Ligand source activities (1 row/activity)



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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Potency)		 # tested GPCRs
(Potency)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI
11337 2872 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.
Guide to Pharmacology 440 4 0 4 3.9 O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1 31127149
124085867 2872 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.
Guide to Pharmacology 440 4 0 4 3.9 O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1 31127149
5312830 187 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
5567 187 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
CHEMBL1230670 187 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
DB07302 187 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715


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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Affinity)		 # tested GPCRs
(Affinity)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI