Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
grpr_mouse 3.50x50 139 TM3 R => G N/A N/A Benya RV et al (1995)
grpr_mouse 6.34x34 264 TM6 A => E N/A N/A Benya RV et al (1995)
grpr_mouse 3.50x50 139 TM3 R => G N/A N/A Benya RV et al (1994)
grpr_mouse 6.34x34 264 TM6 A => E N/A N/A Benya RV et al (1994)
grpr_mouse 6.58x58 288 TM6 R => H N/A N/A Akeson M et al (1997)
grpr_mouse 3.32x32 121 TM3 Q => R N/A N/A Akeson M et al (1997)
grpr_mouse 2.63x62 100 TM2 S => T N/A N/A Akeson M et al (1997)
grpr_mouse 105 ECL1 D => E N/A N/A Akeson M et al (1997)
grpr_mouse 3.28x28 117 TM3 I => L N/A N/A Akeson M et al (1997)
grpr_mouse 4.56x56 172 TM4 L => F N/A N/A Akeson M et al (1997)
grpr_mouse 292 ECL3 Y => S N/A N/A Akeson M et al (1997)
grpr_mouse 45.52x52 199 ECL2 P => S N/A N/A Akeson M et al (1997)
grpr_mouse 7.38x37 308 TM7 A => S N/A N/A Akeson M et al (1997)
grpr_mouse 4.64x65 180 TM4 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 181 ECL2 D => A N/A N/A Lin Y et al (2000)
grpr_mouse 5.39x40 212 TM5 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 5.42x43 215 TM5 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 5.43x44 216 TM5 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.40x40 270 TM6 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.48x48 278 TM6 W => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.51x51 281 TM6 N => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.55x55 285 TM6 Y => A N/A N/A Lin Y et al (2000)
grpr_mouse 7.43x42 313 TM7 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 5 N-term N => Q N/A N/A Benya RV et al (2000)
grpr_mouse 20 N-term N => Q N/A N/A Benya RV et al (2000)
grpr_mouse 24 N-term N => Q N/A N/A Benya RV et al (2000)
grpr_mouse 2.61x60 98 TM2 D => A N/A N/A Donohue PJ et al (1999)
grpr_mouse 2.61x60 98 TM2 D => R N/A N/A Donohue PJ et al (1999)
grpr_mouse 2.63x62 100 TM2 S => T N/A N/A Akeson M et al (1997)
grpr_mouse 105 ECL1 D => E N/A N/A Akeson M et al (1997)
grpr_mouse 3.28x28 117 TM3 I => L N/A N/A Akeson M et al (1997)
grpr_mouse 3.32x32 121 TM3 Q => R N/A N/A Akeson M et al (1997)
grpr_mouse 3.50x50 139 TM3 R => G N/A N/A Benya RV et al (1995)
grpr_mouse 4.56x56 172 TM4 L => F N/A N/A Akeson M et al (1997)
grpr_mouse 4.64x65 180 TM4 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 181 ECL2 D => A N/A N/A Lin Y et al (2000)
grpr_mouse 182 ECL2 L => V N/A N/A Tokita K et al (2002)
grpr_mouse 183 ECL2 H => A N/A N/A Tokita K et al (2002)
grpr_mouse 184 ECL2 P => R N/A N/A Tokita K et al (2002)
grpr_mouse 185 ECL2 F => I N/A N/A Tokita K et al (2002)
grpr_mouse 191 ECL2 N => E N/A N/A Benya RV et al (2000)
grpr_mouse 191 ECL2 N => Q N/A N/A Benya RV et al (2000)
grpr_mouse 45.51x51 198 ECL2 A => I N/A N/A Tokita K et al (2002)
grpr_mouse 45.52x52 199 ECL2 P => S N/A N/A Akeson M et al (1997)
grpr_mouse 5.39x40 212 TM5 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 5.42x43 215 TM5 S => A N/A N/A Lin Y et al (2000)
grpr_mouse 5.43x44 216 TM5 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.40x40 270 TM6 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.48x48 278 TM6 W => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.51x51 281 TM6 N => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.55x55 285 TM6 Y => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.58x58 288 TM6 R => H N/A N/A Akeson M et al (1997)
grpr_mouse 292 ECL3 Y => S N/A N/A Akeson M et al (1997)
grpr_mouse 293 ECL3 S => K N/A N/A Tokita K et al (2001)
grpr_mouse 295 ECL3 V => I N/A N/A Tokita K et al (2001)
grpr_mouse 297 ECL3 T => P N/A N/A Tokita K et al (2001)
grpr_mouse 7.32x31 302 TM7 F => M N/A N/A Tokita K et al (2001)
grpr_mouse 7.33x32 303 TM7 V => I N/A N/A Tokita K et al (2001)
grpr_mouse 7.34x33 304 TM7 T => V N/A N/A Tokita K et al (2001)
grpr_mouse 7.35x34 305 TM7 S => T N/A N/A Tokita K et al (2001)
grpr_mouse 7.38x37 308 TM7 A => S N/A N/A Akeson M et al (1997)
grpr_mouse 7.39x38 309 TM7 R => A N/A N/A Donohue PJ et al (1999)
grpr_mouse 7.39x38 309 TM7 R => D N/A N/A Donohue PJ et al (1999)
grpr_mouse 7.43x42 313 TM7 F => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.51x51 281 TM6 N => A N/A N/A Lin Y et al (2000)
grpr_mouse 6.51x51 281 TM6 N => A N/A N/A Lin Y et al (2000)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 K S M R ICL1ECL1 D R W L F ECL1ICL2 P M D I Q A S H ICL2ECL2 D L H P F H V K D T N Q T F I S C A P Y P H S ECL2ICL3 P V E G ICL3ECL3 Y S E V D T ECL3N-term M A P N N C S H L N L D V D P F L S C N D T F N Q S L S P P K M D N W F H N-termC-term C Q P G L M N R S H S T G R S T T C M T S F K S T N P S A T F S L I N R N I C H E G Y V C-term P G F I Y V I P A V Y G L I I V I G L I G N I T L I K I F C T V N V P N L F I S S L A L G D L L L L V T C A P V D A S K Y L A G R I G C K L I P F I Q L T S V G V S V F T L T A L S A D R Y K A I V R A L M K I C L K A A L I W I V S M L L A I P E A V F S N E L H P K I H S M A S F L V F Y V I P L A I I S V Y Y Y F I A R N L I Q S A Y N L N I H V K K Q I E S R K R L A K T V L V F V G L F A F C W L P N H V I Y L Y R S Y H S M L H F V T S I C A R L L A F T N S C V N P F A L Y L L S K S F N T F R K Q Q L L C
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
I N G I L G I V I I L G Y V A P I V Y I 1 S S L A L G D L L L L T V C A P V D A S K 2 A T L T F V S V G V S T L Q I F P I L K 3 I C L K A A L I W I V S M L L A I P E 4 Y Y V S I I A L P I V Y F V L F S A M S H 5 L V F V G L F A F C W L P N H V I Y L Y 6 F P N V C S N T F A L L R A C I S T V 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
BB2 receptor
TM2
2x60 2.61x60 D98
2x62 2.63x62 S100
TM3
3x28 3.28x28 I117
3x32 3.32x32 Q121
3x50 3.50x50 R139
TM4
4x56 4.56x56 L172
4x65 4.64x65 S180
TM5
5x40 5.39x40 S212
5x43 5.42x43 S215
5x44 5.43x44 F216
TM6
6x34 6.34x34 A264
6x40 6.40x40 F270
6x48 6.48x48 W278
6x51 6.51x51 N281
6x55 6.55x55 Y285
6x58 6.58x58 R288
TM7
7x31 7.32x31 F302
7x32 7.33x32 V303
7x33 7.34x33 T304
7x34 7.35x34 S305
7x37 7.38x37 A308
7x38 7.39x38 R309
7x42 7.43x42 F313