC)c1	nan
	CHEMBL1569365	49738	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	3.7	COc1cc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc(OC)c1	nan
	1146106	49762	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	5	5.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(Cl)cc3)n2)cc1	nan
	CHEMBL1569521	49762	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	5	5.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(Cl)cc3)n2)cc1	nan
	1433832	49784	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	4	1	4	2.5	N#Cc1cc2ccccc2nc1SCC(=O)NC1CC1	nan
	CHEMBL1569775	49784	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	4	1	4	2.5	N#Cc1cc2ccccc2nc1SCC(=O)NC1CC1	nan
	660750	49788	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	1	5	2.9	Cn1nnnc1-c1cc(Br)ccc1NC(=O)c1ccccc1	nan
	CHEMBL1569814	49788	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	1	5	2.9	Cn1nnnc1-c1cc(Br)ccc1NC(=O)c1ccccc1	nan
	16020020	49847	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	5	0	5	4.2	CCOC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)cc2)c1C	nan
	CHEMBL1570342	49847	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	5	0	5	4.2	CCOC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)cc2)c1C	nan
	893344	49848	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	3.3	Cn1nnc2cc(NC(=O)Nc3cccc(Cl)c3)ccc21	nan
	CHEMBL1570344	49848	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	3.3	Cn1nnc2cc(NC(=O)Nc3cccc(Cl)c3)ccc21	nan
	7692920	49915	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	3.0	O=C(Nc1nnc(S(=O)(=O)Cc2ccc(F)cc2)s1)c1ccccc1F	nan
	CHEMBL1570825	49915	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	3.0	O=C(Nc1nnc(S(=O)(=O)Cc2ccc(F)cc2)s1)c1ccccc1F	nan
	16015598	49979	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	6.0	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccccc3)on2)cc1	nan
	CHEMBL1571539	49979	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	6.0	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccccc3)on2)cc1	nan
	16015076	50042	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	6	4.0	COC(=O)c1ccccc1NC(=O)CSc1cc(-c2ccccc2)nc(C)n1	nan
	CHEMBL1572102	50042	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	6	4.0	COC(=O)c1ccccc1NC(=O)CSc1cc(-c2ccccc2)nc(C)n1	nan
	663126	50104	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	6	5.1	Clc1ccc(OCc2nn3c(C4CCCCC4)nnc3s2)c(Cl)c1	nan
	CHEMBL1572687	50104	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	6	5.1	Clc1ccc(OCc2nn3c(C4CCCCC4)nnc3s2)c(Cl)c1	nan
	2318048	50128	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	7	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1OC	nan
	CHEMBL1572874	50128	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	7	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1OC	nan
	135492018	50150	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135635832	50150	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135914561	50150	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	CHEMBL1573000	50150	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135870946	50174	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	8	1.6	COc1ccc(C(=O)COC(=O)CCNC2=NS(=O)(=O)c3ccccc32)c(OC)c1	nan
	CHEMBL1573236	50174	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	8	1.6	COc1ccc(C(=O)COC(=O)CCNC2=NS(=O)(=O)c3ccccc32)c(OC)c1	nan
	16011872	50178	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	0	6	7.1	Cc1cccc(-c2nc(Cn3c(SCc4cccc(C(F)(F)F)c4)nc4ccncc43)c(C)o2)c1	nan
	CHEMBL1573276	50178	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	0	6	7.1	Cc1cccc(-c2nc(Cn3c(SCc4cccc(C(F)(F)F)c4)nc4ccncc43)c(C)o2)c1	nan
	16019020	50191	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1573442	50191	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	4599423	50237	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	3	1	5.2	S=C(NCc1ccc2[nH]c3c(c2c1)CCCC3)Nc1ccccc1Cl	nan
	CHEMBL1573942	50237	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	3	1	5.2	S=C(NCc1ccc2[nH]c3c(c2c1)CCCC3)Nc1ccccc1Cl	nan
	16014814	50280	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.2	Cc1cccc(NC(=O)c2c(C)cc(C)nc2SCC(=O)c2ccccc2)c1	nan
	CHEMBL1574276	50280	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.2	Cc1cccc(NC(=O)c2c(C)cc(C)nc2SCC(=O)c2ccccc2)c1	nan
	921918	50397	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	0	5	4.8	Fc1ccc(-n2c(-c3cccs3)nc3nc4ccccc4nc32)cc1	nan
	CHEMBL1575663	50397	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	0	5	4.8	Fc1ccc(-n2c(-c3cccs3)nc3nc4ccccc4nc32)cc1	nan
	1960193	50452	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	4	3.9	Cn1c(NC(=O)c2ccccc2)c(-c2ccccn2)c(=O)c2ccccc21	nan
	CHEMBL1576207	50452	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	4	3.9	Cn1c(NC(=O)c2ccccc2)c(-c2ccccn2)c(=O)c2ccccc21	nan
	5846704	50461	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	9	1	5	3.9	CCN(CC)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1576280	50461	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	9	1	5	3.9	CCN(CC)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	935443	50471	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	2	5.1	Cc1ccc(NC(S)=Nc2cc(-c3ccccc3)[nH]n2)cc1Cl	nan
	CHEMBL1576343	50471	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	2	5.1	Cc1ccc(NC(S)=Nc2cc(-c3ccccc3)[nH]n2)cc1Cl	nan
	3228917	50540	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	5	4.7	CCc1cccc(C)c1NC(=O)CSc1[nH]c(-c2ccccc2F)nc2ncnc1-2	nan
	CHEMBL1576889	50540	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	5	4.7	CCc1cccc(C)c1NC(=O)CSc1[nH]c(-c2ccccc2F)nc2ncnc1-2	nan
	709545	50575	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	2.9	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)no1	nan
	CHEMBL1577228	50575	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	2.9	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)no1	nan
	3917007	50683	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	2.9	O=C1COc2ccc(C(=O)COC(=O)CCSc3ccccc3)cc2N1	nan
	CHEMBL1578153	50683	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	2.9	O=C1COc2ccc(C(=O)COC(=O)CCSc3ccccc3)cc2N1	nan
	20884721	50870	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.7	COc1cccc2c1cc1c(=O)n(CC(=O)NCc3ccccn3)nc(C)n12	nan
	CHEMBL1579740	50870	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.7	COc1cccc2c1cc1c(=O)n(CC(=O)NCc3ccccn3)nc(C)n12	nan
	1292507	50914	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	7	4.4	Cc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3sc(C)c(C)c3c2=O)cc1	nan
	CHEMBL1580140	50914	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	7	4.4	Cc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3sc(C)c(C)c3c2=O)cc1	nan
	2347564	51134	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	9	1.6	Cc1nn(-c2ccccc2)c2sc(C(=O)c3c(N)n(C)c(=O)n(C)c3=O)cc12	nan
	CHEMBL1581991	51134	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	9	1.6	Cc1nn(-c2ccccc2)c2sc(C(=O)c3c(N)n(C)c(=O)n(C)c3=O)cc12	nan
	1454917	51164	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1cccc(C)c1)C1CC1)c1nnnn12	nan
	CHEMBL1582197	51164	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1cccc(C)c1)C1CC1)c1nnnn12	nan
	7080789	51230	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	3	4	3.3	Cc1ccc2cc(CCNC(=O)C(=O)c3c[nH]c4ccccc34)c(O)nc2c1	nan
	CHEMBL1582792	51230	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	3	4	3.3	Cc1ccc2cc(CCNC(=O)C(=O)c3c[nH]c4ccccc34)c(O)nc2c1	nan
	1420394	51248	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	4	5.2	Cc1ccc2cc(CN(C(=O)c3cccs3)c3ccccc3)c(O)nc2c1	nan
	CHEMBL1583002	51248	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	4	5.2	Cc1ccc2cc(CN(C(=O)c3cccs3)c3ccccc3)c(O)nc2c1	nan
	2012958	51295	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	4.1	Cc1nc(SCC(=O)NCc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1583344	51295	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	4.1	Cc1nc(SCC(=O)NCc2ccccc2)c2oc3ccccc3c2n1	nan
	2810452	51321	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	0	6	3.5	Cc1cc(C)c(-n2nnnc2SC2Cc3ccccc3C2=O)c(C)c1	nan
	CHEMBL1583573	51321	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	0	6	3.5	Cc1cc(C)c(-n2nnnc2SC2Cc3ccccc3C2=O)c(C)c1	nan
	4102688	51407	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	5	2.6	Cc1cccc(NC(=O)c2cnc3sccn3c2=O)c1C	nan
	CHEMBL1584232	51407	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	5	2.6	Cc1cccc(NC(=O)c2cnc3sccn3c2=O)c1C	nan
	15944711	51410	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	5	3.9	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccccc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1584268	51410	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	5	3.9	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccccc3)c(=O)c3cc(F)ccc32)cc1	nan
	2981373	51660	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	4	4.3	Cc1nc(Nc2cccc(C(F)(F)F)c2)nc2c1C(=O)CC(C)C2	nan
	CHEMBL1586327	51660	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	4	4.3	Cc1nc(Nc2cccc(C(F)(F)F)c2)nc2c1C(=O)CC(C)C2	nan
	6404569	51799	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	0	3	5.4	c1ccc(Cc2nnc(Sc3ccccc3)c3ccccc23)cc1	nan
	CHEMBL1587518	51799	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	0	3	5.4	c1ccc(Cc2nnc(Sc3ccccc3)c3ccccc23)cc1	nan
	16189382	51951	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1cccc(N(C)C(=O)c2cc3c(O)nc4ccc(C)cc4c3s2)c1	nan
	CHEMBL1588813	51951	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1cccc(N(C)C(=O)c2cc3c(O)nc4ccc(C)cc4c3s2)c1	nan
	5770860	51993	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	2	6	2.4	CCOC(=O)CNC(=O)c1sc(NC(=O)/C=C/c2ccccc2)nc1C	nan
	CHEMBL1589172	51993	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	2	6	2.4	CCOC(=O)CNC(=O)c1sc(NC(=O)/C=C/c2ccccc2)nc1C	nan
	2428876	51996	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	4	2.7	O=C(COc1ccc2ccccc2c1)Nc1cccc2c1C(=O)NC2=O	nan
	CHEMBL1589183	51996	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	4	2.7	O=C(COc1ccc2ccccc2c1)Nc1cccc2c1C(=O)NC2=O	nan
	16007870	52079	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	8	1	4	4.9	Cc1ccc(CCNC(=O)CSCc2nc(-c3ccc(C)cc3)oc2C)cc1	nan
	CHEMBL1589908	52079	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	8	1	4	4.9	Cc1ccc(CCNC(=O)CSCc2nc(-c3ccc(C)cc3)oc2C)cc1	nan
	6418319	52096	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	5.7	O=C(CSc1nnc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)n1)NC1CCCC1	nan
	CHEMBL1590097	52096	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	5.7	O=C(CSc1nnc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)n1)NC1CCCC1	nan
	16025990	52107	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	2.2	Cc1c(Cl)cccc1NC(=O)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1590252	52107	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	2.2	Cc1c(Cl)cccc1NC(=O)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	16030611	52124	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCc3ccccc32)c1	nan
	CHEMBL1590504	52124	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCc3ccccc32)c1	nan
	16009482	52125	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	7	3.9	COc1ccccc1C(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1590536	52125	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	7	3.9	COc1ccccc1C(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	16015095	52126	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	6	5.5	CCOc1ccccc1NC(=O)c1sc(-n2nc(C)c(CCC(C)C)c2C)nc1C	nan
	CHEMBL1590548	52126	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	6	5.5	CCOc1ccccc1NC(=O)c1sc(-n2nc(C)c(CCC(C)C)c2C)nc1C	nan
	16019575	52134	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	5	1	9	4.6	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1590659	52134	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	5	1	9	4.6	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	4249793	52141	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	2	4	1.8	COc1ccccc1C(=O)Nc1ccc2c(c1)C(=O)NC2=O	nan
	CHEMBL1590747	52141	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	2	4	1.8	COc1ccccc1C(=O)Nc1ccc2c(c1)C(=O)NC2=O	nan
	16016850	52149	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	2	3	5.9	COc1ccc2c(Sc3ccccc3)c(C(=O)NCC(C)c3ccccc3)[nH]c2c1	nan
	CHEMBL1590842	52149	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	2	3	5.9	COc1ccc2c(Sc3ccccc3)c(C(=O)NCC(C)c3ccccc3)[nH]c2c1	nan
	16025801	52183	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	1	7	2.9	COc1cccc(CNc2nccn(-c3ccc(OC)c(OC)c3)c2=O)c1	nan
	CHEMBL1591265	52183	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	1	7	2.9	COc1cccc(CNc2nccn(-c3ccc(OC)c(OC)c3)c2=O)c1	nan
	7533419	52222	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	8	1	6	3.5	CCOc1ccc(-c2nnc(SCC(=O)NCc3ccccc3)o2)cc1	nan
	CHEMBL1591699	52222	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	8	1	6	3.5	CCOc1ccc(-c2nnc(SCC(=O)NCc3ccccc3)o2)cc1	nan
	16030248	52243	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	5	3.7	O=C(CSc1nnc(-c2ccccc2Cl)[nH]1)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1591982	52243	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	5	3.7	O=C(CSc1nnc(-c2ccccc2Cl)[nH]1)N1CCN(c2ccc(F)cc2)CC1	nan
	16021788	52253	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	3.3	O=C(NCc1ccccc1)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1592133	52253	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	3.3	O=C(NCc1ccccc1)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	16008534	52292	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.2	CCOC(=O)C(Cc1ccccc1)NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)c(C)c2)c1C	nan
	CHEMBL1592680	52292	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.2	CCOC(=O)C(Cc1ccccc1)NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)c(C)c2)c1C	nan
	16012042	52294	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	5	4.6	O=C(Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O)NCCc1ccc(Cl)cc1	nan
	CHEMBL1592702	52294	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	5	4.6	O=C(Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O)NCCc1ccc(Cl)cc1	nan
	15991036	52307	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	6.7	COc1ccc(Cl)cc1C(=O)Nc1ccc2oc(-c3ccc(C(C)(C)C)cc3)nc2c1	nan
	CHEMBL1592855	52307	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	6.7	COc1ccc(Cl)cc1C(=O)Nc1ccc2oc(-c3ccc(C(C)(C)C)cc3)nc2c1	nan
	16026106	52322	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	5	3.9	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccco2)CC1	nan
	CHEMBL1593080	52322	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	5	3.9	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccco2)CC1	nan
	16009361	52325	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	1	6	4.3	CCOc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1593099	52325	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	1	6	4.3	CCOc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16030919	52330	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.7	CCc1ccc(NC(=O)CSc2ccc3nc(-c4ccc(OC)cc4)cn3n2)cc1	nan
	CHEMBL1593184	52330	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.7	CCc1ccc(NC(=O)CSc2ccc3nc(-c4ccc(OC)cc4)cn3n2)cc1	nan
	16033356	52335	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.5	COc1ccc(CC(=O)Nc2ccc(-c3nc4ccccc4s3)c(C)c2)cc1	nan
	CHEMBL1593249	52335	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.5	COc1ccc(CC(=O)Nc2ccc(-c3nc4ccccc4s3)c(C)c2)cc1	nan
	16015767	52364	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	0	5	3.9	Cc1ccc(CN(C(=O)COc2ccccc2[N+](=O)[O-])c2ccccn2)cc1	nan
	CHEMBL1593732	52364	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	0	5	3.9	Cc1ccc(CN(C(=O)COc2ccccc2[N+](=O)[O-])c2ccccn2)cc1	nan
	15990880	52369	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	3	5.6	Cc1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)c(C)c1	nan
	CHEMBL1593807	52369	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	3	5.6	Cc1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)c(C)c1	nan
	3623411	52381	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.0	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(C)cc3)c3ccccc3n2)cc1	nan
	CHEMBL1593971	52381	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.0	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(C)cc3)c3ccccc3n2)cc1	nan
	16030473	52452	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n2c1	nan
	CHEMBL1594609	52452	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n2c1	nan
	2328630	52466	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	6	1	6	2.9	CCOC(=O)c1c(C)[nH]c(C(=O)CSc2nccc(C)n2)c1C	nan
	CHEMBL1594696	52466	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	6	1	6	2.9	CCOC(=O)c1c(C)[nH]c(C(=O)CSc2nccc(C)n2)c1C	nan
	16027342	52520	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.1	Cc1cc(=O)n(Cc2cccc(F)c2)c2c1c(C)nn2-c1cccc(F)c1	nan
	CHEMBL1595156	52520	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.1	Cc1cc(=O)n(Cc2cccc(F)c2)c2c1c(C)nn2-c1cccc(F)c1	nan
	16021494	52527	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	4	3.9	CSc1ncc(C(=O)NCc2ccc(F)cc2)c(-c2ccccc2)n1	nan
	CHEMBL1595189	52527	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	4	3.9	CSc1ncc(C(=O)NCc2ccc(F)cc2)c(-c2ccccc2)n1	nan
	4584398	52629	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	1	2	4.7	Cn1c(C(=O)Nc2ccc(Cl)cc2)cc2cc(Cl)ccc21	nan
	CHEMBL1596148	52629	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	1	2	4.7	Cn1c(C(=O)Nc2ccc(Cl)cc2)cc2cc(Cl)ccc21	nan
	16016964	52661	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	4	4.7	Cc1cc(C)c2c(-n3cccc3)c(C(=O)NCCc3ccccc3)sc2n1	nan
	CHEMBL1596415	52661	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	4	4.7	Cc1cc(C)c2c(-n3cccc3)c(C(=O)NCCc3ccccc3)sc2n1	nan
	891582	52686	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	0	5	3.8	Cc1cccc(-n2ncc3c(N4CCc5ccccc54)ncnc32)c1	nan
	CHEMBL1596656	52686	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	0	5	3.8	Cc1cccc(-n2ncc3c(N4CCc5ccccc54)ncnc32)c1	nan
	2138637	52689	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	2	6	3.5	CC(=O)NCCNc1nc2c(-c3cccc(C(F)(F)F)c3)nnn2c2ccccc12	nan
	CHEMBL1596664	52689	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	2	6	3.5	CC(=O)NCCNc1nc2c(-c3cccc(C(F)(F)F)c3)nnn2c2ccccc12	nan
	4062063	52755	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	3	8	-0.4	CN(CCO)S(=O)(=O)c1ccc2c(c1)C(=NN)c1cc(S(=O)(=O)N(C)CCO)ccc1-2	nan
	CHEMBL1597275	52755	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	3	8	-0.4	CN(CCO)S(=O)(=O)c1ccc2c(c1)C(=NN)c1cc(S(=O)(=O)N(C)CCO)ccc1-2	nan
	1611638	52848	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	2	10	3.2	CCOC(=O)Cc1csc(NC(=O)CSc2nc(N)c3c(C)c(C)sc3n2)n1	nan
	CHEMBL1598169	52848	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	2	10	3.2	CCOC(=O)Cc1csc(NC(=O)CSc2nc(N)c3c(C)c(C)sc3n2)n1	nan
	16010773	52851	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.2	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cc(C)cc3C)c2=O)cc1	nan
	CHEMBL1598197	52851	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.2	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cc(C)cc3C)c2=O)cc1	nan
	2958808	52853	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	2	4	3.7	Cc1nc(NC(=S)NC(=O)COc2ccccc2Cl)ccc1Br	nan
	CHEMBL1598226	52853	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	2	4	3.7	Cc1nc(NC(=S)NC(=O)COc2ccccc2Cl)ccc1Br	nan
	921716	52910	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	4.9	Cc1ccc(O)c(C2=Nc3ccccc3N=C(c3ccco3)C2)c1	nan
	CHEMBL1598745	52910	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	4.9	Cc1ccc(O)c(C2=Nc3ccccc3N=C(c3ccco3)C2)c1	nan
	3284133	52918	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	10	2	6	4.2	CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(C(=O)Nc2sc3c(c2C(N)=O)CCN(C(C)C)C3)cc1	nan
	CHEMBL1598836	52918	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	10	2	6	4.2	CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(C(=O)Nc2sc3c(c2C(N)=O)CCN(C(C)C)C3)cc1	nan
	7326265	52969	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	2	5	3.5	CC(=O)Nc1ccc(C(=O)Nc2nnc(CCc3ccccc3)s2)cc1	nan
	CHEMBL1599247	52969	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	2	5	3.5	CC(=O)Nc1ccc(C(=O)Nc2nnc(CCc3ccccc3)s2)cc1	nan
	16009345	52984	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	0	6	4.0	COc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	CHEMBL1599358	52984	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	0	6	4.0	COc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	16024944	53023	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	4.8	Cc1cccc(N2CCN(c3ccc(C(=O)O)cc3NC(=O)c3ccccc3F)CC2C)c1	nan
	CHEMBL1599731	53023	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	4.8	Cc1cccc(N2CCN(c3ccc(C(=O)O)cc3NC(=O)c3ccccc3F)CC2C)c1	nan
	6536107	53068	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	5.2	Cc1ccc(-c2csc(/C=C3\SC(C)C(=O)N3CC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1600183	53068	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	5.2	Cc1ccc(-c2csc(/C=C3\SC(C)C(=O)N3CC(=O)Nc3ccccc3F)n2)cc1	nan
	733979	53078	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	1	4	2.5	CC(=O)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1	nan
	CHEMBL1600285	53078	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	1	4	2.5	CC(=O)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1	nan
	2999237	53083	4	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	2.8	CCCCn1c(-c2ccsc2)nc2c1c(=O)[nH]c(=O)n2CCC	nan
	CHEMBL1600302	53083	4	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	2.8	CCCCn1c(-c2ccsc2)nc2c1c(=O)[nH]c(=O)n2CCC	nan
	3946061	53125	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	3.2	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NCc5ccccc5)cnc4c3cc2CO1	nan
	CHEMBL1600688	53125	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	3.2	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NCc5ccccc5)cnc4c3cc2CO1	nan
	16019821	53128	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1600701	53128	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	648853	53136	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	1	4	3.2	Cc1ccc(C(=O)Nc2nc3ccccc3c(=O)s2)cc1	nan
	CHEMBL1600749	53136	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	1	4	3.2	Cc1ccc(C(=O)Nc2nc3ccccc3c(=O)s2)cc1	nan
	1326969	53196	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	4	5.1	Cc1ccc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)c(C)c1	nan
	CHEMBL1601297	53196	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	4	5.1	Cc1ccc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)c(C)c1	nan
	20949434	53199	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	2	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CC(=O)N4)CC2)cc1	nan
	CHEMBL1601336	53199	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	2	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CC(=O)N4)CC2)cc1	nan
	16015783	53210	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	6	1	6	6.2	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(Cl)cc4)oc4ccccc34)no2)cc1	nan
	CHEMBL1601476	53210	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	6	1	6	6.2	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(Cl)cc4)oc4ccccc34)no2)cc1	nan
	3579351	53249	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	0	7	4.2	COc1ccc(-n2c(SCC(=O)C(C)(C)C)nc3ccsc3c2=O)cc1	nan
	CHEMBL1601921	53249	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	0	7	4.2	COc1ccc(-n2c(SCC(=O)C(C)(C)C)nc3ccsc3c2=O)cc1	nan
	16034721	53315	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	7	4.3	Cc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4)cc3nc2s1	nan
	CHEMBL1602585	53315	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	7	4.3	Cc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4)cc3nc2s1	nan
	3938730	53355	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	2	4	6.4	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)NCc3ccc(Cl)cc3)sc2n1	nan
	CHEMBL1602945	53355	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	2	4	6.4	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)NCc3ccc(Cl)cc3)sc2n1	nan
	3343394	53435	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	2	1	6	5.1	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccc(Br)cc2)CO1	nan
	CHEMBL1603651	53435	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	2	1	6	5.1	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccc(Br)cc2)CO1	nan
	5223767	53436	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	4	3.3	Cc1cc2cc(CNC(=O)Cc3ccc([N+](=O)[O-])cc3)ccc2n1C	nan
	CHEMBL1603656	53436	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	4	3.3	Cc1cc2cc(CNC(=O)Cc3ccc([N+](=O)[O-])cc3)ccc2n1C	nan
	16030948	53453	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.1	O=C(CSc1ccc2nc(-c3ccccc3)cn2n1)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1603757	53453	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.1	O=C(CSc1ccc2nc(-c3ccccc3)cn2n1)Nc1ccccc1C(F)(F)F	nan
	2791873	53485	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.0	CCOC(=O)c1cnc2ccc(Br)cc2c1NCC(C)O	nan
	CHEMBL1603951	53485	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.0	CCOC(=O)c1cnc2ccc(Br)cc2c1NCC(C)O	nan
	16014801	53597	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	4.1	Cc1cccc(CSc2nc(=O)c3c(n2C)NC(=O)CC3c2cc(F)cc(F)c2)c1	nan
	CHEMBL1605009	53597	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	4.1	Cc1cccc(CSc2nc(=O)c3c(n2C)NC(=O)CC3c2cc(F)cc(F)c2)c1	nan
	135435545	53612	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	2	4	2.3	NC1=C(c2nc3ccccc3[nH]2)C(=O)CN1c1ccccc1	nan
	CHEMBL1605162	53612	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	2	4	2.3	NC1=C(c2nc3ccccc3[nH]2)C(=O)CN1c1ccccc1	nan
	1511904	53627	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	4	3.8	O=C(O)c1cn(-c2ccc(N3CCCC3)c(F)c2)c2c(F)c(F)c(F)cc2c1=O	nan
	CHEMBL1605292	53627	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	4	3.8	O=C(O)c1cn(-c2ccc(N3CCCC3)c(F)c2)c2c(F)c(F)c(F)cc2c1=O	nan
	1961588	53704	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	3	0	6	4.9	Cn1c2ccccc2c(=O)c2c(=O)n(Cc3ccco3)c(-c3ccc(Cl)cc3Cl)nc21	nan
	CHEMBL1605870	53704	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	3	0	6	4.9	Cn1c2ccccc2c(=O)c2c(=O)n(Cc3ccco3)c(-c3ccc(Cl)cc3Cl)nc21	nan
	16001902	53719	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	3.3	Cc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3cccc4nsnc34)C2)cc1C	nan
	CHEMBL1605982	53719	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	3.3	Cc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3cccc4nsnc34)C2)cc1C	nan
	16031132	53807	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	5	4.5	CN(C)c1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	CHEMBL1606681	53807	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	5	4.5	CN(C)c1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	2931173	53813	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	2	3	4.9	CCCCn1c(N=C(S)Nc2ccccc2)nc2ccccc21	nan
	CHEMBL1606716	53813	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	2	3	4.9	CCCCn1c(N=C(S)Nc2ccccc2)nc2ccccc21	nan
	1481761	53929	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	4.1	COc1ccc(-c2c(C)nc3c(-c4ccc(F)cc4)cnn3c2N)cc1	nan
	CHEMBL1607515	53929	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	4.1	COc1ccc(-c2c(C)nc3c(-c4ccc(F)cc4)cnn3c2N)cc1	nan
	16030158	53965	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	7	3.2	Cc1nn(CC(=O)NCc2ccc(N(C)C)cc2)c(=O)c2c(C)n(-c3ccc(Cl)cc3)nc12	nan
	CHEMBL1607845	53965	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	7	3.2	Cc1nn(CC(=O)NCc2ccc(N(C)C)cc2)c(=O)c2c(C)n(-c3ccc(Cl)cc3)nc12	nan
	786570	53979	36	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	1	1	3	3.8	O=c1c2cc(Br)ccc2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1608028	53979	36	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	1	1	3	3.8	O=c1c2cc(Br)ccc2[nH]c(=S)n1-c1ccccc1	nan
	744022	54076	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	4	1	4	3.8	COCc1cc(C)nc(Nc2ccc(C)c(C)c2)c1C#N	nan
	CHEMBL1608862	54076	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	4	1	4	3.8	COCc1cc(C)nc(Nc2ccc(C)c(C)c2)c1C#N	nan
	20868577	54093	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(C)nc5ccccc5c4o3)CC2)cc1	nan
	CHEMBL1609003	54093	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(C)nc5ccccc5c4o3)CC2)cc1	nan
	16015522	54099	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	3.5	COc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCOCC4)sc3c2)cc1	nan
	CHEMBL1609032	54099	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	3.5	COc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCOCC4)sc3c2)cc1	nan
	3128209	54187	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	8	1.5	NS(=O)(=O)c1ccc(Nc2ccc([N+](=O)[O-])c3nonc23)cc1	nan
	CHEMBL1609744	54187	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	8	1.5	NS(=O)(=O)c1ccc(Nc2ccc([N+](=O)[O-])c3nonc23)cc1	nan
	16026888	54257	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	0	8	3.6	COc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1610338	54257	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	0	8	3.6	COc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16015736	54281	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	4	3.3	Cc1ccc(C(C)C)c(OCC(=O)N2CCN(CCc3ccncc3)CC2)c1	nan
	CHEMBL1610516	54281	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	4	3.3	Cc1ccc(C(C)C)c(OCC(=O)N2CCN(CCc3ccncc3)CC2)c1	nan
	2220915	54355	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	5	4.9	COc1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)cc1OC	nan
	CHEMBL1611237	54355	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	5	4.9	COc1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)cc1OC	nan
	16030297	54383	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	5	4.9	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCc2ccccc21	nan
	CHEMBL1611407	54383	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	5	4.9	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCc2ccccc21	nan
	903550	54427	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	4	1	5	2.5	CCOC(=O)c1sc(NC(=O)CC)c(C#N)c1C	nan
	CHEMBL1611829	54427	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	4	1	5	2.5	CCOC(=O)c1sc(NC(=O)CC)c(C#N)c1C	nan
	2804057	54455	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	206	0	2	2	3.1	Cc1c(C)c(C)c2[nH]c(S)nc2c1C	nan
	CHEMBL1612138	54455	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	206	0	2	2	3.1	Cc1c(C)c(C)c2[nH]c(S)nc2c1C	nan
	16019436	54522	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(C)c(CSc2ccc3nnc(CCNS(=O)(=O)c4ccccc4)n3n2)c1	nan
	CHEMBL1612674	54522	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(C)c(CSc2ccc3nnc(CCNS(=O)(=O)c4ccccc4)n3n2)c1	nan
	4152434	54536	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	5	5.7	CC(C)c1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1612783	54536	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	5	5.7	CC(C)c1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	16034221	54572	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	1.1	CCOC(=O)N1CCN(S(=O)(=O)N2CCCC(C(=O)NCc3cc(OC)ccc3OC)C2)CC1	nan
	CHEMBL1613162	54572	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	1.1	CCOC(=O)N1CCN(S(=O)(=O)N2CCCC(C(=O)NCc3cc(OC)ccc3OC)C2)CC1	nan
	3238969	54576	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	1	4	5.6	O=C(Nc1ccc2oc(-c3ccccc3Cl)nc2c1)c1cncc(Br)c1	nan
	CHEMBL1613230	54576	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	1	4	5.6	O=C(Nc1ccc2oc(-c3ccccc3Cl)nc2c1)c1cncc(Br)c1	nan
	16033448	54587	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	Cc1cc(C)c(NC(=O)c2nc3ccccc3nc2N2CCCCC2)c(C)c1	nan
	CHEMBL1613324	54587	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	Cc1cc(C)c(NC(=O)c2nc3ccccc3nc2N2CCCCC2)c(C)c1	nan
	2138172	54592	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	3.1	C=CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	CHEMBL1613374	54592	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	3.1	C=CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	17585635	54871	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	73401607	54871	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1311226	54871	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1617414	54871	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	424003	55007	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	CHEMBL1359356	55007	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	CHEMBL1618556	55007	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	719481	55017	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	CHEMBL1379055	55017	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	CHEMBL1618658	55017	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	1453026	55364	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	CHEMBL1442637	55364	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	CHEMBL1621750	55364	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	5044272	55612	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1524152	55612	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1623691	55612	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	3149296	55644	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	5768586	55644	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	CHEMBL1508982	55644	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	CHEMBL1623968	55644	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	1956404	55669	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	CHEMBL1556245	55669	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	CHEMBL1624228	55669	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	3602384	55803	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	CHEMBL1602214	55803	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	CHEMBL1625426	55803	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	2151347	71622	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	0	4	3.3	C#CCn1/c(=N/C(=O)c2ccco2)sc2cccc(Cl)c21	nan
	CHEMBL1973713	71622	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	0	4	3.3	C#CCn1/c(=N/C(=O)c2ccco2)sc2cccc(Cl)c21	nan
	741794	71928	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	4	3.1	Cc1c(C(C)(C)C)s/c(=N/C(=O)c2ccccc2O)n1C	nan
	CHEMBL1983034	71928	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	4	3.1	Cc1c(C(C)(C)C)s/c(=N/C(=O)c2ccccc2O)n1C	nan
	9583974	72189	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	2	7	5.1	COc1cccc(/C=N/NC(=O)c2oc3nc(-c4ccccc4)cc(-c4ccco4)c3c2N)c1	nan
	CHEMBL1991618	72189	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	2	7	5.1	COc1cccc(/C=N/NC(=O)c2oc3nc(-c4ccccc4)cc(-c4ccco4)c3c2N)c1	nan
	135498048	72272	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	3	2	6	0.8	Cc1nonc1C(=O)N/N=C/c1ccc(O)cc1	nan
	CHEMBL1994596	72272	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	3	2	6	0.8	Cc1nonc1C(=O)N/N=C/c1ccc(O)cc1	nan
	1362920	95313	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(OCC(=O)Nc2ccc(-c3nc4cc(C)cc(C)c4o3)cc2)cc1	nan
	CHEMBL258549	95313	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(OCC(=O)Nc2ccc(-c3nc4cc(C)cc(C)c4o3)cc2)cc1	nan
	2150885	107118	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	5	3.3	COc1ccc(OC)c2c1s/c(=N\C(=O)C1CCCCC1)n2C	nan
	CHEMBL3189890	107118	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	5	3.3	COc1ccc(OC)c2c1s/c(=N\C(=O)C1CCCCC1)n2C	nan
	3604296	107280	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	2.1	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	CHEMBL3191753	107280	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	2.1	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	1389664	107476	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	0	8	3.2	COc1cc(/C=c2\sc3nc(=O)c(-c4ccccc4)nn3c2=O)ccc1OCCC(C)C	nan
	CHEMBL3193918	107476	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	0	8	3.2	COc1cc(/C=c2\sc3nc(=O)c(-c4ccccc4)nn3c2=O)ccc1OCCC(C)C	nan
	2321009	107550	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	0	4	3.4	Cc1ccc2c(c1)s/c(=N/C(=O)c1cccs1)n2C	nan
	CHEMBL3194826	107550	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	0	4	3.4	Cc1ccc2c(c1)s/c(=N/C(=O)c1cccs1)n2C	nan
	3245289	107555	11	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	0	8	2.0	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(OC)ccc21	nan
	CHEMBL3194890	107555	11	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	0	8	2.0	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(OC)ccc21	nan
	4668650	107827	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	1.5	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(N)(=O)=O)ccc21	nan
	CHEMBL3197833	107827	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	1.5	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(N)(=O)=O)ccc21	nan
	2150918	107882	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	6	3.0	COc1ccc(C)c2s/c(=N\C(=O)c3cccc(N4C(=O)CCC4=O)c3)n(C)c12	nan
	CHEMBL3198311	107882	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	6	3.0	COc1ccc(C)c2s/c(=N\C(=O)c3cccc(N4C(=O)CCC4=O)c3)n(C)c12	nan
	135460447	107895	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	3	3	6	1.9	Nc1c(Cl)ncnc1N/N=C/c1ccc(O)cc1	nan
	CHEMBL3198494	107895	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	3	3	6	1.9	Nc1c(Cl)ncnc1N/N=C/c1ccc(O)cc1	nan
	6184027	108173	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	12	1	9	0.8	COCCCn1c(=O)/c(=C\c2ccc(OC(F)F)c(OC)c2)s/c1=C(/C#N)C(=O)NCCOC	nan
	CHEMBL3207685	108173	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	12	1	9	0.8	COCCCn1c(=O)/c(=C\c2ccc(OC(F)F)c(OC)c2)s/c1=C(/C#N)C(=O)NCCOC	nan
	2150849	108205	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	7	3.3	COc1cc(C(=O)/N=c2\sc3c(C)ccc(OC)c3n2C)cc(OC)c1OC	nan
	CHEMBL3208227	108205	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	7	3.3	COc1cc(C(=O)/N=c2\sc3c(C)ccc(OC)c3n2C)cc(OC)c1OC	nan
	5122885	108334	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccccc2Br)n(C)c1C	nan
	CHEMBL3209816	108334	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccccc2Br)n(C)c1C	nan
	9631393	108427	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	3.2	O=C(N/N=C/c1ccc2nccnc2c1)c1ccc(Br)cc1	nan
	CHEMBL3211205	108427	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	3.2	O=C(N/N=C/c1ccc2nccnc2c1)c1ccc(Br)cc1	nan
	4128025	108441	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	0	6	2.4	COc1cccc(C(=O)/N=c2\sc3cc(S(C)(=O)=O)ccc3n2C)c1	nan
	CHEMBL3211378	108441	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	0	6	2.4	COc1cccc(C(=O)/N=c2\sc3cc(S(C)(=O)=O)ccc3n2C)c1	nan
	7161820	108461	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	5	2.7	CCOC(=O)Cn1/c(=N/C(=O)CC)sc2c(C)cc(C)cc21	nan
	CHEMBL3211674	108461	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	5	2.7	CCOC(=O)Cn1/c(=N/C(=O)CC)sc2c(C)cc(C)cc21	nan
	2150987	108671	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	0	5	2.5	CCCC(=O)/N=c1\sc2c(OC)ccc(OC)c2n1C	nan
	CHEMBL3214516	108671	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	0	5	2.5	CCCC(=O)/N=c1\sc2c(OC)ccc(OC)c2n1C	nan
	3213263	112101	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	CHEMBL3197118	112101	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	CHEMBL3302243	112101	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	6540428	184271	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	CHEMBL3989558	184271	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	CHEMBL485253	184271	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	846186	192759	24	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	3	3	3.0	Cc1nc2ccc(-c3nc4cc(N)ccc4[nH]3)cc2[nH]1	nan
	CHEMBL525103	192759	24	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	3	3	3.0	Cc1nc2ccc(-c3nc4cc(N)ccc4[nH]3)cc2[nH]1	nan
	2850154	196209	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	2	1	2.1	CC1=CC(c2ccccc2)NC(=S)N1	nan
	CHEMBL572806	196209	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	2	1	2.1	CC1=CC(c2ccccc2)NC(=S)N1	nan
	138884	198309	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	4	4.2	COc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(OC)c3)c2)c1	nan
	CHEMBL595273	198309	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	4	4.2	COc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(OC)c3)c2)c1	nan
	16020583	200682	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	0	5	4.2	Cn1cc(S(=O)(=O)c2cccc(Cl)c2)c(=O)c2cc(F)c(N3CCCCC3)cc21	nan
	CHEMBL610622	200682	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	0	5	4.2	Cn1cc(S(=O)(=O)c2cccc(Cl)c2)c(=O)c2cc(F)c(N3CCCCC3)cc21	nan
	1361408	21182	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	6.1	O=C(Nc1ccc(-c2nc3cc(Cl)ccc3o2)cc1)c1cc2ccccc2o1	nan
	CHEMBL1314585	21182	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	6.1	O=C(Nc1ccc(-c2nc3cc(Cl)ccc3o2)cc1)c1cc2ccccc2o1	nan
	1369231	21307	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	2	5	5.5	O=C(COc1ccc(Cl)cc1)Nc1ccc(-c2nc3cc(Cl)ccc3o2)c(O)c1	nan
	CHEMBL1316173	21307	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	2	5	5.5	O=C(COc1ccc(Cl)cc1)Nc1ccc(-c2nc3cc(Cl)ccc3o2)c(O)c1	nan
	16033420	21702	3	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1ccc(NC(=O)c2nc3ccccc3n(C)c2=O)cc1	nan
	CHEMBL1320318	21702	3	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1ccc(NC(=O)c2nc3ccccc3n(C)c2=O)cc1	nan
	16019599	22193	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	8	4.5	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)c(C)c1	nan
	CHEMBL1324615	22193	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	8	4.5	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)c(C)c1	nan
	16033879	22262	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	8	3.2	CCOC(=O)c1ccc(Nc2nn3c(=O)c4ccccc4nc3s2)cc1	nan
	CHEMBL1325210	22262	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	8	3.2	CCOC(=O)c1ccc(Nc2nn3c(=O)c4ccccc4nc3s2)cc1	nan
	1115824	22987	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	CHEMBL1331382	22987	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	460749	23331	9	None	-11	6	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	7	0.7	Cn1nc(-c2ccc(Cl)cc2)nc2c(=O)n(C)c(=O)nc1-2	nan
	CHEMBL1334062	23331	9	None	-11	6	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	7	0.7	Cn1nc(-c2ccc(Cl)cc2)nc2c(=O)n(C)c(=O)nc1-2	nan
	16746586	24314	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	3	8	0.2	CCCN=C1C(=O)C2=C(C(O)=C1C)N1CC3NC3[C@@]1(OC)C2COC(N)=O	nan
	CHEMBL1342436	24314	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	3	8	0.2	CCCN=C1C(=O)C2=C(C(O)=C1C)N1CC3NC3[C@@]1(OC)C2COC(N)=O	nan
	2128809	26823	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	5	1	6	3.2	Cc1cc(C)c(C(=O)CSc2nnc(O)n2C2CC2)cc1C	nan
	CHEMBL1365084	26823	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	5	1	6	3.2	Cc1cc(C)c(C(=O)CSc2nnc(O)n2C2CC2)cc1C	nan
	15988395	26951	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	2	3	3.4	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Cl)cc3)c(=O)[nH]c2C1	nan
	CHEMBL1366158	26951	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	2	3	3.4	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Cl)cc3)c(=O)[nH]c2C1	nan
	2168191	27855	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.8	Cc1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	CHEMBL1372901	27855	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.8	Cc1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	4578108	28867	8	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	5	2.4	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc2ncsc2c1	nan
	CHEMBL1381180	28867	8	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	5	2.4	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc2ncsc2c1	nan
	15988012	29774	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1388847	29774	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	16024702	32069	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	9	1	7	4.3	COCCn1c(SCC(=O)c2ccc(C)cc2C)nc2cc(C(=O)NC3CCCC3)ccc2c1=O	nan
	CHEMBL1410231	32069	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	9	1	7	4.3	COCCn1c(SCC(=O)c2ccc(C)cc2C)nc2cc(C(=O)NC3CCCC3)ccc2c1=O	nan
	16025307	32960	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccccc1CNC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	CHEMBL1417794	32960	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccccc1CNC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	4658659	35136	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	5	4.9	CCOC(=O)CSc1nc(-c2ccc(Cl)cc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1437587	35136	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	5	4.9	CCOC(=O)CSc1nc(-c2ccc(Cl)cc2)cc(C(F)(F)F)c1C#N	nan
	16018194	40364	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	4	4.1	O=C(CCCn1c(=O)c2cccn2c2ccccc21)NCc1ccccc1Br	nan
	CHEMBL1483956	40364	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	4	4.1	O=C(CCCn1c(=O)c2cccn2c2ccccc21)NCc1ccccc1Br	nan
	1046621	40438	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	3	1	6	5.4	Cc1c(Cl)cccc1NC(=O)c1cc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2n1	nan
	CHEMBL1484483	40438	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	3	1	6	5.4	Cc1c(Cl)cccc1NC(=O)c1cc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2n1	nan
	16025305	43856	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1515325	43856	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	2119988	44339	14	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	6	4.7	CCOC(=O)c1sc2nc(Cc3ccc(Cl)cc3)nc(S)c2c1C	nan
	CHEMBL1520325	44339	14	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	6	4.7	CCOC(=O)c1sc2nc(Cc3ccc(Cl)cc3)nc(S)c2c1C	nan
	3368526	46919	16	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	6	3.9	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Br)cc2)o1	nan
	CHEMBL1543365	46919	16	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	6	3.9	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Br)cc2)o1	nan
	16020714	52080	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	6	3.8	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1ccc(OC)cc1)cn2CC	nan
	CHEMBL1589919	52080	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	6	3.8	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1ccc(OC)cc1)cn2CC	nan
	1164393	52098	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	6	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	CHEMBL1590134	52098	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	6	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	2254266	107575	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	0	6	4.7	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\Cc1ccccc1	nan
	CHEMBL3195210	107575	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	0	6	4.7	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\Cc1ccccc1	nan
	7424526	40147	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	7	0.0	COCCNC(=O)C(=O)Nc1c2c(nn1-c1ccccc1)CS(=O)(=O)C2	nan
	CHEMBL1482031	40147	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	7	0.0	COCCNC(=O)C(=O)Nc1c2c(nn1-c1ccccc1)CS(=O)(=O)C2	nan
	4890321	19493	8	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	2	6	3.7	Cc1ccc(NC2=NC(c3ccc(F)cc3)n3c(nc(C)cc3=O)N2)c(C)c1	nan
	CHEMBL1300954	19493	8	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	2	6	3.7	Cc1ccc(NC2=NC(c3ccc(F)cc3)n3c(nc(C)cc3=O)N2)c(C)c1	nan
	7119211	21257	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.6	COc1ccc(-c2nc(CCNC(=O)c3c(F)cccc3Cl)cs2)cc1	nan
	CHEMBL1315624	21257	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.6	COc1ccc(-c2nc(CCNC(=O)c3c(F)cccc3Cl)cs2)cc1	nan
	16028928	21384	4	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	2	6	3.0	COC(=O)c1ccc(NC(=O)C(=O)NCCc2csc(-c3ccc(F)cc3)n2)cc1	nan
	CHEMBL1317331	21384	4	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	2	6	3.0	COC(=O)c1ccc(NC(=O)C(=O)NCCc2csc(-c3ccc(F)cc3)n2)cc1	nan
	16009640	21962	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	4.5	CCOc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1322592	21962	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	4.5	CCOc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	15988993	22196	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	4	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	CHEMBL1324637	22196	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	4	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	682221	25164	17	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	4	3	8	0.2	CC(C)OC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1349621	25164	17	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	4	3	8	0.2	CC(C)OC(=O)CNc1nnc(S)nc1O	nan
	16009655	25860	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	4.4	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1355671	25860	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	4.4	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	16019300	26996	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	6	1	10	4.6	COc1cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)cc(OC)c1	nan
	CHEMBL1366490	26996	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	6	1	10	4.6	COc1cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)cc(OC)c1	nan
	16024750	29011	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1382499	29011	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	5302633	30729	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	6	2	5	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	CHEMBL1398493	30729	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	6	2	5	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	16009653	35385	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	4	5.2	Cc1ccccc1OCC(=O)Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12	nan
	CHEMBL1439712	35385	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	4	5.2	Cc1ccccc1OCC(=O)Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12	nan
	3522635	38767	7	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	CHEMBL1468421	38767	7	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	16018176	39755	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.2	COc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	CHEMBL1478735	39755	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.2	COc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	3432810	39912	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	4	5.7	O=C(Nc1ccc(-c2nc3ccccc3s2)c(O)c1)c1ccc(Br)cc1	nan
	CHEMBL1479998	39912	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	4	5.7	O=C(Nc1ccc(-c2nc3ccccc3s2)c(O)c1)c1ccc(Br)cc1	nan
	1234246	41091	10	None	-1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	1	1	5	3.0	Cc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	CHEMBL1489869	41091	10	None	-1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	1	1	5	3.0	Cc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	6800739	44287	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	4.6	CCc1ccc2n(-c3ccc(OC)cc3)c([S-])c(C(=O)Nc3cc(C)cc(C)c3)[n+]2c1	nan
	CHEMBL1519802	44287	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	4.6	CCc1ccc2n(-c3ccc(OC)cc3)c([S-])c(C(=O)Nc3cc(C)cc(C)c3)[n+]2c1	nan
	1744296	48112	22	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	4	6.7	N#Cc1c(-c2ccccc2)cc(-c2ccccc2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	CHEMBL1555056	48112	22	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	4	6.7	N#Cc1c(-c2ccccc2)cc(-c2ccccc2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	15988419	52250	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	2	3	3.5	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Br)cc3)c(=O)[nH]c2C1	nan
	CHEMBL1592108	52250	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	2	3	3.5	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Br)cc3)c(=O)[nH]c2C1	nan
	1863779	71875	15	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	8	2.4	CC1=CC=CN2C(=O)C(=C\c3sc(S)nc3O)/C(=N/CCCN3CCOCC3)N=C12	nan
	CHEMBL1981539	71875	15	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	8	2.4	CC1=CC=CN2C(=O)C(=C\c3sc(S)nc3O)/C(=N/CCCN3CCOCC3)N=C12	nan
	755656	172111	46	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2cccs2)nc2ccc(Br)cc12	nan
	CHEMBL450135	172111	46	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2cccs2)nc2ccc(Br)cc12	nan
	5808	176196	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	CHEMBL1257092	176196	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	CHEMBL460574	176196	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	4905097	26717	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	6	1	5	2.2	CCCC(=O)Nc1ccc2c(c1)nc1n2CCN(CCOC)C1	nan
	CHEMBL1364140	26717	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	6	1	5	2.2	CCCC(=O)Nc1ccc2c(c1)nc1n2CCN(CCOC)C1	nan
	995260	30837	13	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	CHEMBL1399507	30837	13	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	15990423	32025	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	5.3	CCOc1ccccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1409911	32025	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	5.3	CCOc1ccccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	16024826	32697	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccc(F)cc5)CC4)ccc3c2)CC1	nan
	CHEMBL1415463	32697	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccc(F)cc5)CC4)ccc3c2)CC1	nan
	3242125	38683	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	1.7	COc1ccc(OC)c(CNC(=O)C2CCN(C(=O)N(C)C)CC2)c1	nan
	CHEMBL1467628	38683	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	1.7	COc1ccc(OC)c(CNC(=O)C2CCN(C(=O)N(C)C)CC2)c1	nan
	3501359	42500	17	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	8	2.6	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3n(CC3CCCO3)c2=N)cc1	nan
	CHEMBL1501993	42500	17	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	8	2.6	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3n(CC3CCCO3)c2=N)cc1	nan
	1234242	46292	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	6	3.1	CCOc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	CHEMBL1538068	46292	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	6	3.1	CCOc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	20921619	23365	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	2.9	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccc(C)cc3)s2)cc1OC	nan
	CHEMBL1334300	23365	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	2.9	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccc(C)cc3)s2)cc1OC	nan
	16024792	24868	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	CHEMBL1347118	24868	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	5762489	25196	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	1	3	4.6	N#C/C(=C/c1ccc(OCc2ccccc2)cc1)C(=O)NC1CCCCC1	nan
	CHEMBL1349947	25196	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	1	3	4.6	N#C/C(=C/c1ccc(OCc2ccccc2)cc1)C(=O)NC1CCCCC1	nan
	652632	26775	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	0	8	3.7	COc1cccc(C(=O)CSc2nnc(-c3cc(OC)cc(OC)c3)o2)c1	nan
	CHEMBL1364667	26775	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	0	8	3.7	COc1cccc(C(=O)CSc2nnc(-c3cc(OC)cc(OC)c3)o2)c1	nan
	4137748	27207	1	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	1	4	4.0	Cc1cc(NC(=O)c2ccccc2F)nc2c1c(=O)oc1ccccc12	nan
	CHEMBL1368254	27207	1	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	1	4	4.0	Cc1cc(NC(=O)c2ccccc2F)nc2c1c(=O)oc1ccccc12	nan
	701063	28023	17	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.7	COc1ccc(Cl)cc1-c1nnc(S)o1	nan
	CHEMBL1374054	28023	17	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.7	COc1ccc(Cl)cc1-c1nnc(S)o1	nan
	16024750	29011	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1382499	29011	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	1051489	29136	14	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(NC(=O)CSc2nc(-c3ccc(C)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1383601	29136	14	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(NC(=O)CSc2nc(-c3ccc(C)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	2185557	29478	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	0	6	3.7	COc1ccc(C(=O)/C=C2/Sc3cc4c(cc3N2C)OCO4)cc1	nan
	CHEMBL1386474	29478	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	0	6	3.7	COc1ccc(C(=O)/C=C2/Sc3cc4c(cc3N2C)OCO4)cc1	nan
	16017568	30434	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccccc3)s2)c1	nan
	CHEMBL1394623	30434	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccccc3)s2)c1	nan
	16025297	30468	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	582	8	1	8	5.3	COc1cc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc(OC)c1	nan
	CHEMBL1395000	30468	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	582	8	1	8	5.3	COc1cc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc(OC)c1	nan
	2092877	30990	6	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	3.1	CS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4CCCC4=O)cc3)sc2c1	nan
	CHEMBL1400998	30990	6	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	3.1	CS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4CCCC4=O)cc3)sc2c1	nan
	681250	33630	15	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	3	3.7	N#Cc1cc2c(nc1SCc1ccccc1)CCC2	nan
	CHEMBL1423417	33630	15	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	3	3.7	N#Cc1cc2c(nc1SCc1ccccc1)CCC2	nan
	2994363	37301	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	4	2.3	CN1C(=O)c2ccc(C(=O)Nc3ccc(Br)cn3)cc2C1=O	nan
	CHEMBL1456212	37301	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	4	2.3	CN1C(=O)c2ccc(C(=O)Nc3ccc(Br)cn3)cc2C1=O	nan
	54679694	37911	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	8	2	6	3.5	C=CCn1c(=O)c(C(=O)NCCc2ccc(Cl)cc2)c(O)c2cc(OC)c(OC)cc21	nan
	CHEMBL1461466	37911	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	8	2	6	3.5	C=CCn1c(=O)c(C(=O)NCCc2ccc(Cl)cc2)c(O)c2cc(OC)c(OC)cc21	nan
	16814136	38534	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	11	1.1	CCCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1466491	38534	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	11	1.1	CCCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16017049	39436	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	6	4.4	CCC(C(=O)N1CCN(c2ccccc2F)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1475149	39436	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	6	4.4	CCC(C(=O)N1CCN(c2ccccc2F)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	655498	40360	3	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	7	1	5	3.5	CCOc1ccc2cc(C#N)c(SCC(=O)NC(C)CC)nc2c1	nan
	CHEMBL1483885	40360	3	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	7	1	5	3.5	CCOc1ccc2cc(C#N)c(SCC(=O)NC(C)CC)nc2c1	nan
	16019676	40802	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	CHEMBL1487718	40802	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	1305684	40814	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1487797	40814	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	4008999	40904	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	4	6.7	CCCCOc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cc2C)cc1	nan
	CHEMBL1488396	40904	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	4	6.7	CCCCOc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cc2C)cc1	nan
	976779	41285	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	4	1	4	2.5	COc1ccc(S(=O)(=O)Nc2ccccn2)c(C)c1C	nan
	CHEMBL1491184	41285	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	4	1	4	2.5	COc1ccc(S(=O)(=O)Nc2ccccn2)c(C)c1C	nan
	1457998	42225	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	6	2.3	Cc1cc(C)n2c(SCC(=O)NC3CCCCC3)nnc2n1	nan
	CHEMBL1499565	42225	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	6	2.3	Cc1cc(C)n2c(SCC(=O)NC3CCCCC3)nnc2n1	nan
	1555503	43452	19	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	6	3	8	0.6	CCCCOC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1510408	43452	19	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	6	3	8	0.6	CCCCOC(=O)CNc1nnc(S)nc1O	nan
	1484666	43574	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	0	6	4.2	COc1ccc(Oc2nc(SC)nc3ccsc23)cc1	nan
	CHEMBL1511350	43574	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	0	6	4.2	COc1ccc(Oc2nc(SC)nc3ccsc23)cc1	nan
	23760140	44105	1	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	9	5	5	-1.6	CC(=O)N[C@@H](CC(=O)N[C@H](CCC(=O)O)C(=O)O)C(=O)O	nan
	CHEMBL1518212	44105	1	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	9	5	5	-1.6	CC(=O)N[C@@H](CC(=O)N[C@H](CCC(=O)O)C(=O)O)C(=O)O	nan
	4385342	44413	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	7	1	6	3.2	CCOC(=O)c1sc(NC(=O)CCc2ccc(OC)cc2)nc1C	nan
	CHEMBL1520883	44413	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	7	1	6	3.2	CCOC(=O)c1sc(NC(=O)CCc2ccc(OC)cc2)nc1C	nan
	2552702	46320	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.2	O=C(OCc1cc([N+](=O)[O-])cc2c1OCOC2)c1ccccn1	nan
	CHEMBL1538293	46320	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.2	O=C(OCc1cc([N+](=O)[O-])cc2c1OCOC2)c1ccccn1	nan
	16021074	48011	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	1	4	4.3	Cc1cc(C)cc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1553439	48011	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	1	4	4.3	Cc1cc(C)cc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	16034749	48012	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	2	1	4	4.7	CC1Cn2cc(C(=O)Nc3ccccc3C(F)(F)F)c(=O)c3c(Cl)ccc(c32)O1	nan
	CHEMBL1553466	48012	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	2	1	4	4.7	CC1Cn2cc(C(=O)Nc3ccccc3C(F)(F)F)c(=O)c3c(Cl)ccc(c32)O1	nan
	16019427	48035	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	9	5.0	COc1ccccc1Nc1nc2c(S(=O)(=O)c3ccc(C(C)C)cc3)nnn2c2ccsc12	nan
	CHEMBL1553892	48035	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	9	5.0	COc1ccccc1Nc1nc2c(S(=O)(=O)c3ccc(C(C)C)cc3)nnn2c2ccsc12	nan
	16024639	49502	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	5	4.1	CCc1ccc(C(=O)c2cn(CC(=O)NCc3ccc(C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1567298	49502	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	5	4.1	CCc1ccc(C(=O)c2cn(CC(=O)NCc3ccc(C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16017791	50264	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	5	2.6	Cc1cc(C)cc(-n2ccn(CC(=O)c3ccc(F)cc3)c(=O)c2=O)c1	nan
	CHEMBL1574186	50264	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	5	2.6	Cc1cc(C)cc(-n2ccn(CC(=O)c3ccc(F)cc3)c(=O)c2=O)c1	nan
	935556	50989	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	6	1	5	3.7	O=C(O)c1cccc(CSc2nnc(Cc3ccccc3)o2)c1	nan
	CHEMBL1580776	50989	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	6	1	5	3.7	O=C(O)c1cccc(CSc2nnc(Cc3ccccc3)o2)c1	nan
	3441236	52327	3	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.2	O=c1c2ccccc2nc2sc(Nc3ccc(F)cc3)nn12	nan
	CHEMBL1593132	52327	3	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.2	O=c1c2ccccc2nc2sc(Nc3ccc(F)cc3)nn12	nan
	7199916	52513	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	8	3.5	Cc1cc(NC(=O)CSc2ncnc3c2cnn3-c2cccc(Cl)c2)no1	nan
	CHEMBL1595048	52513	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	8	3.5	Cc1cc(NC(=O)CSc2ncnc3c2cnn3-c2cccc(Cl)c2)no1	nan
	865684	53866	12	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	4	4.2	COc1ccccc1Nc1nc2cc(C)ccc2cc1C#N	nan
	CHEMBL1607092	53866	12	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	4	4.2	COc1ccccc1Nc1nc2cc(C)ccc2cc1C#N	nan
	135421676	108564	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	135599408	108564	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	137179849	108564	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	CHEMBL3212907	108564	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	23874512	55094	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1397465	55094	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1619312	55094	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	16019610	10748	10	None	-50	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	4	1	8	5.0	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	CHEMBL1172404	10748	10	None	-50	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	4	1	8	5.0	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	20923126	22900	2	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1C	nan
	CHEMBL1330832	22900	2	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1C	nan
	1425004	23053	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	216	3	3	8	-0.5	COC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1331930	23053	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	216	3	3	8	-0.5	COC(=O)CNc1nnc(S)nc1O	nan
	16024792	24868	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	CHEMBL1347118	24868	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	15989825	25868	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.9	Cc1ccc(CNc2nc3ccc(C)cc3n3nnnc23)cc1	nan
	CHEMBL1355740	25868	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.9	Cc1ccc(CNc2nc3ccc(C)cc3n3nnnc23)cc1	nan
	930238	26546	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	1	5	4.1	CC(C)c1nc2sc3c(S)ncnc3c2c2c1CCC2	nan
	CHEMBL1362595	26546	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	1	5	4.1	CC(C)c1nc2sc3c(S)ncnc3c2c2c1CCC2	nan
	15988284	27457	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccccc3)nnc12	nan
	CHEMBL1370040	27457	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccccc3)nnc12	nan
	7245805	30614	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	1.8	Cc1ccc(CNC(=O)Cn2ccn(-c3ccc(F)cc3)c(=O)c2=O)cc1	nan
	CHEMBL1396990	30614	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	1.8	Cc1ccc(CNC(=O)Cn2ccn(-c3ccc(F)cc3)c(=O)c2=O)cc1	nan
	16025341	30717	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	8	1	6	5.0	O=C(CSc1ncc2c(n1)-c1cc(Cl)ccc1N(Cc1ccccc1)S2(=O)=O)NCCc1ccccc1	nan
	CHEMBL1398424	30717	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	8	1	6	5.0	O=C(CSc1ncc2c(n1)-c1cc(Cl)ccc1N(Cc1ccccc1)S2(=O)=O)NCCc1ccccc1	nan
	995260	30837	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	CHEMBL1399507	30837	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	3243282	34417	2	None	2	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	1	4	4.3	CCCCn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	CHEMBL1429998	34417	2	None	2	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	1	4	4.3	CCCCn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	1007107	35525	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	3	1	4	5.8	Cc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	CHEMBL1441054	35525	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	3	1	4	5.8	Cc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	16800714	38716	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	9	0.4	CCCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1468004	38716	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	9	0.4	CCCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	814519	39180	24	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	201	0	2	3	2.4	Sc1[nH]cnc2c3ccccc3nc1-2	nan
	CHEMBL1471924	39180	24	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	201	0	2	3	2.4	Sc1[nH]cnc2c3ccccc3nc1-2	nan
	44142305	39394	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	5	3.1	Cn1cncc1C#Cc1ccc2cc(C3(O)CCCCC3)oc(=O)c2c1	nan
	CHEMBL1474528	39394	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	5	3.1	Cn1cncc1C#Cc1ccc2cc(C3(O)CCCCC3)oc(=O)c2c1	nan
	2138538	48604	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1ccc(CCNc2nc3c(-c4cccc(C)c4)nnn3c3ccccc23)cc1OC	nan
	CHEMBL1559550	48604	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1ccc(CCNc2nc3c(-c4cccc(C)c4)nnn3c3ccccc23)cc1OC	nan
	16028162	49136	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3ccc(F)cc3)cc21	nan
	CHEMBL1564507	49136	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3ccc(F)cc3)cc21	nan
	7720817	51073	0	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	1	5	2.9	Sc1nncn2c1cc1oc3ccccc3c12	nan
	CHEMBL1581464	51073	0	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	1	5	2.9	Sc1nncn2c1cc1oc3ccccc3c12	nan
	1909591	51805	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	3.4	Oc1c2nc3ccc(Br)cc3c-2ncn1Cc1ccncc1	nan
	CHEMBL1587545	51805	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	3.4	Oc1c2nc3ccc(Br)cc3c-2ncn1Cc1ccncc1	nan
	15988964	52218	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCCN(C)CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1591653	52218	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCCN(C)CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	44143234	52366	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	16	3	12	2.5	CCCC[N+](CCCC)(CCCC)CCCC.Nc1ncnc2c1ncn2[C@@H]1O[C@H](COS(=O)(=O)[O-])[C@@H](O)[C@H]1O	nan
	CHEMBL1593759	52366	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	16	3	12	2.5	CCCC[N+](CCCC)(CCCC)CCCC.Nc1ncnc2c1ncn2[C@@H]1O[C@H](COS(=O)(=O)[O-])[C@@H](O)[C@H]1O	nan
	660350	55141	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	CHEMBL1413816	55141	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	CHEMBL1619747	55141	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	24892704	71437	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	0	8	2.4	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1967784	71437	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	0	8	2.4	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2cc(C(=O)OC)ccc21	nan
	2815701	104957	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	4	2.6	Cc1ccc(S(=O)(=O)NC(=O)Nc2ccc(N(C)C)cc2)cc1	nan
	CHEMBL312032	104957	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	4	2.6	Cc1ccc(S(=O)(=O)NC(=O)Nc2ccc(N(C)C)cc2)cc1	nan
	664514	46194	11	None	3	2	Human	6.1	pPotency	=	6.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	0	7	3.0	CCOC(=O)CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1537230	46194	11	None	3	2	Human	6.1	pPotency	=	6.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	0	7	3.0	CCOC(=O)CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	4679126	22449	14	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	9	4.3	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1327057	22449	14	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	9	4.3	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	16030531	23897	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	4	4.9	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	CHEMBL1338691	23897	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	4	4.9	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	1371049	24176	11	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	3.6	COc1ccc(Cl)cc1C(=O)Nc1nc2ccc(S(C)(=O)=O)cc2s1	nan
	CHEMBL1341278	24176	11	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	3.6	COc1ccc(Cl)cc1C(=O)Nc1nc2ccc(S(C)(=O)=O)cc2s1	nan
	3236027	24893	10	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	7	3.9	COc1ccc(N2CCN(c3ccc(NC(=O)c4ccc5c(c4)OCO5)cc3C#N)CC2)cc1	nan
	CHEMBL1347313	24893	10	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	7	3.9	COc1ccc(N2CCN(c3ccc(NC(=O)c4ccc5c(c4)OCO5)cc3C#N)CC2)cc1	nan
	1208330	25104	16	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	0	5	4.6	CCN(CC)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	CHEMBL1349151	25104	16	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	0	5	4.6	CCN(CC)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	3414203	25987	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	5	2.9	Cn1/c(=N\C(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)sc2cc(F)ccc21	nan
	CHEMBL1357194	25987	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	5	2.9	Cn1/c(=N\C(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)sc2cc(F)ccc21	nan
	1920995	26649	8	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	3	4.1	Cc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1363550	26649	8	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	3	4.1	Cc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	15988900	27996	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	7	5.1	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Br)cc3)on2)sc(C(C)=O)c1C	nan
	CHEMBL1373810	27996	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	7	5.1	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Br)cc3)on2)sc(C(C)=O)c1C	nan
	1450216	29859	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	4.2	Cc1ccc(C)c2nc(SCC(=O)NCc3cccs3)c(C#N)cc12	nan
	CHEMBL1389491	29859	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	4.2	Cc1ccc(C)c2nc(SCC(=O)NCc3cccs3)c(C#N)cc12	nan
	3330912	30528	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	5	5.9	CCOc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1395727	30528	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	5	5.9	CCOc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	16033852	30879	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	6	4.1	O=c1c2ccccc2nc2sc(Nc3cccc(C(F)(F)F)c3)nn12	nan
	CHEMBL1399988	30879	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	6	4.1	O=c1c2ccccc2nc2sc(Nc3cccc(C(F)(F)F)c3)nn12	nan
	20923127	30901	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCC(C)C1	nan
	CHEMBL1400119	30901	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCC(C)C1	nan
	692203	31383	16	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	5	4.5	O=C(Oc1ccccc1)Oc1ccc2c(c1)oc(=O)c1ccccc12	nan
	CHEMBL1404472	31383	16	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	5	4.5	O=C(Oc1ccccc1)Oc1ccc2c(c1)oc(=O)c1ccccc12	nan
	16745677	31813	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	9	0	9	6.0	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1408237	31813	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	9	0	9	6.0	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1Cc1ccc2c(c1)OCO2	nan
	16010801	34867	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	3.1	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1OC	nan
	CHEMBL1433929	34867	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	3.1	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1OC	nan
	4107570	39541	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	4	4.8	COc1ccc2c(c1)-c1nc(NC(=O)c3ccc(Cl)cc3)sc1CC2	nan
	CHEMBL1476611	39541	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	4	4.8	COc1ccc2c(c1)-c1nc(NC(=O)c3ccc(Cl)cc3)sc1CC2	nan
	16009524	39567	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	7	4.3	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1C	nan
	CHEMBL1476936	39567	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	7	4.3	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1C	nan
	7184626	40374	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	3.0	CCOc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1484029	40374	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	3.0	CCOc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4423184	43907	11	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	8	2.6	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1516075	43907	11	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	8	2.6	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(C(=O)OC)ccc21	nan
	2946893	44251	12	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	1	7	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	CHEMBL1519514	44251	12	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	1	7	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	2808378	10274	26	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	2.9	CC(=O)c1sccc1NC(=O)c1ccccc1C(=O)O	nan
	CHEMBL1162443	10274	26	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	2.9	CC(=O)c1sccc1NC(=O)c1ccccc1C(=O)O	nan
	2085722	22235	2	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	7	1.6	CCCNC(=O)COC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1324965	22235	2	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	7	1.6	CCCNC(=O)COC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	2918454	23836	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	4.1	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(F)cc2)nc1C	nan
	CHEMBL1338266	23836	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	4.1	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(F)cc2)nc1C	nan
	4902571	24023	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	8	4.3	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(C)cc2)s1	nan
	CHEMBL1339921	24023	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	8	4.3	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(C)cc2)s1	nan
	15990443	25945	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	5.8	COc1cc(Cl)c(C)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1356755	25945	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	5.8	COc1cc(Cl)c(C)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3442498	26959	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	1	8	1.9	Cc1nnc(NC(=O)CSc2ccc([N+](=O)[O-])cn2)s1	nan
	CHEMBL1366225	26959	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	1	8	1.9	Cc1nnc(NC(=O)CSc2ccc([N+](=O)[O-])cn2)s1	nan
	18561048	28209	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1375333	28209	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	5098091	29500	3	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	4	5.6	COc1ccc(-c2sc(C(=O)c3ccc(Cl)cc3Cl)cc2CC(=O)O)cc1	nan
	CHEMBL1386663	29500	3	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	4	5.6	COc1ccc(-c2sc(C(=O)c3ccc(Cl)cc3Cl)cc2CC(=O)O)cc1	nan
	1112430	36194	18	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	6	3.3	CCOC(=O)c1cccc(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	CHEMBL1447146	36194	18	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	6	3.3	CCOC(=O)c1cccc(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	734580	36796	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	3	1	4	2.2	CC(=O)c1sc(NC(=O)C(C)C)nc1C	nan
	CHEMBL1451957	36796	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	3	1	4	2.2	CC(=O)c1sc(NC(=O)C(C)C)nc1C	nan
	18561036	37577	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1458644	37577	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	16195440	38259	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.7	CCn1c(=O)c2cc(C(=O)Nc3cccc(C(C)=O)c3)sc2c2ccccc21	nan
	CHEMBL1464378	38259	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.7	CCn1c(=O)c2cc(C(=O)Nc3cccc(C(C)=O)c3)sc2c2ccccc21	nan
	16008699	39357	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	9	2.5	CCOc1ccc(-c2nc(C(N)=O)c3c(n2)n(-c2ccc4c(c2)OCO4)c(=O)n3CC)cc1	nan
	CHEMBL1474027	39357	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	9	2.5	CCOc1ccc(-c2nc(C(N)=O)c3c(n2)n(-c2ccc4c(c2)OCO4)c(=O)n3CC)cc1	nan
	2746740	41543	5	None	2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	2	6	5.5	O=C(Nc1ccc(Cl)cc1)Nc1ccccc1Sc1ncc([N+](=O)[O-])s1	nan
	CHEMBL1493199	41543	5	None	2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	2	6	5.5	O=C(Nc1ccc(Cl)cc1)Nc1ccccc1Sc1ncc([N+](=O)[O-])s1	nan
	17469833	42651	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	6	3.0	COc1ccccc1NC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	CHEMBL1503328	42651	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	6	3.0	COc1ccccc1NC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	17581208	42829	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1ccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)cc1	nan
	CHEMBL1505004	42829	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1ccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)cc1	nan
	3207506	43086	4	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1ccc2nc(SCC(=O)NCc3cccs3)c(C#N)cc2c1	nan
	CHEMBL1507076	43086	4	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1ccc2nc(SCC(=O)NCc3cccs3)c(C#N)cc2c1	nan
	16018870	44336	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	4	0	7	6.2	Cc1oc(-c2ccc(Cl)cc2)nc1CSc1nnc(C)n2c1cc1sccc12	nan
	CHEMBL1520274	44336	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	4	0	7	6.2	Cc1oc(-c2ccc(Cl)cc2)nc1CSc1nnc(C)n2c1cc1sccc12	nan
	1130973	46611	6	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.1	Cc1ccccc1OCC(=O)Nc1sc(C(=O)Nc2cccc(C)c2C)c(C)c1C#N	nan
	CHEMBL1540811	46611	6	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.1	Cc1ccccc1OCC(=O)Nc1sc(C(=O)Nc2cccc(C)c2C)c(C)c1C#N	nan
	724891	47036	26	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	5	3.5	O=C(O)CSc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1544233	47036	26	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	5	3.5	O=C(O)CSc1ncnc2scc(-c3ccccc3)c12	nan
	1004390	47557	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	5	4.1	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3ccccc3)n2)c1	nan
	CHEMBL1548754	47557	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	5	4.1	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3ccccc3)n2)c1	nan
	1450522	48499	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	3.2	COc1ccc2cc(C#N)c(SCC(=O)N3CC(=O)Nc4ccccc43)nc2c1	nan
	CHEMBL1558667	48499	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	3.2	COc1ccc2cc(C#N)c(SCC(=O)N3CC(=O)Nc4ccccc43)nc2c1	nan
	16021094	48840	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	4.3	CCc1cccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1561841	48840	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	4.3	CCc1cccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	4585955	50275	6	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	6	1	9	4.4	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)CC1	nan
	CHEMBL1574238	50275	6	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	6	1	9	4.4	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)CC1	nan
	16025788	52088	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	4	5.7	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4c(C)cc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1590035	52088	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	4	5.7	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4c(C)cc5ccccc54)s3)CC2)cc1	nan
	7184644	52192	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	2	8	0.2	CC(=O)NCCNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1591356	52192	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	2	8	0.2	CC(=O)NCCNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	16010575	52261	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	3.2	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c(C)c1	nan
	CHEMBL1592228	52261	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	3.2	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c(C)c1	nan
	101430	95973	18	None	-1949	5	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	4	9	0.2	OC[C@H]1O[C@@H](n2cnc3c(Nc4ccccc4)ncnc32)[C@H](O)[C@@H]1O	nan
	CHEMBL262083	95973	18	None	-1949	5	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	4	9	0.2	OC[C@H]1O[C@@H](n2cnc3c(Nc4ccccc4)ncnc32)[C@H](O)[C@@H]1O	nan
	12501	3386	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Determined in a cell-based cAMP assay.Determined in a cell-based cAMP assay.	Guide to Pharmacology		None	None	None		None	33555858
	12501	3386	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Determined in a cell-based cAMP assay.Determined in a cell-based cAMP assay.	Guide to Pharmacology		None	None	None		None	36443381
	1989	3241	0	None	17	3	Human	10.4	pEC50	=	10.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	18434306
	56593349	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	56593349	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	56593349	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	8322	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	8322	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	8322	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	CHEMBL3716980	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	CHEMBL3716980	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	CHEMBL3716980	2524	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	11898	1096	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	33555858
	8346	200	0	None	165	2	Human	8.2	pEC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21878627
	11462	3679	0	None	-	1	Human	9.1	pEC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	30594862
	134813895	201	0	None	-	1	Human	9.8	pEC50	=	9.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	8349	201	0	None	-	1	Human	9.8	pEC50	=	9.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	1988	3242	0	None	-	1	Human	8.8	pEC50	None	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	16411781
	4371	706	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20043231
	4371	706	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	24812057

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	162654489	180043	0	None	-	1	Rat	9.3	pEC50	=	9.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180043	0	None	-	1	Rat	9.3	pEC50	=	9.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162672610	182424	0	None	-	0	Rat	9.1	pEC50	=	9.1	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182424	0	None	-	0	Rat	9.1	pEC50	=	9.1	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162664297	181489	0	None	-	0	Rat	8.3	pEC50	=	8.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781560	181489	0	None	-	0	Rat	8.3	pEC50	=	8.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654489	180043	0	None	-	1	Human	9.0	pKi	=	9.0	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180043	0	None	-	1	Human	9.0	pKi	=	9.0	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162662592	181377	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4780098	181377	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	12502	2376	0	None	24	2	Human	10.1	pKd	=	10.1	Binding	Binding affinity determined by SPR.Binding affinity determined by SPR.	Guide to Pharmacology		None	None	None		None	36780899
	12502	2376	0	None	-24	2	Mouse	8.7	pKd	=	8.7	Binding	Binding affinity determined by SPR.Binding affinity determined by SPR.	Guide to Pharmacology		None	None	None		None	36780899
	8346	200	0	None	9	2	Human	7.0	pKd	=	7.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21878627
	3874	1567	0	None	-	1	Human	9.0	pKd	=	9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19343240
	3874	1567	0	None	-	1	Human	9.3	pKd	=	9.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	22425984
	1993	3240	0	None	-	1	Human	7.3	pKd	None	7.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1992	3238	0	None	15	2	Human	9.1	pKd	None	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1994	3239	0	None	39	2	Human	9.4	pKd	None	9.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	9321	558	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	30155023
	9321	558	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	32295457
	4371	706	0	None	-	1	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20043231
	4371	706	0	None	-	1	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	24812057
	1995	2005	0	None	-16982	2	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23303914
	134813895	201	0	None	-	1	Human	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	8349	201	0	None	-	1	Human	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	1989	3241	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	12506116
	1989	3241	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1989	3241	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	18434306
	1990	3244	0	None	-14	4	Human	7.8	pKi	None	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	12506116
	1990	3244	0	None	-14	4	Human	7.8	pKi	None	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866

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Main reference

Ligand source activities (1 row/activity)